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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66618 products of "Inhibitors"

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  • 3-O-β-D-Glucopyranosylplatycodigenin

    CAS:
    <p>3-O-beta-D-Glucopyranosylplatycodigenin is isolated from the roots of Platycodon grandiflorum.</p>
    Formula:C36H58O12
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:682.84
  • (+)-JQ-1

    CAS:
    <p>(+)-JQ-1 (JQ1) is a BET bromine domain inhibitor that inhibits BRD4 (1/2) (IC50=77/33 nM) with specificity and reversibility.</p>
    Formula:C23H25ClN4O2S
    Purity:97.57% - ≥95%
    Color and Shape:Solid
    Molecular weight:456.99
  • TSPC

    CAS:
    <p>TSPC is an inhibitor for GA perception by in vitro and in planta evaluations.</p>
    Formula:C9H5N3O2S2
    Purity:98.58%
    Color and Shape:Solid
    Molecular weight:251.28
  • Solifenacin

    CAS:
    Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,
    Formula:C23H26N2O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:362.46
  • Corynoxeine

    CAS:
    <p>Corynoxeine inhibits ERK1/2, curbs VSMC growth induced by PDGF-BB, and may prevent vascular diseases and restenosis post-angioplasty.</p>
    Formula:C22H26N2O4
    Purity:98.61% - 99.73%
    Color and Shape:Solid
    Molecular weight:382.45
  • GS-441524

    CAS:
    <p>GS-441524 treatment of cats with naturally occurring feline infectious peritonitis.</p>
    Formula:C12H13N5O4
    Purity:98.78% - 99.75%
    Color and Shape:Solid
    Molecular weight:291.26
  • Pyridoxal 5'-phosphate monohydrate

    CAS:
    <p>Pyridoxal 5'-phosphate monohydrate is an active vitamin B6 metabolite</p>
    Formula:C8H12NO7P
    Purity:98.94% - 99.05%
    Color and Shape:Slightly Yellow Powder
    Molecular weight:265.16
  • Pemirolast

    CAS:
    <p>Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.</p>
    Formula:C10H8N6O
    Color and Shape:Solid
    Molecular weight:228.21
  • H3B-5942

    CAS:
    <p>H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).</p>
    Formula:C31H34N4O2
    Purity:99.21% - ≥95%
    Color and Shape:Solid
    Molecular weight:494.63
  • Tetradehydrothalictrifoline

    CAS:
    <p>Tetradehydrothalictrifoline is a nature product.</p>
    Formula:C21H20NO4
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:350.39
  • NRC-2694 hydrochloride

    CAS:
    <p>NRC-2694 hydrochloride is an epidermal growth factor receptor (EGFR) antagonist potentially for the treatment of solid tumors.</p>
    Formula:C24H27ClN4O3
    Color and Shape:Solid
    Molecular weight:454.95
  • Phenethyl ferulate

    CAS:
    <p>Phenethyl ferulate is a chemopreventive against colon cancer, enhancing apoptosis in tumors and inhibiting COX/5-LOX (IC50: 4.35/5.75 μM).</p>
    Formula:C18H18O4
    Purity:99.88% - 99.91%
    Color and Shape:Solid
    Molecular weight:298.33
  • MSX-127

    CAS:
    <p>MSX-127 elicites positive response in peptide CXCR4.</p>
    Formula:C16H24N2O4
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:308.37
  • (S)-Afatinib

    CAS:
    <p>(S)-Afatinib (BIBW2992) is an irreversible EGFR family inhibitor with IC50s of 0.5/0.4/10/14/1 nM for EGFRwt, L858R, L858R/T790M, HER2, and HER4, respectively.</p>
    Formula:C24H25ClFN5O3
    Purity:99.22% - >99.99%
    Color and Shape:Off-White Solid
    Molecular weight:485.94
  • 26RFa acetate


    26RFa acetate is a hypothalamic neuropeptide with orexigenic activity in mammals[1].
    Formula:C129H201N37O38
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:2878.2
  • Abafungin

    CAS:
    <p>Abafungin (Bay w 6341) is an antifungal agent with a broad-spectrum.</p>
    Formula:C21H22N4OS
    Purity:98.11%
    Color and Shape:Solid
    Molecular weight:378.49
  • Conivaptan hydrochloride

    CAS:
    <p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>
    Formula:C32H26N4O2·HCl
    Purity:98.33% - 99.86%
    Color and Shape:Solid
    Molecular weight:535.04
  • SYR127063

    CAS:
    <p>SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a reactive conformation.</p>
    Formula:C23H20ClF3N4O3
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:492.88
  • Fasudil hydrochloride hydrate

    CAS:
    <p>Fasudil HCl hydrate is a ROCK inhibitor that hinders mature CCM development and lowers portal pressure in cirrhotic rats.</p>
    Formula:C28H38Cl2N6O5S2
    Color and Shape:Solid
    Molecular weight:673.67
  • TRV-120027 TFA


    <p>TRV-120027 TFA is an angiotensin II–mediated vasoconstriction inhibitor and increases cardiomyocyte contractility.</p>
    Formula:C45H68F3N13O12
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:1040.1
  • Brexpiprazole HCl

    CAS:
    <p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>
    Formula:C25H27N3O2S·xHCl
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:433.6
  • Chebulic acid

    CAS:
    <p>Chebulic acid, a phenolcarboxylic acid compound isolated from Terminalia chebula, has potent anti-oxidant activity,which breaks the cross-links of proteins</p>
    Formula:C14H12O11
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:356.24
  • Sodium Glucoheptonate

    CAS:
    <p>Sodium Glucoheptonate: Used in Tc-99m radio-labeling, brain/kidney imaging, brain-tumor detection, metal cleaning, and etching.</p>
    Formula:C7H13NaO8
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:248.16
  • Saracatinib

    CAS:
    <p>Saracatinib (AZD0530) (AZD0530) is an effective Src inhibitor (IC50: 2.7 nM), and effective to Lck, Fyn, Lyn, Blk, Fgr and c-Yes.</p>
    Formula:C27H32ClN5O5
    Purity:98% - 99.63%
    Color and Shape:Solid
    Molecular weight:542.03
  • Smadl/5 ubiquitinatio activator 1

    CAS:
    <p>1-ethyl-6-fluoroquinoline derivative; used in molecular structures; inhibits SMURF1.</p>
    Formula:C25H26FN3O4
    Purity:98.71%
    Color and Shape:Solid
    Molecular weight:451.49
  • Deferitazole magnesium

    CAS:
    <p>Deferitazole magnesium is a potential chelator for iron overload treatment.</p>
    Formula:C18H25MgNO8S
    Color and Shape:Solid
    Molecular weight:439.76
  • SR8278

    CAS:
    <p>SR8278 is an REV-ERBα antagonist(EC50 = 0.47 μM), blocking activation of the receptor by the synthetic agonist GSK 4112</p>
    Formula:C18H19NO3S2
    Purity:99.44% - 99.73%
    Color and Shape:Solid
    Molecular weight:361.48
  • Thalidomide-O-amido-C6-NH2 TFA

    CAS:
    Thalidomide-O-amido-C6-NH2 TFA (Cereblon Ligand-Linker Conjugates 11 TFA), a synthesized E3 ligase ligand-linker conjugate containing a Thalidomide-based
    Formula:C46H53F6N8O16
    Purity:95.16%
    Color and Shape:Solid
    Molecular weight:1087.95
  • 2-(4-methoxyphenyl)-2-oxoethyl 2-hydroxy-5-methylbenzoate

    CAS:
    <p>Pro-neurotropic drug boosts brain acetylcholine synthesis and release, inhibits breakdown.</p>
    Formula:C17H16O5
    Purity:98.68%
    Color and Shape:Solid
    Molecular weight:300.31
  • Grapiprant

    CAS:
    Grapiprant (AAT-007) is a selective EP4 receptor antagonist.
    Formula:C26H29N5O3S
    Purity:99.49% - 99.843%
    Color and Shape:Solid
    Molecular weight:491.61
  • Vandetanib

    CAS:
    Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 and EGFR.
    Formula:C22H24BrFN4O2
    Purity:99.7% - >99.99%
    Color and Shape:White Solid
    Molecular weight:475.35
  • Eflornithine hydrochloride hydrate

    CAS:
    Eflornithine hydrochloride hydrate (DFMO hydrochloride hydrate) is an ornithine decarboxylase (ODC) inhibitor with antitumor activity. Cost-effective and quality-assured.
    Formula:C6H15ClF2N2O3
    Purity:99% - 99.61%
    Color and Shape:White Solid
    Molecular weight:236.64
  • Dodecyl gallate

    CAS:
    <p>Dodecyl gallate (Progallin LA) is the ester of gallic acid and dodecanol. As a food additive, it is used as a preservative and antioxidant.</p>
    Formula:C19H30O5
    Purity:99.74%
    Color and Shape:White Or Creamy-White Odourless Solid
    Molecular weight:338.44
  • VK-II-36

    CAS:
    <p>VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.</p>
    Formula:C26H26N2O5
    Purity:99.12%
    Color and Shape:Solid
    Molecular weight:446.49
  • β-catenin-IN-2

    CAS:
    <p>β-catenin-IN-2 is a potent inhibitor of β-catenin that can be used in colorectal cancer research.</p>
    Formula:C15H14FN3
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:255.29
  • (Z)-LFM-A13

    CAS:
    (Z)-LFM-A13(IC50=2.5 μM), a specific Bruton's tyrosine kinase (BTK), is more than 100-fold specificity than other protein kinases, such as JAK1, JAK2, HCK, EGFR, and IRK.
    Formula:C11H8Br2N2O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:360
  • APS-2-79

    CAS:
    <p>APS-2-79: KSR-dependent MEK inhibitor, blocks ATP biotin at KSR2, IC50 of 120 nM, disrupts Ras-MAPK signaling.</p>
    Formula:C23H21N3O3
    Color and Shape:Solid
    Molecular weight:387.43
  • DOPEXAMINE

    CAS:
    <p>Dopexamine is a dopaminergic agonist</p>
    Formula:C22H32N2O2
    Purity:99.42%
    Color and Shape:Solid
    Molecular weight:356.5
  • Bayogenin

    CAS:
    <p>Bayogenin is an alfalfa saponin, Bayogenin shows moderate potency of glycogen phosphorylase inhibition.</p>
    Formula:C30H48O5
    Purity:99.69% - 99.76%
    Color and Shape:Solid
    Molecular weight:488.7
  • TM5007

    CAS:
    <p>TM5007 is a poent inhibitor of plasminogen activator inhibitor-1 (PAI-1; IC50 of 29 uM).</p>
    Formula:C24H20N2O6S4
    Purity:96.91%
    Color and Shape:Solid
    Molecular weight:560.69
  • Syringaresinol diglucoside

    CAS:
    <p>Syringaresinol diglucoside (Syringaresinol-di-O-glucoside) protects the animals from the stress-induced decreases in sex behaviours and in rectal temperature.</p>
    Formula:C34H46O18
    Purity:98.59% - 99.77%
    Color and Shape:Solid
    Molecular weight:742.72
  • Pentamidine dimesylate

    CAS:
    <p>Pentamidine dimesylate blocks (Ca)S100B-p53, aiding p53 activity against melanoma.</p>
    Formula:C20H28N4O5S
    Color and Shape:Solid
    Molecular weight:436.53
  • Cilobradine

    CAS:
    <p>Cilobradine is an HCN Channel blocker; an open channel blocker of neuronal Ih and related cardiac If channels.</p>
    Formula:C28H38N2O5
    Color and Shape:Solid
    Molecular weight:482.61
  • AMG-208

    CAS:
    <p>AMG-208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.</p>
    Formula:C22H17N5O2
    Purity:98.56%
    Color and Shape:Solid
    Molecular weight:383.4
  • 4-Isopropylbenzyl Alcohol

    CAS:
    <p>4-Isopropylbenzyl Alcohol (Cuminic alcohol) is a natural product,with insecticidal effect.</p>
    Formula:C10H14O
    Purity:99.01%
    Color and Shape:Less To Pale Yellow Clear Liquid Colorless To Pale Yellow Clear Liquid
    Molecular weight:150.22
  • I-49 free base


    I-49 free base (Pyrido[4,3-d]pyrimidin-7(6H)-one, 2-methyl-4-[[(1R)-1-[2-methyl-3-(trifluoromethyl)phenyl]ethyl]amino]-6-(tetrahydro-2H-pyran-4-yl)-) is a novel
    Formula:C23H26ClF3N4O2
    Purity:99.64% - 99.88%
    Color and Shape:Solid
    Molecular weight:482.92
  • N-Oleoyl glycine

    CAS:
    <p>N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated Akt</p>
    Formula:C20H37NO3
    Purity:97.43%
    Color and Shape:Solid
    Molecular weight:339.51
  • Dynasore

    CAS:
    <p>Dynasore, a cell-permeable dynamin inhibitor, blocks GTPase of dynamin 1/2 and Drp1 (IC50: 15 μM) without affecting other small GTPases.</p>
    Formula:C18H14N2O4
    Purity:95.85% - 99.22%
    Color and Shape:Solid
    Molecular weight:322.31
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Formula:C17H16FN3
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:281.33
  • Palmatine

    CAS:
    <p>Palmatine, also known as Burasaine, inhibits dopamine production and may treat flavivirus, jaundice, dysentery, hypertension, and liver issues.</p>
    Formula:C21H22NO4
    Purity:96.28% - 99.49%
    Color and Shape:Solid
    Molecular weight:352.4