Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65580 products of "Quinazoline and Quinoline Derivatives"
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Nitrendipine
CAS:<p>Nitrendipine is a vasodilating calcium channel blocker and antihypertensive that preserves kidney function and promotes sodium excretion.</p>Formula:C18H20N2O6Purity:99% - 99.55%Color and Shape:SolidMolecular weight:360.36Nitisinone
CAS:<p>Nitisinone (SC0735)(SC0735) is an enzyme 4-hydroxyphenylpyruvate dioxygenase inhibitor.</p>Formula:C14H10F3NO5Purity:99.63%Color and Shape:SolidMolecular weight:329.23Mebeverine hydrochloride
CAS:<p>Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut</p>Formula:C25H35NO5Purity:99.81% - 99.81%Color and Shape:SolidMolecular weight:429.55Butenafine hydrochloride
CAS:<p>Butenafine hydrochloride (KP363 Hydrochloride) is a synthetic benzylamine antifungal, inhibiting the synthesis of sterols by inhibiting squalene epoxidase.</p>Formula:C23H27N·HClPurity:99.66% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:353.93Ketanserin
CAS:<p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43Lenvatinib
CAS:<p>Lenvatinib (E7080) is a multi-target receptor tyrosine kinase inhibitor that inhibits VEGFR1-3, FGFR1-4, KIT, PDGFR, and RET, and has oral activity.</p>Formula:C21H19ClN4O4Purity:98.46% - 99.69%Color and Shape:SolidMolecular weight:426.85Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Formula:C17H18F3NOPurity:99.07% - 99.28%Color and Shape:SolidMolecular weight:309.33Incyclinide
CAS:<p>Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.</p>Formula:C19H17NO7Purity:97.99%Color and Shape:SolidMolecular weight:371.34Ramatroban
CAS:<p>Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.</p>Formula:C21H21FN2O4SPurity:98.75% - >99.99%Color and Shape:Crystalline SolidMolecular weight:416.47Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formula:C21H24N4O2SPurity:99.64%Color and Shape:Light Yellow To Yellow SolidMolecular weight:396.51UT-34
CAS:<p>UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s of 211.7 nM, 262.4 nM and 215.7 nM for wild</p>Formula:C15H12F4N4O2Purity:98.12%Color and Shape:SolidMolecular weight:356.27Flubendazole
CAS:<p>Flubendazole (Flumoxane) is available OTC in Europe that is an anthelmintic using to treat worm infection in humans.</p>Formula:C16H12FN3O3Purity:98.47% - 99.30%Color and Shape:White To Pale Yellow PowderMolecular weight:313.28Amiodarone hydrochloride
CAS:<p>Amiodarone HCl: Antianginal, class III antiarrhythmic. Lengthens heart muscle action, slows heart rate, reduces vascular resistance.</p>Formula:C25H29I2NO3·HClPurity:99.82% - ≥95%Color and Shape:White To Cream Crystalline PowderMolecular weight:681.78Tropisetron hydrochloride
CAS:<p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>Formula:C17H21ClN2O2Purity:99.72% - 99.83%Color and Shape:SolidMolecular weight:320.82Reserpine
CAS:<p>Reserpine, an alkaloid from Rauwolfia roots, depletes neurotransmitters, used in treating hypertension and psychosis, but side effects restrict use.</p>Formula:C33H40N2O9Purity:98.85% - 99.81%Color and Shape:White Or Pale Buff To Slightly Yellowish Powder With A Bitter Taste (Ntp 1992)Molecular weight:608.68Pimethixene
CAS:<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Formula:C19H19NSPurity:97.50%Color and Shape:SolidMolecular weight:293.43Ozagrel
CAS:<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Formula:C13H12N2O2Purity:97.90% - 99.38%Color and Shape:White PowderMolecular weight:228.25Oxcarbazepine
CAS:<p>Oxcarbazepine (GP 47680), an anti-epileptic, reduces CNS disorganized electrical activity.</p>Formula:C15H12N2O2Purity:98.46%Color and Shape:Crystals From Ethanol SolidMolecular weight:252.27Solabegron
CAS:<p>Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-AR</p>Formula:C23H23ClN2O3Purity:97.89%Color and Shape:SolidMolecular weight:410.891-Pyrrolidineethanol, β-methyl-α-phenyl-, (αR,βS)-
CAS:Formula:C13H19NOPurity:98%Color and Shape:SolidMolecular weight:205.2961Erlotinib
CAS:<p>Erlotinib (NSC-718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of non-small cell lung cancer.</p>Formula:C22H23N3O4Purity:98.19% - 99.98%Color and Shape:White To Off-White PowderMolecular weight:393.44Celecoxib
CAS:<p>Celecoxib (SC 58635) is a Nonsteroidal Anti-inflammatory Drug. The mechanism of action of celecoxib is as a Cyclooxygenase Inhibitor.</p>Formula:C17H14F3N3O2SPurity:99.44% - 99.98%Color and Shape:White PowderMolecular weight:381.37Fenofibric acid
CAS:<p>Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.</p>Formula:C17H15ClO4Purity:99.36%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:318.75Alfuzosin hydrochloride
CAS:<p>Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).</p>Formula:C19H27N5O4·HClPurity:99.78%Color and Shape:White To Off-White SolidMolecular weight:425.91Moclobemide
CAS:<p>Moclobemide (Ro111163) is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.</p>Formula:C13H17ClN2O2Purity:99.51% - 99.59%Color and Shape:White To Off-White SolidMolecular weight:268.74Telmisartan
CAS:<p>Telmisartan (BIBR 277) is an Angiotensin 2 Receptor Blocker. The mechanism of action of telmisartan is as an Angiotensin 2 Receptor Antagonist.</p>Formula:C33H30N4O2Purity:99.88% - 99.97%Color and Shape:White Or Off White Crystalline PowderMolecular weight:514.62Robenidine hydrochloride
CAS:<p>Robenidine hydrochloride (Robenidine Hydrochoride) is an anticoccidial agent mainly used in poultry.</p>Formula:C15H14Cl3N5Purity:>99.99%Color and Shape:Off-White SolidMolecular weight:370.66Dasatinib
CAS:<p>Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.</p>Formula:C22H26ClN7O2SPurity:99.59% - 99.86%Color and Shape:Pale-Yellow SolidMolecular weight:488.01Nifuratel
CAS:<p>Nifuratel (SAP 113) is a local antiprotozoal and antifungal agent that may also be given orally.</p>Formula:C10H11N3O5SPurity:99.76% - 99.87%Color and Shape:Fresh Yellow Crystalline Or Yellow PowderMolecular weight:285.28Thio-TEPA
CAS:<p>Thio-TEPA (Tiofosyl) is a polyfunctional, organophosphorus alkylating agent with antineoplastic activity.</p>Formula:C6H12N3PSPurity:98.45% - 99.07%Color and Shape:White Crystals Or PowderMolecular weight:189.22Menbutone
CAS:<p>Menbutone, a choleretic and oxobutyric acid derivative, peaks in plasma in 1hr, effects last ~10hrs.</p>Formula:C15H14O4Purity:97.48%Color and Shape:CoaMolecular weight:258.27Paliperidone
CAS:<p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>Formula:C23H27FN4O3Purity:95% - 99.08%Color and Shape:Off White To Light Orange Coloured SolidMolecular weight:426.48Tilorone dihydrochloride
CAS:<p>Tilorone dihydrochloride is an orally active interferon inducer, and has antineoplastic and anti-inflammatory actions.</p>Formula:C25H36Cl2N2O3Purity:98% - 99.86%Color and Shape:Orange Yellow Crystal PowderMolecular weight:483.47Sildenafil citrate
CAS:<p>Sildenafil citrate, a PDE5 inhibitor for erectile dysfunction and occasionally pulmonary hypertension.</p>Formula:C28H38N6O11SPurity:99.59% - 99.97%Color and Shape:White SolidMolecular weight:666.70Niraparib (R-enantiomer)
CAS:<p>Niraparib R-enantiomer (MK 4827 R-enantiomer) is an inhibitor of PARP1(IC50 of 2.4 nM).</p>Formula:C19H20N4OPurity:99.83%Color and Shape:SolidMolecular weight:320.39Vildagliptin
CAS:<p>Vildagliptin (LAF237), an oral DPP-4 inhibitor with hypoglycemic effects, is metabolized and excreted in urine.</p>Formula:C17H25N3O2Purity:97.81% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:303.40Zinc pyrithione
CAS:<p>Zinc pyrithione (OM-1563), an antibacterial and antifungal agent can disrupt membrane transport by blocking the proton pump.</p>Formula:C10H8N2O2S2ZnPurity:99.09% - 99.47%Color and Shape:Off-White To Tan PowderMolecular weight:317.71Medrysone
CAS:<p>Medrysone is a synthetic glucocorticoid for topical use with anti-inflammatory and anti-allergic effects, altering gene expression to reduce inflammation.</p>Formula:C22H32O3Purity:97.72% - 99.91%Color and Shape:SolidMolecular weight:344.49Adenine
CAS:<p>Adenine: a purine nucleobase vital for ATP, NAD, FAD production, and DNA/RNA synthesis.</p>Formula:C5H5N5Purity:99.39% - 99.95%Color and Shape:SolidMolecular weight:135.13Clonidine hydrochloride
CAS:<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Formula:C9H10Cl3N3Purity:99.16% - 99.86%Color and Shape:SolidMolecular weight:266.55Mirtazapine
CAS:<p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>Formula:C17H19N3Purity:99.98%Color and Shape:SolidMolecular weight:265.35Deracoxib
CAS:<p>Deracoxib (SC 46) is a selective COX-2 inhibitor, non-steroidal, non-narcotic anti-inflammatory drug with an IC50 of 70-150 μM for osteosarcoma cells.</p>Formula:C17H14F3N3O3SPurity:98.94% - 99.81%Color and Shape:SolidMolecular weight:397.37Mexiletine hydrochloride
CAS:<p>Mexiletine hydrochloride is a lidocaine-like antiarrhythmic (Class IB) and anesthetic, stabilizing heartbeats by inhibiting sodium in cardiac cells.</p>Formula:C11H18ClNOPurity:99.88%Color and Shape:White To Off-White SolidMolecular weight:215.72Azelnidipine
CAS:<p>Azelnidipine (UR-12592) is a dihydropyridine used as calcium channel blocker.</p>Formula:C33H34N4O6Purity:99.78%Color and Shape:Light Yellowish PowderMolecular weight:582.65Orbifloxacin
CAS:<p>Orbifloxacin (CP-104354) is a broad-spectrum fluoroquinolone antibiotic.</p>Formula:C19H20F3N3O3Purity:99.46% - 99.58%Color and Shape:SolidMolecular weight:395.38Hydralazine hydrochloride
CAS:<p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>Formula:C8H9ClN4Purity:99.85% - 99.86%Color and Shape:Yellow Crystals White Crystalline SolidMolecular weight:196.64Fluphenazine dihydrochloride
CAS:<p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>Formula:C22H28Cl2F3N3OSPurity:99.23%Color and Shape:Off-White SolidMolecular weight:510.44Tafenoquine Succinate
CAS:<p>Tafenoquine Succinate (WR 238605 (Succinate)) is an 8-aminoquinoline. and is an agent of anti-malarial prophylactic.</p>Formula:C28H34F3N3O7Purity:99.77%Color and Shape:SolidMolecular weight:581.58Amiloride hydrochloride
CAS:<p>Amiloride hydrochloride (Amiloride HCl) 是上皮钠通道和尿激酶型纤溶酶原激活物受体的抑制剂，也是 polycystin-2通道阻断剂。</p>Formula:C6H9Cl2N7OPurity:99.72% - 99.95%Color and Shape:Physical Description Crystalline Solid Or Very Light Yellow Powder (Ntp 1992)Molecular weight:266.09Dutasteride
CAS:<p>Dutasteride (GI 198745) is a 5-alpha-reductase inhibitor that inhibits both type-1 and type2 isoforms of the enzyme and is used to treat benign prostatic</p>Formula:C27H30F6N2O2Purity:99.58%Color and Shape:White Crystalline SolidMolecular weight:528.53
