Apoptose
Os inibidores da apoptose são compostos que previnem ou retardam o processo de morte celular programada, conhecido como apoptose. Esses inibidores são vitais no estudo dos mecanismos de sobrevivência celular e são usados para investigar doenças onde a apoptose é desregulada, como câncer, distúrbios neurodegenerativos e doenças autoimunes. Ao modular a apoptose, esses inibidores podem ajudar no desenvolvimento de terapias destinadas a controlar a morte celular. Na CymitQuimica, oferecemos uma ampla seleção de inibidores da apoptose de alta qualidade para apoiar sua pesquisa em biologia celular, oncologia e áreas relacionadas.
Subcategorias de "Apoptose"
- ASK(6 produtos)
- BCL(11 produtos)
- Caspase(125 produtos)
- FOXO1(3 produtos)
- IAP(66 produtos)
- Mdm2(12 produtos)
- PD-1/PD-L1(125 produtos)
- PDK(9 produtos)
- PERK(25 produtos)
- Serina/treonina quinase(15 produtos)
- Survivina(13 produtos)
- TNF(92 produtos)
- c-RET(51 produtos)
- p53(62 produtos)
Exibir 6 mais subcategorias
Foram encontrados 5599 produtos de "Apoptose"
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Ethyl 3,4-dihydroxybenzoate
CAS:<p>Ethyl 3,4-dihydroxybenzoate (EDHB): a prolyl hydroxylase inhibitor attenuates acute hypobaric hypoxia mediated vascular leakage in brain.</p>Fórmula:C9H10O4Pureza:99.88%Cor e Forma:White Crystal Or PowderPeso molecular:182.17PF-3758309 hydrochloride
CAS:<p>PF-3758309 hydrochloride (PF-03758309 hydrochloride) , is a PAK4 inhibitor, is also a n orally bioavailable small-molecule inhibitor of p21-activated kinase 4 (</p>Fórmula:C25H31ClN8OSPureza:98.83% - >99.99%Cor e Forma:SolidPeso molecular:527.08Liproxstatin-1
CAS:<p>Liproxstatin-1 is a potent and selective inhibitor of iron death (IC50=22 nM).</p>Fórmula:C19H21ClN4Pureza:97.11% - 99.44%Cor e Forma:SolidPeso molecular:340.85PP121
CAS:<p>PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.</p>Fórmula:C17H17N7Pureza:98.45% - 99.67%Cor e Forma:SolidPeso molecular:319.36MK-8745
CAS:<p>MK-8745 is a potent and selective Aurora A inhibitor.</p>Fórmula:C20H19ClFN5OSPureza:99.09% - 99.79%Cor e Forma:SolidPeso molecular:431.91Panobinostat
CAS:<p>Panobinostat (NVP-LBH589) is a broad-spectrum HDAC inhibitor (IC50=5 nM) with oral activity and non-selectivity.</p>Fórmula:C21H23N3O2Pureza:97.2% - 99.81%Cor e Forma:Yellow SolidPeso molecular:349.43HS-1793
CAS:<p>HS-1793, resveratrol-like, reduces HIF-1, VEGF in hypoxia, and curbs human breast cancer growth in mouse model.</p>Fórmula:C16H12O3Pureza:98.16% - 99.82%Cor e Forma:SolidPeso molecular:252.26Cucurbitacin B
CAS:<p>Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.</p>Fórmula:C32H46O8Pureza:97.1% - 99.33%Cor e Forma:SolidPeso molecular:558.7FX1
CAS:<p>FX1 is an effective and selective BCL6 inhibitor (IC50: 35 μM).</p>Fórmula:C14H9ClN2O4S2Pureza:97.59%Cor e Forma:SolidPeso molecular:368.82SP600125
CAS:<p>SP600125 (JNK Inhibitor II) is a JNK inhibitor that inhibits JNK1, JNK2, and JNK3 (IC50=40/40/90 nM) with oral potency, reversibility, and ATP-competitive</p>Fórmula:C14H8N2OPureza:97.63% - 99.82%Cor e Forma:SolidPeso molecular:220.23ASK1-IN-2
CAS:<p>ASK1-IN-2: oral ASK1 inhibitor, IC50 32.8 nM, potential ulcerative colitis treatment.</p>Fórmula:C19H17FN6OPureza:98.79%Cor e Forma:SolidPeso molecular:364.38GSK-923295
CAS:<p>GSK923295 is a selective allosteric inhibitor of CENP-E kinesin motor ATPase(Ki=3.2 nM).</p>Fórmula:C32H38ClN5O4Pureza:96.22% - 98.02%Cor e Forma:SolidPeso molecular:592.13Mimosine
CAS:<p>L-Mimosine (Leucenol) is an antineoplastic alanine-substituted pyridine derivative isolated from Leucena glauca and acts as an iron chelator.</p>Fórmula:C8H10N2O4Pureza:99.2% - 99.84%Cor e Forma:Crystals From Water SolidPeso molecular:198.18Etomoxir sodium salt
CAS:<p>Etomoxir sodium salt ((R)-Etomoxir sodium salt) is a carnitine palmitoyltransferase 1a (CPT-1a) inhibitor that blocks fatty acid synthesis.</p>Fórmula:C15H18ClO4·NaPureza:99.34% - 99.82%Cor e Forma:SolidPeso molecular:320.741A-116
CAS:<p>1A-116 is a specific Rac1 inhibitor.</p>Fórmula:C16H16F3N3Pureza:99.71%Cor e Forma:SolidPeso molecular:307.31CCT 137690
CAS:<p>CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).</p>Fórmula:C26H31BrN8OPureza:98.51% - 99.89%Cor e Forma:SolidPeso molecular:551.48COTI-2
CAS:<p>COTI-2, an orally available thiosemicarbazone, is an activator of mutant forms of the p53 protein with potential antineoplastic activity.</p>Fórmula:C19H22N6SPureza:99% - 99.55%Cor e Forma:SolidPeso molecular:366.48C-DIM12
CAS:<p>C-DIM12 boosts Nurr1 gene expression, heightens Nurr1 protein in neurons, and improves survival against 6-OHDA.</p>Fórmula:C23H17ClN2Pureza:97.72% - ≥95%Cor e Forma:SolidPeso molecular:356.85Tomatine
CAS:<p>Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.</p>Fórmula:C50H83NO21Pureza:98.42% - 99.94%Cor e Forma:White To Light YellowPeso molecular:1034.19MG-101
CAS:<p>MG-101 (Calpain inhibitor I) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.</p>Fórmula:C20H37N3O4Pureza:98% - ≥98%Cor e Forma:SolidPeso molecular:383.53L-685458
CAS:<p>L-685458 (L-685,458) is a specific and potent inhibitor of A beta PP gamma-secretase activity with Ki of 17 nM.</p>Fórmula:C39H52N4O6Pureza:99.62% - 99.80%Cor e Forma:SolidPeso molecular:672.85Serdemetan
CAS:<p>Serdemetan (JNJ-26854165) is an orally bioavailable HDM2 antagonist with potential antineoplastic activity.</p>Fórmula:C21H20N4Pureza:98% - 99.51%Cor e Forma:SolidPeso molecular:328.41Kahweol
CAS:<p>Kahweol has anticarcinogenic, anti-angiogenic,and anti-inflammatory activities, it can block the LPS-induced activation of NF-kappaB by preventing IkappaB</p>Fórmula:C20H26O3Pureza:99.26% - 99.86%Cor e Forma:Off-White To Yellow SolidPeso molecular:314.42Oleic acid
CAS:<p>Oleic acid, a common unsaturated fat, is used in oleates, lotions, and as a pharma solvent.</p>Fórmula:C18H34O2Pureza:97.14% - 99.91%Cor e Forma:Colorless Or Nearly Colorless Liq (Above 5-7 Deg C) Oleic Acid Is A Colorless To Pale Yellow Liquid With A Mild Odor Floats On Water (Uscg 1999)Peso molecular:282.46RA-9
CAS:<p>RA-9 is a potent and selective proteasome-associated inhibitor of deubiquitinating enzymes (DUBs), with favorable toxicity profile and anticancer activity.</p>Fórmula:C19H15N3O5Pureza:98.15%Cor e Forma:SolidPeso molecular:365.34GSK 872 hydrochloride
CAS:<p>GSK872 HCl（1346546-69-7 free base） (GSK2399872A) is an effective and specific RIP3 kinase inhibitor.</p>Fórmula:C19H18ClN3O2S2Pureza:99%Cor e Forma:SolidPeso molecular:419.94B-AP15
CAS:<p>B-AP15 (NSC-687852) selectively inhibits 26S proteasome enzymes Usp14 and UCHL5, blocking their activity.</p>Fórmula:C22H17N3O6Pureza:91.43% - 98.77%Cor e Forma:SolidPeso molecular:419.39Niraparib
CAS:<p>Niraparib (MK-4827) inhibits PARP1/PARP2 (IC50: 3.8/2.1 nM), effective on BRCA mutant cancers, 330x less effective on PARP3, V-PARP, Tank1.</p>Fórmula:C19H20N4OPureza:98% - 99.91%Cor e Forma:SolidPeso molecular:320.39R406
CAS:<p>R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn.</p>Fórmula:C22H23FN6O5·C6H6O3SPureza:97.67% - 98.82%Cor e Forma:SolidPeso molecular:628.63PS 48
CAS:<p>PS 48 has been shown to be a PKB Kinase (PDK1) activator (Kd: 10.3 μM). This compound selectively binds to the PIF-binding pocket of PKB Kinase (PDK1).</p>Fórmula:C17H15ClO2Pureza:99.96% - ≥95%Cor e Forma:SolidPeso molecular:286.75Mito-LND
CAS:<p>Mito-LND (Mito-Loidamine) is an orally active and mitochondria-targeted inhibitor of oxidative phosphorylation.</p>Fórmula:C43H45BrCl2N3OPPureza:97.25% - 98.34%Cor e Forma:SolidPeso molecular:801.62Xevinapant
CAS:<p>Xevinapant (Debio-1143) is a potent Smac mimetic and an antagonist of IAP, binding to XIAP-BIR3, cIAP1-BIR3 and cIAP2-BIR3.</p>Fórmula:C32H43N5O4Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:561.71Rosiglitazone
CAS:<p>Rosiglitazone (BRL49653) is a PPARγ agonist, TRPC5 activator, and TRPM3 inhibitor with oral activity.</p>Fórmula:C18H19N3O3SPureza:98.61% - 99.87%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:357.43Alisertib Sodium
CAS:<p>Alisertib Sodium (MLN 8237 Sodium)is a selective Aurora A inhibitor that causes G2/M phase arrest and chromosomal misalignment, leading to tumour cell apoptosis.</p>Fórmula:C27H19ClFN4NaO4Pureza:99.77%Cor e Forma:SolidPeso molecular:540.91(R)-(-)-Gossypol acetic acid
CAS:<p>(R)-(-)-Gossypol acetic acid binds Bcl-2, Bcl-xL, Mcl-1 (Ki: 0.32, 0.48, 0.18 μM); no BIR3/BID inhibition. Phase 2.</p>Fórmula:C30H30O8·C2H4O2Pureza:98.88% - 99.5%Cor e Forma:SolidPeso molecular:578.61Etalocib
CAS:<p>Etalocib (LY293111) is a potent diaryl ether inhibitor blocking LTB4 receptor and 5'-lipoxygenase, with antineoplastic properties.</p>Fórmula:C33H33FO6Pureza:98.21%Cor e Forma:SolidPeso molecular:544.63-Dehydrotrametenolic acid
CAS:<p>3-Dehydrotrametenolic acid is a potential anticancer agent against H-ras transformed tumor and a promising candidate for a new type of insulin-sensitizing drug.</p>Fórmula:C30H46O3Pureza:98.5% - 99.25%Cor e Forma:SolidPeso molecular:454.68K34C
CAS:<p>K34C is a selective inhibitor of Integrin α5β1, which inhibits cell survival and migration, promotes apoptosis, inhibits invasion.</p>Fórmula:C26H29N3O4Pureza:99.66%Cor e Forma:SolidPeso molecular:447.53Ginkgolide B
CAS:<p>Ginkgolide B (BN-52021) is a PAFR antagonist(IC50=3.6 μM) isolated from Ginkgo biloba.</p>Fórmula:C20H24O10Pureza:98.66% - 99.81%Cor e Forma:White Crystal PowderPeso molecular:424.4Toyocamycin
CAS:<p>Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (</p>Fórmula:C12H13N5O4Pureza:98.1% - 98.17%Cor e Forma:SolidPeso molecular:291.26Dp44mT
CAS:<p>Dp44mT, a effective iron chelator, has selective antitumor activity.</p>Fórmula:C14H15N5SPureza:99% - 99.02%Cor e Forma:SolidPeso molecular:285.37trans-Chalcone
CAS:<p>trans-Chalcone (Chalkone) is an aromatic ketone that forms the central core for a variety of important biological compounds, which are known collectively as</p>Fórmula:C15H12OPureza:99.89%Cor e Forma:SolidPeso molecular:208.26Icaritin
CAS:<p>Icaritin (Anhydroicaritin) has hormone regulation activity and cardiovascular function improvement activity.</p>Fórmula:C21H20O6Pureza:97.69% - 99.76%Cor e Forma:SolidPeso molecular:368.38Se-Methylselenocysteine
CAS:<p>Se-Methylselenocysteine (Se-MSC) is a potent chemopreventive agent in many test systems and has been shown to inhibit tumor promotion and induce apoptosis.</p>Fórmula:C4H9NO2SePureza:99.49% - 99.87%Cor e Forma:White To Slightly Yellow PowderPeso molecular:182.08PTC-028
CAS:<p>PTC-028 selectively suppresses cancer cells whereas normal cells remain unaffected.</p>Fórmula:C19H12F5N5Pureza:97.61% - 98.12%Cor e Forma:SolidPeso molecular:405.32Angiotensin II human acetate
CAS:<p>Angiotensin II human acetate (DRVYIHPF acetate) is a vasoconstrictor that mainly acts on the AT1 receptor.</p>Fórmula:C52H75N13O14Pureza:98.89% - 99.78%Cor e Forma:SolidPeso molecular:1106.2BIBR 1532
CAS:<p>BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay).</p>Fórmula:C21H17NO3Pureza:98.49% - 98.90%Cor e Forma:SolidPeso molecular:331.36MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Cor e Forma:SolidPeso molecular:470.51Rapanone
CAS:<p>Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2.</p>Fórmula:C19H30O4Pureza:99.56%Cor e Forma:SolidPeso molecular:322.44RHPS4
CAS:<p>RHPS4 (RHPS 4 methosulfate) is a potent inhibitor of Telomerase at submicromolar.</p>Fórmula:C22H17F2N2·CH3O4SPureza:99.72%Cor e Forma:SolidPeso molecular:458.48Leachianone A
CAS:<p>Leachianone A (Isokurarinone) is a potential antitoxic agent, it shows inhibitory effects on cadmium- Induced cytotoxicity.</p>Fórmula:C26H30O6Pureza:98.53% - 99.79%Cor e Forma:SolidPeso molecular:438.51L-Glutamic acid monosodium salt
CAS:<p>L-Glutamic acid monosodium salt (MSG) (Monosodium glutamate) is an activator of mGlu1 receptor.</p>Fórmula:C5H8NO4·NaPureza:99.93%Cor e Forma:White Solid CrystallinePeso molecular:169.11Kevetrin hydrochloride
CAS:<p>Kevetrin hydrochloride (4-Isothioureidobutyronitrile hydrochloride) is a small molecule and activator of the tumor suppressor protein p53, with potential</p>Fórmula:C5H10ClN3SPureza:99.32% - 99.93%Cor e Forma:SolidPeso molecular:179.673-O-Acetyloleanolic acid
CAS:<p>3-O-acetyloleanolic acid dose-dependently inhibited the viability of HCT-116 cells.</p>Fórmula:C32H50O4Pureza:98% - 99.57%Cor e Forma:SolidPeso molecular:498.74Curcumol
CAS:<p>Curcumol ((-)-Curcumol), a pure monomer isolated extracted from Rhizoma Curcumaeis, has antitumor activities.</p>Fórmula:C15H24O2Pureza:98.99% - 99.87%Cor e Forma:SolidPeso molecular:236.35Everolimus
CAS:<p>Everolimus (SDZ-RAD) is a potent mTOR inhibitor that binds to FKBP-12. It is used alone or in combination with calcineurin inhibitors.</p>Fórmula:C53H83NO14Pureza:97.76% - 99.78%Cor e Forma:Off-White To Light Yellow PowdPeso molecular:958.22Ursonic Acid
CAS:<p>Ursonic Acid (TOS-BB-0966) belongs to the family of Ursane Triterpenes whose structure is based on the pentacyclic ursane skeleton.</p>Fórmula:C30H46O3Pureza:98.90% - >99.99%Cor e Forma:SolidPeso molecular:454.68Dinoprost tromethamine salt
CAS:<p>Dinoprost tromethamine salt (PGF2α THAM) is a naturally occurring prostaglandin used in medicine to induce labor and as an abortifacient.</p>Fórmula:C24H45NO8Pureza:99.73%Cor e Forma:Natural Form Crystals SolidPeso molecular:475.62Sanguinarine
CAS:<p>Sanguinarine (Pseudochelerythrine) is a specific inhibitor of Rac1b with anti-microbial, anti-oxidant and anti-inflammatory properties.</p>Fórmula:C20H14NO4Pureza:99.04% - 99.76%Cor e Forma:SolidPeso molecular:332.33Clovamide
CAS:<p>Trans-Clovamide (trans-Clovamide) is a naturally occurring caffeoyl conjugate identified in the antioxidant polyphenolic fraction of cocoa (T.</p>Fórmula:C18H17NO7Pureza:97.12% - 97.68%Cor e Forma:SolidPeso molecular:359.33Salermide
CAS:<p>Salermide is an inhibitor of Sirt1 and Sirt2, causing strong cancer-specific apoptotic cell death.</p>Fórmula:C26H22N2O2Pureza:97.09% - 99.55%Cor e Forma:SolidPeso molecular:394.47Piperlongumine
CAS:<p>Piperlongumine (Piplartine) is a natural alkaloid from Piper longum L.</p>Fórmula:C17H19NO5Pureza:97.03% - 99.90%Cor e Forma:SolidPeso molecular:317.34ODQ
CAS:<p>ODQ is an effective and selective soluble guanylyl cyclase (sGC) inhibitor.</p>Fórmula:C9H5N3O2Pureza:98.98%Cor e Forma:Off-White To Light Yellow PowderPeso molecular:187.15Epothilone B
CAS:<p>Epothilone B (EPO 906) is a compound isolated from the myxobacterium Sorangium cellulosum.</p>Fórmula:C27H41NO6SPureza:99.79% - 99.84%Cor e Forma:White PowderPeso molecular:507.68Atractylenolide II
CAS:<p>Atractylenolide II inhibits STAT3, activates p38, deactivates ERK/Akt, and induces p53-dependent cytotoxicity against melanoma.</p>Fórmula:C15H20O2Pureza:99.89% - 99.93%Cor e Forma:SolidPeso molecular:232.32Pitavastatin calcium
CAS:<p>Pitavastatin calcium (NK-104), a inhibitor of HMG-CoA reductase, lowers both total cholesterol and low-density lipoprotein cholesterol in animals and humans.</p>Fórmula:C50H46CaF2N2O8Pureza:98.89% - >99.99%Cor e Forma:White To Off-White PowderPeso molecular:880.98D4476
CAS:<p>D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).</p>Fórmula:C23H18N4O3Pureza:99.7% - 99.96%Cor e Forma:SolidPeso molecular:398.41Capsazepine
CAS:<p>Capsazepine, a TRPV1 antagonist (IC50: 562 nM), blocks capsaicin-induced heat pain.</p>Fórmula:C19H21ClN2O2SPureza:98% - 99.78%Cor e Forma:White To Off-White PowderPeso molecular:376.9L-Glutamic acid
CAS:<p>L-Glutamic acid is an agonist of glutamate receptors, including metabotropic glutamate receptors (mGluR), AMPA, NMDA, and KA. High-Quality, Low-Cost!</p>Fórmula:C5H9NO4Pureza:99.14% - 99.55%Cor e Forma:White Solid CrystallinePeso molecular:147.13SC144
CAS:<p>SC144 is an orally active small-molecule gp130 inhibitor.</p>Fórmula:C16H11FN6OPureza:99.20%Cor e Forma:SolidPeso molecular:322.3PND-1186
CAS:<p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>Fórmula:C25H26F3N5O3Pureza:99.14% - 99.75%Cor e Forma:SolidPeso molecular:501.5SIRT7 inhibitor 97491
CAS:<p>SIRT7 inhibitor 97491 is an HDAC inhibitor with high specificity for SIRT7 (IC50 = 325 nM). SIRT7 inhibitor 97491 promotes apoptosis through caspase pathway.</p>Fórmula:C15H12ClN3OPureza:99.79%Cor e Forma:SolidPeso molecular:285.73Bafetinib
CAS:<p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>Fórmula:C30H31F3N8OPureza:94.16% - 99.68%Cor e Forma:SolidPeso molecular:576.62PHT-427
CAS:<p>PHT-427 (CS-0223) is a dual Akt (Ki: 2.7 μM) and PDPK1 (Ki: 5.2 μM) inhibitor (high-affinity binding for the PH domains of Akt and PDPK1).</p>Fórmula:C20H31N3O2S2Pureza:97.54% - >99.99%Cor e Forma:SolidPeso molecular:409.61KPT-251
CAS:<p>KPT-251 is a selective nuclear export inhibitor.</p>Fórmula:C14H7F6N5OPureza:98.54%Cor e Forma:SolidPeso molecular:375.23Menin-MLL inhibitor MI-2
CAS:<p>Menin-MLL inhibitor MI-2 (MI2) is a potent menin-MLL interaction inhibitor with IC50 of 446 nM.</p>Fórmula:C18H25N5S2Pureza:97.46%Cor e Forma:SolidPeso molecular:375.55Benzyl isothiocyanate
CAS:<p>BITC, found in cruciferous veggies, exhibits anticancer, antimicrobial, and immunomodulatory effects.</p>Fórmula:C8H7NSPureza:99.25% - 99.83%Cor e Forma:Clear Yellow LiquidPeso molecular:149.21T0901317
CAS:<p>T0901317 is a potent and selective agonist for both LXR and FXR, with EC50 of ~50 nM and 5 μM, respectively; it inhibits nuclear factor/κB (NF/κB).</p>Fórmula:C17H12F9NO3SPureza:98% - 99.64%Cor e Forma:SolidPeso molecular:481.33DCH36_06
CAS:<p>DCH36_06 ((5E)-1-(3-chloro-4-methylphenyl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-ylidene]-2-thioxodihydropyrimidine-4,6(1H,5H)-dione) as a bona fide is a potent</p>Fórmula:C18H13ClN2O3SPureza:97.78%Cor e Forma:SolidPeso molecular:372.83Onvansertib
CAS:<p>Onvansertib (NMS-1286937) is a PLK1 inhibitor with high selectivity and oral activity. Onvansertib has antitumor activity. Cost-effective and quality-assured.</p>Fórmula:C24H27F3N8O3Pureza:98.3% - 99.88%Cor e Forma:SolidPeso molecular:532.52Tofacitinib
CAS:<p>Tofacitinib (Tasocitinib) is an orally Janus kinase inhibitor. Tofacitinib is used for the treatment of rheumatoid arthritis. Cost effective and quality assured.</p>Fórmula:C16H20N6OPureza:99% - >99.99%Cor e Forma:SolidPeso molecular:312.37PHA-793887
CAS:<p>PHA-793887 has been used in trials studying the treatment of Advanced/Metastatic Solid Tumors.</p>Fórmula:C19H31N5O2Pureza:98.02% - >99.99%Cor e Forma:SolidPeso molecular:361.48EPI-001
CAS:<p>EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.</p>Fórmula:C21H27ClO5Pureza:99% - 99.67%Cor e Forma:SolidPeso molecular:394.897,8-Dihydroxyflavone
CAS:<p>7,8-Dihydroxyflavone (7,8-DHF) is a naturally-occurring flavone and exist in Tridax procumbens, Godmania aesculifolia, and primula tree leaves.</p>Fórmula:C15H10O4Pureza:98.48% - 99.81%Cor e Forma:SolidPeso molecular:254.24INH6
CAS:<p>INH6, an effective Hec1 inhibitor, selectively disrupts the Hec1/Nek2 interaction and induces chromosome mis-alignment.</p>Fórmula:C19H18N2OSPureza:98.81%Cor e Forma:SolidPeso molecular:322.42Trigonelline
CAS:<p>Trigonelline (Trigenolline), an alkaloid with potential antidiabetic activity, is present in considerable amounts in coffee.</p>Fórmula:C7H7NO2Pureza:97.585% - 99.49%Cor e Forma:Prisms Aqueous From Alcohol + Water SolidPeso molecular:137.14Tetramethylcurcumin
CAS:<p>Tetramethylcurcumin is a novel curcumin analog, is an effective inhibitors of STAT3 phosphorylation, DNA binding activity, and transactivation in vitro.it also</p>Fórmula:C25H28O6Pureza:97.69% - 99.94%Cor e Forma:SolidPeso molecular:424.49Tauroursodeoxycholate sodium
CAS:<p>Tauroursodeoxycholate sodium (TUDC) is an endoplasmic reticulum (ER) stress inhibitor, used for the treatment of gallstones and liver cirrhosis.</p>Fórmula:C26H44NNaO6SPureza:97.90%Cor e Forma:SolidPeso molecular:521.69Cinobufagin
CAS:<p>Cinobufagin (Cinobufagine) is a selective Na+/K+-ATPase inhibitor. The activity of Cinobufagin is same as ouabain.</p>Fórmula:C26H34O6Pureza:97.77% - 99.97%Cor e Forma:SolidPeso molecular:442.54Euphorbia Factor L2
CAS:<p>Euphorbia Factor L2 alleviates lipopolysaccharide-induced acute lung injury and inflammation through inhibits NF-κB activation.</p>Fórmula:C38H42O9Pureza:99.53% - 99.96%Cor e Forma:SolidPeso molecular:642.73LYN-1604 dihydrochloride
CAS:<p>LYN-1604 is a novel ULK1 activator.It inducing cell death involved in ATF3, RAD21, and caspase3, accompanied by autophagy and apoptosis.</p>Fórmula:C33H45Cl4N3O2Pureza:98.95% - 99.92%Cor e Forma:SolidPeso molecular:657.54Azadirachtin
CAS:<p>Azadirachtin has antifungal activity, used as an insecticide.</p>Fórmula:C35H44O16Pureza:98.11% - 99.713%Cor e Forma:SolidPeso molecular:720.71SBE13 Hydrochloride
CAS:<p>SBE13 Hydrochloride (SBE 13 HCl) is an effective and specific PLK1 inhibitor (IC50: 0.2 nM); no inhibition om Aurora A kinase, Plk2/3.</p>Fórmula:C24H28Cl2N2O4Pureza:99.00% - ≥95%Cor e Forma:SolidPeso molecular:479.4Polyphyllin VI
CAS:<p>1. Polyphyllin VI has hemostasis , expectorant , bacteriostasis, anticytotoxic, anti pregnancy kill sperm effects.</p>Fórmula:C39H62O13Pureza:99.69% - 99.72%Cor e Forma:SolidPeso molecular:738.9TCS JNK 5a
CAS:<p>TCS JNK 5a (SC202671) is an effective, specific inhibitor of JNK3(pIC50= 6.7), JNK2(pIC50=6.5).</p>Fórmula:C20H16N2OSPureza:99.22% - 99.51%Cor e Forma:SolidPeso molecular:332.42Ruxolitinib
CAS:<p>Ruxolitinib (INCB018424) is a JAK1/2 inhibitor (IC50=3.3/2.8 nM) that is potent and selective.</p>Fórmula:C17H18N6Pureza:99.4% - >99.99%Cor e Forma:SolidPeso molecular:306.36Eribulin mesylate
CAS:<p>Eribulin mesylate (E7389), a microtubule inhibitor, treats metastatic breast cancer by halting cell division.</p>Fórmula:C41H63NO14SPureza:97.02% - >99.99%Cor e Forma:SolidPeso molecular:826XI-006
CAS:<p>NSC-207895 (XI-006) suppresses MDMX with IC50 of 2.5 μM, leading to enhanced p53 stabilization/activation and DNA damage, and regulates MDM2, an E3 ligase.</p>Fórmula:C11H13N5O4Pureza:99.51%Cor e Forma:SolidPeso molecular:279.25Cabozantinib
CAS:<p>Cabozantinib (XL184) is a multi-targeted tyrosine kinase receptor inhibitor that inhibits VEGFR2, c-Met, Kit, Axl, and Flt3 (IC50=0.035/1.3/4.6/7/11.3 nM).</p>Fórmula:C28H24FN3O5Pureza:99.68% - 99.88%Cor e Forma:SolidPeso molecular:501.51Urolithin C
CAS:<p>Urolithin C is a gut metabolite of ellagic acid. Urolithin C induces apoptosis in PC12 cells through a mitochondria-mediated pathway.</p>Fórmula:C13H8O5Pureza:98.01% - 99.53%Cor e Forma:SolidPeso molecular:244.2Piperazine Erastin
CAS:<p>Piperazine erastin is an analog of erastin. It causes an iron-dependent form of non-apoptotic cell death termed ferroptosis.</p>Fórmula:C35H41ClN6O4Pureza:99.52%Cor e Forma:SolidPeso molecular:645.19Importazole
CAS:<p>Importazole is an inhibitor of the nuclear transport receptor importin-β.</p>Fórmula:C20H22N4Pureza:99.6% - >99.99%Cor e Forma:SolidPeso molecular:318.42AP-III-a4
CAS:<p>AP-III-a4 (ENOblock) (ENOblock) is the first nonsubstrate analogue inhibitor of enolase with IC50 of 0.576 μM.</p>Fórmula:C31H43FN8O3Pureza:98.24% - 99.90%Cor e Forma:SolidPeso molecular:594.72PRIMA-1
CAS:<p>PRIMA-1 (NSC-281668) is a mutant p53 reactivator. It induces apoptosis and inhibits growth of human tumors with mutant p53.</p>Fórmula:C9H15NO3Pureza:99.22%Cor e Forma:SolidPeso molecular:185.22GSK2656157
CAS:<p>GSK2656157 is a highly specific and ATP-competitive PERK inhibitor (IC50: 0.9 nM) in a cell-free assay.</p>Fórmula:C23H21FN6OPureza:98.59% - >99.99%Cor e Forma:SolidPeso molecular:416.45PROCYANIDIN C1
CAS:<p>Procyanidin C1 is a natural polyphenol. It reduces Bcl-2 protein levels.Cost-effective and quality-assured.</p>Fórmula:C45H38O18Pureza:97.01% - 99.86%Cor e Forma:SolidPeso molecular:866.77ICCB-19 hydrochloride
CAS:<p>ICCB-19 hydrochloride (ICCB-19 HCl) is an inhibitor of TRADD (TNFRSF1A Associated Via Death Domain). It binds to a pocket on the TRADD-N.</p>Fórmula:C12H22ClN3OSPureza:99.3%Cor e Forma:SolidPeso molecular:291.84ON1231320
CAS:<p>ON1231320 (GBO-006) is a Polo-like kinase 2 (PLK2) inhibitor.</p>Fórmula:C22H15F2N5O3SPureza:97.31%Cor e Forma:SolidPeso molecular:467.45Pictilisib
CAS:<p>Pictilisib (GDC-0941) (GDC-0941) is a potent pan inhibitor of class I catalytic subunits of PI3K (IC50s: 3/33/3/75 nM for p110α/β/δ/γ).</p>Fórmula:C23H27N7O3S2Pureza:98.69% - 99.97%Cor e Forma:SolidPeso molecular:513.64BAI1
CAS:<p>BAI1 (Bax channel blocker) is a potent inhibitor of Bax-mediated mitochondrial cytochrome C release (IC50: 0.52 μM).</p>Fórmula:C19H21Br2N3OPureza:97.74%Cor e Forma:SolidPeso molecular:467.2STM2457
CAS:<p>View and buy STM2457 from TargetMol.STM2457 is a first-in-class, highly potent, selective and orally active inhibitor of METTL3.Cited in 2 publications.</p>Fórmula:C25H28N6O2Pureza:97.44% - 98.90%Cor e Forma:SolidPeso molecular:444.53Cidofovir
CAS:<p>Cidofovir ((S)-HPMPC) 通过特异性抑制病毒 DNA 合成来抑制病毒复制。</p>Fórmula:C8H14N3O6PPureza:99.24% - 99.76%Cor e Forma:Fluffy White PowderPeso molecular:279.19Galanthamine
CAS:<p>Galanthamine (Galantamine) is an acetylcholinesterase (AChE)inhibitor(IC50 : 500 nM), can reduce brain damage induced by hypoxia-ischemia.</p>Fórmula:C17H21NO3Pureza:98.03% - 99.87%Cor e Forma:Off-White SolidPeso molecular:287.35LQZ-7I
CAS:<p>LQZ-7I is an inhibitor of surviving-targeting. It orally effectively inhibits xenograft tumor growth and induces survivin loss in tumors</p>Fórmula:C20H14F2N4Pureza:99.81% - 99.87%Cor e Forma:SolidPeso molecular:348.35Liensinine
CAS:<p>1. Liensinine, a kind of isoquinoline alkaloid, can antagonize the ventricular arrhythmias.</p>Fórmula:C37H42N2O6Pureza:98.92% - 99.93%Cor e Forma:White-Like PowderPeso molecular:610.74Adaphostin
CAS:<p>Adaphostin (NSC-680410) is a p210Bcr/Abl tyrosine kinase inhibitor with IC50 of 14 μM.</p>Fórmula:C24H27NO4Pureza:98.29%Cor e Forma:SolidPeso molecular:393.48Cabozantinib hydrochloride
CAS:<p>Cabozantinib hydrochloride (XL184) is a potent pan-tyrosine kinases inhibitor that inhibits VEGFR2, c-Met, Kit, Axl, and Flt4 (IC50s: 0.035, 1.3, 4.6, 7 and 6</p>Fórmula:C28H25ClFN3O5Pureza:99.97%Cor e Forma:SolidPeso molecular:537.96Malachite green oxalate
CAS:<p>Malachite green oxalate is a triphenylmethane dye which can be used to detect the release of phosphate in enzymatic reactions.</p>Fórmula:C23H25N2·C2HO4C2H2O4Cor e Forma:Dark Green Crystals With A Metallic LusterPeso molecular:463.51HYPOCRELLIN B
CAS:<p>HYPOCRELLIN B, from Hypocrella bambusae, breaks DNA, triggers apoptosis in ovarian cells, and stops Staphylococcus growth via ROS.</p>Fórmula:C30H24O9Pureza:98% - 98.87%Cor e Forma:SolidPeso molecular:528.51Raddeanin A
CAS:<p>Raddeanin A is a natural triterpenoid saponin from Cyperus japonicus that inhibits histone deacetylase.Cost-effective and quality-assured.</p>Fórmula:C47H76O16Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:897.1Karanjin
CAS:<p>Karanjin, a flavonoid from karanja seeds, boosts GLUT4, AMPK in muscles, and triggers cancer cell apoptosis.</p>Fórmula:C18H12O4Pureza:99.01%Cor e Forma:SolidPeso molecular:292.29Mivebresib
CAS:<p>Mivebresib (ABBV-075) is a potent BET inhibitor with antitumor effects, disrupting gene expression and MYC, TMPRSS2-ETS proteins.</p>Fórmula:C22H19F2N3O4SPureza:98.74% - 99.32%Cor e Forma:SolidPeso molecular:459.47Madecassoside
CAS:<p>Madecassoside (Asiaticoside A) is a pentacyclic triterpene extracted from Centella asitica (L.) with anti-inflammatory, anti-oxidative and anti-aging activities</p>Fórmula:C48H78O20Pureza:99.46% - 99.85%Cor e Forma:White PowderPeso molecular:975.12PFK-158
CAS:<p>PFK-158 is an effective and specific inhibitor PFKFB3.</p>Fórmula:C18H11F3N2OPureza:95.49% - 99.16%Cor e Forma:SolidPeso molecular:328.29Z-FA-FMK
CAS:<p>Z-FA-FMK can irreversibly inhibit cysteine protease and also inhibit effector caspases.</p>Fórmula:C21H23FN2O4Pureza:98.84% - 99.68%Cor e Forma:SolidPeso molecular:386.422-methoxycinnamaldehyde
CAS:<p>2-methoxycinnamaldehyde is a natural compound of Cinnamomum cassia,has been widely studied with regard to its antitumor activity.</p>Fórmula:C10H10O2Pureza:98%Cor e Forma:Physical Description Yellow Crystals (Ntp 1992)Peso molecular:162.19Desoxyrhaponticin
CAS:<p>Deoxyrhaponticin may reduce post-meal blood sugar and inhibit cancer cell growth.</p>Fórmula:C21H24O8Pureza:99.97% - ≥95%Cor e Forma:SolidPeso molecular:404.41SU9516
CAS:<p>SU9516 is a potent CDK2 inhibitor, with an IC50 of 22 nM, and also has inhibitory effects on CDK1 and CDK4, with IC50s of 40 nM and 200 nM, respectively.</p>Fórmula:C13H11N3O2Pureza:99.34% - 99.87%Cor e Forma:SolidPeso molecular:241.25Erastin
CAS:<p>Erastin is an iron death activator that acts on the mitochondrial VDAC in a ROS- and iron-dependent manner, anti-tumor. High-Quality, Low-Cost!</p>Fórmula:C30H31ClN4O4Pureza:98% - 99.75%Cor e Forma:SolidPeso molecular:547.04PKCβ inhibitor 1
CAS:<p>PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2,</p>Fórmula:C24H21N5O2Pureza:99.33%Cor e Forma:SolidPeso molecular:411.46L-Ascorbic acid sodium salt
CAS:<p>L-Ascorbic acid sodium salt (Vitamin C sodium salt) is a more bioavailable form of vitamin C that is an alternative to taking ascorbic acid as a supplement.</p>Fórmula:C6H7NaO6Pureza:98.73% - 99.75%Cor e Forma:Less Solid PowderPeso molecular:198.11Zinc Protoporphyrin
CAS:<p>Zinc Protoporphyrin is an oral HO-1 inhibitor that reduces PG's protection against H2O2 and has anti-cancer properties.</p>Fórmula:C34H32N4O4ZnPureza:95.43% - 99.27%Cor e Forma:SolidPeso molecular:626.02A-1155463
CAS:<p>A-1155463, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and >1000-fold weaker binding to BCL-2, BCL-W and MCL-1.</p>Fórmula:C35H32FN5O4S2Pureza:96.1% - 99%Cor e Forma:SolidPeso molecular:669.79LY-294002 hydrochloride
CAS:<p>LY-294002 HCl (NSC 697286) is a stable PI3K inhibitor (IC50: 0.5-0.97 µM) and prevents autophagosome formation.</p>Fórmula:C19H17NO3·HClPureza:99.95%Cor e Forma:SolidPeso molecular:343.81PI-1840
CAS:<p>PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.</p>Fórmula:C22H26N4O3Pureza:98.82%Cor e Forma:SolidPeso molecular:394.47Cynaroside
CAS:<p>Cynaroside (Luteolin 7-O-Glucoside) is a flavone, a flavonoid-like chemical compound. It has an anti-oxidant effect, inhibiting lipid and protein oxidation.</p>Fórmula:C21H20O11Pureza:98% - >99.99%Cor e Forma:SolidPeso molecular:448.38Soyasapogenol B
CAS:<p>Soyasapogenol B has anti-cancer, hypocholesterolemic, anticomplementary, hepatoprotective effects, it inhibits proliferation of cultured Hep-G2.</p>Fórmula:C30H50O3Pureza:99.51% - 99.81%Cor e Forma:SolidPeso molecular:458.72Linderalactone
CAS:<p>1. Linderalactone showed significant inhibitory effects on superoxide anion generation by human neutrophils in response to fMLP/CB, values of IC5 is 8.48 μg/mL.</p>Fórmula:C15H16O3Pureza:99.79%Cor e Forma:SolidPeso molecular:244.29TVB-3166
CAS:<p>TVB-3166: reversible, selective FASN inhibitor, induces apoptosis, hinders xenograft growth (IC50: 42 nM FASN, 81 nM palmitate synthesis).</p>Fórmula:C24H24N4OPureza:99.53% - 99.57%Cor e Forma:SolidPeso molecular:384.47Sirtinol
CAS:<p>Sirtinol is a selective SIRT1/2 inhibitor (IC50: 131/38 μM).</p>Fórmula:C26H22N2O2Pureza:97.12% - 99.96%Cor e Forma:SolidPeso molecular:394.47Embelin
CAS:<p>Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM).</p>Fórmula:C17H26O4Pureza:97.07% - 99.88%Cor e Forma:SolidPeso molecular:294.39CPI1189
CAS:<p>CPI1189 (REN-1189) is a TNF-a release inhibitor potentially for the treatment of sciatica and postherpetic neuralgia.</p>Fórmula:C13H18N2O2Pureza:98.34% - 99.51%Cor e Forma:SolidPeso molecular:234.29Betulin
CAS:<p>Betulin (betulinol) (lup-20(29)-ene-3β, 28-diol) is an abundant, naturally occurring triterpene.</p>Fórmula:C30H50O2Pureza:98.52% - 99.88%Cor e Forma:White Crystalline PowderPeso molecular:442.72GSK 3 Inhibitor IX
CAS:<p>GSK 3 Inhibitor IX (6-BIO) is a selective reversible, ATP-competitive inhibitor of GSK-3α/β and CDK1-cyclinB complex.</p>Fórmula:C16H10BrN3O2Pureza:98% - 99.72%Cor e Forma:SolidPeso molecular:356.17FR 180204
CAS:<p>FR 180204 is a potent and selective ATP-competitive inhibitor of ERK1 and ERK2.</p>Fórmula:C18H13N7Pureza:98% - 99.74%Cor e Forma:SolidPeso molecular:327.34Calycosin
CAS:<p>Calycosin modulates estrogen receptors, induces apoptosis in cancers, and shows skin-lightening by inhibiting tyrosinase (IC50: 38.4µM).</p>Fórmula:C16H12O5Pureza:99.91% - >99.99%Cor e Forma:White PowderPeso molecular:284.26Selonsertib
CAS:<p>Selonsertib (GS-4997), an oral ASK1 inhibitor, may have anti-inflammatory, anti-fibrotic, and anti-cancer effects.</p>Fórmula:C24H24FN7OPureza:95.04% - 99.53%Cor e Forma:SolidPeso molecular:445.49Trametinib
CAS:<p>Trametinib (GSK1120212), an ATP-noncompetitive MEK 1/2 inhibitor (IC50: 0.7/0.9 nM), weakly inhibits >180 kinases.</p>Fórmula:C26H23FIN5O4Pureza:98% - 99.96%Cor e Forma:SolidPeso molecular:615.39Wogonin
CAS:<p>Wogonin (Vogonin) is a cell-permeable and orally available flavonoid that displays anti-inflammatory and anticancer properties.</p>Fórmula:C16H12O5Pureza:98% - 99.8%Cor e Forma:Yellow CrystalPeso molecular:284.26Formosanin C
CAS:<p>Formosanin C (Polyphyllin B) is a compound isolated from Rhizoma Paridis, showed pro-apoptosis and immunoregulation with antitumor activity.</p>Fórmula:C51H82O20Pureza:99.75% - >99.99%Cor e Forma:SolidPeso molecular:1015.18Cyasterone
CAS:<p>Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, via regulating EGFR signaling pathway, it may be a promising</p>Fórmula:C29H44O8Pureza:99.32% - 99.70%Cor e Forma:SolidPeso molecular:520.65Quisinostat
CAS:<p>Quisinostat (JNJ-26481585), a second-gen HDAC inhibitor, is most potent for HDAC1 (IC50 0.11 nM) and selectively affects HDACs 2, 4, 10, and 11.</p>Fórmula:C21H26N6O2Pureza:96.01% - ≥98%Cor e Forma:SolidPeso molecular:394.47α-Hederin
CAS:<p>Alpha-Hederin (Tauroside E) is a water-soluble pentacyclic triterpenoid saponin found in the seeds of Nigella sativa, with hemolytic and apoptotic properties.</p>Fórmula:C41H66O12Pureza:99.44% - 99.89%Cor e Forma:SolidPeso molecular:750.96BMS-536924
CAS:<p>BMS-536924 (BMS 536924) is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for</p>Fórmula:C25H26ClN5O3Pureza:99.02%Cor e Forma:SolidPeso molecular:479.96Genistein
CAS:<p>Genistein (NPI 031L) is a natural soy isoflavone, a multi-targeted tyrosine kinase inhibitor. Genistein has antitumor effects. Cost effective and quality assured.</p>Fórmula:C15H10O5Pureza:98.22% - 99.64%Cor e Forma:Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether SolidPeso molecular:270.24(1E,6E)-Bis(demethoxy)curcumin
CAS:<p>(1E,6E)-Bis(demethoxy)curcumin (Curcumin III) is a natural demethoxy derivative of curcumin,with anti-inflammatory and anti-cancer activities.</p>Fórmula:C19H16O4Pureza:97.45%Cor e Forma:SolidPeso molecular:308.33AZ 628
CAS:<p>AZ628 is a new pan-Raf inhibitor for BRAF, BRAFV600E, and c-Raf-1 with IC50 of 105 nM, 34 nM and 29 nM, also inhibits VEGFR2, DDR2, Lyn, Flt1, FMS, etc.</p>Fórmula:C27H25N5O2Pureza:99.50%Cor e Forma:SolidPeso molecular:451.52Chelidonine
CAS:<p>Chelidonine from Chelidonium majus triggers HeLa cell apoptosis, may reverse MDR, boost chemotherapeutics against leukemia, and inhibit cancer cell metastasis.</p>Fórmula:C20H19NO5Pureza:98% - 99.61%Cor e Forma:SolidPeso molecular:353.37Tasisulam
CAS:<p>Tasisulam (LY573636) is an apoptosis inducer and an antitumor agent via the intrinsic pathway.</p>Fórmula:C11H6BrCl2NO3S2Pureza:99% - >99.99%Cor e Forma:SolidPeso molecular:415.11Wedelolactone
CAS:<p>Wedelolactone (IKK Inhibitor II) inhibits NF-κB-mediated gene transcription in cells by blocking the phosphorylation and degradation of IκBα.</p>Fórmula:C16H10O7Pureza:98.07% - 99.87%Cor e Forma:SolidPeso molecular:314.25Goserelin acetate
CAS:<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Fórmula:C61H88N18O16Pureza:99.77% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:1329.46PKR-IN-C16
CAS:<p>PKR-IN-C16: inhibits PKR autophosphorylation and translation blockade; binds ATP site; IC50 of 186-210 nM; protects cells from ER stress damage.</p>Fórmula:C13H8N4OSPureza:97.8%Cor e Forma:SolidPeso molecular:268.29Neferine
CAS:<p>Neferine: anti-tumor, enhances DOX efficacy, prevents diabetic vasculopathy; mediates via CYP3A4, GSH depletion, blocks ROS/Akt/NF-κB.</p>Fórmula:C38H44N2O6Pureza:98.81% - 99.65%Cor e Forma:SolidPeso molecular:624.77Momordin Ic
CAS:<p>Momordin Ic (Momordin 1c) might represent a potential anticancer activity, by inducing apoptosis through oxidative stress-regulated mitochondrial dysfunction</p>Fórmula:C41H64O13Pureza:98% - 99.69%Cor e Forma:SolidPeso molecular:764.94Sal003
CAS:<p>Sal003, an effective cell-permeable analog, inhibitis the eIF2α phosphatase.</p>Fórmula:C18H15Cl4N3OSPureza:99.17% - 99.77%Cor e Forma:SolidPeso molecular:463.21Hypericin
CAS:<p>Hypericin (Cyclosan) is a natural anthraquinone compound. Hypericin exhibits antimicrobial, antiviral, antitumor, and antidepressant effects. Cost-effective and quality-assured.</p>Fórmula:C30H16O8Pureza:99.05% - ≥98%Cor e Forma:Red-Coloured Anthraquinone-DerivativePeso molecular:504.44Afatinib
CAS:<p>Afatinib (BIBW 2992) is an irreversible and orally EGFR family inhibitor that inhibits EGFR and HER2. Afatinib has antitumor activity. Cost effective and quality assured.</p>Fórmula:C24H25ClFN5O3Pureza:98.56% - 99.9%Cor e Forma:Off-White SolidPeso molecular:485.94Salvigenin
CAS:<p>Salvigenin is a potent hMAO-A inhibitor, has neuroprotective, antitumor and immunomodulatory effects.</p>Fórmula:C18H16O6Pureza:99.17% - 99.78%Cor e Forma:SolidPeso molecular:328.32Gardenin B
CAS:<p>Gardenin B exhibits superior antiproliferative activity against lung, breast, colon, hepatic and leukaemia cell lines as well as in keratinocytes .</p>Fórmula:C19H18O7Pureza:98.80% - 99.74%Cor e Forma:SolidPeso molecular:358.34Delanzomib
CAS:<p>Delanzomib (CEP-18770) is an oral proteasome inhibitor with an IC50 of 3.8 nM, targeting chymotrypsin-like activity with minimal effect on other activities.</p>Fórmula:C21H28BN3O5Pureza:95.52% - 99.46%Cor e Forma:SolidPeso molecular:413.28Telekin
CAS:<p>Telekin, a sesquiterpene lactone from Carpesium divaricatum, strongly inhibits cancer cell growth.</p>Fórmula:C15H20O3Pureza:99.86% - 99.97%Cor e Forma:SolidPeso molecular:248.32AT7519
CAS:<p>AT7519 is a CDK1/2/4/6/9 inhibitor (IC50: 10-210 nM). It is less effective to CDK3 and little active to CDK7.</p>Fórmula:C16H17Cl2N5O2Pureza:98.88% - 99.65%Cor e Forma:SolidPeso molecular:382.24Malabaricone B
CAS:<p>Malabaricone B is a Spice-derived phenolic, it induces mitochondrial damage in lung cancer cells via a p53-independent pathway.</p>Fórmula:C21H26O4Pureza:99.84% - 99.91%Cor e Forma:SolidPeso molecular:342.43(E/Z)-TG003
CAS:<p>(E/Z)-TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor.</p>Fórmula:C13H15NO2SPureza:98% - 99.04%Cor e Forma:SolidPeso molecular:249.33ENMD-2076
CAS:<p>ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα.</p>Fórmula:C21H25N7Pureza:97.63% - ≥95%Cor e Forma:SolidPeso molecular:375.47m-3M3FBS
CAS:<p>m-3M3FBS is a phospholipase C (PLC) activator.</p>Fórmula:C16H16F3NO2SPureza:99.66%Cor e Forma:SolidPeso molecular:343.36Polygalacin D
CAS:<p>Polygalacin D shows anti- proliferation, anti-inflammary, and hepatoprotective activities, it can inhibit the expression of lipopolysaccharide (LPS)-induced</p>Fórmula:C57H92O27Pureza:98.95% - ≥98%Cor e Forma:SolidPeso molecular:1209.4Choline
CAS:<p>Choline is a ubiquitous water soluble nutrient, often associated with the B vitamins</p>Fórmula:C5H15NO2Pureza:99.97% - ≥98%Cor e Forma:LiquidPeso molecular:121.18MPTP hydrochloride
CAS:<p>MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability.</p>Fórmula:C12H16ClNPureza:96.35% - >99.99%Cor e Forma:SolidPeso molecular:209.72CHR-6494 TFA
CAS:<p>CHR-6494 TFA: potent haspin inhibitor (IC50=2 nM), blocks H3T3 phosphorylation, triggers apoptosis in cancer cells. Used for cancer research.</p>Fórmula:C18H17F3N6O2Pureza:99.50%Cor e Forma:SolidPeso molecular:406.36Obatoclax Mesylate
CAS:Obatoclax Mesylate (GX15-070) is a Bcl-2 antagonist (Ki: 0.22 μM) and can induce apoptosis with up-regulation of Bim, induced cytochrome c release, andFórmula:C20H19N3O·CH4O3SPureza:99.58% - 99.88%Cor e Forma:SolidPeso molecular:413.49Ibandronate sodium monohydrate
CAS:<p>Ibandronate sodium monohydrate (BM-210955) is a highly potent nitrogen-containing bisphosphonate used for the treatment of osteoporosis.</p>Fórmula:C9H24NNaO8P2Pureza:99.62%Cor e Forma:White Crystalline PowderPeso molecular:359.23Neobavaisoflavone
CAS:<p>Neobavaisoflavone: DNA polymerase inhibitor, potential for treating bone loss, anti-inflammatory, reduces ROS, RNS, cytokines in macrophages.</p>Fórmula:C20H18O4Pureza:99.31% - 99.87%Cor e Forma:SolidPeso molecular:322.35RGX-202
CAS:<p>RGX-202 (β-GPA) is an orally active inhibitor of the SLC6A8 transport protein. RGX-202 is a creatine analog that alters skeletal muscle energy expenditure.</p>Fórmula:C4H9N3O2Pureza:99.67% - 99.8%Cor e Forma:SolidPeso molecular:131.13PD173955
CAS:<p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>Fórmula:C21H16Cl2N4OSPureza:98.52% - 98.99%Cor e Forma:SolidPeso molecular:443.35Nobiletin
CAS:<p>Nobiletin: a citrus-derived flavone with anti-inflammatory and anti-cancer properties; water-insoluble, very weak acid.</p>Fórmula:C21H22O8Pureza:98.65% - 99.76%Cor e Forma:SolidPeso molecular:402.39Bioymifi
CAS:<p>Bioymifi (DR5 Activator), a novel TRAIL activator, binds to DR5's ECD, inducing DR5 aggregation and stimulating cell apoptosis. Cost-effective and quality-assured.</p>Fórmula:C22H12BrN3O4SPureza:98% - 99.79%Cor e Forma:SolidPeso molecular:494.32Oncrasin-1
CAS:<p>Oncrasin 1 is a potent inhibitor of anticancer that kills various human lung cancer cells with K-Ras mutations at low or submicromolar concentrations</p>Fórmula:C16H12ClNOPureza:99.75%Cor e Forma:SolidPeso molecular:269.73TREM2-IN-1
CAS:<p>TREM2-IN-1 (OPA) is a platinum-based TREM2 inhibitor with anti-cancer and anti-tumor activity, inhibiting the immune-regulatory activity of TREM2 on macrophages</p>Fórmula:C46H68N2O20PtPureza:98.56%Cor e Forma:SolidPeso molecular:1164.12Enzastaurin
CAS:<p>Enzastaurin (LY317615) (LY317615) is an effective PKCβ selective inhibitor (IC50: 6 nM), 6- to 20-fold selectivity against PKCα/γ/ε.</p>Fórmula:C32H29N5O2Pureza:98% - >99.99%Cor e Forma:SolidPeso molecular:515.6CA-5f
CAS:<p>CA-5f is a potent late-stage macroautophagy/autophagy inhibitor via inhibiting autophagosome-lysosome fusion.</p>Fórmula:C24H24N2O3Pureza:99.69%Cor e Forma:SolidPeso molecular:388.46Trabectedin
CAS:<p>Trabectedin (Ecteinascidin 743) has potent antitumor activity and the potential for soft tissue sarcoma and ovarian cancer research.</p>Fórmula:C39H43N3O11SPureza:≥98%Cor e Forma:SolidPeso molecular:761.84Etidronic acid
CAS:<p>Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.</p>Fórmula:C2H8O7P2Pureza:99.93% - ≥95%Cor e Forma:Liquid SyrupPeso molecular:206.03Roquinimex
CAS:<p>Roquinimex (FCF89) (Linomide) is a quinoline derivative immunostimulant which increases NK cell activity and macrophage cytotoxicity; inhibits angiogenesis and</p>Fórmula:C18H16N2O3Pureza:97.69%Cor e Forma:SolidPeso molecular:308.33Epoxiconazole
CAS:<p>Epoxiconazole (BAS-480F) is a 14-α demethylase inhibitor. It inhibits ergosterol synthesis and fungal cell wall formation.</p>Fórmula:C17H13ClFN3OPureza:98.57%Cor e Forma:Solid PowderPeso molecular:329.76BAY 87-2243
CAS:<p>BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).</p>Fórmula:C26H26F3N7O2Pureza:98% - 99.95%Cor e Forma:SolidPeso molecular:525.53PATULIN
CAS:<p>Patulin (Claviform) is a mycotoxin produced by a variety of molds commonly found in rotting apples, including Aspergillus and Penicillium.</p>Fórmula:C7H6O4Pureza:99.91% - 99.98%Cor e Forma:Compact Prisms Or Thick Plates From Ether Or Chloroform White CrystallinePeso molecular:154.12Semaglutide
CAS:<p>Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).</p>Fórmula:C187H291N45O59Pureza:96.92% - 99.78%Cor e Forma:SolidPeso molecular:4114
