Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,519 products)
- Apoptosis(5,786 products)
- Cell Cycle/Checkpoint(4,444 products)
- Chromatin/Epigenetics(2,235 products)
- Cytoskeletal Signaling(1,382 products)
- DNA Damage/DNA Repair(2,823 products)
- Endocrinology/Hormones(3,499 products)
- Enzyme(3,639 products)
- GPCR/G-Protein(8,314 products)
- Immunology and Inflammation(3,516 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,199 products)
- Membrane Transporter/Ion Channel(2,786 products)
- Metabolism(9,417 products)
- Microbiology/Virology(6,967 products)
- Neuroscience(9,920 products)
- Other Inhibitors(37,931 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,399 products)
- Proteases/Proteasome(1,596 products)
- Stem Cell and Derivatives(832 products)
- Tyrosine Kinase/Adaptors(2,015 products)
- Ubiquitination(1,646 products)
Show 16 more subcategories
Found 66627 products of "Inhibitors"
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Golgicide A-2
CAS:<p>GCA-2 is a potent enantiomer of GCA, selectively and efficiently kills An. stephensi larvae, useful for dengue research.</p>Formula:C17H14F2N2Color and Shape:SolidMolecular weight:284.31Metrizoic acid
CAS:<p>Metrizoic acid is an ionic contrast medium. Metrizoic acid displays high osmolality and has a risk of inducing allergic reactions.</p>Formula:C12H11I3N2O4Purity:98%Color and Shape:SolidMolecular weight:627.9402Muzolimine
CAS:<p>Muzolimine: a long-acting, high-capacity diuretic for kidney failure/hypertension; withdrawn due to serious neurological side effects.</p>Formula:C11H11Cl2N3OColor and Shape:SolidMolecular weight:272.13STING agonist-23
CAS:<p>CF502 (STING agonist-23) is a non-nucleotide that activates STING pathway, boosts immune responses, and shows activity against SARS-CoV.</p>Formula:C33H35N13O4Color and Shape:SolidMolecular weight:677.72TD-106
CAS:<p>TD-106 is a modulator of cereblon (CRBN), and can be used for targeted protein degradation. BRD4 PROTACs with TD-106 induce BRD4 degradation.</p>Formula:C12H11N5O3Purity:98%Color and Shape:SolidMolecular weight:273.25Ref: TM-T13104
Discontinued product2-Nitrosopyridine
CAS:<p>2-Nitrosopyridine: used in antibiotic synthesis, Click/Diels-Alder reactions, excellent dienophile.</p>Formula:C5H4N2OColor and Shape:SolidMolecular weight:108.1Phosal 50 PG
CAS:<p>Phosal 50 PG is a co-solvent used as an emulsifier and stabilizer in the pharmaceutical and cosmetic industries.Phosal 50 PG is used as a dietary supplement.</p>Purity:98%Color and Shape:SolidSEMBL
CAS:<p>SEMBL, a novel inhibitor of DNA binding of NF-kappaB component p65 in vitro, inhibits NF-kappaB and cellular invasion in ovarian carcinoma ES-2 cells.</p>Formula:C12H11NO4Purity:98%Color and Shape:SolidMolecular weight:233.22Valiloxibic acid
CAS:<p>Valiloxibic acid is a prodrug for GHB, a natural psychoactive neurotransmitter and weak GABAB agonist.</p>Formula:C9H17NO4Color and Shape:SolidMolecular weight:203.238HT-2 Toxin
CAS:<p>HT-2 Toxin, a deacetylated metabolite of T-2 toxin, impairs protein synthesis and hinders cell proliferation in plants.</p>Formula:C22H32O8Purity:98%Color and Shape:SolidMolecular weight:424.49Loviride
CAS:<p>Loviride, a reverse transcriptase inhibitor with IC50 of 0.3 μM, blocks HIV-1/2 and SIV in MT-4 cells.</p>Formula:C17H16Cl2N2O2Color and Shape:SolidMolecular weight:351.23Ref: TM-T15776
Discontinued productSIRT-IN-3
CAS:<p>SIRT-IN-3: potent SIRT1 inhibitor (IC50=17μM), 4x selective over SIRT2, 14x over SIRT3 (IC50s: 74μM & 235μM).</p>Formula:C13H12N2OColor and Shape:SolidMolecular weight:212.25Indium(III) isopropoxide
CAS:<p>Indium(III) Isopropoxide: a catalyst for Oppenauer oxidation, turns benzylic alcohols to aldehydes/ketones.</p>Formula:C3H8InOPurity:98%Color and Shape:SolidMolecular weight:174.914Ref: TM-T19372
Discontinued productCysteinylglycine TFA
CAS:<p>Cysteinylglycine TFA is an endogenous metabolite. It is used in disease diagnosis.</p>Formula:C7H11F3N2O5SColor and Shape:SolidMolecular weight:292.23sodium 4-pentynoate
CAS:<p>sodium 4-pentynoate is a alkynylacetate analogue.</p>Formula:C5H5NaO2Purity:98%Color and Shape:SolidMolecular weight:120.083-Hydroxyhippuric acid
CAS:<p>3-Hydroxyhippuric acid is an acyl glycine, which are normally minor metabolites of fatty acids.</p>Formula:C9H9NO4Color and Shape:SolidMolecular weight:195.173,5-Diphenyl pyridine
CAS:<p>Heterocyclic compounds-pyridine,</p>Formula:C17H13NColor and Shape:SolidMolecular weight:231.29Ref: TM-TNU0677
Discontinued product3-Methylcrotonylglycine
CAS:<p>3-Methylcrotonylglycine is an acyl glycine, a normal amino acid metabolite found in urine.</p>Formula:C7H11NO3Purity:98%Color and Shape:SolidMolecular weight:157.17(S)-Rasagiline
CAS:<p>(S)-Rasagiline is rasagiline S-isomer, and is an agent of anti-Parkinson.</p>Formula:C12H13NColor and Shape:SolidMolecular weight:171.24Ref: TM-T13252
Discontinued product(S,S)-Valifenalate
CAS:<p>(S,S)-Valifenalate is an acylamino acid fungicide and is used to control a wide range of fungi belonging to the class of Oomycetes.</p>Formula:C19H27ClN2O5Color and Shape:SolidMolecular weight:398.88PDK1-IN-RS2
CAS:<p>PDK1-IN-RS2, a PIFtide mimic, selectively inhibits PDK1, blocking S6K1 activation (Kd: 9 μM).</p>Formula:C15H9ClN2O2S3Purity:98%Color and Shape:SolidMolecular weight:380.89Ref: TM-T16450
Discontinued productGRK2 Inhibitor
CAS:<p>GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).</p>Formula:C12H9NO6Color and Shape:SolidMolecular weight:263.2Deoxypseudouridine
CAS:<p>Deoxypseudouridine is a nucleotide analog.</p>Formula:C9H12N2O5Color and Shape:SolidMolecular weight:228.2Ref: TM-T13645
Discontinued product5-OxoETE
CAS:<p>5-OxoETE, a dehydrogenase-oxidized 5-HETE, raises neutrophil Ca²⁺ (EC50=2nM) & drives eosinophil migration & MAPK pathway.</p>Formula:C20H30O3Purity:98.59%Color and Shape:SolidMolecular weight:318.454',5'-Dibromofluorescein
CAS:<p>4',5'-Dibromofluorescein (Eosinic acid) is a fluorescent dye that can be used as a ligand for protein characterization by spectroscopic analysis.</p>Formula:C20H10Br2O5Color and Shape:Orange Solid PowderMolecular weight:490.10Ceritinib D7
CAS:<p>Ceritinib D7 (LDK378 D7) is a deuterium-labeled Ceritinib. Ceritinib is an ATP-competitive inhibitor of ALK tyrosine kinase.</p>Formula:C28H36ClN5O3SPurity:98%Color and Shape:SolidMolecular weight:565.18Canagliflozin-d4
CAS:<p>Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.</p>Formula:C24H25FO5SPurity:98%Color and Shape:SolidMolecular weight:448.54Aniline-2,4-diphosphonic acid tetraethyl ester;
CAS:<p>Intermediates and building blocks - phosphorous compounds; nucleophile</p>Formula:C14H25NO6P2Color and Shape:SolidMolecular weight:365.3Ref: TM-TNU0723
Discontinued productL-690330
CAS:<p>L-690330 inhibits human/bovine inositol monophosphatase; Ki: 0.19-0.42 μM. 10x potency vs. mouse/rat IMPase.</p>Formula:C8H12O8P2Color and Shape:SolidMolecular weight:298.12Ref: TM-T15685
Discontinued productTFLLR-NH2 2TFA(197794-83-5(free base))
<p>TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).</p>Formula:C35H55F6N9O10Purity:99.56%Color and Shape:SolidMolecular weight:875.87NLX-204 hydrochloride(2170405-10-2 free base)
<p>NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).</p>Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Elamipretide
CAS:<p>Elamipretide (SS-31, MTP-131, Bendavia) is a mitochondria-focused peptide that curbs toxic ROS and stabilizes cardiolipin.</p>Formula:C32H49N9O5Purity:98.53% - 99.85%Color and Shape:SolidMolecular weight:639.79Pamoic acid
CAS:<p>Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.</p>Formula:C23H16O6Purity:99.99%Color and Shape:Fine Yellow PowderMolecular weight:388.37Ethyl 4-hydroxyphenylacetate
CAS:<p>Ethyl 4-hydroxyphenylacetate is a selective inhibitor of monoamine oxidase A.</p>Formula:C10H12O3Purity:99.89%Color and Shape:Slightly Yellow LiquidMolecular weight:180.2Tropinone
CAS:<p>Tropinone used as an intermediate in the synthesis of atropine sulfate, and is a decane alkaloid.</p>Formula:C8H13NOPurity:99.90%Color and Shape:Beige To Brown Crystalline PowderMolecular weight:139.19Elamipretide 2TFA
CAS:<p>Elamipretide 2TFA (RX-31 2TFA) is a novel mitochondrion-targeted antioxidant.</p>Formula:C36H51F6N9O9Purity:>99.99%Color and Shape:SolidMolecular weight:867.84Ref: TM-T8831
Discontinued productElamipretide Triacetate
CAS:<p>Elamipretide TriTFA, a tetrapeptide, targets mitochondria, associates with cardiolipin, studied for treating Leber's Optic Neuropathy.</p>Formula:C38H61N9O11Purity:>99.99%Color and Shape:SolidMolecular weight:819.942-Methyl-5-HT hydrochloride
CAS:<p>2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.</p>Formula:C11H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:226.7Compound T69202(SC)
CAS:<p>NBQX (FG9202), an AMPA/kainate receptor blocker, counters glutamate toxicity; water-soluble as disodium salt, has anticonvulsant properties.</p>Formula:C12H6N4Na2O6SColor and Shape:SolidMolecular weight:380.2415L-(+)-Abrine
CAS:<p>L-(+)-Abrine (L-N-Methyltryptophan) is a toxic protein found in the jequirity seed.,can be used as a biomarker for abrin exposure.</p>Formula:C12H14N2O2Purity:98.71% - ≥95%Color and Shape:White PowderMolecular weight:218.25Coumaran
CAS:<p>Coumaran (2,3-Dihydrobenzofuran) is an acetylcholinesterase (AChE) inhibitor isolated from leaves of L. camara. Coumaran(2,3-Dihydrobenzofuran) can be used as a biopesticide. 2,3-dihydrobenzofuran is a member of the class of 1-benzofurans that is the 2,3-dihydroderivative of benzofuran. It has a role as a metabolite.</p>Formula:C8H8OPurity:99.61%Color and Shape:LiquidMolecular weight:120.15MTP 131 acetate
CAS:<p>MTP 131 (acetate) is a small mitochondrially-targeted tetrapeptide.</p>Formula:C34H53N9O7Purity:99.9%Color and Shape:SolidMolecular weight:699.844-Hydroxy-6-methylcoumarin
CAS:<p>4-Hydroxy-6-methylcoumarin (4-HMC) is a naturally occurring phenolic compound, a derivative of coumarin, found in a variety of plants, fungi, and bacteria. It has anti-inflammatory and anti-tumor activity.4-HMC is used as a flavoring agent, preservative and antioxidant in the food industry.</p>Formula:C10H8O3Purity:99.95%Color and Shape:White PowderMolecular weight:176.17p-Toluic Acid
CAS:<p>p-Toluic Acid (4-Methylbenzoic acid) belongs to the class of organic compounds known as benzoic acids. 4-Methylbenzoic acid has been primarily detected in saliva. Within the cell, 4-methylbenzoic acid is primarily located in the cytoplasm.</p>Formula:C8H8O2Purity:99.44%Color and Shape:Physical Description White Powder Sublimes (Ntp 1992)Molecular weight:136.15Cebranopadol
CAS:<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Formula:C24H27FN2OPurity:98.32% - 99.78%Color and Shape:SolidMolecular weight:378.48Oxindole
CAS:<p>Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.</p>Formula:C8H7NOPurity:99.34%Color and Shape:Off-White Crystalline PowderMolecular weight:133.15Danoprevir sodium
CAS:<p>Danoprevir sodium is an NS3/4A protease inhibitor used in the treatment of Hepatitis C</p>Formula:C35H45FN5NaO9SColor and Shape:SolidMolecular weight:753.82Rosmanol
CAS:<p>Rosmanol has antioxidant, anti-inflammatory, CNS effects; induces apoptosis in cancer cells; modulates GABAA receptors.</p>Formula:C20H26O5Purity:98.82% - 99.79%Color and Shape:SolidMolecular weight:346.424-Methoxycoumarine
CAS:<p>4-Methoxycoumarine has antitumour effects.</p>Formula:C10H8O3Purity:99.88%Color and Shape:SolidMolecular weight:176.1710Z-Nonadecenoic acid
CAS:<p>10Z-Nonadecenoic acid is a long-chain fatty acid with anti-tumor activity.</p>Formula:C19H36O2Purity:99.43%Color and Shape:SolidMolecular weight:296.49Dimethylamine hydrochloride
CAS:<p>Dimethylamine hydrochloride, found in urine, comes from food compound TMAO and NO synthesis inhibitor ADMA, processed by DDAH enzyme.</p>Formula:C2H8ClNPurity:98% - 99.89%Color and Shape:White Solid CrystallineMolecular weight:81.54Sculponeatin O
CAS:<p>Sculponeatin O may have protective effects on the lipid peroxidation-damaged live cells.</p>Formula:C28H40O4Purity:95.00%Color and Shape:SolidMolecular weight:440.614-Hydroxybenzyl cyanide
CAS:<p>4-Hydroxybenzyl cyanide (4-Hydroxyphenylacetonitrile) shows strong antioxidative activity.</p>Formula:C8H7NOPurity:98.13%Color and Shape:Light Brown SolidMolecular weight:133.157-Methoxy-1-tetralone
CAS:<p>7-Methoxy-1-tetralone may have insecticidal activity.</p>Formula:C11H12O2Purity:99.93%Color and Shape:White CrystalMolecular weight:176.21SR17018
CAS:<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Formula:C19H18Cl3N3OPurity:99.89%Color and Shape:SolidMolecular weight:410.72SR-4370
CAS:<p>SR-4370 is an HDAC inhibitor. SR- 4370 exhibited IC50 values of 0.5 μM, 0.1 μM and 0.06 μM towards HDAC1, HDAC2 and HDAC3, resp.</p>Formula:C17H18F2N2OPurity:99.50%Color and Shape:SolidMolecular weight:304.33Decyl-TPP bromide
CAS:<p>Decyl-TPP bromide ((1-Decyl)triphenylphosphonium bromide) may be used as an intermediate for chemical synthesis and an inactive control or as a reference to</p>Formula:C28H36BrPPurity:98%Color and Shape:SolidMolecular weight:483.46CTB
CAS:<p>CTB (Cholera Toxin B subunit) is an activator of p300 histone acetyltransferase and induces apoptosis in MCF-7 cells.</p>Formula:C16H13ClF3NO2Purity:99.82%Color and Shape:SolidMolecular weight:343.73Lupinine
CAS:<p>Lupinine is an alkaloid capable of counteracting ethanol anesthesia. Lupinine is an AChE and BChE inhibitor and potential CD69 activator found in species of Loranthus, Calia, and Lupinus. It may also inhibit heparin.</p>Formula:C10H19NOPurity:99.95%Color and Shape:SolidMolecular weight:169.26Desidustat
CAS:<p>Desidustat is an inhibitor of HIF hydroxylase.</p>Formula:C16H16N2O6Purity:98%Color and Shape:SolidMolecular weight:332.31Isonicotinic acid
CAS:<p>Isonicotinic acid is a metabolite of Isoniazid.Isonicotinic acid is a useful isomer of nicotinic acid. Isoniazid is converted to Isonicotinic acid by hydrazinolysis, with the biotransformation also to be catalyzed by cytochrome P450 enzymes, such as CYP2C.</p>Formula:C6H5NO2Purity:99.68%Color and Shape:White To Off-White Crystalline SolidMolecular weight:123.11AM-2232
CAS:<p>AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.</p>Formula:C24H20N2OPurity:99.37%Color and Shape:SolidMolecular weight:352.43IGFBP-1 Protein, Rat, Recombinant
<p>IGF-binding proteins prolong the half-life of the IGFs and have been shown to either inhibit or stimulate the growth promoting effects of the IGFs on cell culture. They alter the interaction of IGFs with their cell surface receptors. Promotes cell migration. IGFBP-1 Protein, Rat, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.9 kDa and the accession number is P21743.</p>Molecular weight:26.9 kDa (predicted)ARGX-112
CAS:<p>Temtokibart is a humanized IgG1 λ2 antibody that specifically targets IL22RA1, and is expressed by cells that are deficient in the glutamine synthetase gene.</p>Color and Shape:Odour LiquidCOR-001
CAS:<p>Ziltivekimab (COR-001) is a human IL-6 antibody, lowers CRP, and may treat inflammation and heart issues in CKD.</p>Purity:95%Color and Shape:Odour LiquidOkadaic acid
CAS:<p>Okadaic acid, a polyether marine toxin, is a highly potent and selective protein phosphatase (PP) inhibitor.</p>Formula:C44H68O13Purity:98%Color and Shape:White Crystals Or PowderMolecular weight:805Questiomycin A derivatives 18 TFA
<p>Questiomycin A derivative 18 TFA exhibits antibacterial, anticancer properties and inhibits GRP78.</p>Formula:C16H12F3N3O5Purity:98.45%Color and Shape:SoildMolecular weight:383.07Lp-PLA2-IN-16
CAS:<p>Lp-PLA2-IN-16 (Example 1) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential applications in Alzheimer's disease research [1].</p>Formula:C22H17F5N4O3Purity:98%Color and Shape:SolidMolecular weight:480.39AMPK activator C2
CAS:<p>AMPK activator C2 is an AMPK allosteric activator.</p>Formula:C7H6NO6PPurity:98%Color and Shape:SolidMolecular weight:231.1EGFR-IN-82
CAS:<p>EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of 0.09 nM for EGFR L858R/T790M/C797S and 0.06 nM for EGFR Del19/</p>Formula:C32H41BrN9O2PPurity:98%Color and Shape:SolidMolecular weight:694.6CH-100
CAS:<p>CH-100 is a Chinese herbal medicine previously used in the treatment of human hepatitis C.</p>Formula:C14H22ClNO3Color and Shape:SolidMolecular weight:287.78SR14150
CAS:<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Formula:C21H30N2OPurity:98%Color and Shape:SolidMolecular weight:326.48Ceronapril
CAS:<p>Ceronapril (SQ 29852) is an orally active and potent angiotensin-converting enzyme (ACE) inhibitor (IC50 : 36 nM) for the study of dementia and hypertension.</p>Formula:C21H33N2O6PPurity:97.94%Color and Shape:SolidMolecular weight:440.47Ref: TM-T25226
Discontinued productAnti-NASH agent 1
CAS:<p>Anti-NASH Agent 1 (Compound 3d), derived from Elafibranor, serves as a strong PPAR-α/δ agonist aimed at treating nonalcoholic steatohepatitis (NASH).</p>Formula:C26H33NO4Purity:98%Color and Shape:SolidMolecular weight:423.54HBV-IN-34
CAS:<p>HBV-IN-34 (compound 17i) is a potent inhibitor of HBsAg production, demonstrating remarkable in vitro anti-HBV efficacy with EC50 values of 0.018 μM for HBV DNA</p>Formula:C21H19F2N7Purity:98%Color and Shape:SolidMolecular weight:407.42SB251023
CAS:<p>SB251023 is an agonist of β3-adrenoceptor.</p>Formula:C28H34NO6PColor and Shape:SolidMolecular weight:511.55MitoE10
CAS:<p>MitoE10 is an effective mitochondrial targeting antioxidant.</p>Formula:C42H55O5PSColor and Shape:SolidMolecular weight:702.92FGFR1 inhibitor-10
CAS:<p>FGFR1 inhibitor-10 (Compound 4i), with an IC50 of 28 nM, effectively inhibits FGFR1 phosphorylation.</p>Formula:C26H30F3N7O2SPurity:98%Color and Shape:SolidMolecular weight:561.62ALPK1-IN-2
CAS:<p>ALPK1-IN-2 is a potent inhibitor of ALPK1 (α-kinase 1) (IC50: 95 nM). ALPK1-IN-2 inhibits NF-κB (IC50: 1.31 μM).</p>Formula:C20H18F2N4O2SColor and Shape:SolidMolecular weight:416.44(E)-Crotylbarbital
CAS:<p>(E)-Crotylbarbital, a Crotylbarbital isomer, is a sedative with hypnotic, anticonvulsant properties, aiding sleep and mental stability.</p>Formula:C10H14N2O3Purity:99.94%Color and Shape:SolidMolecular weight:210.23Fostedil
CAS:<p>Fostedil enhances heart function, maintains blood flow during partial/total coronary occlusions, and lowers aortic pressure.</p>Formula:C18H20NO3PSPurity:98%Color and Shape:SolidMolecular weight:361.4Fotemustine
CAS:<p>Fotemustine: antineoplastic, chloroethylates DNA, blocks synthesis, causes cell arrest/apoptosis, lipophilic, crosses blood-brain barrier.</p>Formula:C9H19ClN3O5PColor and Shape:SolidMolecular weight:315.69FM-24 HCl
CAS:<p>FM-24 HCl is a long acting beta-adrenergic receptor antagonist.</p>Formula:C19H30ClNO2Color and Shape:SolidMolecular weight:339.9PKUMDL-LTQ-301
CAS:<p>PKUMDL-LTQ-301 is a potent inhibitor of HipA toxin. PKUMDL-LTQ-301 also inhibits E. coli persistence.</p>Formula:C30H28N2O4Purity:98%Color and Shape:SolidMolecular weight:480.55D(-)-Octopamine CSA salt
CAS:<p>D(-)-Octopamine CSA salt is an agonist of octopamine receptors.</p>Formula:C18H27NO6SPurity:98%Color and Shape:SolidMolecular weight:385.48CGP 44532
CAS:<p>CGP 44532 a GABAB receptor agonist.</p>Formula:C4H12NO3PPurity:98%Color and Shape:SolidMolecular weight:153.12Saxitoxinol
CAS:<p>Saxitoxinol is an analog of saxitoxin, a known voltage-gated sodium channel blocker.</p>Formula:C10H17N7O3Purity:98%Color and Shape:SolidMolecular weight:283.29IDX-375
CAS:<p>IDX-375, a HCV NS5B polymerase inhibitor, is used potentially for the treatment of HCV infection.</p>Formula:C29H50N5O7PSPurity:98%Color and Shape:SolidMolecular weight:643.78Cebranopadol ((1α,4α)stereoisomer)
CAS:<p>Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.</p>Formula:C24H27FN2OPurity:98%Color and Shape:SolidMolecular weight:378.48CK176
CAS:<p>CK176 is an HIV-1 inhibitor, 11x more effective than I-XW-053 in human PBMCs.</p>Formula:C21H12IN3O2Purity:98%Color and Shape:SolidMolecular weight:465.24AKOS-22
CAS:<p>AKOS-22: potent VDAC1 inhibitor, Kd=15.4 μM; prevents mitochondrial dysfunction and apoptosis.</p>Formula:C22H21ClF3N3O3Purity:98%Color and Shape:SolidMolecular weight:467.87DPX-3778
CAS:<p>DPX-3778, a triethanolamine salt, boosts tobacco callus growth 4-5x at 0.124-2.48 μM and slows aging with IAA and kinetin.</p>Formula:C16H23ClN4O6Color and Shape:SolidMolecular weight:402.83GR 218,231
CAS:<p>GR 218,231 is a selective antagonist of D3 dopamine receptor.</p>Formula:C24H33NO3SPurity:98%Color and Shape:SolidMolecular weight:415.59Pazinaclone
CAS:<p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>Formula:C25H23ClN4O4Purity:97.79% - 99.07%Color and Shape:SolidMolecular weight:478.93Lp-PLA2-IN-15
CAS:<p>Lp-PLA2-IN-15 (example 2) is an inhibitor of lipoprotein-associated phospholipase A2 (Lp-PLA2) with potential application in Alzheimer's disease research [1].</p>Formula:C22H17F5N4O3Purity:98%Color and Shape:SolidMolecular weight:480.39KP372-1
CAS:<p>KP372-1, an Akt inhibitor, blocks PI3K signaling, arrests cell growth, and triggers apoptosis in head/neck squamous cell carcinoma.</p>Formula:C20H8N12O2Color and Shape:SolidMolecular weight:448.36Oxitropium Bromide
CAS:<p>Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.</p>Formula:C19H26BrNO4Purity:98%Color and Shape:SolidMolecular weight:412.32PSB-6426
CAS:<p>PSB-6426 is the first potent and selective human nucleoside triphosphate diphosphohydrolase-2 inhibitor.</p>Formula:C22H29N4O10PPurity:98%Color and Shape:SolidMolecular weight:540.46Bromadoline maleate
CAS:<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Formula:C19H25BrN2O5Purity:98%Color and Shape:SolidMolecular weight:441.322JAK2-IN-9
CAS:<p>Compound A8, known as JAK2-IN-9, is a selective JAK2 inhibitor with an IC50 of 5 nM.</p>Formula:C20H24N6O2SPurity:98%Color and Shape:SolidMolecular weight:412.51PPARγ-IN-2
CAS:<p>"PPARγ-IN-2 (Compound 5a), a PPARγ inhibitor, exhibits an EC50 of 0.106 μM in inhibiting TG accumulation in 3T3-L1 preadipocytes.</p>Formula:C19H21N5OPurity:98%Color and Shape:SolidMolecular weight:335.4Erythrityl Tetranitrate
CAS:<p>Erythrityl Tetranitrate, a vasodilator similar to nitroglycerin, was first in "sustained release" tablets; may cause "nitro headache."</p>Formula:C4H6N4O12Color and Shape:SolidMolecular weight:302.11Mavodelpar free base
CAS:<p>Mavodelpar free acid (REN001 free acid) is an selective agonist of PPARδ.</p>Formula:C31H30FNO5Purity:98%Color and Shape:SolidMolecular weight:515.57PS372424 HCl
CAS:<p>PS372424 activates CXCR3, triggers ERK phosphorylation, and inhibits CXCL11's effect on CD45+ cell migration in humanized mice.</p>Formula:C33H45ClN6O4Color and Shape:SolidMolecular weight:625.21PAD4-IN-2
CAS:<p>PAD4-IN-2 (compound 5i) is a PAD4 inhibitor with an IC50 value of 1.94 μM, shown to suppress tumor growth in mice through specific inhibition of the PAD4-H3cit-</p>Formula:C20H23BClN7O6Color and Shape:SolidMolecular weight:503.7BET-IN-15
CAS:<p>BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2.</p>Formula:C21H18F2N4O3SPurity:98%Color and Shape:SolidMolecular weight:444.45Radafaxine hydrochloride
CAS:<p>Radafaxine hydrochloride is an inhibitor of DAT and NET transporters, and nAChR family modulator.</p>Formula:C13H19Cl2NO2Purity:98%Molecular weight:292.2anti-TNBC agent-2
CAS:<p>Anti-TNBC agent-2 (3j), a purine derivative, acts as an anti-triple negative breast cancer (TNBC) therapeutic.</p>Formula:C28H37ClFN7OPurity:98%Color and Shape:SolidMolecular weight:542.09DprE1-IN-8
CAS:<p>DprE1-IN-8 is a potent inhibitor of DprE1, exhibiting an IC50 of less than 0.75 μM.</p>Formula:C19H12F3N5O4SPurity:98%Color and Shape:SolidMolecular weight:463.39Lp-PLA2-IN-12
CAS:<p>Lp-PLA2-IN-12 (compound 19), an Lp-PLA2 inhibitor, is utilized in researching neurodegenerative diseases including Alzheimer's disease (AD), glaucoma, age-</p>Formula:C24H23F2N5O3Purity:98%Color and Shape:SolidMolecular weight:467.47H 35-25
CAS:<p>H 35-25 is a beta 2-antagonist.</p>Formula:C13H21NOColor and Shape:SolidMolecular weight:207.31Neurokinin antagonist 1
CAS:<p>Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.</p>Formula:C38H40N4O3Purity:>99.99%Color and Shape:SolidMolecular weight:600.75(S)-Coriolic acid
CAS:<p>(S)-Coriolic acid, a 15-LOX metabolite and signaling molecule, modulates cell growth, tumor adhesion, receptor expression, and can cause mitochondrial damage.</p>Formula:C18H32O3Purity:97.67% - 98.04%Color and Shape:SolidMolecular weight:296.44ALPK1-IN-1
CAS:<p>ALPK1-IN-1 (A001) strongly inhibits ALPK1, key for innate immunity & NF-κB signaling via TIFA/TRAF.</p>Formula:C25H32N6O2SColor and Shape:SolidMolecular weight:480.63Benzovindiflupyr
CAS:<p>Benzovindiflupyr: a fungicide that inhibits SDH (IC50=5.2nM), halts S. sclerotiorum growth (EC50=0.011μg/ml), and protects crops like eggplants.</p>Formula:C18H15Cl2F2N3OColor and Shape:SolidMolecular weight:398.23CXCR4-IN-1
CAS:<p>CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, applicable for the research of various conditions such as cancer, HIV, diabetic</p>Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54BChE-IN-17
CAS:<p>BChE-IN-17 (compound 6n) is a potent, selective inhibitor of butyrylcholinesterase (BChE), demonstrating inhibitory half-maximal inhibitory concentrations (</p>Formula:C23H23BrN2O4S2Color and Shape:SolidMolecular weight:535.47Aminobutane bisphosphonate
CAS:<p>Aminobutane bisphosphonate curbs bone loss; may manage hypercalcemia in cancer.</p>Formula:C4H13NO6P2Color and Shape:SolidMolecular weight:233.1Glutaminyl Cyclase Inhibitor 4
CAS:<p>Glutaminyl Cyclase Inhibitor 4 is a potent, selective glutaminyl cyclase (QC) inhibitor (IC50: 6.1 nM). It is a potent anti-Alzheimer’s agent.</p>Formula:C22H33N5O3Purity:98%Color and Shape:SolidMolecular weight:415.53Culmerciclib
CAS:<p>Culmerciclib is a cell cycle protein-dependent kinase (CDK) inhibitor that exhibits antitumour effects.</p>Formula:C24H27FN8Color and Shape:SolidMolecular weight:446.52anti-TNBC agent-3
CAS:<p>Anti-TNBC agent-3 (compound 3g) is a compound that induces apoptosis and possesses anti-cancer cell proliferation properties.</p>Formula:C29H39F2N7OColor and Shape:SolidMolecular weight:539.66Albuterol stearate
CAS:<p>Albuterol stearate, a salt form of Albuterol, is a selective beta2 agonist for treating asthma and COPD, with 29x preference for beta2 over beta1.</p>Formula:C31H57NO5Purity:98%Color and Shape:SolidMolecular weight:523.799Fosfonet sodium
CAS:<p>Fosfonet sodium is a sodium salt of phosphonoacetic acid, effective against herpesviruses by inhibiting viral DNA polymerase.</p>Formula:C2H4NaO5PColor and Shape:SolidMolecular weight:162.01UBP1112
CAS:<p>group III mGlu receptor antagonist</p>Formula:C10H14NO5PPurity:98%Color and Shape:SolidMolecular weight:259.2YM 298198 Hydrochloride
CAS:<p>YM 298198 HCl: non-competitive mGlu1 antagonist, Ki=19 nM. Inactive on mGlu2-7, stronger than CPCCOEt.</p>Formula:C18H22N4OSColor and Shape:SolidMolecular weight:342.46Phenazolam
CAS:<p>Phenazolam is an analytical reference standard categorized as a benzodiazepine. [1] This product is intended for research and forensic applications.</p>Formula:C17H12BrClN4Color and Shape:SolidMolecular weight:387.66Trimetoquinol HCl hydrate
CAS:<p>Trimetoquinol hydrochloride possesses differential and selective beta-adrenergic properties.</p>Formula:C19H26ClNO6Color and Shape:SolidMolecular weight:399.87Dioxifedrine
CAS:<p>Dioxifedrine is a beta-2 -adrenergic agonist with bronchodilator activity.</p>Formula:C10H15NO3Color and Shape:SolidMolecular weight:197.23HPK1-IN-18
CAS:<p>HPK1-IN-18: Potent, specific inhibitor of HPK1, a MAP4K enzyme, for cancer research and treatment.</p>Formula:C24H24N4Color and Shape:LiquidMolecular weight:368.47PL265
CAS:<p>PL265 is a long-acting dual ENKephalinase inhibitor (DENKi) with analgesic potential.</p>Formula:C27H35N2O9PPurity:98%Color and Shape:SolidMolecular weight:562.55Gacyclidine
CAS:<p>Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal cord.</p>Formula:C16H25NSPurity:99.85% - 99.92%Color and Shape:SolidMolecular weight:263.44MEN11467
CAS:<p>MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.</p>Formula:C38H40N4O3Purity:>99.99%Color and Shape:SolidMolecular weight:600.75URAT1 inhibitor 5
CAS:<p>URAT1 Inhibitor 5 (compound 16) serves as a powerful inhibitor of URAT1 and is utilized in hyperuricemia research [1].</p>Formula:C18H14BrN3O2SColor and Shape:SolidMolecular weight:416.29Canlitinib
CAS:<p>Canlitinib, a tyrosine kinase inhibitor, holds potential for cancer research.</p>Formula:C33H31F2N3O7Purity:98%Color and Shape:SolidMolecular weight:619.61CGP 56999A
CAS:<p>CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.</p>Formula:C19H30NO5PPurity:98%Color and Shape:SolidMolecular weight:383.42MDL-811
CAS:<p>MDL-811, an allosteric activator of SIRT6, markedly enhances the deacetylation of histone H3 at lysine residues 9, 18, and 56 (H3K9Ac, H3K18Ac, and H3K56Ac),</p>Formula:C25H25BrCl2FN3O5S2Purity:98%Color and Shape:SolidMolecular weight:681.42Syk-IN-8
CAS:<p>Syk-IN-8 (compound 19q) functions as a Syk inhibitor with demonstrated antiproliferative effects on a variety of hematological tumor cells.</p>Formula:C23H26N10Purity:98%Color and Shape:SolidMolecular weight:442.52Anti-MI/R injury agent 1
CAS:<p>Anti-MI/R injury agent 1 (compound 18), derived from Panaxatriol, represents an orally administered, potent agent against myocardial ischemia/reperfusion (MI/R</p>Formula:C32H49NO6Color and Shape:SolidMolecular weight:543.73L 689037
CAS:<p>L 689037 is an inhibitor of leukotriene biosynthesis.</p>Formula:C36H37ClN2O4Purity:98%Color and Shape:SolidMolecular weight:597.14Py-MAA-Val-Cit-PAB-MMAE
CAS:<p>Py-MAA-Val-Cit-PAB-MMAE (AAJ8D6-PY-Val-Cit-MMAE) serves as an ADC linker for Zapadcine-3a, a broad-spectrum anti-TRAILR2 ADC with antineoplastic properties.</p>Formula:C72H111N13O16SColor and Shape:SolidMolecular weight:1446.79Azilsartan mepixetil potassium
CAS:<p>Azilsartan medoxomil potassium (QR-01019K), an angiotensin II receptor antagonist, exhibits a potent and sustained antihypertensive effect, along with a more</p>Formula:C36H33KN6O8Color and Shape:SolidMolecular weight:716.78BCR-ABL-IN-8
CAS:<p>BCR-ABL-IN-8 (compound 26f) is a BCR-ABL inhibitor featuring a trimethoxy group [1].</p>Formula:C30H33N7O5Purity:98%Color and Shape:SolidMolecular weight:571.63Antitumor agent-104
CAS:<p>Antitumor Agent-104 (Compound 9) serves as an antineoplastic by impeding DNA repair mechanisms in tumor cells, primarily through the inhibition of PARP1 enzyme</p>Formula:C31H33FN6O3Purity:98%Color and Shape:SolidMolecular weight:556.63SARS-CoV-2-IN-68
CAS:<p>SARS-CoV-2-IN-68 (compound 6C) is a covalent inhibitor of both SARS-CoV-2 PLpro and Mpro, exhibiting potent antiviral properties by targeting the Zn-finger</p>Formula:C14H12N2OSePurity:98%Color and Shape:SolidMolecular weight:303.22Antibacterial agent 157
CAS:<p>Compound B12 (Antibacterial agent 157) is a fungicidal agent that can impact protein synthesis in Botrytis cinerea.</p>Formula:C26H23BrF4N2O3Color and Shape:SolidMolecular weight:567.37PI3Kδ-IN-13
CAS:<p>PI3Kδ-IN-13 (compound 89), with an IC50 value of 2.6 nM, is an inhibitor of PI3Kδ, applicable for researching diseases involving cell proliferation, including</p>Formula:C27H39N7O4S2Color and Shape:SolidMolecular weight:589.77Immune cell migration-IN-1
CAS:<p>Immune cell migration-IN-1 (compound 2) serves as a potent inhibitor of immune cell migration, with potential research applications for mitigating conditions</p>Formula:C30H25ClN4O6SColor and Shape:SolidMolecular weight:605.06URAT1&XO inhibitor 1
CAS:<p>URAT1&XO Inhibitor 1 (compound 29) serves as a dual inhibitor with IC50 values of approximately 10 μM for URAT1 and 1.01 μM for Xanthine Oxidase.</p>Formula:C20H13N5O3SPurity:98%Color and Shape:SolidMolecular weight:403.41BTK-IN-25
CAS:<p>BTK-IN-25 (compound 71) is a potent BTK inhibitor, demonstrating an IC50 of 0.77 nM against BTK(C481S) and achieving an IC50 of 1 nM in DOHH2 cells [1].</p>Formula:C28H27F2N3O5Purity:98%Color and Shape:SolidMolecular weight:523.53FLT3-IN-19
CAS:<p>FLT3-IN-19 (Comp 50) is a potent, selective inhibitor of FLT3, demonstrating an IC50 value of 0.213 nM, and is applicable in research pertaining to acute</p>Formula:C22H26N8OColor and Shape:SolidMolecular weight:418.49CIAC001
CAS:<p>CIAC001, a pyruvate kinase PKM2 inhibitor, exhibits anti-neuroinflammatory properties.</p>Formula:C20H25N3O2Color and Shape:SolidMolecular weight:339.43Xilmenolone
CAS:<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Formula:C26H37N3O2Purity:98%Color and Shape:SolidMolecular weight:423.59STAT3-IN-18
CAS:<p>STAT3-IN-18 (compound SPP), a platinum (IV) complex featuring an axial ligand from sandalwood, suppresses the JAK2-STAT3 pathway in breast cancer (BC) cells and</p>Formula:C18H24Cl2N2O6PtPurity:98%Color and Shape:SolidMolecular weight:630.38MOR agonist-1
CAS:<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Formula:C22H26ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:404.91LM2I
CAS:<p>LM2I, a derivative of Spinosyn A (SPA), serves both as an argininosuccinate synthase (ASS1) enzyme activator and a tumor inhibitor through direct interaction</p>Formula:C47H77N3O11Color and Shape:SolidMolecular weight:860.13DiaFluo
CAS:<p>DiaFluo is a probe for protein S-sulfinylation from cells.</p>Formula:C32H32N4O9SColor and Shape:SolidMolecular weight:648.69Ref: TM-T31416
Discontinued productAntibacterial agent 160
CAS:<p>Antibacterial Agent 160 is a potent antibacterial agent that rapidly eradicates bacteria and inhibits the formation of bacterial biofilms.</p>Formula:C29H27ClFN3O6Color and Shape:SolidMolecular weight:567.99FOXM1-IN-2
CAS:<p>FOXM1-IN-2, a FOXM1 inhibitor, exhibits antineoplastic activity [1].</p>Formula:C48H47F4N7O12SColor and Shape:SolidMolecular weight:1021.99Mal-VC-PAB-PNP-CDN-A
CAS:<p>Mal-VC-PAB-PNP-CDN-A is a conjugate comprised of an agent and a linker, utilized in antibody-drug conjugates (ADC) [1] [2].</p>Formula:C51H67N17O20P2Color and Shape:SolidMolecular weight:1300.13S1P1 agonist 6
CAS:<p>Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive</p>Formula:C25H26F3NO3Purity:98%Color and Shape:SolidMolecular weight:445.47I-BET282
CAS:<p>BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).</p>Formula:C25H30N4O4Purity:98%Color and Shape:SolidMolecular weight:450.53BTK-IN-27
CAS:<p>BTK-IN-27 (example 8), a potent BTK inhibitor with an IC50 of 0.2 nM, demonstrates anti-proliferative effects in TMD8 cells with an IC50 of less than 5 nM.</p>Formula:C31H35N7O2Purity:98%Color and Shape:SolidMolecular weight:537.66Civorebrutinib
CAS:<p>Civorebrutinib (WS-413) is an inhibitor of Bruton's tyrosine kinase that exhibits antineoplastic activity [1].</p>Formula:C23H22ClN7O2Color and Shape:SolidMolecular weight:463.92Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan
CAS:<p>Mal-cyclohexane-Gly-Gly-Phe-Gly-Exatecan is a linker molecule employed in the synthesis of antibody-drug conjugates (ADCs), demonstrating potent antitumor</p>Formula:C55H60FN9O13Color and Shape:SolidMolecular weight:1074.12Cap-dependent endonuclease-IN-9
CAS:<p>Cap-dependent endonuclease-IN-9, a strong influenza inhibitor, shows low toxicity, good pharmacokinetics, and dynamic action.</p>Formula:C29H22F2N4O7SPurity:98%Color and Shape:SolidMolecular weight:608.57VMAT2-IN-2 tosylate
CAS:<p>VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].</p>Formula:C27H36F3NO6SPurity:98%Color and Shape:SolidMolecular weight:559.64Antitumor photosensitizer-1
CAS:<p>Antitumor Photosensitizer-1 (Compound 8) is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-toxicity,</p>Formula:C42H51N5O6Color and Shape:SolidMolecular weight:721.88Davelizomib
CAS:<p>Davelizomib is a proteasome inhibitor that exhibits antineoplastic activity [1].</p>Formula:C21H26BF2N3O7Purity:98%Color and Shape:SolidMolecular weight:481.25JAK-IN-34
CAS:<p>JAK-IN-34 (compound 11n) is a potent inhibitor of Janus kinases (JAKs), demonstrating IC50 values of 0.40 nM for JAK1, 0.83 nM for JAK2, 2.10 nM for JAK3,</p>Formula:C27H26N6OPurity:98%Color and Shape:SolidMolecular weight:450.53ATR-IN-24
CAS:<p>ATR-IN-24 (Compound 1) is an ATR inhibitor with demonstrated anticancer activity [1].</p>Formula:C23H26N6O2Purity:98%Color and Shape:SolidMolecular weight:418.49MDVN1003
CAS:<p>MDVN1003 inhibits BTK & PI3Kδ in B cells, blocking NHL growth; it kills lymphoma cells, not erythroblasts.</p>Formula:C22H20FN7OPurity:98%Color and Shape:SolidMolecular weight:417.44RIOK2-IN-2
CAS:<p>RIOK2-IN-2 (8) functions as an inhibitor of RIOK2, exhibiting IC50 values of 3.02 μM in MKN-1 cells and 5.34 μM in MOLT4 cells [1].</p>Formula:C27H23F3N6O2Color and Shape:SolidMolecular weight:520.51diMal-O-CH2COOH
CAS:<p>DiMal-O-CH2COOH is a cleavable linker utilized in antibody-drug conjugates (ADCs).</p>Formula:C13H12N2O7Color and Shape:SolidMolecular weight:308.24Antitumor photosensitizer-2
CAS:<p>Compound 11, also known as Antitumor Photosensitizer-2, is a potent photosensitizer with remarkable photodynamic anti-tumor properties and minimal skin photo-</p>Formula:C40H47N5O7Color and Shape:SolidMolecular weight:709.83(αR)-Cyclopropaneacetamide-Exatecan
CAS:<p>(αR)-Cyclopropaneacetamide-Exatecan (compound 2-A), an Exenotecan derivative, serves as a cytotoxic agent that effectively inhibits the proliferation of U87MG</p>Formula:C29H28FN3O6Color and Shape:SolidMolecular weight:533.55APG-2449
CAS:<p>APG-2449 is an orally active inhibitor targeting ALK, ROS1, and FAK, demonstrating antitumor efficacy in mouse models of non-small cell lung cancer (NSCLC) [1].</p>Formula:C33H42ClN5O4SPurity:98%Color and Shape:SolidMolecular weight:640.24Tauro-Obeticholic Acid sodium
CAS:<p>Tauro-obeticholic acid, a farnesoid X receptor (FXR) agonist and semisynthetic derivative of chenodeoxycholic acid, is an active metabolite of obeticholic acid.</p>Formula:C28H48NO6S·NaColor and Shape:SolidMolecular weight:549.74Omeprazole acid
CAS:<p>Omeprazole treats GERD, ulcers, Zollinger-Ellison syndrome, prevents GI bleeding; it's a proton pump inhibitor.</p>Formula:C34H32N6Na2O10S2Color and Shape:SolidMolecular weight:794.76Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE
CAS:<p>Compound S6, Mc-Alanyl-Alanyl-Asparagine-PAB-MMAE, is a potent anticancer agent specifically activated by the tumor microenvironment; it demonstrates efficacy</p>Formula:C67H101N11O16Purity:98%Color and Shape:SolidMolecular weight:1316.58Sakura 6
CAS:<p>Sakura 6, a synthetic serotonin transporter (SERT)-binding peptide, enhances the interaction between SERT and neuronal nitric oxide synthase.</p>Formula:C31H45N5O7Color and Shape:SolidMolecular weight:599.73AEF0117
CAS:<p>AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.</p>Formula:C29H40O3Purity:99.58%Color and Shape:SolidMolecular weight:436.63ROCK2-IN-6
CAS:<p>ROCK2-IN-6 (Comp A) is a selective inhibitor of ROCK2, applicable in the study and treatment of ROCK-mediated, autoimmune, and inflammatory diseases [1].</p>Formula:C26H21F2N7OPurity:98%Color and Shape:SolidMolecular weight:485.49JAK1-IN-10
CAS:<p>JAK1-IN-10 (compound 9), a cyano-substituted cyclic hydrazine derivative, functions as a potent and selective inhibitor of JAK1 [1].</p>Formula:C15H17N7Purity:98%Color and Shape:SolidMolecular weight:295.34Bi-Mc-VC-PAB-MMAE
CAS:<p>Bi-Mc-VC-PAB-MMAE is an agent-linker conjugate for antibody-drug conjugates (ADCs), featuring the linker (Fmoc-Val-Cit-PAB) and the potent tubulin inhibitor (</p>Formula:C71H104N12O18Color and Shape:SolidMolecular weight:1413.66Belfosdil
CAS:<p>Belfosdil is a blocker of antihypertensive calcium channel.</p>Formula:C27H50O7P2Purity:98%Color and Shape:SolidMolecular weight:548.63YK-029A
CAS:<p>YK-029A, an orally active EGFR mutant inhibitor, targets both EGFR T790M and EGFRex20ins mutations.</p>Formula:C27H32N8O2Purity:98%Color and Shape:SolidMolecular weight:500.6JAK-IN-27
CAS:<p>JAK-IN-27, also known as compound 1, is an orally active, potent inhibitor of the JAKS family kinases, displaying inhibitory concentrations (IC50s) of 3.0 nM</p>Formula:C20H21F2N7OPurity:98%Color and Shape:SolidMolecular weight:413.42And1-IN-1
CAS:<p>And1-IN-1, also known as compound III, is a potent inhibitor of And1 [1].</p>Formula:C15H11BCl2O2Color and Shape:SolidMolecular weight:304.96S-72
CAS:<p>S-72 acts as a microtubule polymerization inhibitor, effective in cell-free assays at concentrations of 1, 3, and 10 µM.</p>Formula:C20H22N4O3SColor and Shape:SolidMolecular weight:398.50JAK1-IN-11
CAS:<p>JAK1-IN-11 (compound 11) serves as a potent inhibitor of Janus kinases, exhibiting nanomolar inhibitory concentrations with IC50 values of 0.02 nM (JAK1) and 0.</p>Formula:C26H36N6O4SPurity:98%Color and Shape:SolidMolecular weight:528.67Igermetostat
CAS:<p>Igermetostat, an EZH2 inhibitor, is utilized both in vivo and in vitro for cancer research [1].</p>Formula:C32H46N4O4Purity:98%Color and Shape:SolidMolecular weight:550.73HBV-IN-38
CAS:<p>HBV-IN-38 (Example 193), an HBV DNA inhibitor with an EC50 value of ≤100 nM, serves as a research tool for investigating viral infections [1].</p>Formula:C18H16F3N5O4S2Purity:98%Color and Shape:SolidMolecular weight:487.48HPK1-IN-38
CAS:<p>HPK1-IN-38 (compound 15) is an inhibitor of MAP4K1/HPK1, suitable for research into disorders related to HPK1 [1].</p>Formula:C29H29N5O3Color and Shape:SolidMolecular weight:495.57PF-05236216 hydrochloride
CAS:<p>PF-05236216 hydrochloride: Brain-penetrant, potent CK1δ/ε inhibitor affecting mouse circadian rhythms.</p>Formula:C18H15FN4OColor and Shape:SolidMolecular weight:322.34LT-540-717
CAS:<p>LT-540-717 (compound 32), a potent FLT3 inhibitor (IC50=0.62 nM), exhibits antiproliferative activity and effectively inhibits various acquired FLT3 mutations,</p>Formula:C24H24N8O2Color and Shape:SolidMolecular weight:456.5Yhhu6669
CAS:<p>Yhhu6669 is an anti-HBV agent that suppresses viral DNA and replication by promoting DNA-free capsid assembly, effectively reducing HBV DNA and HBcAg levels in</p>Formula:C29H28ClFN6O3Purity:98%Color and Shape:SolidMolecular weight:563.02IDO/Tubulin-IN-2
CAS:<p>IDO/Tubulin-IN-2 inhibits TDO/tubulin, effective on U87, HepG2, A549, HCT-116, LO2 cancer cells; IC50 values 0.036-1.04 μM, boosts antitumor action.</p>Formula:C48H40N6O10Color and Shape:SolidMolecular weight:860.87Tibremciclib
CAS:<p>Tibremciclib is a cyclin-dependent kinase 4 (CDK4) inhibitor that exhibits antineoplastic properties [1].</p>Formula:C28H32F2N8Purity:98%Color and Shape:SolidMolecular weight:518.6FAP-IN-2
CAS:<p>FAP-IN-2 is a 99mTc-labeled, isonitrile-containing derivative of a fibroblast activation protein (FAPI) inhibitor suitable for tumor imaging [1].</p>Formula:C24H28F2N6O3Color and Shape:SolidMolecular weight:486.51ALPK1-IN-3
CAS:<p>ALPK1-IN-3,serves as an ALPK1 inhibitor that dampens proinflammatory gene expression in the kidney and enhances survival in animal models of sepsis-induced</p>Formula:C20H16F2N4OSPurity:98%Color and Shape:SolidMolecular weight:398.43
