Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65578 products of "Quinazoline and Quinoline Derivatives"
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Elexacaftor
CAS:<p>Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.</p>Formula:C26H34F3N7O4SPurity:98.87% - 99.87%Color and Shape:SolidMolecular weight:597.65Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurity:99.84% - 99.92%Color and Shape:White SolidMolecular weight:332.87Deracoxib
CAS:<p>Deracoxib (SC 46) is a selective COX-2 inhibitor, non-steroidal, non-narcotic anti-inflammatory drug with an IC50 of 70-150 μM for osteosarcoma cells.</p>Formula:C17H14F3N3O3SPurity:98.94% - 99.81%Color and Shape:SolidMolecular weight:397.37Pranlukast
CAS:<p>Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.</p>Formula:C27H23N5O4Purity:99.41%Color and Shape:Off-White SolidMolecular weight:481.5Trelagliptin
CAS:<p>Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.</p>Formula:C18H20FN5O2Purity:98.88%Color and Shape:SolidMolecular weight:357.38Trimetazidine dihydrochloride
CAS:<p>Trimetazidine, an anti-ischemic agent, enhances myocardial glucose use, inhibits fat metabolism, and helps with angina.</p>Formula:C14H24Cl2N2O3Purity:99.58%Color and Shape:Crystalline SolidMolecular weight:339.258Tetrahydrozoline
CAS:<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Formula:C13H16N2Purity:97.85% - 99.77%Color and Shape:SolidMolecular weight:200.28Primaquine diphosphate
CAS:<p>Primaquine diphosphate is the phosphate salt form of primaquine, a synthetic, 8-aminoquinoline derivative with antimalarial properties.</p>Formula:C15H21N3O·2H3PO4Purity:98.06% - 99.73%Color and Shape:Orange PowderMolecular weight:455.34Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Formula:C20H23ClN2O5Purity:99.97%Color and Shape:Off-White SolidMolecular weight:406.86Chlorhexidine dihydrochloride
CAS:Chlorhexidine dihydrochloride (NSC-185) is a disinfectant and topical anti-infective agent used also as mouthwash to prevent oral plaque.Formula:C22H32Cl4N10Purity:97.51% - 98.32%Color and Shape:White To Pale Yellow PowderMolecular weight:578.38Ritodrine hydrochloride
CAS:<p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>Formula:C17H21NO3·HClPurity:99% - 99.52%Color and Shape:SolidMolecular weight:323.82Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Formula:C22H22FN3O2Purity:97.16% - 98%Color and Shape:SolidMolecular weight:379.43Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Formula:C31H38N2OPurity:97.49%Color and Shape:SolidMolecular weight:454.65Phenformin hydrochloride
CAS:<p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>Formula:C10H16ClN5Purity:97.11% - 99.80%Color and Shape:Lactic AcidosisMolecular weight:241.72Ramelteon
CAS:<p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>Formula:C16H21NO2Purity:97.21% - 99.92%Color and Shape:Crystalline SolidMolecular weight:259.34Bromopride
CAS:<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Formula:C14H22BrN3O2Purity:99.95%Color and Shape:SolidMolecular weight:344.25Moclobemide
CAS:<p>Moclobemide (Ro111163) is a reversible inhibitor of monoamine oxidase type A; (RIMA); (see MONOAMINE OXIDASE INHIBITORS) that has antidepressive properties.</p>Formula:C13H17ClN2O2Purity:99.51% - 99.59%Color and Shape:White To Off-White SolidMolecular weight:268.74Cloperastine hydrochloride
CAS:<p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>Formula:C20H25Cl2NOPurity:97.74% - 99.42%Color and Shape:SolidMolecular weight:366.33Valemetostat
CAS:<p>Valemetostat (DS-3201) is a first-in-class EZH1/2 dual inhibitor, which can be used to study T-cell lymphoma.Cost-effective and quality-assured.</p>Formula:C26H34ClN3O4Purity:98.38% - 99.08%Color and Shape:SolidMolecular weight:488.02Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Formula:C15H17NO2Purity:99.92%Color and Shape:White SolidMolecular weight:243.3Dronedarone hydrochloride
CAS:<p>Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.</p>Formula:C31H44N2O5S·HClPurity:99.61%Color and Shape:SolidMolecular weight:593.22Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formula:C21H24N4O2SPurity:99.64%Color and Shape:Light Yellow To Yellow SolidMolecular weight:396.51Diphenmanil methylsulfate
CAS:<p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>Formula:C20H24N·CH3O4SPurity:98% - 99.27%Color and Shape:SolidMolecular weight:389.51Ketanserin
CAS:<p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>Formula:C22H22FN3O3Purity:99.19% - 99.73%Color and Shape:SolidMolecular weight:395.43Ofloxacin
CAS:<p>Ofloxacin (Oxaldin) is a fluoroquinolone antibacterial antibiotic.</p>Formula:C18H20FN3O4Purity:99.33% - 99.87%Color and Shape:Off-White SolidMolecular weight:361.37Imrecoxib
CAS:<p>Imrecoxib (BAP-909) is a novel and selective cyclooxygenase 2 (COX-2) inhibitor (IC50: 18 nM).</p>Formula:C21H23NO3SPurity:99.87%Color and Shape:SolidMolecular weight:369.48Loxapine succinate
CAS:<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Formula:C22H24ClN3O5Purity:99.69%Color and Shape:White To Of-White SolidMolecular weight:445.9Arimoclomol maleate
CAS:<p>Arimoclomol maleate (BRX-220) (BRX-220) is a heat shock protein (HSP) co-inducer.</p>Formula:C18H24ClN3O7Purity:99.44% - 99.98%Color and Shape:SolidMolecular weight:429.85Maprotiline hydrochloride
CAS:<p>Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.</p>Formula:C20H24ClNPurity:99.68% - 99.84%Color and Shape:White PowderMolecular weight:313.864Sorafenib
CAS:<p>Sorafenib (Bay 43-9006) is a multikinase inhibitor that inhibits Raf-1, B-Raf, VEGFR2, VEGFR3, VEGFR4, PDGFRβ, FLT3, c-Kit, and others (IC50=6/22/90/15/20/20/57</p>Formula:C21H16ClF3N4O3Purity:98% - 99.89%Color and Shape:SolidMolecular weight:464.82Amisulpride
CAS:<p>Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.</p>Formula:C17H27N3O4SPurity:99.97%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:369.48Balofloxacin
CAS:<p>Balofloxacin, a quinolone antibiotic, can inhibit the synthesis of bacterial DNA by interfering with the DNA gyrase.</p>Formula:C20H24FN3O4Purity:99.62% - 99.98%Color and Shape:Crystalline SolidMolecular weight:389.42Pentoxifylline
CAS:<p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>Formula:C13H18N4O3Purity:99.26% - 99.93%Color and Shape:SolidMolecular weight:278.31Quinoxyfen
CAS:<p>Quinoxyfen has antimicrobial activity and can be used to study powdery mildew.</p>Formula:C15H8Cl2FNOPurity:99.61%Color and Shape:LiquidMolecular weight:308.13Terbutaline Sulfate
CAS:Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.Formula:C12H19NO3H2SO4Purity:99.47% - 99.94%Color and Shape:Crystalline PowderMolecular weight:274.32Decoquinate
CAS:<p>Decoquinate (Deccox) is a coccidiostat for poultry.</p>Formula:C24H35NO5Purity:97.10%Color and Shape:Pale Yellow CrystalsMolecular weight:417.54Mianserin hydrochloride
CAS:<p>Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.</p>Formula:C18H21ClN2Purity:99.63% - 99.82%Color and Shape:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMolecular weight:300.83Nefopam hydrochloride
CAS:<p>Nefopam hydrochloride (Nefopam HCl) is the hydrochloride salt form of nefopam, a centrally-acting, non-opioid benzoxazocine with analgesic activity.</p>Formula:C17H20ClNOPurity:99.32% - 99.85%Color and Shape:SolidMolecular weight:289.81,3-Propanediol, 2-amino-1-(4-nitrophenyl)-, (1S,2S)-
CAS:Formula:C9H12N2O4Purity:98%Color and Shape:SolidMolecular weight:212.2026Atazanavir
CAS:<p>Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.</p>Formula:C38H52N6O7Purity:98% - 99.95%Color and Shape:Crystalline SolidMolecular weight:704.86Blonanserin
CAS:<p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>Formula:C23H30FN3Purity:99.85%Color and Shape:SolidMolecular weight:367.5Diazoxide
CAS:<p>Diazoxide (Proglycem) is a benzothiadiazine derivative that is a peripheral vasodilator used for hypertensive emergencies.</p>Formula:C8H7ClN2O2SPurity:99% - 99.83%Color and Shape:SolidMolecular weight:230.67Isoxsuprine hydrochloride
CAS:<p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>Formula:C18H24ClNO3Purity:99.38%Color and Shape:Crystals From Water SolidMolecular weight:337.84Sarafloxacin hydrochloride
CAS:<p>Sarafloxacin hydrochloride (A-56620 (hydrochloride)), a quinolone antibiotic drug, is a hydrochloride salt form of sarafloxacin.</p>Formula:C20H18ClF2N3O3Purity:97.33% - 97.44%Color and Shape:White To Yellow Crystalline SolidMolecular weight:421.83Pictilisib dimethanesulfonate
CAS:<p>Pictilisib dimethanesulfonate (GDC-0941 2 MeSO3H salt) is a potent inhibitor of PI3Kα/δ with IC50 of 3 nM, with modest selectivity against p110β (11-fold) and</p>Formula:C25H35N7O9S4Purity:99.63%Color and Shape:SolidMolecular weight:705.85Tizanidine hydrochloride
CAS:<p>Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.</p>Formula:C9H9Cl2N5SPurity:99.96%Color and Shape:Solid WhiteMolecular weight:290.17Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:463.79Prazosin hydrochloride
CAS:<p>Prazosin HCl, a synthetic antiadrenergic, treats hypertension, heart failure, and more by relaxing blood vessels with an unclear mechanism.</p>Formula:C19H22ClN5O4Purity:99.88% - >99.99%Color and Shape:White To Tan Powder Off-White To Yellow PowderMolecular weight:419.86Propylthiouracil
CAS:<p>Propylthiouracil (6-n-Propylthiouracil) is a thyroid peroxidase inhibitor and also a 5' -deiodinase inhibitor.</p>Formula:C7H10N2OSPurity:99.24%Color and Shape:White Crystalline Powder Of Starch-Like Appearance To Eye And To Touch Saturated Solution Is Neutral Or Slightly Acid To Litmus (Ntp 1992)Molecular weight:170.23Lisinopril dihydrate
CAS:<p>Lisinopril dihydrate （MK-521) is an orally bioavailable, long-acting angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.</p>Formula:C21H35N3O7Purity:98.83% - 99.22%Color and Shape:White To Off-White Crystalline PowderMolecular weight:441.52
