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Tyrosine Kinase/Adaptors
Subcategories of "Tyrosine Kinase/Adaptors"
ALK
c-Fms
c-Kit
c-Met/HGFR
c-RET
CSF-1R
EGFR
Ephrin Receptor
Fibroblast Growth Factor Receptor (FGFR)
FLT
Hck
HER
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
Show 15 more subcategories
Products of "Tyrosine Kinase/Adaptors"
Tyrphostin AG528
CAS:133550-49-9
Formula:
C18H14N2O3
Purity:
>97.0%(HPLC)
Color and Shape:
Light yellow to Amber to Dark green powder to crystal
Molecular weight:
306.32
Estimated delivery in United States, on Thursday 27 Jan 2022
SB 431542
CAS:301836-41-9
Formula:
C22H16N4O3
Purity:
>97.0%(HPLC)
Color and Shape:
White to Orange to Green powder to crystal
Molecular weight:
384.40
Estimated delivery in United States, on Thursday 27 Jan 2022
AEE 788
CAS:497839-62-0
Formula:
C27H32N6
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
440.60
Estimated delivery in United States, on Thursday 27 Jan 2022
Afatinib
CAS:850140-72-6
Formula:
C24H25ClFN5O3
Purity:
>97.0%(HPLC)(N)
Color and Shape:
White to Orange to Green powder to crystal
Molecular weight:
485.94
Estimated delivery in United States, on Thursday 27 Jan 2022
PD 173074
CAS:219580-11-7
Formula:
C28H41N7O3
Purity:
>95.0%(HPLC)
Color and Shape:
White to Yellow to Orange powder to crystal
Molecular weight:
523.68
Estimated delivery in United States, on Thursday 27 Jan 2022
Methyl 2,5-Dihydroxycinnamate
CAS:63177-57-1
Formula:
C10H10O4
Purity:
>96.0%(HPLC)
Color and Shape:
Very Pale Yellow - Yellow Solid
Molecular weight:
194.19
Estimated delivery in United States, on Thursday 27 Jan 2022
Genistein
CAS:446-72-0
Formula:
C15H10O5
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
270.24
Estimated delivery in United States, on Thursday 27 Jan 2022
SU 1498
CAS:168835-82-3
Formula:
C25H30N2O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Orange to Green powder to crystal
Molecular weight:
390.53
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin A1
CAS:2826-26-8
Formula:
C11H8N2O
Purity:
>98.0%(GC)
Color and Shape:
Light orange to Yellow to Green powder to crystal
Molecular weight:
184.20
Estimated delivery in United States, on Thursday 27 Jan 2022
Mubritinib
CAS:366017-09-6
Formula:
C25H23F3N4O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Gray to Brown powder to crystal
Molecular weight:
468.48
Estimated delivery in United States, on Thursday 27 Jan 2022
CL-387785
CAS:194423-06-8
Formula:
C18H13BrN4O
Purity:
>98.0%(GC)
Color and Shape:
White to Orange to Green powder to crystal
Molecular weight:
381.23
Estimated delivery in United States, on Thursday 27 Jan 2022
PD 158780
CAS:171179-06-9
Formula:
C14H12BrN5
Purity:
>97.0%(HPLC)
Color and Shape:
White to Yellow to Green powder to crystal
Molecular weight:
330.19
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin RG 13022
CAS:136831-48-6
Formula:
C16H14N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Yellow to Green powder to crystal
Molecular weight:
266.30
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin AG 494
CAS:133550-35-3
Formula:
C16H12N2O3
Purity:
>98.0%(HPLC)(N)
Color and Shape:
Light yellow to Amber to Dark green powder to crystal
Molecular weight:
280.28
Estimated delivery in United States, on Thursday 27 Jan 2022
SKLB1002
CAS:1225451-84-2
Formula:
C13H12N4O2S2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
320.39
Estimated delivery in United States, on Thursday 27 Jan 2022
Dacomitinib
CAS:1110813-31-4
Formula:
C24H25ClFN5O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
469.95
Estimated delivery in United States, on Thursday 27 Jan 2022
PQ401
CAS:196868-63-0
Formula:
C18H16ClN3O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Yellow to Orange powder to crystal
Molecular weight:
341.80
Estimated delivery in United States, on Thursday 27 Jan 2022
PP 2
CAS:172889-27-9
Formula:
C15H16ClN5
Purity:
>97.0%(HPLC)(T)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
301.78
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin A9
CAS:10537-47-0
Formula:
C18H22N2O
Purity:
>98.0%(GC)
Color and Shape:
Light orange to Yellow to Green powder to crystal
Molecular weight:
282.39
Estimated delivery in United States, on Thursday 27 Jan 2022
MNS
CAS:1485-00-3
Formula:
C9H7NO4
Purity:
>98.0%(GC)
Color and Shape:
Light yellow to Yellow to Green powder to crystal
Molecular weight:
193.16
Estimated delivery in United States, on Thursday 27 Jan 2022
Gefitinib
CAS:184475-35-2
Formula:
C22H24ClFN4O3
Purity:
>98.0%(HPLC)(T)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
446.91
Estimated delivery in United States, on Thursday 27 Jan 2022
Piceatannol
CAS:10083-24-6
Formula:
C14H12O4
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light red powder to crystal
Molecular weight:
244.25
Estimated delivery in United States, on Thursday 27 Jan 2022
Imatinib Mesylate
CAS:220127-57-1
Formula:
C29H31N7OCH4O3S
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
589.72
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin AG 835
CAS:133550-37-5
Formula:
C18H16N2O3
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Amber to Dark green powder to crystal
Molecular weight:
308.34
Estimated delivery in United States, on Thursday 27 Jan 2022
LFM-A13
CAS:62004-35-7
Formula:
C11H8Br2N2O2
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
360.01
Estimated delivery in United States, on Thursday 27 Jan 2022
Butein
CAS:487-52-5
Formula:
C15H12O5
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
272.26
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin AG 1478
CAS:153436-53-4
Formula:
C16H14ClN3O2
Purity:
>98.0%(HPLC)
Color and Shape:
Light orange to Yellow to Green powder to crystal
Molecular weight:
315.76
Estimated delivery in United States, on Thursday 27 Jan 2022
Daphnetin
CAS:486-35-1
Formula:
C9H6O4
Purity:
>90.0%(HPLC)
Color and Shape:
White to Light yellow to Light red powder to crystal
Molecular weight:
178.14
Estimated delivery in United States, on Thursday 27 Jan 2022
Regorafenib
CAS:755037-03-7
Formula:
C21H15ClF4N4O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
482.82
Estimated delivery in United States, on Thursday 27 Jan 2022
JK-P3
CAS:942655-44-9
Formula:
C18H17N3O3
Purity:
>98.0%(HPLC)(T)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
323.35
Estimated delivery in United States, on Thursday 27 Jan 2022
Curcumin (Natural)
CAS:458-37-7
Formula:
C21H20O6
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
368.39
Estimated delivery in United States, on Thursday 27 Jan 2022
AG-1296
CAS:146535-11-7
Formula:
C16H14N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Orange to Green powder to crystal
Molecular weight:
266.30
Estimated delivery in United States, on Thursday 27 Jan 2022
PD-161570
CAS:192705-80-9
Formula:
C26H35Cl2N7O
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
532.51
Estimated delivery in United States, on Thursday 27 Jan 2022
Lapatinib
CAS:231277-92-2
Formula:
C29H26ClFN4O4S
Purity:
>98.0%(HPLC)(T)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
581.06
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin RG 14620
CAS:136831-49-7
Formula:
C14H8Cl2N2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
275.13
Estimated delivery in United States, on Thursday 27 Jan 2022
BMS-599626
CAS:714971-09-2
Formula:
C27H27FN8O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
530.56
Estimated delivery in United States, on Thursday 27 Jan 2022
SB-505124
CAS:694433-59-5
Formula:
C20H21N3O2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystaline
Molecular weight:
335.41
Estimated delivery in United States, on Thursday 27 Jan 2022
Pelitinib
CAS:257933-82-7
Formula:
C24H23ClFN5O2
Purity:
>97.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
467.93
Estimated delivery in United States, on Thursday 27 Jan 2022
RPI 1
CAS:269730-03-2
Formula:
C17H15NO4
Purity:
>95.0%(HPLC)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
297.31
Estimated delivery in United States, on Thursday 27 Jan 2022
Curcumin (Synthetic)
CAS:458-37-7
Formula:
C21H20O6
Purity:
>97.0%(T)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
368.39
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin A23
CAS:118409-57-7
Formula:
C10H6N2O2
Purity:
>98.0%(GC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
186.17
Estimated delivery in United States, on Thursday 27 Jan 2022
WHI-P154
CAS:211555-04-3
Formula:
C16H14BrN3O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Yellow to Orange powder to crystal
Molecular weight:
376.21
Estimated delivery in United States, on Thursday 27 Jan 2022
Imatinib
CAS:152459-95-5
Formula:
C29H31N7O
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
493.62
Estimated delivery in United States, on Thursday 27 Jan 2022
NVP-BHG 712
CAS:940310-85-0
Formula:
C26H20F3N7O
Purity:
>95.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
503.49
Estimated delivery in United States, on Thursday 27 Jan 2022
TCS 359
CAS:301305-73-7
Formula:
C18H20N2O4S
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Brown powder to crystal
Molecular weight:
360.43
Estimated delivery in United States, on Thursday 27 Jan 2022
SB-525334
CAS:356559-20-1
Formula:
C21H21N5
Purity:
>98.0%(HPLC)
Color and Shape:
White to Yellow to Orange powder to crystal
Molecular weight:
343.43
Estimated delivery in United States, on Thursday 27 Jan 2022
GW 2580
CAS:870483-87-7
Formula:
C20H22N4O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
366.42
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin AG 879
CAS:148741-30-4
Formula:
C18H24N2OS
Purity:
>98.0%(HPLC)
Color and Shape:
Light yellow to Yellow to Orange powder to crystal
Molecular weight:
316.46
Estimated delivery in United States, on Thursday 27 Jan 2022
Pazopanib Hydrochloride
CAS:635702-64-6
Formula:
C21H23N7O2SHCl
Purity:
>95.0%(HPLC)(T)
Color and Shape:
White to Almost white powder to crystal
Molecular weight:
473.98
Estimated delivery in United States, on Thursday 27 Jan 2022
PD 153035 Hydrochloride
CAS:183322-45-4
Formula:
C16H14BrN3O2HCl
Purity:
>97.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
396.67
Estimated delivery in United States, on Thursday 27 Jan 2022
Tyrphostin AG 490
CAS:133550-30-8
Formula:
C17H14N2O3
Purity:
>98.0%(HPLC)(T)
Color and Shape:
Slightly Pale Yellow - Yellow Solid
Molecular weight:
294.31
Estimated delivery in United States, on Thursday 27 Jan 2022
KX1004
CAS:518058-84-9
KX1-004, a potential protective drug for NIHL, is an effective small molecule inhibitor of Src-PTK.
Formula:
C16H13FN2O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
284.29
Estimated delivery in United States, on Monday 7 Feb 2022
Icotinib Hydrochloride
CAS:1204313-51-8
Icotinib Hydrochloride is the hydrochloride salt form of icotinib, an orally available quinazoline-based inhibitor of …
Formula:
C22H22ClN3O4
Molecular weight:
427.88
Estimated delivery in United States, on Monday 7 Feb 2022
BMS536924
CAS:468740-43-4
BMS-536924 is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for …
Formula:
C25H26ClN5O3
Purity:
99.19%
Color and Shape:
solid
Molecular weight:
479.96
Estimated delivery in United States, on Monday 7 Feb 2022
Dacomitinib
CAS:1110813-31-4
Dacomitinib(PF299804; PF-00299804) is a highly selective, orally bioavailable small-molecule inhibitor of the HER family of …
Formula:
C24H25ClFN5O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
469.94
Estimated delivery in United States, on Monday 7 Feb 2022
AMG337
CAS:1173699-31-4
AMG-337 is an effective and highly specific ATP-competitive MET kinase inhibitor. In enzymatic assays, AMG-337 …
Formula:
C23H22FN7O3
Purity:
99.90%
Color and Shape:
solid
Molecular weight:
463.46
Estimated delivery in United States, on Monday 7 Feb 2022
Rociletinib
CAS:1374640-70-6
Rociletinib is an orally available small molecule, irreversible inhibitor of epidermal growth factor receptor (EGFR) …
Formula:
C27H28F3N7O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
555.55
Estimated delivery in United States, on Monday 7 Feb 2022
Daphnetin
CAS:486-35-1
Daphnetin, a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: …
Formula:
C9H6O4
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
178.14
Estimated delivery in United States, on Monday 7 Feb 2022
PF-562271 besylate
CAS:939791-38-5
PF-562271 (besylate) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, …
Formula:
C21H20F3N7O3S·C6H6O3S
Purity:
99.01%
Color and Shape:
solid
Molecular weight:
665.66
Estimated delivery in United States, on Monday 7 Feb 2022
OSI420
CAS:183320-51-6
OSI-420 (Desmethyl Erlotinib, CP-473420) is an active metabolite of erlotinib which is an orally active …
Formula:
C21H21N3O4·HCl
Purity:
98.0%
Molecular weight:
415.87
Estimated delivery in United States, on Monday 7 Feb 2022
AG18
CAS:118409-57-7
AG-18 inhibits EGFR with IC50 of 35 μM.
Formula:
C10H6N2O2
Purity:
99.19%
Color and Shape:
Yellow-Tan Solid
Molecular weight:
186.17
Estimated delivery in United States, on Monday 7 Feb 2022
Savolitinib
CAS:1313725-88-0
Savolitinib (AZD-6094) is an effective, selective, and orally bioavailable c-Met inhibitor (IC50s: 5 nM/3 nM …
Formula:
C17H15N9
Purity:
98.03%
Color and Shape:
solid
Molecular weight:
345.36
Estimated delivery in United States, on Monday 7 Feb 2022
TrkA-IN-1
CAS:1680179-43-4
TrkA-IN-1 is a potent and selective inhibitor of Tropomyosin-related kinase A (TrkA) (IC50: 99 nM …
Formula:
C25H20N4O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
392.45
Estimated delivery in United States, on Monday 7 Feb 2022
N-Desethylsunitinib hydrochloride
CAS:1261432-05-6
N-Desethylsunitinib hydrochloride is a major and pharmacologically active metabolite of sunitinib, which is potent, ATP-competitive …
Formula:
C20H24ClFN4O2
Molecular weight:
406.88
Estimated delivery in United States, on Monday 7 Feb 2022
BMS777607
CAS:1025720-94-8
BMS-777607 is a Met-related inhibitor for c-Met/Axl/Ron/Tyro3 (IC50: 3.9/1.1/1.8/4.3 nM). BMS-777607 has been investigated for …
Formula:
C25H19ClF2N4O4
Purity:
99.74%
Color and Shape:
solid
Molecular weight:
512.89
Estimated delivery in United States, on Monday 7 Feb 2022
Lenvatinib mesylate
CAS:857890-39-2
Lenvatinib mesylate is an oral and multi-targeted inhibitor of VEGFR1-3, FGFR1-4, PDGFR, KIT, and RET, …
Formula:
C22H23ClN4O7S
Purity:
99.79%
Color and Shape:
solid
Molecular weight:
522.96
Estimated delivery in United States, on Monday 7 Feb 2022
BGB-102
CAS:807640-87-5
BGB-102 is a potent multi-kinase inhibitor against HER2, EGFR, and HER4 (IC50s: 18 nM, 9.6 …
Formula:
C22H25BrN4O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
457.36
Estimated delivery in United States, on Monday 7 Feb 2022
Capmatinib xHCl
CAS:1029714-89-3
Capmatinib xHCl is a potent, orally active, selective, and ATP competitive c-Met kinase inhibitor, potently …
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
N/A
Estimated delivery in United States, on Monday 7 Feb 2022
CH6953755
CAS:2055918-71-1
CH6953755 is a potent, orally active and selective inhibitor of YES1 kinase (IC50: 1.8 nM). …
Formula:
C26H22F2N6O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
552.55
Estimated delivery in United States, on Monday 7 Feb 2022
ALW-II-41-27
CAS:1186206-79-0
ALW-II-41-27, an Eph receptor tyrosine kinase inhibitor, is used for cancer therapy.
Formula:
C32H32F3N5O2S
Purity:
99.52%
Color and Shape:
solid
Molecular weight:
607.7
Estimated delivery in United States, on Monday 7 Feb 2022
RO495
CAS:1258296-60-4
RO495, a potent inhibitor of TYK2, inhibits TYK2 with IC50 of 1.5nM as tested in …
Formula:
C17H14Cl2N6O
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
389.2
Estimated delivery in United States, on Monday 7 Feb 2022
SU6656
CAS:330161-87-0
SU 6656 is a selective inhibitor of Src family kinases, with IC50 of 280 nM, …
Formula:
C19H21N3O3S
Purity:
97.00%
Color and Shape:
solid
Molecular weight:
371.45
Estimated delivery in United States, on Monday 7 Feb 2022
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD
CAS:40732-48-7
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE, also known as cGMP, is a cellular regulatory agent and has been …
Formula:
C10H11N5NaO7P
Purity:
99.53%
Color and Shape:
White Powder / White To Off-White Solid
Molecular weight:
367.19
Estimated delivery in United States, on Monday 7 Feb 2022
Endoxifen Z-isomer
CAS:112093-28-4
Endoxifen (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity …
Formula:
C25H27NO2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
373.49
Estimated delivery in United States, on Monday 7 Feb 2022
AG-1557 hydrochloride (189290-58-2(free base))
AG-1557 is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: 8.194).
Formula:
C16H15ClIN3O2
Purity:
98.95%
Color and Shape:
solid
Molecular weight:
443.66
Estimated delivery in United States, on Monday 7 Feb 2022
Mutated EGFR-IN-2
CAS:2050906-97-1
Mutated EGFR-IN-2 is an inhibitor of mutant-selective EGFR.
Formula:
C29H35FN8O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
562.64
Estimated delivery in United States, on Monday 7 Feb 2022
Picropodophyllotoxin
CAS:17434-18-3
Picropodophyllin is a cyclolignan alkaloid found in the mayapple plant family (Podophyllum peltatum), and a …
Formula:
C22H22O8
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
414.41
Estimated delivery in United States, on Monday 7 Feb 2022
Osimertinib dimesylate
CAS:2070014-82-1
Osimertinib dimesylate is an irreversible and mutant selective EGFR inhibitor (IC50s: 12 and 1 nM …
Formula:
C30H41N7O8S2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
691.82
Estimated delivery in United States, on Monday 7 Feb 2022
Zinc bacitracin
CAS:1405-89-6
Bacitracin Zinc is an antibiotic that interferes with the dephosphorylation of C55-isoprenyl pyrophosphate, interference for …
Formula:
C66H101N17O16SZn
Purity:
63.98%
Color and Shape:
Solid
Molecular weight:
1486.07
Estimated delivery in United States, on Monday 7 Feb 2022
Nampt-IN-1
CAS:1698878-14-6
Nampt-IN-1 (LSN3154567) is a potent and selective NAMPT inhibitor. Nampt-IN-1 inhibits purified NAMPT with an …
Formula:
C20H25N3O5S
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
419.49
Estimated delivery in United States, on Monday 7 Feb 2022
PD153035 hydrochloride
CAS:183322-45-4
PD153035 hydrochloride (ZM 252868; AG 1517) is a effective and selective inhibitor of EGFR (Ki: …
Formula:
C16H15BrClN3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
396.67
Estimated delivery in United States, on Monday 7 Feb 2022
Ginsenoside Rg5
CAS:186763-78-0
1. Ginsenoside Rg5 could be a beneficial agent for the treatment of Alzheimer's disease. 2. …
Formula:
C42H70O12
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
767.01
Estimated delivery in United States, on Monday 7 Feb 2022
PKG Substrate acetate81187-14-6 free base)
PKG Substrate acetate is a selective substrate for cGMP-dependent protein kinase (PKG).PKG Substrate is a …
Formula:
C37H71N17O13
Molecular weight:
962.08
Estimated delivery in United States, on Monday 7 Feb 2022
Butein
CAS:487-52-5
Butein, a plant polyphenol, is isolated from Rhus verniciflua. It can inhibit the activation of …
Formula:
C15H12O5
Purity:
99.85%
Color and Shape:
solid
Molecular weight:
272.25
Estimated delivery in United States, on Monday 7 Feb 2022
Merestinib
CAS:1206799-15-6
LY2801653 is an orally available, small molecule inhibitor of the proto-oncogene c-Met (Ki: 2 nM) …
Formula:
C30H22F2N6O3
Purity:
95.00%
Color and Shape:
solid
Molecular weight:
552.54
Estimated delivery in United States, on Monday 7 Feb 2022
AG1557
CAS:189290-58-2
AG-1557 is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: 8.194).
Formula:
C16H14IN3O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
407.21
Estimated delivery in United States, on Monday 7 Feb 2022
Tie2 kinase inhibitor
CAS:948557-43-5
Tie2 kinase inhibitor, an optimized compound of SB-203580, is selective to Tie2 with IC50 of …
Formula:
C26H21N3O2S
Purity:
99.82%
Color and Shape:
solid
Molecular weight:
439.53
Estimated delivery in United States, on Monday 7 Feb 2022
DBPR112
CAS:1226549-49-0
DBPR112 has an IC50 of 15 nM and 48 nM for EGFRWT and EGFRL858R / …
Formula:
C32H31N5O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
533.62
Estimated delivery in United States, on Monday 7 Feb 2022
eCF506
CAS:1914078-41-3
eCF506 is a potent and selective inhibitor of SRC (IC50 < 0.5 nM)
Formula:
C26H38N8O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
510.63
Estimated delivery in United States, on Monday 7 Feb 2022
c-Fms-IN-8
CAS:1255303-58-2
c-Fms-IN-8 is a colony-stimulating factor-1 receptor (CSF-1R, c-FMS) Type II inhibitor (IC50: 9.1 nM). It …
Formula:
C27H30N2O5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
462.54
Estimated delivery in United States, on Monday 7 Feb 2022
HA-100
CAS:84468-24-6
HA-100 is an inhibitor of protein kinase
Formula:
C13H15N3O2S
Purity:
99.69%
Color and Shape:
Pale Yellow Crystalline Solid
Molecular weight:
277.34
Estimated delivery in United States, on Monday 7 Feb 2022
CREBtide acetate(149155-45-3 free base)
CREBtide acetate is a synthetic substrate for PKA (Km=3.9 µM), which is based on the …
Formula:
C75H133N29O21
Molecular weight:
1777.07
Estimated delivery in United States, on Monday 7 Feb 2022
Gefitinib-based PROTAC 3
CAS:2230821-27-7
Gefitinib-based PROTAC 3, conjugating an EGFR binding element to a VHL ligand via a linker, …
Formula:
C47H57ClFN7O8S
Purity:
98.25%
Color and Shape:
Solid
Molecular weight:
934.51
Estimated delivery in United States, on Monday 7 Feb 2022
WZ3146
CAS:1214265-56-1
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750) with IC50 of 2 nM …
Formula:
C24H25ClN6O2
Purity:
98.95%
Color and Shape:
solid
Molecular weight:
464.95
Estimated delivery in United States, on Monday 7 Feb 2022
Bemcentinib
CAS:1037624-75-1
R428 is a selective inhibitor of Axl (IC50: 14 nM) and has been investigated for …
Formula:
C30H34N8
Purity:
99.80%
Color and Shape:
solid
Molecular weight:
506.64
Estimated delivery in United States, on Monday 7 Feb 2022
Dacomitinib hydrate
CAS:1042385-75-0
Dacomitinib hydrate is a highly selective and second-generation small-molecule inhibitor of the pan-epidermal growth factor …
Formula:
C24H27ClFN5O3
Purity:
98.05%
Molecular weight:
487.96
Estimated delivery in United States, on Monday 7 Feb 2022
CP724714
CAS:383432-38-0
CP-724714 is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against EGFR, …
Formula:
C27H27N5O3
Purity:
98.82%
Color and Shape:
solid
Molecular weight:
469.54
Estimated delivery in United States, on Monday 7 Feb 2022
c-Fms-IN-2
CAS:791587-67-2
c-Fms-IN-2 is an inhibitor of FMS kinase (IC50: 0.024 μM).
Formula:
C19H21N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
339.39
Estimated delivery in United States, on Monday 7 Feb 2022
7-Hydroxy-4-chromone
CAS:59887-89-7
7-Hydroxychromone is a Src kinase inhibitor (IC50 of <300 μM).
Formula:
C9H6O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
162.14
Estimated delivery in United States, on Monday 7 Feb 2022
PF-06733804
CAS:1873373-33-1
PF-06733804 is a potent inhibitor of pan-Trk in cell-based assays (IC50s: 8.4 nM, 6.2 nM, …
Formula:
C20H19F5N4O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
474.38
Estimated delivery in United States, on Monday 7 Feb 2022
