Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,904 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,137 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,423 products)
- Other Inhibitors(35,848 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66516 products of "Inhibitors"
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Lometrexol
CAS:Lometrexol (LY 264618) is an antifolate that inhibits GARFT, blocks purine synthesis, induces apoptosis, and has anticancer properties.Formula:C21H25N5O6Purity:97.76% - 99.56%Color and Shape:SolidMolecular weight:443.45Ref: TM-T15826
1mg84.00€5mg178.00€10mg295.00€25mg505.00€50mg747.00€100mg1,035.00€200mg1,378.00€1mL*10mM (DMSO)203.00€INCB054329
CAS:INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.Formula:C19H16N4O3Purity:99.52%Color and Shape:SolidMolecular weight:348.36NRX-103094
CAS:NRX-103094 boosts β-catenin binding to SCFβ-TrCP ligase with EC50 62 nM and Kd 0.6 nM.Formula:C20H11Cl2F3N2O4SPurity:99.13%Color and Shape:SolidMolecular weight:503.28BCL6-IN-3
CAS:BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.Formula:C24H31ClF2N6O2Purity:98.17%Color and Shape:SolidMolecular weight:508.99Ref: TM-T10487
1mg109.00€5mg241.00€10mg355.00€25mg532.00€50mg745.00€100mg1,018.00€500mgTo inquire1mL*10mM (DMSO)370.00€Dazostinag disodium
CAS:Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.Formula:C21H20F2N8Na2O10P2S2Purity:98.84% - 99.96%Color and Shape:SolidMolecular weight:754.48BAY-3827
CAS:BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.Formula:C27H25FN6OPurity:99.90%Color and Shape:SolidMolecular weight:468.53Ref: TM-T73350
1mg52.00€5mg113.00€10mg177.00€25mg334.00€50mg560.00€100mg792.00€500mg1,575.00€1mL*10mM (DMSO)117.00€Enbezotinib
CAS:Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.Formula:C21H21FN6O3Purity:99.84%Color and Shape:SolidMolecular weight:424.43Ref: TM-T62285
1mg77.00€5mg166.00€10mg253.00€25mg414.00€50mg567.00€100mg745.00€1mL*10mM (DMSO)182.00€SDZ 220-040
CAS:SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂，可诱导根系生长的部分无重力模式 。Formula:C16H16Cl2NO6PPurity:98.13%Color and Shape:SolidMolecular weight:420.18NRX-252114
CAS:NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).Formula:C22H12Cl2F3N3O2SPurity:99.70%Color and Shape:SolidMolecular weight:510.32KU-60019
CAS:KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).
Formula:C30H33N3O5SPurity:98.05% - 98.50%Color and Shape:SolidMolecular weight:547.67Tigemonam
CAS:Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.Formula:C12H15N5O9S2Purity:97.71% - >99.99%Color and Shape:SolidMolecular weight:437.41LY2979165
CAS:LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.Formula:C13H22N6O6SPurity:98.41%Color and Shape:SolidMolecular weight:390.42ELOVL1-IN-2
CAS:ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).Formula:C18H15FN2OPurity:99.94%Color and Shape:SolidMolecular weight:294.32DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).Formula:C22H24FN3O3Purity:98.22% - 99.74%Color and Shape:SolidMolecular weight:397.44Umibecestat
CAS:Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.Formula:C19H15ClF7N5O2Purity:99.88%Color and Shape:SolidMolecular weight:513.8Ref: TM-T13253
1mg163.00€5mg334.00€10mg485.00€25mg807.00€50mg1,099.00€100mg1,485.00€1mL*10mM (DMSO)376.00€Darizmetinib
CAS:Darizmetinib (HRX215) is an MKK4 inhibitor.Formula:C21H17F2N5O3SPurity:98.03% - 99.57%Color and Shape:SolidMolecular weight:457.45Ref: TM-T72956
1mg69.00€2mg89.00€5mg147.00€10mg224.00€25mg324.00€50mg400.00€100mg587.00€1mL*10mM (DMSO)148.00€AM103
CAS:AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).Formula:C36H38N3NaO4SPurity:99.75%Color and Shape:SolidMolecular weight:631.76GLPG0974
CAS:GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.Formula:C25H25ClN2O4SPurity:99.8%Color and Shape:SolidMolecular weight:484.99Cap-dependent endonuclease-IN-1
CAS:Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.Formula:C27H22F2N2O6SPurity:99.53% - 99.61%Color and Shape:SolidMolecular weight:540.54CP-642931
CAS:CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.Formula:C17H25N7OPurity:99.67% - >99.99%Color and Shape:SolidMolecular weight:343.43Evixapodlin
CAS:Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.Formula:C34H36Cl2N8O4Purity:97.02%Color and Shape:SolidMolecular weight:691.61Ref: TM-T36487
1mg111.00€5mg264.00€10mg424.00€25mg747.00€50mg1,008.00€100mg1,359.00€200mg1,833.00€1mL*10mM (DMSO)405.00€Treprostinil diethanolamine
CAS:Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,Formula:C27H45NO7Purity:99.86%Color and Shape:SolidMolecular weight:495.65AKT Kinase Inhibitor
CAS:AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.Formula:C16H19N7O3Purity:97.83% - 99.13%Color and Shape:SolidMolecular weight:357.37Ref: TM-T10276
1mg129.00€5mg313.00€10mg537.00€25mg840.00€50mg1,125.00€100mg1,521.00€1mL*10mM (DMSO)341.00€Tuvusertib
CAS:Tuvusertib (M1774), an oral ATR inhibitor (Ki<1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.Formula:C16H12F2N8OPurity:98.44% - 99.66%Color and Shape:SolidMolecular weight:370.32Ref: TM-T10406
1mg58.00€5mg124.00€10mg187.00€25mg363.00€50mg505.00€100mg717.00€1mL*10mM (DMSO)142.00€D75-4590
CAS:D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.Formula:C21H27N5Purity:98.56% - 98.85%Color and Shape:SolidMolecular weight:349.47Ref: TM-T61194
5mg39.00€10mg62.00€25mg122.00€50mg187.00€100mg269.00€200mg358.00€1mL*10mM (DMSO)46.00€AChE-IN-26
CAS:AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).
Formula:C21H21BrN2O3Purity:99.24% - 99.85%Color and Shape:SoildMolecular weight:429.31MAO-B-IN-17
CAS:MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.Formula:C17H17F2NO2Purity:99.41%Color and Shape:SoildMolecular weight:305.32O-Propargyl-Puromycin
CAS:O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.Formula:C24H29N7O5Purity:97.83% - 99.29%Color and Shape:SolidMolecular weight:495.53NRX-1532
NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.Formula:C16H11F3N4O2Purity:98.95% - 99.94%Color and Shape:SolidMolecular weight:348.28Ref: TM-T61172
1mg147.00€5mg358.00€10mg597.00€25mg1,153.00€50mg1,549.00€100mg2,088.00€500mg4,185.00€1mL*10mM (DMSO)394.00€Pocenbrodib
CAS:Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.Formula:C28H32FN3O6Purity:98.48% - 99.54%Color and Shape:SolidMolecular weight:525.57BODIPY FL prazosin
CAS:BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.
Formula:C28H32BF2N7O3Purity:97.27%Color and Shape:SolidMolecular weight:563.41Vecabrutinib
CAS:Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.Formula:C22H24ClF4N7O2Purity:99.74%Color and Shape:SolidMolecular weight:529.92Ref: TM-T17220
1mg82.00€5mg177.00€10mg289.00€25mg470.00€50mg623.00€100mg874.00€1mL*10mM (DMSO)207.00€Zotizalkib
CAS:TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.Formula:C21H20F3N5O3Purity:98.7%Color and Shape:SolidMolecular weight:447.41Ref: TM-T9414
1mg114.00€5mg268.00€10mg439.00€25mg879.00€50mg1,395.00€100mg1,873.00€1mL*10mM (DMSO)303.00€LLY-283
CAS:LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.Formula:C17H18N4O4Purity:99.49%Color and Shape:SolidMolecular weight:342.35GSK3368715 dihydrochloride
CAS:GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.Formula:C20H40Cl2N4O2Purity:99.66% - 99.66%Color and Shape:SolidMolecular weight:439.46KI696
CAS:KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.Formula:C28H30N4O6SPurity:99.74%Color and Shape:SolidMolecular weight:550.63Ref: TM-T11758L
1mg137.00€5mg281.00€10mg423.00€25mg707.00€50mg1,018.00€100mg1,468.00€200mg1,963.00€1mL*10mM (DMSO)341.00€DRB18
CAS:DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.Formula:C22H23ClN2O2Purity:99.54%Color and Shape:SolidMolecular weight:382.88Ref: TM-T22317
1mg89.00€5mg215.00€10mg340.00€25mg687.00€50mg1,108.00€100mg1,485.00€500mg2,962.00€1mL*10mM (DMSO)236.00€BMS 299897
CAS:BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.Formula:C24H21ClF3NO4SPurity:99.82%Color and Shape:SolidMolecular weight:511.94FABPs ligand 6
CAS:FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.Formula:C28H27FN2O3Purity:97.45%Color and Shape:SolidMolecular weight:458.52BLU2864
CAS:BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.Formula:C24H19F3N4O2Purity:97.58% - 99.92%Color and Shape:SoildMolecular weight:452.43(+)-Tetrabenazine
CAS:(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-foldFormula:C19H27NO3Purity:98.69%Color and Shape:SolidMolecular weight:317.42EZM0414
CAS:EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.Formula:C22H29FN4O2Purity:99.58%Color and Shape:SolidMolecular weight:400.49SY-5609
CAS:SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.Formula:C23H26F3N6OPPurity:99.34% - >99.99%Color and Shape:SolidMolecular weight:490.46Ref: TM-T36038
1mg139.00€2mg200.00€5mg343.00€10mg553.00€25mgTo inquire50mgTo inquire1mL*10mM (DMSO)373.00€CK2 inhibitor 2
CAS:CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.Formula:C21H17ClN4O2Purity:99.02%Color and Shape:SolidMolecular weight:392.84Ref: TM-T35557
1mg62.00€5mg138.00€10mg215.00€25mg425.00€50mg637.00€100mg853.00€200mg1,153.00€1mL*10mM (DMSO)152.00€PD 151746
CAS:PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.Formula:C11H8FNO2SPurity:98.63% - ≥95%Color and Shape:SolidMolecular weight:237.25SR 11302
CAS:SR 11302 is an inhibitor of activator protein-1 (AP-1).Formula:C26H32O2Purity:98.65%Color and Shape:SolidMolecular weight:376.53Ref: TM-T23384
1mg93.00€5mg137.00€10mg205.00€25mg356.00€50mg587.00€100mg888.00€1mL*10mM (DMSO)150.00€10-Methoxycamptothecin
CAS:10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.Formula:C21H18N2O5Purity:98.36%Color and Shape:SolidMolecular weight:378.38BAY-8400
BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy inFormula:C21H17F2N5OPurity:99.53%Color and Shape:SolidMolecular weight:393.39Ref: TM-T9498
1mg80.00€5mg147.00€10mg215.00€25mg439.00€50mg750.00€100mg1,009.00€1mL*10mM (DMSO)161.00€BRD0639
CAS:BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Formula:C21H22ClN5O4SPurity:99.85%Color and Shape:SolidMolecular weight:475.95Durlobactam sodium salt
CAS:Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.Formula:C8H10N3NaO6SPurity:97.01% - 99.03%Color and Shape:SolidMolecular weight:299.23
