Enzyme Modulators
Enzyme modulators are compounds that can enhance or inhibit the activity of enzymes, thereby regulating the rate of biochemical reactions. These modulators play a critical role in controlling metabolic pathways, cell signaling, and various physiological processes. Enzyme modulators are widely used in research and drug development to study enzyme functions and to develop therapeutic agents. At CymitQuimica, we offer a comprehensive range of high-quality enzyme modulators to support your research in enzyme regulation and drug discovery.
Subcategories of "Enzyme Modulators"
Found 690 products for "Enzyme Modulators". Showing the first 500.
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Fluvastatin sodium salt - Bio-X ™
CAS:Fluvastatin is a statin that lowers blood cholesterol and triglycerides by inhibiting HMG-CoA reductase, an enzyme that plays a critical role in the synthesis of cholesterol. Fluvastatin has also been shown to reduce the incidence of myocardial infarction, and to reduce atherosclerotic lesions in animal models, reducing the incidence of cardiovascular disease. Fluvastatin also has been shown to inhibit the activation of toll-like receptor 4 (TLR4) by lipopolysaccharide (LPS), which may be related to its anti-inflammatory effects. Furthermore, through lowering blood cholesterol, Fluvastatin also inhibits tubulointerstitial injury and prevents renal damage caused by high concentrations of the lipid.Formula:C24H25FNNaO4Purity:Min. 98%Molecular weight:433.45 g/molTAK 243
CAS:A potent inhibitor of ubiquitin activating enzyme E1. Lowers ubiquitin conjugates in cells, thereby disrupting cell signalling, cell cycle progression and repair of DNA damage. Anti-tumor effects have been demonstrated in vitro and in vivo. TAK 243 has been used to study the biology of ubiquitins and its potential as anti-cancer therapy.Formula:C19H20F3N5O5S2Purity:Min. 95%Color and Shape:White Off-White PowderMolecular weight:519.52 g/molN-[3-(1,3-Benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-N',N'-dimethyl-propane-1,3-diamine
Selective inhibitor of the mutated RET variant RETV804M, which is the anticipated drug-resistant RET mutant that can occur in tumours treated with kinase inhibitors. The compound has a biochemical IC50 of 0.02 µM and selectivity for purified RETV804M over purified RET and KDR of 3.7 and 110, respectively. The efficacy of the compound was shown also in cell cultures with IC50 of 4.4 µM, and cell assay selectivity for RETV804M over RET and KDR of 0.89 and 2.3, respectively.Formula:C18H21N5O2Purity:Min. 98 Area-%Color and Shape:PowderMolecular weight:339.39 g/molAnagrelide HCl - Bio-X ™
CAS:Anagrelide is a thrombocytopenic drug that is used to treat thrombocythemia and related conditions. This drug works by decreasing the platelet count by suppressing transcription factors that are necessary for the maturation of platelets. This drug is also a phosphodiesterase III inhibitor.Formula:C10H7Cl2N3O•HClPurity:Min. 95%Color and Shape:PowderMolecular weight:292.55 g/molMEK162
CAS:Inhibitor of MEK1/2 kinase enzymes; antineoplasticFormula:C17H15BrF2N4O3Purity:Min. 95%Color and Shape:White/Off-White SolidMolecular weight:441.23 g/molUNC 0379
CAS:Inhibitor of the histone methyltransferase SETD8 that supresses methylation of the K20 residue in histone 4. UNC 0379 treatment of human glioma reduced recruitment of 53BP1 protein to double strand breaks and sensitised cells to radiotherapy without altering cell cycle kinetics.
Formula:C23H35N5O2Purity:Min. 95%Color and Shape:SolidMolecular weight:413.56 g/molDanusertib
CAS:Inhibitor of aurora kinases
Formula:C26H30N6O3Purity:Min. 95%Color and Shape:White PowderMolecular weight:474.57 g/molK252c
CAS:Inhibitor of protein kinase PKCFormula:C20H13N3OPurity:Min. 95%Color and Shape:PowderMolecular weight:311.34 g/molPemetrexed disodium salt - Bio-X ™
CAS:Pemetrexed is an antifolate drug that is used to treat mesothelioma and non-small cell lung cancer. It is used during chemotherapy and sometimes used in conjunction with cisplatin. This drug disrupts folate-dependent metabolic activities essential for cell replication. In vitro studies have shown that Pemetrexed inhibits thymidylate synthase.Formula:C20H19N5Na2O6Purity:Min. 95%Color and Shape:PowderMolecular weight:471.37 g/molMoexipril HCl - Bio-X ™
CAS:Moexipril is an angiotensin converting enzyme inhibitor that is used for the treatment of hypertension. This drug is a prodrug for moexiprilat and works by relaxing the blood vessels causing them to widen and lowering blood pressure. Moexipril has been shown to be effective in treating metabolic disorders such as congestive heart failure.Formula:C27H34N2O7Purity:Min. 95%Color and Shape:PowderMolecular weight:498.57 g/molNVP AAM 077 tetrasodium hydrate
CAS:NMDA receptor antagonistFormula:C17H13BrN3Na4O5P·xH2OPurity:Min. 95%Color and Shape:Light yellow to light green solid.Molecular weight:542.14Pazopanib - Bio-X ™
CAS:Pazopanib is an antineoplastic agent that is used to treat advanced renal cell cancer and advanced soft tissues sarcoma. This drug is a multitargeted tyrosine kinase inhibitor against vascular endothelial growth factor receptor 1, 2, 3 and c-kit. As a result, it increases tumor apoptosis and decreases tumor blood flow.
Formula:C21H23N7O2SPurity:Min. 95%Color and Shape:PowderMolecular weight:437.52 g/molCobimetinib
CAS:Inhibitor of MEK kinase
Formula:C21H21F3IN3O2Purity:Min. 95%Color and Shape:White PowderMolecular weight:531.31 g/molTolrestat
CAS:Aldose reductase AKR1B10 inhibitor; hepatotoxic
Formula:C16H14F3NO3SPurity:Min. 95%Molecular weight:357.35 g/molSunitinib malate - Bio-X ™
CAS:Sunitinib is a receptor tyrosine kinase inhibitor and a chemotherapeutic agent used for the treatment of renal cell carcinoma. This drug can also be used to treat gastrointestinal tumors that are resistant to imatinib. Sunitinib inhibits VEGFR1, VEGFR2, VEGFR3, PDGFR and KIT tyrosine kinases.Formula:C22H27FN4O2·C4H6O5Purity:Min. 95%Color and Shape:PowderMolecular weight:532.56 g/molEAI045
CAS:Inhibitor of EGFR receptor
Formula:C19H14FN3O3SPurity:Min. 95%Color and Shape:White Off-White PowderMolecular weight:383.4 g/molCP 43
CAS:Inhibitor of TAOK1 and TAOK2 kinasesFormula:C25H24N2O2Purity:Min. 95%Color and Shape:SolidMolecular weight:384.47 g/molDexrazoxane - Bio-X ™
CAS:Dexrazoxane is a cytoprotective drug that is used in chemotherapy to provide cardio-protection against anthracycline toxicity. It is an antimitotic agent with immunosuppressive properties. Dexrazoxane works by binding to iron in the cell, preventing it from being released. Dexrazoxane is also a catalytic inhibitor of topoisomerase II.Formula:C11H16N4O4Purity:Min. 95%Color and Shape:PowderMolecular weight:268.27 g/molD 4476
CAS:Inhibitor of protein kinase CK1Formula:C23H18N4O3Purity:Min. 95%Molecular weight:398.41 g/molRucaparib
CAS:Inhibitor of poly (ADP-ribose) polymerase enzyme; antineoplastic
Formula:C19H18FN3OPurity:Min. 98 Area-%Color and Shape:Yellow PowderMolecular weight:323.36 g/mol
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