
Inhibitors
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,904 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,137 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,423 products)
- Other Inhibitors(35,848 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Found 66516 products of "Inhibitors"
ELOVL1-IN-2
CAS:ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).Formula:C18H15FN2OPurity:99.94%Color and Shape:SolidMolecular weight:294.32Emprumapimod
CAS:Emprumapimod, an oral p38α MAPK inhibitor, targets RPMI-8226 cells, curbs LPS-induced IL-6; IC50: 100 pM; for cardiomyopathy, acute pain.Formula:C24H29F2N5O3Purity:99.21% - >99.99%Color and Shape:SolidMolecular weight:473.52Umibecestat
CAS:Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.Formula:C19H15ClF7N5O2Purity:99.88%Color and Shape:SolidMolecular weight:513.8Ref: TM-T13253
1mg163.00€5mg334.00€10mg485.00€25mg807.00€50mg1,099.00€100mg1,485.00€1mL*10mM (DMSO)376.00€SDZ 220-040
CAS:SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂,可诱导根系生长的部分无重力模式 。Formula:C16H16Cl2NO6PPurity:98.13%Color and Shape:SolidMolecular weight:420.18SJ6986
CAS:SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].Formula:C20H14F3N3O7SPurity:99.73%Color and Shape:SolidMolecular weight:497.4Ref: TM-T41257
5mg52.00€10mg86.00€25mg140.00€50mg245.00€100mg378.00€500mg898.00€1mL*10mM (DMSO)59.00€SB-423562
CAS:SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.Formula:C26H32N2O4Purity:99.22%Color and Shape:SolidMolecular weight:436.54Ref: TM-T12846
1mg37.00€5mg80.00€10mg119.00€25mg210.00€50mg319.00€100mg442.00€200mg605.00€1mL*10mM (DMSO)89.00€Enbezotinib
CAS:Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Formula:C21H21FN6O3Purity:99.84%Color and Shape:SolidMolecular weight:424.43Ref: TM-T62285
1mg77.00€5mg166.00€10mg253.00€25mg414.00€50mg567.00€100mg745.00€1mL*10mM (DMSO)182.00€(+)-Tetrabenazine
CAS:(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFormula:C19H27NO3Purity:98.69%Color and Shape:SolidMolecular weight:317.42PF-07258669
CAS:PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.Formula:C25H27FN6O2Purity:99.9%Color and Shape:SolidMolecular weight:462.52BMS 299897
CAS:BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.Formula:C24H21ClF3NO4SPurity:99.82%Color and Shape:SolidMolecular weight:511.94Aldometanib
CAS:Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.Formula:C27H43Cl2IN2Purity:99.32% - 99.55%Color and Shape:SolidMolecular weight:593.46ALOX15-IN-2
CAS:ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.Formula:C23H29N3O4SPurity:99.98%Color and Shape:SolidMolecular weight:443.56Ref: TM-T62606
1mg46.00€5mg90.00€10mg160.00€25mg313.00€50mg537.00€100mg767.00€500mg1,558.00€1mL*10mM (DMSO)100.00€CCF0058981
CAS:CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.
Formula:C24H19ClN6OPurity:98.94%Color and Shape:SoildMolecular weight:442.9Ref: TM-T60095
1mg46.00€2mg60.00€5mg92.00€10mg160.00€25mg324.00€50mg449.00€100mg562.00€500mgTo inquireSYM2206
CAS:SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediatedFormula:C20H22N4O3Purity:99.8%Color and Shape:SolidMolecular weight:366.41SB-224289 hydrochloride
CAS:SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Formula:C32H33ClN4O3Purity:98.99% - 99.96%Color and Shape:SolidMolecular weight:557.08Milademetan
CAS:Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.Formula:C30H34Cl2FN5O4Purity:>99.99%Color and Shape:SolidMolecular weight:618.53Ref: TM-T12040
1mg93.00€5mg167.00€10mg260.00€25mg492.00€50mg802.00€100mg1,378.00€1mL*10mM (DMSO)221.00€L-371,257
CAS:L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.Formula:C28H33N3O6Purity:99.79%Color and Shape:SolidMolecular weight:507.58DRB18
CAS:DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.Formula:C22H23ClN2O2Purity:99.54%Color and Shape:SolidMolecular weight:382.88Ref: TM-T22317
1mg89.00€5mg215.00€10mg340.00€25mg687.00€50mg1,108.00€100mg1,485.00€500mg2,962.00€1mL*10mM (DMSO)236.00€MIV-247
CAS:MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.Formula:C17H24F3N3O4Purity:99.27%Color and Shape:SolidMolecular weight:391.39STK-15
CAS:STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.Formula:C34H29NO5Purity:98.05%Color and Shape:SolidMolecular weight:531.6Treprostinil diethanolamine
CAS:Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,Formula:C27H45NO7Purity:99.86%Color and Shape:SolidMolecular weight:495.65FABPs ligand 6
CAS:FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Formula:C28H27FN2O3Purity:97.45%Color and Shape:SolidMolecular weight:458.52GLPG0974
CAS:GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.Formula:C25H25ClN2O4SPurity:99.8%Color and Shape:SolidMolecular weight:484.99AChE/BChE-IN-10
CAS:AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.
Formula:C26H30N2O2Purity:99.55% - 99.88%Color and Shape:SoildMolecular weight:402.53BMS453
CAS:BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.Formula:C27H24O2Purity:99.93%Color and Shape:SolidMolecular weight:380.48Cap-dependent endonuclease-IN-1
CAS:Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.Formula:C27H22F2N2O6SPurity:99.53% - 99.61%Color and Shape:SolidMolecular weight:540.54AZD-5672
CAS:AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.Formula:C32H38F2N2O5S2Purity:98.1%Color and Shape:SolidMolecular weight:632.78Ref: TM-T30260
1mg192.00€5mg434.00€10mg610.00€25mg888.00€50mg1,243.00€100mg1,693.00€1mL*10mM (DMSO)530.00€Dual FAAH/sEH-IN-1
CAS:Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.
Formula:C25H22ClN3O3S2Purity:99.89%Color and Shape:SolidMolecular weight:512.04D75-4590
CAS:D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.Formula:C21H27N5Purity:98.56% - 98.85%Color and Shape:SolidMolecular weight:349.47Ref: TM-T61194
5mg39.00€10mg62.00€25mg122.00€50mg187.00€100mg269.00€200mg358.00€1mL*10mM (DMSO)46.00€KI696
CAS:KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.Formula:C28H30N4O6SPurity:99.74%Color and Shape:SolidMolecular weight:550.63Ref: TM-T11758L
1mg137.00€5mg281.00€10mg423.00€25mg707.00€50mg1,018.00€100mg1,468.00€200mg1,963.00€1mL*10mM (DMSO)341.00€Zotizalkib
CAS:TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.Formula:C21H20F3N5O3Purity:98.7%Color and Shape:SolidMolecular weight:447.41Ref: TM-T9414
1mg114.00€5mg268.00€10mg439.00€25mg879.00€50mg1,395.00€100mg1,873.00€1mL*10mM (DMSO)303.00€Cbl-b-IN-3
CAS:Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.Formula:C30H34F3N5OPurity:97.63%Color and Shape:SolidMolecular weight:537.62Ref: TM-T63790
1mg66.00€5mg145.00€10mg192.00€25mg364.00€50mg558.00€100mg893.00€1mL*10mM (DMSO)172.00€NRX-1532
NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.Formula:C16H11F3N4O2Purity:98.95% - 99.94%Color and Shape:SolidMolecular weight:348.28Ref: TM-T61172
1mg147.00€5mg358.00€10mg597.00€25mg1,153.00€50mg1,549.00€100mg2,088.00€500mg4,185.00€1mL*10mM (DMSO)394.00€Obicetrapib
CAS:Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.Formula:C32H31F9N4O5Purity:99.26% - >99.99%Color and Shape:SolidMolecular weight:722.6Glycosyltransferase-IN-1
Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.Formula:C19H21N5OPurity:99.76%Color and Shape:SolidMolecular weight:335.4AZD 3147
CAS:AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).
Formula:C24H31N5O4S2Purity:99.99%Color and Shape:SolidMolecular weight:517.66PREP inhibitor-1
CAS:PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.Formula:C22H28N4O2Purity:98.78%Color and Shape:SoildMolecular weight:380.48BAY-3827
CAS:BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.Formula:C27H25FN6OPurity:99.90%Color and Shape:SolidMolecular weight:468.53Ref: TM-T73350
1mg52.00€5mg113.00€10mg177.00€25mg334.00€50mg560.00€100mg792.00€500mg1,575.00€1mL*10mM (DMSO)117.00€Pocenbrodib
CAS:Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.Formula:C28H32FN3O6Purity:98.48% - 99.54%Color and Shape:SolidMolecular weight:525.57Elacytarabine
CAS:Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.Formula:C27H45N3O6Purity:97.69%Color and Shape:SolidMolecular weight:507.66JTK-109
CAS:JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.Formula:C37H33ClFN3O4Purity:98.48% - 99.68%Color and Shape:SolidMolecular weight:638.13Ref: TM-T27696
1mg296.00€5mg718.00€10mg982.00€25mg1,485.00€50mg2,008.00€100mg2,637.00€1mL*10mM (DMSO)1,108.00€EZM0414
CAS:EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.Formula:C22H29FN4O2Purity:99.58%Color and Shape:SolidMolecular weight:400.49GSK3368715 dihydrochloride
CAS:GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.Formula:C20H40Cl2N4O2Purity:99.66% - 99.66%Color and Shape:SolidMolecular weight:439.46XMD-17-51 Trifluoroacetate
CAS:XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.Formula:C23H25F3N8O3Purity:99.65%Color and Shape:SolidMolecular weight:518.49CK2 inhibitor 2
CAS:CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Formula:C21H17ClN4O2Purity:99.02%Color and Shape:SolidMolecular weight:392.84Ref: TM-T35557
1mg62.00€5mg138.00€10mg215.00€25mg425.00€50mg637.00€100mg853.00€200mg1,153.00€1mL*10mM (DMSO)152.00€ARN19702
CAS:ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.Formula:C21H22FN3O3S2Purity:99.86%Color and Shape:SolidMolecular weight:447.55Ref: TM-T9528
1mg52.00€5mg113.00€10mg177.00€25mg350.00€50mg560.00€100mg880.00€200mg1,189.00€500mg1,765.00€1mL*10mM (DMSO)124.00€(E/Z)-GSK5182
CAS:GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Formula:C27H31NO3Purity:97.58%Color and Shape:SolidMolecular weight:417.54Ref: TM-T7709
1mg77.00€5mg167.00€10mg260.00€25mg477.00€50mg707.00€100mg1,063.00€1mL*10mM (DMSO)177.00€10-Methoxycamptothecin
CAS:10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.Formula:C21H18N2O5Purity:98.36%Color and Shape:SolidMolecular weight:378.38LY3143921 hydrate
CAS:LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].Formula:C16H14FN5O2Purity:98.43%Color and Shape:SolidMolecular weight:327.31Durlobactam sodium salt
CAS:Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.Formula:C8H10N3NaO6SPurity:97.01% - 99.03%Color and Shape:SolidMolecular weight:299.23FGI-106 tetrahydrochloride
CAS:FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as EbolaFormula:C28H42Cl4N6Purity:99.68%Color and Shape:SolidMolecular weight:604.48Ref: TM-T11281L
1mg82.00€5mg161.00€10mg245.00€25mg406.00€50mg572.00€100mg772.00€200mg1,035.00€1mL*10mM (DMSO)207.00€Rineterkib
CAS:Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.Formula:C26H27BrF3N5O2Purity:99.73%Color and Shape:SolidMolecular weight:578.42Ref: TM-T11224
1mg87.00€5mg170.00€10mg318.00€25mg538.00€50mg765.00€100mg1,035.00€1mL*10mM (DMSO)224.00€Rolapitant hydrochloride
CAS:Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Formula:C25H27ClF6N2O2Purity:98.35% - 99.79%Color and Shape:SolidMolecular weight:536.94Ref: TM-T3724
1mg153.00€5mg365.00€10mg520.00€25mg780.00€50mg1,054.00€100mg1,425.00€200mg1,882.00€1mL*10mM (DMSO)439.00€Gemcitabine elaidate hydrochloride
CAS:CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.
Formula:C27H44ClF2N3O5Purity:98.50% - 99.6%Color and Shape:SolidMolecular weight:564.11PD 151746
CAS:PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.Formula:C11H8FNO2SPurity:98.63% - ≥95%Color and Shape:SolidMolecular weight:237.25TGFβRI-IN-3
CAS:TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.Formula:C28H23N3O2SPurity:99.85%Color and Shape:SoildMolecular weight:465.57Ref: TM-T9523
1mg84.00€5mg177.00€10mg281.00€25mg552.00€50mg859.00€100mg1,234.00€500mg2,457.00€1mL*10mM (DMSO)177.00€BAY-8400
BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy inFormula:C21H17F2N5OPurity:99.53%Color and Shape:SolidMolecular weight:393.39Ref: TM-T9498
1mg80.00€5mg147.00€10mg215.00€25mg439.00€50mg750.00€100mg1,009.00€1mL*10mM (DMSO)161.00€Sinefungin
CAS:Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viralFormula:C15H23N7O5Purity:98% - 98.12%Color and Shape:SolidMolecular weight:381.39BRD0639
CAS:BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Formula:C21H22ClN5O4SPurity:99.85%Color and Shape:SolidMolecular weight:475.95SR 11302
CAS:SR 11302 is an inhibitor of activator protein-1 (AP-1).Formula:C26H32O2Purity:98.65%Color and Shape:SolidMolecular weight:376.53Ref: TM-T23384
1mg93.00€5mg137.00€10mg205.00€25mg356.00€50mg587.00€100mg888.00€1mL*10mM (DMSO)150.00€JAK2-IN-7
CAS:JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.Formula:C26H33N7OPurity:99.54%Color and Shape:SolidMolecular weight:459.59Ref: TM-T35900
1mg138.00€5mg334.00€10mg597.00€25mg1,234.00€50mg1,648.00€100mg2,232.00€1mL*10mM (DMSO)339.00€INCB086550
CAS:INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 <= 10 nM.Formula:C41H39N7O4Purity:98.49%Color and Shape:SolidMolecular weight:693.79Sebetralstat
CAS:Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.
Formula:C26H26FN5O4Purity:99.85%Color and Shape:SolidMolecular weight:491.51FX-11
CAS:FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.Formula:C22H22O4Purity:98.95% - 98.95%Color and Shape:SolidMolecular weight:350.41LSZ-102
CAS:LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.Formula:C25H17F3O4SPurity:98.56%Color and Shape:SolidMolecular weight:470.46Clorophene
CAS:Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.Formula:C13H11ClOPurity:99.87%Color and Shape:White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)Molecular weight:218.68GAS6 Protein, Human, Recombinant (His)
GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.
Purity:>99.90%Color and Shape:SoildMolecular weight:72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)TCblR Protein, Human, Recombinant (His)
TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.
Color and Shape:SolidMolecular weight:32-58 KDa (reducing condition)TEM1/CD248 Protein, Mouse, Recombinant (His)
TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.
Color and Shape:SolidMolecular weight:73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.Relacorilant
CAS:Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.
Formula:C27H22F4N6O3SPurity:98.53% - 99%Color and Shape:SolidMolecular weight:586.563-Acetylcoumarin
CAS:3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.
Formula:C11H8O3Purity:99.41%Color and Shape:Yellow Crystalline PowderMolecular weight:188.18α-Terpineol
CAS:Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.
Formula:C10H18OPurity:97.55%Color and Shape:Colorless LiquidMolecular weight:154.252'-Hydroxy-4'-methylacetophenone
CAS:2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.
Formula:C9H10O2Purity:99.88%Color and Shape:Black LiquidMolecular weight:150.174-Ethoxycoumarin
CAS:4-Ethoxycoumarin has antimicrobial activity.
Formula:C11H10O3Purity:99.64%Color and Shape:SolidMolecular weight:190.2EGFR-IN-7
CAS:EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.
Formula:C32H41BrN9O2PPurity:95.32% - 99.64%Color and Shape:SolidMolecular weight:694.63-Methoxyphenylacetic acid
CAS:3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot
Formula:C9H10O3Purity:98.61%Color and Shape:White SolidMolecular weight:166.17(-)-Isopulegol
CAS:Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.
Formula:C10H18OPurity:99.89%Color and Shape:LiquidMolecular weight:154.25PRGL493
CAS:PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.Formula:C25H21N7O2Purity:98.80% - 99.11%Color and Shape:SolidMolecular weight:451.48Ref: TM-T35666
Discontinued productAnisylacetone
CAS:Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.
Formula:C11H14O2Purity:99.74%Color and Shape:LiquidMolecular weight:178.23m-PEG1-acid
CAS:M-PEG1-acid, a soluble PEG derivative, has a terminal carboxylic acid for forming amide bonds with primary amines using activators like EDC, DCC.
Formula:C4H8O3Purity:98%Color and Shape:SolidMolecular weight:104.10Mitoquinone-cyclodextrin
CAS:Mitoquinone-cyclodextrin is a mitochondria-targeted, 1:1 mix of Mitoquinone mesylate and cyclodextrin, aiming to combat oxidative damage.
Formula:C80H117O42PSColor and Shape:SolidMolecular weight:1813.81MRS2802
CAS:MRS2802 is a P2Y14 receptor agonist, its EC50 value for P2Y14 receptor is 63 nM.Formula:C10H14F2N2O11P2Purity:98%Color and Shape:SolidMolecular weight:438.169DFHBI-2T
CAS:DFHBI-2T, a membrane-permeable fluorescence probe activated by RNA aptamers (ex/em=500 nm/523 nm), is utilized for imaging RNA within live cells.Formula:C12H7F5N2O2Color and Shape:SolidMolecular weight:306.192Cap-dependent endonuclease-IN-22
CAS:Cap-dependent endonuclease-IN-22 is a powerful inhibitor of cap-dependent endonuclease (CEN) [1].
Formula:C37H37ClF2N6O7S2Color and Shape:SolidMolecular weight:815.31Melarsonyl dipotassium
CAS:Melarsonyl dipotassium, also known as melarsonic acid dipotassium, is a potent anthelmintic agent with the ability to effectively inhibit parasites.
Formula:C13H13AsK2N6O4S2Color and Shape:SolidMolecular weight:534.52Yimitasvir diphosphate
CAS:Yimitasvir (Emitasvir) diphosphate,一种针对丙型肝炎病毒(HCV)非结构蛋白5A (NS5A)的口服活性抑制剂,适用于慢性丙型肝炎病毒感染的研究。
Formula:C49H64N8O14P2Color and Shape:SolidMolecular weight:1051.03OVA Peptide 323-339
OVA Peptide (323-339) is an Ovalbumin epitope crucial for hypersensitivity in BALB/c mice.
Formula:C74H120N26O25Purity:98%Color and Shape:SolidMolecular weight:1773.91SHP2 protein degrader-1
CAS:SHP2 degrader-1: highly efficient, induces SHP2 degradation & cell apoptosis, shows promise in SHP2-related disease research.
Formula:C42H51Cl2N11O8Color and Shape:SolidMolecular weight:908.84Coumberone
CAS:Coumberone, a fluorogenic probe, is reduced by AKR1C family to fluorescent coumberol; vital for AKR1C research.Formula:C22H19NO3Color and Shape:SolidMolecular weight:345.398MitoPY1
CAS:a fluorescent probe for imaging hydrogen peroxide (H2O2) in mitochondria of living cellsFormula:C52H53BN2O5PPurity:98%Color and Shape:SolidMolecular weight:827.77Thalidomide-NH-PEG2-C2-NH-Boc
CAS:Thalidomide-based cereblon ligand-linker for selective dBRD9 synthesis, enabling BAF complex study.
Formula:C24H32N4O8Color and Shape:SolidMolecular weight:504.53(D)-PPA 1
CAS:PD-1/PD-L1 binder, Kd 0.51 μM; blocks interaction in flow cytometry at 1 mg/mL; inhibits tumors, extends mouse survival.
Formula:C70H98N20O21Purity:98%Color and Shape:SolidMolecular weight:1555.67Gd-NMC-3
CAS:Gd-NMC-3, a bimodal imaging probe, exhibits high resolution and sensitivity for tumor imaging with favorable biocompatibility, demonstrating significant
Formula:C77H114Gd2N14O24S2Color and Shape:SolidMolecular weight:1998.44PEG2-bis(phosphonic acid)
CAS:PEG2-bis(phosphonic acid) is a PEG Linker.Formula:C6H16O8P2Color and Shape:SolidMolecular weight:278.13PLK1-IN-6
PLK1-IN-6: potent, selective PLK1 inhibitor, IC50 = 0.45 nM, hinders cancer cell growth.
Formula:C28H37N9O3Color and Shape:SolidMolecular weight:547.65Darobactin
CAS:Darobactin is an antibiotic effective against critical Gram-negative pathogens, demonstrating activity both in vitro and in animal infection models [1].
Formula:C47H55N11O12Purity:98%Color and Shape:SolidMolecular weight:966.0118-Hydroxycortisol
CAS:18-Hydroxycortisol: adrenal steroid, cortisol derivative, studied in primary aldosteronism.Formula:C21H30O6Color and Shape:SolidMolecular weight:378.46BODIPY 576/589
CAS:BODIPY 576/589 is a long wavelength biological labeled dye.Formula:C16H14BF2N3O2Color and Shape:SolidMolecular weight:329.11TLQP-21 TFA
TLQP-21 TFA is a VGF-derived peptide, C3aR1 agonist (mouse EC50: 10.3μM; human EC50: 68.8μM), that raises intracellular Ca2+ for nociception research.
Purity:98%Color and Shape:LiquidGLF16 FA
GLF16 FA is a hydrophilic fluorescent SBB analogue for rapid detection of senescent cells using flow cytometry and live cell sorting.Formula:C73H81IN10O5Purity:98.20% - 99.89%Color and Shape:SoildMolecular weight:1305.42Ref: TM-T77767L
Discontinued product

