Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,623 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,759 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,051 products)
- Immunology and Inflammation(3,945 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,149 products)
- Microbiology/Virology(7,672 products)
- Neuroscience(10,549 products)
- Other Inhibitors(35,857 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,693 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,743 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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CAS:SDOX, a prodrug, releases Doxorubicin selectively in high-GSH tumor cells, minimizing harm to healthy tissue.Formula:C69H97NO20S2Purity:98%Color and Shape:SolidMolecular weight:1324.63ACT-280778
CAS:ACT-280778 is a potent L/T calcium channel blocker.Formula:C41H51N3O12Color and Shape:SolidMolecular weight:777.87GLP-1R agonist 12
CAS:GLP-1R agonist 12 (Compound 123) 是一种 GLP-1R 激动剂，能够用于研究糖尿病。Formula:C34H36N6O4Color and Shape:SolidMolecular weight:592.69KF21213
CAS:KF21213 shows a high affinity for the adenosine A2A receptors (Ki=3.0 nM). KF21213 is a highly selective ligand for mapping CNS adenosine A2A receptors.Formula:C19H22N4O3Purity:98%Color and Shape:SolidMolecular weight:354.4OM-1700
CAS:OM-1700 inhibits tankyrase 1 (IC50=127 nM) and 2 (IC50=14 nM); hinders colon cancer cell growth, COLO 320DM (GI50=650 nM).Formula:C25H23FN6O2Color and Shape:SolidMolecular weight:458.49Cyanidin-3,5-O-diglucoside chloride
CAS:Antioxidant, Cyanidin-3,5-diglucoside chloride aids in glaucoma research, counters GLAST decline, degrades via hydrolysis.Formula:C27H31ClO16Purity:98%Color and Shape:Light Green PowderMolecular weight:646.98Ianthelliformisamine B TFA
CAS:Ianthelliformisamine B TFA, an antibiotic enhancer, is used to against resistant Gram-negative bacteria.Formula:C21H27Br2F6N3O6Purity:98%Color and Shape:SolidMolecular weight:691.25GSK-598809
CAS:GSK598809, a D3 receptor antagonist in Phase I trials, may lessen drug cravings by reducing reward cues.Formula:C23H25F4N5OSColor and Shape:SolidMolecular weight:495.54AD 0261
CAS:AD 0261 is a radical scavenger. It has a strong inhibitory action on the generation of lipid peroxides and superoxide anions.Formula:C27H31F2N3OPurity:98%Color and Shape:SolidMolecular weight:451.55PHD-IN-2
CAS:PHD-IN-2 (Compound 91), a potent PHD antagonist with an IC50 of less than 5 nM, effectively stimulates erythropoietin synthesis in HEP3B cells with an EC50 ofFormula:C26H27N7O4Purity:98%Color and Shape:SolidMolecular weight:501.54Phenylarsine oxide
CAS:Phenylarsine Oxide (Oxophenylarsine) is a membrane-permeable tyrosine phosphatase inhibitor with an IC50 value of 18 µM that stimulates 2-deoxyglucose transportFormula:C6H5AsOColor and Shape:SolidMolecular weight:168.03STING Agonist D61
CAS:STING agonist D61 is a compound that activates the stimulator of interferon genes (STING), leading to the induction of IFN3-inducible secreted alkalineFormula:C29H29F3N8O4Color and Shape:SolidMolecular weight:610.60δ-Tocotrienol
CAS:δ-Tocotrienol (Delta-Tocotrienol) is a potential angiogenic inhibitor.Formula:C27H40O2Purity:99.86%Color and Shape:SolidMolecular weight:396.61Ref: TM-TMA2474
1mg46.00€5mg92.00€1mL*10mM (DMSO)101.00€10mg145.00€25mg281.00€50mg423.00€100mg625.00€Ulonivirine
CAS:Ulonivirine is an orally active non-nucleoside reverse transcriptase inhibitor that exhibits high antiviral activity and can be used to study HIV-1 infection.Formula:C18H8ClF6N5O3Color and Shape:SolidMolecular weight:491.73SDH-IN-3
CAS:SDH-IN-3 is a succinate dehydrogenase (SDH) inhibitor, demonstrating potent antifungal activity with an inhibition concentration (IC50) of 7.2 μg/mL and anFormula:C15H11F2N3OSPurity:98%Color and Shape:SolidMolecular weight:319.33Fiboflapon sodium
CAS:Fiboflapon sodium, an oral 5-LOX-activating protein inhibitor, binds FLAP at 2.9 nM, inhibits LTB4 at 76 nM.Formula:C38H43N3NaO4SColor and Shape:SolidMolecular weight:660.83CDK4/6-IN-15
CAS:CDK4/6-IN-15: Oral, selective CDK4/6 inhibitor, halts cancer cell growth, G1 arrest, suppresses Rb phosphorylation.Formula:C21H27FN8SColor and Shape:SolidMolecular weight:442.56VU 0255035
CAS:VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.
Formula:C18H20N6O3S2Purity:98.09% - 98.1%Color and Shape:SolidMolecular weight:432.52WAY-612453
CAS:WAY-612453 is an active compound utilized in researching amyloid diseases and synucleinopathies.Formula:C9H8Cl2N4SColor and Shape:SolidMolecular weight:275.16Verazine
CAS:(-)-Verazine is an antifungal agent isolated from the dried roots and rhizome of Veratrum maackii Regel, which induces DNA damage in the cerebellum and cerebralFormula:C27H43NOColor and Shape:SolidMolecular weight:397.646-Methoxypurine arabinoside
CAS:6-Methoxypurine arabinoside (Ara-m), a potent inhibitor of the varicella-zoster virus (VZV), exhibits 50% inhibitory concentrations (IC50) between 0.5 and 3Formula:C11H14N4O5Color and Shape:SolidMolecular weight:282.25inS3-54A18
CAS:inS3-54A18 is an effective inhibitor of STAT3. inS3-54A18 has anticancer effects.Formula:C23H16ClNO2Purity:99.68%Color and Shape:SolidMolecular weight:373.83Ref: TM-T15582
2mg39.00€5mg62.00€1mL*10mM (DMSO)67.00€10mg87.00€25mg152.00€50mg215.00€100mg304.00€200mg427.00€HPK1-IN-12
CAS:HPK1-IN-12 is a potent inhibitor of HPK1. HPK1-IN-12 has potential for the study of HPK1-related diseases.Formula:C25H24FN5O2Color and Shape:SolidMolecular weight:445.49ASGPR ligand-1
CAS:ASGPR ligand-1 is a compound that targets the asialoglycoprotein receptor (ASGPR) and is utilized in various disease research contexts [1].Formula:C61H110N10O27Color and Shape:SolidMolecular weight:1415.585-HT2 agonist-1
CAS:Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively.Formula:C19H23ClN2O2Purity:98%Color and Shape:SolidMolecular weight:346.85Reverse transcriptase-IN-1
CAS:Reverse transcriptase-IN-1 is a diarylbenzopyrimidine (DABP) analogue and a potent inhibitor of HIV-1 nonnucleoside reverse transcriptase with an IC50of 13.7Formula:C25H17N7O2Purity:99.61%Color and Shape:SolidMolecular weight:447.45Ref: TM-T12715
1mg60.00€5mg124.00€1mL*10mM (DMSO)136.00€10mg173.00€25mg295.00€50mg425.00€100mg583.00€200mg790.00€Muraglitazar glucuronide
CAS:Muraglitazar glucuronide is a Peroxime Proliferator Activated (PPAR) Agonist that has glucose- and lipid-lowering activities.Formula:C35H36N2O13Color and Shape:SolidMolecular weight:692.67eIF4A3-IN-9
CAS:eIF4A3-IN-9, a silvestrol analogue, disrupts eIF4F complex assembly; EC50s: 29/450/80 nM (myc/tub-LUC, MB-231 cells); for cancer research.Formula:C28H27NO8Color and Shape:SolidMolecular weight:505.52Encaleret
CAS:Encaleret( JIT-305) is an antagonist of oral calcium-sensing receptor (CaSR), it is used for the treatment of osteoporosis.Formula:C29H33ClFNO4Color and Shape:SolidMolecular weight:514.03Rosoxacin
CAS:Rosoxacin (Acrosoxacin) shows antibacterial activities against a broad spectrum of Gram-negative bacteria including Neisseria gonorrhoeae (MIC90 = 0.03mg/ml).Formula:C17H14N2O3Purity:99.1%Color and Shape:SolidMolecular weight:294.3Ref: TM-T16789
1mg46.00€5mg93.00€10mg137.00€1mL*10mM (DMSO)152.00€25mg295.00€50mg522.00€100mg743.00€200mg982.00€KRAS G12C inhibitor 28
CAS:KRAS G12C Inhibitor 28 is a compound that effectively inhibits the KRAS G12C mutation, exhibiting potent antitumor effects with an inhibitory concentration (Formula:C33H36F2N5O4PColor and Shape:SolidMolecular weight:635.64BM152054
CAS:BM152054 is a potent PPARγ ligand that induces glucose utilization in peripheral tissues by enhancing insulin action.Formula:C22H18N2O4S3Purity:99.56%Color and Shape:SolidMolecular weight:470.58Cyclophostin
CAS:Cyclophostin is an irreversible inhibitor of acetylcholinesterase (AChE).Formula:C8H11O6PPurity:98%Color and Shape:SolidMolecular weight:234.14Hypusine
CAS:Hypusine is an N-terminal amino alcohol derivative of Lys occurring in bovine brain &Formula:C10H23N3O3Color and Shape:SolidMolecular weight:233.31RB-3
CAS:RB-3, a PRC1 inhibitor, binds to RING1B-BMI1f , with a K d of 2.8 μM.Formula:C24H20ClN3O2Color and Shape:SolidMolecular weight:417.89PDE5-IN-42
CAS:PDE5-IN-42 is a selective inhibitor of second-generation phosphodiesterase type 5 (PDE5).Formula:C23H31N7O3Purity:98%Color and Shape:SolidMolecular weight:453.54UNC9994 hydrochloride
CAS:UNC9994 hydrochloride is a selective β-arrestin-biased D2R agonist, Ki of 79 nM, that stimulates β-arrestin and modulates cAMP.Formula:C21H23Cl3N2OSColor and Shape:SolidMolecular weight:457.84IDO1/2-IN-1
CAS:First potent oral dual IDO1/IDO2 inhibitor with antitumor properties; IC50: 28 nM (IDO1), 144 nM (IDO2).Formula:C16H18BrFN8O4Color and Shape:SolidMolecular weight:485.27Lanabecestat camsylate
CAS:Lanabecestat camsylate is used as a BACE1 Inhibitor.Formula:C36H44N4O5SPurity:98%Color and Shape:SolidMolecular weight:644.83L-ANAP
CAS:L-ANAP is a polarity-sensitive and genetically encodable fluorescent unnatural amino acid.Formula:C15H16N2O3Purity:98%Color and Shape:SolidMolecular weight:272.3RET-IN-25
CAS:RET-IN-25 (compound 6b) is an anticancer RET kinase inhibitor that demonstrates efficacy against medullary thyroid carcinoma (MTC), exhibiting half-maximalFormula:C22H17N3O5SColor and Shape:SolidMolecular weight:435.45Makaluvamine A
CAS:Makaluvamine A comes from the fruiting bodies of Didymium bahiense that act as active anti-cancer agents and DNA topo II inhibitors.Formula:C11H11N3OColor and Shape:SolidMolecular weight:201.22ZLN024
CAS:ZLN024 is an activator of AMPK allosteric.Formula:C13H13BrN2OSPurity:99.751%Color and Shape:SolidMolecular weight:325.22Ref: TM-T13411
1mg93.00€5mg177.00€1mL*10mM (DMSO)178.00€10mg269.00€25mg429.00€50mg610.00€100mg820.00€200mg1,071.00€Aminoguanidine hemisulfate
CAS:Aminoguanidine hemisulfate, an inhibitor of nitric oxide synthases (NOS) and reactive oxygen species (ROS), effectively suppresses ANE-induced ROS production inFormula:CH6N4H2SO4Purity:98%Color and Shape:SolidMolecular weight:123.115Phenethicillin sodium
CAS:Phenethicillin sodium (α-Phenoxyethylpenicillin) is a penicillin-class antibiotic that exhibits antimicrobial activity [1].Formula:C17H19N2NaO5SColor and Shape:SolidMolecular weight:386.41-Deazaadenosine
CAS:1-Deazaadenosine, an adenosine deaminase inhibitor (Ki: 0.66 μM), may treat cancer, particularly lymphoproliferative disorders.Formula:C11H14N4O4Purity:98%Color and Shape:SolidMolecular weight:266.25GS-6201
CAS:GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formula:C21H21F3N6O2Purity:99.78% - 99.94%Color and Shape:SolidMolecular weight:446.43Ref: TM-T15418
1mg34.00€5mg71.00€1mL*10mM (DMSO)78.00€10mg114.00€25mg235.00€50mg380.00€100mg572.00€200mg805.00€Lilopristone
CAS:Lilopristone is an antagonist of progesterone.Formula:C29H37NO3Purity:98%Color and Shape:SolidMolecular weight:447.61Enpp-1-IN-4
CAS:Enpp-1-IN-4: potent enpp-1 inhibitor with potential in cancer research. See patent WO2019177971A1, compound 1.Formula:C19H19N5O5SColor and Shape:SolidMolecular weight:429.45CDK9-IN-29
CAS:CDK9-IN-29 (compound Z11) is a potent inhibitor of CDK9, exhibiting high kinase selectivity and an IC50 value of 3.20 nM.Formula:C29H33F2N5O4Purity:98%Color and Shape:SolidMolecular weight:553.6
