Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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Flomoxef sodium
CAS:Flomoxef sodium, an antibiotic belonging to the oxacephem group, exhibits excellent activity against a broad spectrum of Gram-positive bacteria.Formula:C15H17F2N6NaO7S2Purity:99.28%Color and Shape:SolidMolecular weight:518.44(S)-Tedizolid
CAS:(S)-Tedizolid is the S-enantiomer of Tedizolid. Tedizolid is a novel oxazolidinone with activity against Gram-positive pathogens.Formula:C17H15FN6O3Purity:98%Color and Shape:SolidMolecular weight:370.34ROC-325
CAS:ROC-325: orally active autophagy inhibitor with anticancer effects, induces kidney cancer cell death; selective action.Formula:C28H27ClN4OSPurity:99.26%Color and Shape:SolidMolecular weight:503.06UPF-523
CAS:group I metabotropic glutamate receptors (mGlu1a) antagonistFormula:C11H11NO4Purity:98%Color and Shape:White SolidMolecular weight:221.21mHTT-IN-2
CAS:mHTT-IN-2 (compound 27) is a potent inhibitor of mutant huntingtin protein (mHTT), with an EC50 value of 0.066 μM.Formula:C20H22FN7OPurity:98%Color and Shape:SolidMolecular weight:395.43Detomidine
CAS:Detomidine is a nonnarcotic, synthetic α2-adrenergic agonist. Detomidine produces dose-dependent sedative and analgesic effects.Formula:C12H14N2Purity:98%Color and Shape:White Crystalline PowderMolecular weight:186.25Anti-inflammatory agent 47
CAS:Flo8, an anti-inflammatory and antioxidant agent, effectively suppresses the release of reactive oxygen species (ROS) and nitric oxide (NO) while inhibitingFormula:C25H18N2O3Purity:98%Color and Shape:SolidMolecular weight:394.42NF-κB-IN-8
CAS:NF-κB-IN-8 is a competitive antagonist of LPS for MD-2 binding, and it impedes the expression of inflammatory factors by engaging MD-2.Formula:C24H21N3O3Purity:98%Color and Shape:SolidMolecular weight:399.44BPH-1358 free base
CAS:BPH-1358 inhibits UPPS (IC50: 110 nM) and FPPS (IC50: 1.8 µM), effective against S. aureus (MIC ~250 ng/mL).Formula:C32H28N6O2Purity:98%Color and Shape:SolidMolecular weight:528.6Irbesartan HCl
CAS:Irbesartan: angiotensin II blocker; treats hypertension by inhibiting receptor binding.Formula:C25H29ClN6OPurity:98%Color and Shape:SolidMolecular weight:465PARP-1-IN-2
CAS:PARP-1-IN-2 is a potent PARP1 inhibitor that crosses the blood-brain barrier (IC50: 149 nM).PARP-1-IN-2 showed significant antiproliferative activity against
Formula:C22H15Cl2N3O2Purity:98.82%Color and Shape:SolidMolecular weight:424.28GSK3-IN-3
CAS:GSK3-IN-3 is a mitochondrial autophagy (mitophagy) inducer and GSK-3 inhibitor (IC50: 3.01 μM) that induces parkin-dependent mitochondrial autophagy.
Formula:C24H35N3O4Purity:99.37%Color and Shape:SolidMolecular weight:429.55Glesatinib hydrochloride
CAS:Glesatinib hydrochloride is an orally active and potent dual inhibitor of MET/SMO.Formula:C31H28ClF2N5O3S2Purity:98%Color and Shape:SolidMolecular weight:656.16AMC-01
CAS:AMC-01 has potential antiviral activity and induces dose- and time-dependent inactivation of eIF2-α via phosphorylation of serine residue 51.Formula:C27H27BrN2O6Purity:99.95%Color and Shape:SolidMolecular weight:555.42Bms 188107
CAS:Bms 188107 is a calcium antagonist, it has cardioprotective effects.Formula:C25H26N2O4Purity:98%Color and Shape:SolidMolecular weight:418.48Algestone
CAS:Algestone is a synthetic progestational dihydroxy derivative with anti-inflammatory properties.Formula:C21H30O4Purity:98%Color and Shape:White Or White Crystalline PowderMolecular weight:346.46InhA-IN-3
CAS:InhA-IN-3 (TU13) is a Mycobacterium tuberculosis InhA (enoyl ACP reductase) inhibitor for the study of Mycobacterium tuberculosis infection.Formula:C14H12ClN3O2SPurity:99.48%Color and Shape:SolidMolecular weight:321.78(Rac)-WAY-161503
CAS:(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.Formula:C11H11Cl2N3OPurity:99.51%Color and Shape:SolidMolecular weight:272.13Jineol
CAS:Jineol (NSC-694081) is a quinoline alkaloid from Scolopendra subspinipes. Jineol shows cytotoxic activity against the growth of human tumor cell lines in vitro.Formula:C9H7NO2Purity:99.55%Color and Shape:SolidMolecular weight:161.16Ref: TM-T32291
1mg56.00€5mg133.00€10mg205.00€25mg350.00€50mg515.00€100mg732.00€200mg973.00€1mL*10mM (DMSO)105.00€UR-3216
CAS:UR-3216 is a prodrug, selectively antagonizing GPIIb/IIIa receptors orally, with its active form, UR-2992, binding tightly to platelets.Formula:C27H29N7O7Purity:98%Color and Shape:SolidMolecular weight:563.56MRS1186
CAS:MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).Formula:C16H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:341.75Cinperene
CAS:Cinperene is an atropine-like compound that can block pilocarpine-induced salivation and lacrimation.Formula:C25H28N2O2Purity:98%Color and Shape:SolidMolecular weight:388.5Momelotinib Mesylate
CAS:Momelotinib Mesylate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity versus JAK3.Formula:C24H26N6O5SPurity:98%Color and Shape:SolidMolecular weight:510.57AHR antagonist 5
CAS:Potent, oral AHR blocker from WO2018195397; IC50 < 0.5μM; hinders tumor growth with anti-PD-1.Formula:C25H27Cl3FN7Purity:98%Color and Shape:SolidMolecular weight:550.89HCV-IN-3
CAS:HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor (IC50: 20 μM; Kd: 29 μM).Formula:C13H11F2NOPurity:98%Color and Shape:SolidMolecular weight:235.23RyRs activator 3
CAS:RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.Formula:C23H19BrCl2N6O3Purity:98%Color and Shape:SolidMolecular weight:578.25TC-C 14G
CAS:CB1 receptor inverse agonistFormula:C24H17Cl2F2NO4Purity:98%Color and Shape:SolidMolecular weight:492.3N-Monoacetylcystine
CAS:N-Monoacetylcystine is a paracetamol poisoning antidote. It is used in the treatment of influenza A virus pandemic.Formula:C8H14N2O5S2Purity:98%Color and Shape:SolidMolecular weight:282.34L-NMMA acetate
CAS:L-NMMA acetate inhibits all NOS types (nNOS, eNOS, iNOS); Ki: 0.18, 0.4, 6 µM respectively.Formula:C9H20N4O4Purity:99.72% - 99.80%Color and Shape:White To Off-White SolidMolecular weight:248.28c-Fms-IN-6
CAS:c-Fms-IN-6 is a potent inhibitor of c-FMS (IC50 ≤10 nM for unphosphorylated c-FMS) and also weakly inhibits unphosphorylated c-KIT and PDGFR (IC50: > 1 μM).Formula:C22H25N7O2Purity:98%Color and Shape:SolidMolecular weight:419.48McN5691
CAS:McN5691 is a voltage sensitive calcium channel blocker.Formula:C30H35NO3Purity:98.93% - 99.38%Color and Shape:SolidMolecular weight:457.6Tolciclate
CAS:Tolciclate is an agent of antifungal medication.Formula:C20H21NOSPurity:98%Color and Shape:SolidMolecular weight:323.45L 748780
CAS:L 748780 is a selective inducible COX-2 inhibitor.Formula:C19H14Cl3NO4Purity:98%Color and Shape:SolidMolecular weight:426.68Anabasine hydrochloride
CAS:neuronal nicotinic ACh receptor partial agonistFormula:C10H15ClN2Purity:98%Color and Shape:White To Off-White SolidMolecular weight:198.693Ipsalazide
CAS:Ipsalazide is a novel salicylazosulfapyridine analog for the treatment of inflammatory bowel disease.
Formula:C16H11N3Na2O6Purity:99.43%Color and Shape:SolidMolecular weight:387.25J-2156
CAS:J-2156, a potent SST4 agonist, has ED50s of 3.7 mg/kg for allodynia and 8.0 mg/kg for hyperalgesia in rats; IC50s are 0.05/0.07 nM in human/rat receptors.Formula:C24H28N4O4SPurity:98%Color and Shape:SolidMolecular weight:468.57Fosnetupitant
CAS:Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.Formula:C31H35F6N4O5PPurity:98%Color and Shape:SolidMolecular weight:688.6OT antagonist 1
CAS:OT antagonist 1 is a potent and selective antagonist of Oxytocin(Ki of 50 nM)Formula:C22H22N4O3Purity:98%Color and Shape:SolidMolecular weight:390.44Thrombin Inhibitor 2
CAS:Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.Formula:C19H16ClF3N6O2Purity:98%Color and Shape:SolidMolecular weight:452.82UBP 302
CAS:UBP 302 is a selective GLUK5 kainate receptor antagonist with Kd 402 nM; low GluK2 affinity.Formula:C15H15N3O6Purity:98%Color and Shape:SolidMolecular weight:333.3Aganodine
CAS:Aganodine, a guanidine, activates imidazoline receptors to inhibit norepinephrine release.Formula:C9H10Cl2N4Purity:98%Color and Shape:SolidMolecular weight:245.11CRA-026440
CAS:CRA-026440(PCI-34051) is a highly potent HDAC inhibitor with inhibitory effects on HDAC1, HDAC2, HDAC3, HDAC6, HDAC8 and HDAC10 with Ki values of 4,14,11,15,7Formula:C23H24N4O4Purity:96.42%Color and Shape:SolidMolecular weight:420.46N-(3-Oxooctanoyl)-DL-homoserine lactone
CAS:N-(3-Oxooctanoyl)-DL-homoserine lactone with stereochemistry-dependent growth regulatory activity for roots .Formula:C12H19NO4Purity:98%Color and Shape:SolidMolecular weight:241.28(S)-Coriolic acid
CAS:(S)-Coriolic acid, a 15-LOX metabolite and signaling molecule, modulates cell growth, tumor adhesion, receptor expression, and can cause mitochondrial damage.Formula:C18H32O3Purity:97.67% - 98.04%Color and Shape:SolidMolecular weight:296.44Ref: TM-T37974
100ug (337.33μM*1mL in Ethanol)350.00€500ug (337.33μM*5mL in Ethanol)1,305.00€250ug (337.33μM*2.5mL in Ethanol)702.00€Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Formula:C48H69N13O13S2Purity:97.06%Color and Shape:SolidMolecular weight:1100.27NSC339614 potassium
CAS:NSC339614 potassium is a selective GluN1/GluN2C and GluN1/GluN2D receptors potentiator.Formula:C10H5KN3O6SPurity:98%Color and Shape:SolidMolecular weight:334.32Antitumor agent-115
CAS:Antitumor agent-115 (SS-12) is a potent anti-tumor compound, exhibiting an IC50 range of 0.34 μM-24.14 μM against the 4T1 mouse breast cancer cell line.Formula:C19H38ClNO2Purity:98%Color and Shape:SolidMolecular weight:347.96RSH-7
CAS:RSH-7 is a potent dual inhibitor of BTK and FLT3, with IC50s of 47 and 12 nM, respectively.RSH-7 has antiproliferative and antitumor activities, inducingFormula:C22H25FN8OPurity:99.43%Color and Shape:SolidMolecular weight:436.49Hsp90-Cdc37-IN-1
CAS:Hsp90-Cdc37-IN-1 is an Hsp90-Cdc37 interaction disruptor (IC50: 140 nM) that inhibit cell migration and reverse drug resistance.Formula:C43H57FN2O6SPurity:98%Color and Shape:SolidMolecular weight:748.99SSI-4
CAS:SSI-4 is a Stearoyl CoA desaturase 1 (SCD1) inhibitor that can be labeled with carbon-11 (11C) for use as a ligand in small animal in vivo PET/CT imagingFormula:C19H21ClN4O3Purity:98%Color and Shape:SolidMolecular weight:388.85
