EGFR
PF-6274484
CAS:1035638-91-5
PF-6274484, a high affinity, irreversible covalent inhibitor of EGFR kinase with Ki of 0.14 nM, …
Formula:
C18H14ClFN4O2
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
372.78
Ref: TM-T22396
2mg | 40.00 € | ||
5mg | 60.00 € | ||
10mg | 90.00 € | ||
25mg | 184.00 € | ||
50mg | 343.00 € | ||
100mg | 510.00 € | ||
500mg | 1,112.00 € | ||
1ml*10 (DMSO) | 66.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
CP-724714
CAS:383432-38-0
CP-724714 (CP724714) is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against …
Formula:
C27H27N5O3
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
469.54
Ref: TM-T4014
1mg | 43.00 € | ||
2mg | 57.00 € | ||
5mg | 94.00 € | ||
10mg | 153.00 € | ||
25mg | 267.00 € | ||
50mg | 445.00 € | ||
100mg | 646.00 € | ||
1ml*10 (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AZD8931 diFuMaric acid
CAS:1196531-39-1
AZD8931 is a reversible and ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 (IC50 of …
Formula:
C31H33ClFN5O11
Purity:
99%
Color and Shape:
Solid
Molecular weight:
706.1
Ref: TM-T8751
1mg | 128.00 € | ||
5mg | 282.00 € | ||
10mg | 421.00 € | ||
25mg | 694.00 € | ||
50mg | 975.00 € | ||
100mg | 1,319.00 € | ||
1ml*10 (DMSO) | 418.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
SYR127063
CAS:871026-18-5
SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a …
Formula:
C23H20ClF3N4O3
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
492.88
Ref: TM-T34760
1mg | 128.00 € | ||
5mg | 281.00 € | ||
10mg | 423.00 € | ||
25mg | 694.00 € | ||
50mg | 978.00 € | ||
1ml*10 (DMSO) | 348.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AG490
CAS:133550-30-8
AG490 (Tyrphostin B42) is an inhibitor of EGFR (IC50: 0.1 μM). It is 135-fold more …
Formula:
C17H14N2O3
Purity:
99.7%
Color and Shape:
Yellow Solid
Molecular weight:
294.3
Ref: TM-T2600
10mg | 55.00 € | ||
25mg | 74.00 € | ||
50mg | 90.00 € | ||
100mg | 100.00 € | ||
200mg | 162.00 € | ||
500mg | 278.00 € | ||
1ml*10 (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Chrysophanol
CAS:481-74-3
Chrysophanol (Turkey Rhubarb) is an EGFR/mTOR pathway inhibitor, which can be found in rhubarb, and …
Formula:
C15H10O4
Purity:
99.7%
Color and Shape:
Physical Description Golden Yellow Plates Or Brown Powder Melting Point 196°C
Molecular weight:
254.24
Ref: TM-T2995
50mg | 43.00 € | ||
100mg | 57.00 € | ||
1ml*10 (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Canertinib dihydrochloride
CAS:289499-45-2
Canertinib dihydrochloride (PD-183805 dihydrochloride) is the hydrochloride salt of an orally bio-available quinazoline with potential …
Formula:
C24H27Cl3FN5O3
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
558.86
Ref: TM-T2501
5mg | 38.00 € | ||
10mg | 52.00 € | ||
50mg | 74.00 € | ||
1ml*10 (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
SU5214
CAS:186611-04-1
SU5214 is a modulator of tyrosine kinase signal transduction.
Formula:
C16H13NO2
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
251.28
Ref: TM-T3569
5mg | 60.00 € | ||
10mg | 90.00 € | ||
25mg | 177.00 € | ||
50mg | 276.00 € | ||
100mg | 454.00 € | ||
1ml*10 (DMSO) | 66.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor with pIC50 of 4.4/7.1, almost no …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
367.91
Ref: TM-T6145
5mg | 58.00 € | ||
10mg | 93.00 € | ||
25mg | 168.00 € | ||
50mg | 304.00 € | ||
100mg | 455.00 € | ||
1ml*10 (DMSO) | 94.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
WZ8040
CAS:1214265-57-2
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).
Formula:
C24H25ClN6OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
481.01
Ref: TM-T6734
1mg | 47.00 € | ||
5mg | 92.00 € | ||
10mg | 147.00 € | ||
25mg | 241.00 € | ||
50mg | 358.00 € | ||
100mg | 527.00 € | ||
1ml*10 (DMSO) | 94.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
FIIN-3
CAS:1637735-84-2
FIIN-3 is an irreversible inhibitor of FGFR.
Formula:
C34H36Cl2N8O4
Purity:
97.7%
Color and Shape:
Solid
Molecular weight:
691.61
Ref: TM-T3466
1mg | 60.00 € | ||
2mg | 82.00 € | ||
5mg | 118.00 € | ||
10mg | 185.00 € | ||
25mg | 412.00 € | ||
50mg | 612.00 € | ||
100mg | 867.00 € | ||
1ml*10 (DMSO) | 175.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Vandetanib
CAS:443913-73-3
Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 …
Formula:
C22H24BrFN4O2
Purity:
100%
Color and Shape:
White Solid
Molecular weight:
475.35
Ref: TM-T1656
10mg | 49.00 € | ||
25mg | 68.00 € | ||
50mg | 95.00 € | ||
100mg | 171.00 € | ||
200mg | 231.00 € | ||
500mg | 370.00 € | ||
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
KI8751
CAS:228559-41-9
KI8751 is a potent and selective inhibitor of VEGFR2 with IC50 of 0.9 nM.
Formula:
C24H18F3N3O4
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
469.41
Ref: TM-T2446
2mg | 36.00 € | ||
5mg | 52.00 € | ||
10mg | 84.00 € | ||
25mg | 153.00 € | ||
50mg | 289.00 € | ||
100mg | 508.00 € | ||
200mg | 660.00 € | ||
500mg | 1,003.00 € | ||
1ml*10 (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
PP1
CAS:172889-26-8
PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is …
Formula:
C16H19N5
Purity:
99.97%
Color and Shape:
Off-White To Grey Solid
Molecular weight:
281.36
Ref: TM-T6196
1mg | 40.00 € | ||
2mg | 57.00 € | ||
5mg | 92.00 € | ||
10mg | 122.00 € | ||
25mg | 202.00 € | ||
50mg | 283.00 € | ||
100mg | 440.00 € | ||
500mg | 979.00 € | ||
1ml*10 (DMSO) | 98.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AZD3759 hydrochloride
CAS:1626387-81-2
AZD3759 (hydrochloride) is an effective, orally active and central nervous system-penetrant EGFR inhibitor. At Km …
Formula:
C22H24Cl2FN5O3
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
496.36
Ref: TM-T4249
1mg | 43.00 € | ||
2mg | 54.00 € | ||
5mg | 74.00 € | ||
10mg | 95.00 € | ||
25mg | 163.00 € | ||
50mg | 277.00 € | ||
100mg | 456.00 € | ||
500mg | 1,044.00 € | ||
1ml*10 (DMSO) | 84.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Olafertinib
CAS:1660963-42-7
Olafertinib (RX-518) is a novel mutant-selective, irreversible, orally available EGFR inhibitor. It can overcome T790M-mediated …
Formula:
C29H28F2N6O2
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
530.57
Ref: TM-TQ0255
1mg | 48.00 € | ||
5mg | 94.00 € | ||
10mg | 150.00 € | ||
25mg | 299.00 € | ||
50mg | 441.00 € | ||
100mg | 644.00 € | ||
1ml*10 (DMSO) | 109.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Naquotinib
CAS:1448232-80-1
Naquotinib (ASP8273) (ASP8273) is an orally available, mutant-selective and irreversible EGFR inhibitor; (IC50s: 8-33 nM …
Formula:
C30H42N8O3
Purity:
97.49%
Color and Shape:
Solid
Molecular weight:
562.71
Ref: TM-TQ0092
1mg | 51.00 € | ||
2mg | 66.00 € | ||
5mg | 95.00 € | ||
50mg | To inquire | ||
1ml*10 (DMSO) | 131.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tuxobertinib
CAS:2414572-47-5
Tuxobertinib (BDTX-189) is a potent and selective inhibitor of allosteric EGFR and HER2 oncogenic mutations(KDs …
Formula:
C29H29ClN6O4
Purity:
98.86%
Color and Shape:
Solid
Molecular weight:
561.03
Ref: TM-T9072
2mg | 40.00 € | ||
5mg | 59.00 € | ||
10mg | 94.00 € | ||
25mg | 185.00 € | ||
50mg | 346.00 € | ||
100mg | 514.00 € | ||
200mg | 735.00 € | ||
1ml*10 (DMSO) | 73.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
WS6
CAS:1421227-53-3
WS6, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase …
Formula:
C29H31F3N6O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
568.59
Ref: TM-T2106
1mg | 35.00 € | ||
2mg | 51.00 € | ||
5mg | 71.00 € | ||
10mg | 106.00 € | ||
25mg | 206.00 € | ||
50mg | 379.00 € | ||
100mg | 475.00 € | ||
1ml*10 (DMSO) | 90.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Saracatinib
CAS:379231-04-6
Saracatinib (AZD0530) (AZD0530) is an effective Src inhibitor (IC50: 2.7 nM), and effective to Lck, …
Formula:
C27H32ClN5O5
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
542.03
Ref: TM-T6078
10mg | 64.00 € | ||
25mg | 94.00 € | ||
50mg | 143.00 € | ||
100mg | 224.00 € | ||
1ml*10 (DMSO) | 70.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
(±)-Norcantharidin
CAS:29745-04-8
(±)-Norcantharidin (Endothall anhydride) is a synthetic anticancer compound which is a dual inhibitor for c-Met …
Formula:
C8H8O4
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
168.15
Ref: TM-T5656
1g | 530.00 € | ||
5mg | 44.00 € | ||
10mg | 54.00 € | ||
25mg | 77.00 € | ||
50mg | 103.00 € | ||
100mg | 151.00 € | ||
500mg | 357.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Alflutinib
CAS:1869057-83-9
Alflutinib (ASK120067) is an inhibitor of EGFR, and its targets including EGFR activating mutations and …
Formula:
C28H31F3N8O2
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
568.59
Ref: TM-T22254
1mg | 210.00 € | ||
5mg | 428.00 € | ||
10mg | 610.00 € | ||
25mg | 920.00 € | ||
50mg | 1,295.00 € | ||
100mg | 1,755.00 € | ||
1ml*10 (DMSO) | 550.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
HKI-357
CAS:848133-17-5
HKI-357 is an irreversible dual inhibitor of EGFR and ERBB2 (IC50s: 34 nM and 33 …
Formula:
C31H29ClFN5O3
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
574.05
Ref: TM-T11569
1mg | 78.00 € | ||
5mg | 149.00 € | ||
10mg | 222.00 € | ||
25mg | 452.00 € | ||
50mg | 647.00 € | ||
100mg | 920.00 € | ||
1ml*10 (DMSO) | 185.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
TX1-85-1
CAS:1603845-32-4
TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signaling. TX1-85-1 is an irreversible …
Formula:
C32H36N8O3
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
580.68
Ref: TM-T17182
1mg | 69.00 € | ||
5mg | 125.00 € | ||
10mg | 212.00 € | ||
25mg | 362.00 € | ||
50mg | 532.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
PD168393
CAS:194423-15-9
PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, …
Formula:
C17H13BrN4O
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
369.22
Ref: TM-T6932
1mg | 39.00 € | ||
2mg | 49.00 € | ||
5mg | 66.00 € | ||
10mg | 88.00 € | ||
25mg | 151.00 € | ||
50mg | 219.00 € | ||
100mg | 304.00 € | ||
1ml*10 (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
HG-14-10-04
CAS:1356962-34-9
HG-14-10-04 is a potent and specific ALK inhibitor.
Formula:
C29H34ClN7O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
532.08
Ref: TM-T4015
1mg | 59.00 € | ||
2mg | 87.00 € | ||
5mg | 121.00 € | ||
10mg | 194.00 € | ||
25mg | 274.00 € | ||
50mg | 343.00 € | ||
100mg | 493.00 € | ||
1ml*10 (DMSO) | 141.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Mutant EGFR inhibitor
CAS:1421373-62-7
Mutant EGFR inhibitor is a selective and potent Mutated EGFR inhibitor, inhibits L858R activating mutant, …
Formula:
C27H30ClN7O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
520.03
Ref: TM-T2705
1mg | 36.00 € | ||
2mg | 52.00 € | ||
5mg | 79.00 € | ||
10mg | 95.00 € | ||
25mg | 170.00 € | ||
50mg | 258.00 € | ||
100mg | 371.00 € | ||
500mg | To inquire | ||
1ml*10 (DMSO) | 102.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
ZD-4190
CAS:413599-62-9
ZD-4190 is a compound that inhibits both the vascular endothelial growth factor receptor 2 (VEGFR2) …
Formula:
C19H16BrFN6O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
459.27
Ref: TM-T5475
1mg | 123.00 € | ||
2mg | 179.00 € | ||
5mg | 299.00 € | ||
10mg | 449.00 € | ||
25mg | 714.00 € | ||
50mg | 981.00 € | ||
100mg | 1,318.00 € | ||
1ml*10 (DMSO) | 302.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Methyl 2,5-dihydroxycinnamate
CAS:63177-57-1
Methyl 2,5-dihydroxycinnamate is an EGF receptor-associated tyrosine kinases inhibitor.
Formula:
C10H10O4
Purity:
98.98%
Color and Shape:
Crystalline
Molecular weight:
194.18
Ref: TM-T22974
5mg | 64.00 € | ||
10mg | 99.00 € | ||
25mg | 189.00 € | ||
50mg | 351.00 € | ||
100mg | 522.00 € | ||
1ml*10 (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tucatinib
CAS:937263-43-9
Tucatinib (ONT-380) is a potent and selective HER2 inhibitor (IC50: 8 nM).
Formula:
C26H24N8O2
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
480.52
Ref: TM-T2364
1g | 1,110.00 € | ||
2mg | 40.00 € | ||
5mg | 54.00 € | ||
10mg | 83.00 € | ||
25mg | 127.00 € | ||
50mg | 189.00 € | ||
100mg | 343.00 € | ||
500mg | 812.00 € | ||
1ml*10 (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Butein
CAS:487-52-5
Butein (2’,3,4,4’-tetrahydroxy Chalcone), a plant polyphenol, is isolated from Rhus verniciflua. It can inhibit the …
Formula:
C15H12O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
272.25
Ref: TM-T6427
1mg | 42.00 € | ||
2mg | 55.00 € | ||
5mg | 86.00 € | ||
10mg | 104.00 € | ||
25mg | 210.00 € | ||
50mg | 337.00 € | ||
100mg | 540.00 € | ||
1ml*10 (DMSO) | 86.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Osimertinib
CAS:1421373-65-0
Osimertinib (AZD-9291) is an EGFR third-generation inhibitor that inhibits the T790M resistance mutation produced by …
Formula:
C28H33N7O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
499.61
Ref: TM-T2490
1g | 121.00 € | ||
2mg | 30.00 € | ||
5mg | 45.00 € | ||
10mg | 49.00 € | ||
25mg | 59.00 € | ||
50mg | 70.00 € | ||
100mg | 91.00 € | ||
200mg | 91.00 € | ||
500mg | 100.00 € | ||
1ml*10 (DMSO) | 45.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Beta-Hydroxyisovalerylshikonin
CAS:7415-78-3
Beta-Hydroxyisovalerylshikonin is an inhibitor of protein-tyrosine kinases such as v-Src and EGFR, and has been …
Formula:
C21H24O7
Purity:
98.16%
Color and Shape:
Solid
Molecular weight:
388.41
Ref: TM-TN1440
1mg | 134.00 € | ||
5mg | 395.00 € | ||
10mg | 575.00 € | ||
25mg | 894.00 € | ||
50mg | 1,199.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
EGFR-IN-8
CAS:2407957-87-1
EGFR-IN-8, a dual inhibitor targeting both EGFR and c-Met, shows potential as a promising candidate …
Formula:
C32H23ClF3N7O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
662.02
Ref: TM-T11162
1mg | 74.00 € | ||
5mg | 166.00 € | ||
10mg | 266.00 € | ||
25mg | 440.00 € | ||
50mg | 602.00 € | ||
100mg | 825.00 € | ||
1ml*10 (DMSO) | 235.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
PD153035 hydrochloride
CAS:183322-45-4
PD153035 hydrochloride (ZM 252868) is a effective and selective inhibitor of EGFR (Ki: 5.2 pM, …
Formula:
C16H15BrClN3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
396.67
Ref: TM-T1761
5mg | 35.00 € | ||
10mg | 44.00 € | ||
25mg | 81.00 € | ||
50mg | 142.00 € | ||
100mg | 233.00 € | ||
500mg | 530.00 € | ||
1ml*10 (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
PP 3
CAS:5334-30-5
PP 3 is a Negative control for the Src kinase inhibitor PP 2
Formula:
C11H9N5
Purity:
98.92%
Color and Shape:
Whit To Off-White Solid
Molecular weight:
211.22
Ref: TM-T23176
5mg | 56.00 € | ||
10mg | 83.00 € | ||
25mg | 143.00 € | ||
50mg | 203.00 € | ||
100mg | 306.00 € | ||
500mg | 719.00 € | ||
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Poziotinib
CAS:1092364-38-9
Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).
Formula:
C23H21Cl2FN4O3
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
491.34
Ref: TM-T2630
1mg | 35.00 € | ||
5mg | 69.00 € | ||
10mg | 95.00 € | ||
25mg | 183.00 € | ||
50mg | 323.00 € | ||
100mg | 508.00 € | ||
1ml*10 (DMSO) | 73.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
EAI045
CAS:1942114-09-1
EAI045, an allosteric inhibitor, targets towards drug-resistant EGFR mutants but avoids the wild-type receptor.
Formula:
C19H14FN3O3S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
383.4
Ref: TM-T6824
5mg | 43.00 € | ||
10mg | 58.00 € | ||
25mg | 90.00 € | ||
50mg | 121.00 € | ||
100mg | 193.00 € | ||
1ml*10 (DMSO) | 54.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
ONO-7475
CAS:1646839-59-9
ONO-7475 is an inhibitor with high specificity for anexelekto and MER tyrosine kinase
Formula:
C32H26N4O6
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
562.57
Ref: TM-T8327
1mg | 62.00 € | ||
5mg | 134.00 € | ||
10mg | 206.00 € | ||
25mg | 352.00 € | ||
50mg | 520.00 € | ||
100mg | 733.00 € | ||
1ml*10 (DMSO) | 166.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Poziotinib hydrochloride
CAS:1429757-68-5
Poziotinib hydrochloride irreversibly inhibits EGFR (HER1 or ErbB1), including EGFR mutants, HER2, and HER4, thereby …
Formula:
C23H22Cl3FN4O3
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
527.8
Ref: TM-T8758
5mg | 54.00 € | ||
10mg | 81.00 € | ||
25mg | 124.00 € | ||
50mg | 179.00 € | ||
100mg | 267.00 € | ||
200mg | 401.00 € | ||
500mg | 666.00 € | ||
1ml*10 (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AZ7550
CAS:1421373-99-0
AZ7550, an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).
Formula:
C27H31N7O2
Purity:
97.07%
Color and Shape:
Solid
Molecular weight:
485.58
Ref: TM-T13564
1mg | 129.00 € | ||
5mg | 282.00 € | ||
10mg | 417.00 € | ||
25mg | 689.00 € | ||
50mg | 920.00 € | ||
100mg | 1,287.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tyrphostin A9
CAS:10537-47-0
Tyrphostin A9 (SF 6847) is an Agricultural acaricide, now superseded. Tyrphostin A9 is firstly designed …
Formula:
C18H22N2O
Purity:
99.36%
Color and Shape:
Yellow Solid
Molecular weight:
282.38
Ref: TM-T2479
25mg | 54.00 € | ||
50mg | 63.00 € | ||
100mg | 95.00 € | ||
200mg | 169.00 € | ||
500mg | 374.00 € | ||
1ml*10 (DMSO) | 40.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Dacomitinib
CAS:1110813-31-4
Dacomitinib (PF299)(PF299804; PF-00299804) is a highly selective, orally bioavailable small-molecule inhibitor of the HER family …
Formula:
C24H25ClFN5O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
469.94
Ref: TM-T2483
1mg | 38.00 € | ||
2mg | 49.00 € | ||
5mg | 78.00 € | ||
10mg | 124.00 € | ||
25mg | 170.00 € | ||
50mg | 222.00 € | ||
100mg | 348.00 € | ||
200mg | 435.00 € | ||
500mg | 717.00 € | ||
1ml*10 (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AZ-5104
CAS:1421373-98-9
AZ5104 is a potent EGFR inhibitor.
Formula:
C27H31N7O2
Purity:
99.9%
Color and Shape:
Solid Powder
Molecular weight:
485.58
Ref: TM-T2491
5mg | 57.00 € | ||
10mg | 79.00 € | ||
25mg | 126.00 € | ||
50mg | 188.00 € | ||
100mg | 251.00 € | ||
200mg | 314.00 € | ||
1ml*10 (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Afatinib Dimaleate
CAS:850140-73-7
Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the receptor …
Formula:
C32H33ClFN5O11
Purity:
100%
Color and Shape:
Solid
Molecular weight:
718.08
Ref: TM-T1773
1g | 460.00 € | ||
5mg | 40.00 € | ||
10mg | 58.00 € | ||
25mg | 85.00 € | ||
50mg | 105.00 € | ||
100mg | 138.00 € | ||
200mg | 184.00 € | ||
500mg | 308.00 € | ||
1ml*10 (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Epidermal Growth Factor
CAS:62253-63-8
Epidermal Growth Factor binds to epidermal growth factor receptor (EGFR) and stimulates cell growth and …
Formula:
C270H401N73O83S7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
6222
Ref: TM-T8679
1mg | 129.00 € | ||
2mg | 184.00 € | ||
5mg | 278.00 € | ||
10mg | 421.00 € | ||
25mg | 697.00 € | ||
50mg | 976.00 € | ||
100mg | 1,319.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
CP-380736
CAS:179688-29-0
CP-380736 (PF-00520893) is an epidermal growth factor receptor (EGFR) inhibitor. EGFR is a tyrosine kinase …
Formula:
C14H18N2O5
Purity:
99.91%
Color and Shape:
White To Off-White Solid
Molecular weight:
294.3
Ref: TM-T19814
5mg | 54.00 € | ||
10mg | 81.00 € | ||
25mg | 123.00 € | ||
50mg | 180.00 € | ||
100mg | 267.00 € | ||
200mg | 402.00 € | ||
1ml*10 (DMSO) | 70.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
NSC 228155
CAS:113104-25-9
NSC 228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and …
Formula:
C11H6N4O4S
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
290.25
Ref: TM-T6908
5mg | 50.00 € | ||
10mg | 66.00 € | ||
25mg | 123.00 € | ||
50mg | 215.00 € | ||
100mg | 373.00 € | ||
200mg | 484.00 € | ||
1ml*10 (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
(E)-AG 556
CAS:133550-41-1
AG 556 is a selective inhibitor of EGFR and blocks LPS-induced TNF-α production.
Formula:
C20H20N2O3
Purity:
98%
Color and Shape:
Light Yellow Powder
Molecular weight:
336.38
Ref: TM-T21853
5mg | 51.00 € | ||
10mg | 86.00 € | ||
25mg | 157.00 € | ||
50mg | 231.00 € | ||
100mg | 342.00 € | ||
200mg | 507.00 € | ||
500mg | 801.00 € | ||
1ml*10 (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Alflutinib mesylate
CAS:2130958-55-1
Alflutinib mesylate (AST2818 mesylate) ,is an irreversible tyrosine kinase inhibitor that selectively inhibits EGFR mutations, …
Formula:
C29H35F3N8O5S
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
664.7
Ref: TM-T7175
1mg | 77.00 € | ||
5mg | 160.00 € | ||
10mg | 230.00 € | ||
25mg | 388.00 € | ||
50mg | 576.00 € | ||
100mg | 816.00 € | ||
500mg | 1,662.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tyrphostin 23
CAS:118409-57-7
Tyrphostin 23 (AG18) inhibits EGFR with IC50 of 35 μM.
Formula:
C10H6N2O2
Purity:
99.19%
Color and Shape:
Yellow-Tan Solid
Molecular weight:
186.17
Ref: TM-T2063
10mg | 59.00 € | ||
25mg | 120.00 € | ||
50mg | 221.00 € | ||
100mg | 332.00 € | ||
1ml*10 (DMSO) | 43.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
EGFR-IN-12
CAS:879127-07-8
EGFR-IN-12 (EGFR Inhibitor) is a cell permeable and selective inhibitor of EGFR kinase (IC50: 21 …
Formula:
C21H18F3N5O
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
413.4
Ref: TM-T5168
1mg | 81.00 € | ||
5mg | 156.00 € | ||
10mg | 255.00 € | ||
25mg | 511.00 € | ||
50mg | 727.00 € | ||
100mg | 985.00 € | ||
500mg | 1,977.00 € | ||
1ml*10 (DMSO) | 170.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
WHI-P154
CAS:211555-04-3
WHI-P154 (Jak3 inhibitor ii) is a potent JAK3 inhibitor.
Formula:
C16H14BrN3O3
Purity:
99.6%
Color and Shape:
Solid
Molecular weight:
376.2
Ref: TM-T1985
2mg | 46.00 € | ||
5mg | 65.00 € | ||
10mg | 100.00 € | ||
25mg | 178.00 € | ||
50mg | 331.00 € | ||
100mg | 534.00 € | ||
1ml*10 (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Avitinib maleate
CAS:1557268-88-8
Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.
Formula:
C30H30FN7O6
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
603.61
Ref: TM-T3721
5mg | 72.00 € | ||
10mg | 113.00 € | ||
25mg | 205.00 € | ||
50mg | 346.00 € | ||
100mg | 557.00 € | ||
1ml*10 (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Avitinib
CAS:1557267-42-1
Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth …
Formula:
C26H26FN7O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
487.53
Ref: TM-T3024
2mg | 48.00 € | ||
5mg | 73.00 € | ||
10mg | 113.00 € | ||
25mg | 212.00 € | ||
50mg | 347.00 € | ||
100mg | 513.00 € | ||
1ml*10 (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
BI-4020
CAS:2664214-60-0
BI-4020 is a fourth-generation, orally active, and non-covalent inhibitor of EGFR tyrosine kinase. BI-4020 exhibits …
Formula:
C30H38N8O2
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
542.68
Ref: TM-T10534
1mg | 268.00 € | ||
5mg | 650.00 € | ||
10mg | 925.00 € | ||
25mg | 1,388.00 € | ||
50mg | 1,859.00 € | ||
1ml*10 (DMSO) | 790.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
(S)-Sunvozertinib
CAS:2370013-49-1
(S)-Sunvozertinib (DZD9008) is a rationally designed selective, irreversible EGFR/HER2 inhibitor.
Formula:
C29H35ClFN7O3
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
584.08
Ref: TM-T9304
1mg | 62.00 € | ||
5mg | 134.00 € | ||
10mg | 207.00 € | ||
25mg | 415.00 € | ||
50mg | 612.00 € | ||
100mg | 878.00 € | ||
1ml*10 (DMSO) | 172.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
ALK-IN-1
CAS:1197958-12-5
ALK-IN-1 (AP26113) is a potent ALK inhibitor with IC50 of 0.62 nM in a cell-free …
Formula:
C26H34ClN6O2P
Purity:
100%
Color and Shape:
Solid
Molecular weight:
529.01
Ref: TM-T3059
5mg | 48.00 € | ||
10mg | 70.00 € | ||
25mg | 94.00 € | ||
50mg | 142.00 € | ||
100mg | 230.00 € | ||
200mg | 346.00 € | ||
500mg | 561.00 € | ||
1ml*10 (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Zorifertinib
CAS:1626387-80-1
Zorifertinib (AZD3759) is an orally active, effective and central nervous system-penetrant EGFR inhibitor. The IC50 …
Formula:
C22H23ClFN5O3
Purity:
98.32%
Color and Shape:
White To Off-White Solid
Molecular weight:
459.9
Ref: TM-T3659
10mg | 46.00 € | ||
25mg | 67.00 € | ||
50mg | 96.00 € | ||
100mg | 134.00 € | ||
1ml*10 (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
MTX-211
CAS:1952236-05-3
MTX-211, an inhibitor of EGFR and PI3K, is used for the therapy of cancer and …
Formula:
C20H14Cl2FN5O2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
478.33
Ref: TM-T4296
1mg | 93.00 € | ||
2mg | 161.00 € | ||
5mg | 304.00 € | ||
10mg | 462.00 € | ||
25mg | 765.00 € | ||
50mg | 1,054.00 € | ||
100mg | 1,430.00 € | ||
500mg | 2,775.00 € | ||
1ml*10 (DMSO) | 310.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Desmethyl Erlotinib hydrochloride
CAS:183320-51-6
Desmethyl Erlotinib hydrochloride (OSI 420) is an active metabolite of erlotinib which is an orally …
Formula:
C21H21N3O4·HCl
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
415.87
Ref: TM-T6619
1mg | 59.00 € | ||
2mg | 82.00 € | ||
5mg | 113.00 € | ||
10mg | 184.00 € | ||
25mg | 329.00 € | ||
50mg | 495.00 € | ||
100mg | 704.00 € | ||
1ml*10 (DMSO) | 124.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Allitinib tosylate
CAS:1050500-29-2
Allitinib tosylate (AST-1306) is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of …
Formula:
C31H26ClFN4O5S
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
621.08
Ref: TM-T6331
1mg | 55.00 € | ||
5mg | 118.00 € | ||
10mg | 183.00 € | ||
25mg | 346.00 € | ||
50mg | 517.00 € | ||
100mg | 727.00 € | ||
500mg | 1,538.00 € | ||
1ml*10 (DMSO) | 162.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
RG14620
CAS:136831-49-7
RG14620 (Tyrphostin RG14620) is an epidermal growth factor receptor (EGFR) inhibitor.
Formula:
C14H8Cl2N2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
275.13
Ref: TM-T3554
2mg | 35.00 € | ||
5mg | 52.00 € | ||
10mg | 76.00 € | ||
25mg | 134.00 € | ||
50mg | 255.00 € | ||
100mg | 425.00 € | ||
500mg | 920.00 € | ||
1ml*10 (DMSO) | 58.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AG 555
CAS:133550-34-2
AG 555 (Tyrphostin B46) is an EGFR tyrosine kinase inhibitor.
Formula:
C19H18N2O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
322.36
Ref: TM-T4326
5mg | 46.00 € | ||
10mg | 69.00 € | ||
25mg | 109.00 € | ||
50mg | 166.00 € | ||
100mg | 241.00 € | ||
1ml*10 (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
WHI-P258
CAS:21561-09-1
WHI-P258 is a dimethoxyquinazoline inhibitor of JAK3. This compound binds JAK3 weakly and may be …
Formula:
C16H15N3O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
281.31
Ref: TM-T2035
5mg | 55.00 € | ||
10mg | 86.00 € | ||
25mg | 150.00 € | ||
50mg | 233.00 € | ||
100mg | 391.00 € | ||
500mg | 893.00 € | ||
1ml*10 (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
RG13022
CAS:136831-48-6
RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF …
Formula:
C16H14N2O2
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
266.29
Ref: TM-T3545
2mg | 46.00 € | ||
5mg | 60.00 € | ||
10mg | 87.00 € | ||
25mg | 177.00 € | ||
50mg | 298.00 € | ||
100mg | 470.00 € | ||
1ml*10 (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Osimertinib mesylate
CAS:1421373-66-1
Osimertinib mesylate (Mereletinib mesylate) is an irreversible and mutant selective EGFR inhibitor (IC50s: 12/1 nM …
Formula:
C29H37N7O5S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
595.71
Ref: TM-T3634
1g | 149.00 € | ||
5mg | 49.00 € | ||
10mg | 60.00 € | ||
50mg | 86.00 € | ||
100mg | 94.00 € | ||
200mg | 111.00 € | ||
500mg | 129.00 € | ||
1ml*10 (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AG-1478
CAS:153436-53-4
AG-1478 (NSC-693255) (Tyrphostin AG-1478) is a selective EGFR inhibitor.
Formula:
C16H14ClN3O2
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
315.75
Ref: TM-T2047
5mg | 54.00 € | ||
10mg | 71.00 € | ||
25mg | 115.00 € | ||
50mg | 198.00 € | ||
100mg | 273.00 € | ||
200mg | 355.00 € | ||
1ml*10 (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Neratinib
CAS:698387-09-6
Neratinib (HKI-272) (HKI-272) is an orally available, irreversible tyrosine kinase inhibitor for HER2 and EGFR …
Formula:
C30H29ClN6O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
557.04
Ref: TM-T2325
5mg | 35.00 € | ||
10mg | 51.00 € | ||
25mg | 69.00 € | ||
50mg | 92.00 € | ||
100mg | 122.00 € | ||
200mg | 184.00 € | ||
500mg | 307.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
AG-494
CAS:133550-35-3
AG-494 (Tyrphostin B48) is an inhibitor of epidermal growth factor receptor kinase.
Formula:
C16H12N2O3
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
280.28
Ref: TM-T4205
5mg | 65.00 € | ||
10mg | 93.00 € | ||
25mg | 162.00 € | ||
50mg | 244.00 € | ||
100mg | 387.00 € | ||
1ml*10 (DMSO) | 66.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Withanolide A
CAS:32911-62-9
Withanolide A extends the lifespan in human EGFR-driven cancerous Caenorhabditis elegans.
Formula:
C28H38O6
Purity:
98.49%
Color and Shape:
Solid
Molecular weight:
470.6
Ref: TM-TN2309
1mg | 98.00 € | ||
5mg | 233.00 € | ||
10mg | 357.00 € | ||
25mg | 567.00 € | ||
50mg | 841.00 € | ||
1ml*10 (DMSO) | 366.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
G5-7
CAS:939681-36-4
JAK2 inhibitor G5-7 (JAK2 inhibitor G5-7) is an orally active JAK2 inhibitor, selectively inhibits JAK2-mediated …
Formula:
C22H19F2NO3
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
383.39
Ref: TM-T8742
1mg | 82.00 € | ||
5mg | 158.00 € | ||
10mg | 230.00 € | ||
25mg | 424.00 € | ||
50mg | 613.00 € | ||
100mg | 856.00 € | ||
500mg | 1,700.00 € | ||
1ml*10 (DMSO) | 171.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Benidipine hydrochloride
CAS:91599-74-5
Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker …
Formula:
C28H32ClN3O6
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
542.03
Ref: TM-T6227
1g | 130.00 € | ||
50mg | 36.00 € | ||
100mg | 48.00 € | ||
200mg | 61.00 € | ||
500mg | 90.00 € | ||
1ml*10 (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Desmethyl Erlotinib
CAS:183321-86-0
Desmethyl Erlotinib (CP-473420) is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 …
Formula:
C21H21N3O4
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
379.41
Ref: TM-T6328
1mg | 52.00 € | ||
2mg | 75.00 € | ||
5mg | 114.00 € | ||
10mg | 185.00 € | ||
25mg | 324.00 € | ||
50mg | 489.00 € | ||
100mg | 703.00 € | ||
1ml*10 (DMSO) | 125.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Almonertinib
CAS:1899921-05-1
Almonertinib (HS-10296) is an inhibitor of EGFR activation mutation and tolerant mutation of EGFR T790M, …
Formula:
C30H35N7O2
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
525.64
Ref: TM-T5462
1mg | 88.00 € | ||
5mg | 193.00 € | ||
10mg | 305.00 € | ||
25mg | 514.00 € | ||
50mg | 739.00 € | ||
100mg | 1,016.00 € | ||
500mg | 2,070.00 € | ||
1ml*10 (DMSO) | 245.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Dacomitinib hydrate
CAS:1042385-75-0
Dacomitinib hydrate (PF 299804) is a highly selective and second-generation small-molecule inhibitor of the pan-epidermal …
Formula:
C24H27ClFN5O3
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
487.96
Ref: TM-T19965
1mg | 37.00 € | ||
2mg | 52.00 € | ||
5mg | 78.00 € | ||
10mg | 118.00 € | ||
25mg | 167.00 € | ||
50mg | 223.00 € | ||
100mg | 346.00 € | ||
500mg | 810.00 € | ||
1ml*10 (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tesevatinib
CAS:781613-23-8
Tesevatinib (XL-647) is an orally available, multi-target tyrosine kinase inhibitor (IC50s: 0.3, 16, 1.5, 8.7, …
Formula:
C24H25Cl2FN4O2
Purity:
97.89%
Color and Shape:
Solid
Molecular weight:
491.39
Ref: TM-TQ0166
1mg | 106.00 € | ||
2mg | 152.00 € | ||
5mg | 232.00 € | ||
10mg | 450.00 € | ||
25mg | 737.00 € | ||
50mg | 1,003.00 € | ||
1ml*10 (DMSO) | 250.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
EBE-A22
CAS:229476-53-3
EBE-A22 (PD153035 Analog 63) is a derivative of PD 153035 which can inhibit ErbB-1-phosphorylation, whereas …
Formula:
C17H16BrN3O2
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
374.23
Ref: TM-T3558
1mg | 46.00 € | ||
2mg | 59.00 € | ||
5mg | 91.00 € | ||
10mg | 114.00 € | ||
25mg | 223.00 € | ||
50mg | 339.00 € | ||
100mg | 508.00 € | ||
500mg | 1,087.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Gefitinib-based PROTAC 3
CAS:2230821-27-7
Gefitinib-based PROTAC 3, conjugating an EGFR binding element to a VHL ligand via a linker, …
Formula:
C47H57ClFN7O8S
Purity:
98.25%
Color and Shape:
Solid
Molecular weight:
934.51
Ref: TM-T5437
1mg | 49.00 € | ||
2mg | 69.00 € | ||
5mg | 94.00 € | ||
10mg | 171.00 € | ||
25mg | 278.00 € | ||
50mg | 424.00 € | ||
100mg | 611.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
MAZ51
CAS:163655-37-6
MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.
Formula:
C21H18N2O
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
314.38
Ref: TM-T8496
1mg | 40.00 € | ||
2mg | 56.00 € | ||
5mg | 88.00 € | ||
10mg | 126.00 € | ||
25mg | 242.00 € | ||
50mg | 403.00 € | ||
100mg | 599.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Brigatinib
CAS:1197953-54-0
Brigatinib (AP-26113) is a highly potent and selective ALK inhibitor.
Formula:
C29H39ClN7O2P
Purity:
100%
Color and Shape:
Solid
Molecular weight:
584.09
Ref: TM-T3621
1ml | 65.00 € | ||
2mg | 36.00 € | ||
5mg | 50.00 € | ||
10mg | 66.00 € | ||
25mg | 87.00 € | ||
50mg | 112.00 € | ||
100mg | 163.00 € | ||
200mg | 235.00 € | ||
500mg | 400.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
WZ4002
CAS:1213269-23-8
WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50 of 2 nM/8 …
Formula:
C25H27ClN6O3
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
494.97
Ref: TM-T6238
2mg | 35.00 € | ||
5mg | 51.00 € | ||
10mg | 72.00 € | ||
25mg | 115.00 € | ||
50mg | 183.00 € | ||
100mg | 325.00 € | ||
200mg | 478.00 € | ||
1ml*10 (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tyrphostin A1
CAS:2826-26-8
Tyrphostin A1 (Tyrphostin 1) is an inhibitor of EGFR tyrosine kinase .
Formula:
C11H8N2O
Purity:
99.13%
Color and Shape:
Solid
Molecular weight:
184.19
Ref: TM-T7649
5mg | 35.00 € | ||
10mg | 51.00 € | ||
25mg | 96.00 € | ||
50mg | 121.00 € | ||
100mg | 158.00 € | ||
1ml*10 (DMSO) | 40.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Pelitinib
CAS:257933-82-7
Pelitinib (EKB-569) (EKB-569) is an effective irreversible EGFR inhibitor (IC50: 38.5 nM).
Formula:
C24H23ClFN5O2
Purity:
99.86%
Color and Shape:
Off-White Solid
Molecular weight:
467.92
Ref: TM-T2327
5mg | 55.00 € | ||
10mg | 71.00 € | ||
25mg | 109.00 € | ||
50mg | 133.00 € | ||
100mg | 189.00 € | ||
500mg | 455.00 € | ||
1ml*10 (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
WZ-3146
CAS:1214265-56-1
WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750) with IC50 of 2 nM …
Formula:
C24H25ClN6O2
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
464.95
Ref: TM-T6733
1mg | 52.00 € | ||
2mg | 73.00 € | ||
5mg | 95.00 € | ||
10mg | 176.00 € | ||
25mg | 312.00 € | ||
50mg | 499.00 € | ||
100mg | 713.00 € | ||
1ml*10 (DMSO) | 104.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
CZC-8004
CAS:916603-07-1
CZC-8004 (CZC-00008004) is a pan-kinase(ABL kinase) inhibitor and binds a range of tyrosine kinases.
Formula:
C17H16FN5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
309.34
Ref: TM-T7186
1mg | 47.00 € | ||
5mg | 96.00 € | ||
10mg | 142.00 € | ||
25mg | 291.00 € | ||
50mg | 435.00 € | ||
100mg | 625.00 € | ||
1ml*10 (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Lazertinib
CAS:1903008-80-9
Lazertinib (GNS-1480) is an effective, highly mutant-selective and irreversible EGFR-TKI with IC50 values of 1.7 …
Formula:
C30H34N8O3
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
554.64
Ref: TM-T4485
1mg | 48.00 € | ||
2mg | 64.00 € | ||
5mg | 90.00 € | ||
10mg | 147.00 € | ||
25mg | 253.00 € | ||
50mg | 319.00 € | ||
100mg | 462.00 € | ||
500mg | 1,072.00 € | ||
1ml*10 (DMSO) | 108.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
CNX-2006
CAS:1375465-09-0
CNX-2006 is a novel irreversible mutant-selective EGFR inhibitor with IC50 of < 20 nM, with very …
Formula:
C26H27F4N7O2
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
545.53
Ref: TM-T6008
1mg | 40.00 € | ||
2mg | 52.00 € | ||
5mg | 82.00 € | ||
10mg | 123.00 € | ||
25mg | 219.00 € | ||
50mg | 397.00 € | ||
1ml*10 (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Sapitinib
CAS:848942-61-0
Sapitinib (AZD-8931) , a reversible, ATP competitive inhibitor of EGFR(IC50=4 nM), ErbB2(IC50=3 nM) and ErbB3(IC50=4 …
Formula:
C23H25ClFN5O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
473.93
Ref: TM-T6092
2mg | 38.00 € | ||
5mg | 56.00 € | ||
10mg | 85.00 € | ||
25mg | 109.00 € | ||
50mg | 163.00 € | ||
100mg | 235.00 € | ||
1ml*10 (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Olmutinib
CAS:1353550-13-6
Olmutinib (HM61713, BI 1482694) is an orally available small molecule, a mutant-selective inhibitor of epidermal …
Formula:
C26H26N6O2S
Purity:
99.27%
Color and Shape:
Solid
Molecular weight:
486.59
Ref: TM-T6918
2mg | 39.00 € | ||
5mg | 56.00 € | ||
10mg | 87.00 € | ||
25mg | 134.00 € | ||
50mg | 176.00 € | ||
100mg | 276.00 € | ||
200mg | 454.00 € | ||
1ml*10 (DMSO) | 58.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Cyasterone
CAS:17086-76-9
Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, …
Formula:
C29H44O8
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
520.65
Ref: TM-T3870
1mg | 35.00 € | ||
5mg | 69.00 € | ||
10mg | 109.00 € | ||
25mg | 199.00 € | ||
50mg | 298.00 € | ||
100mg | 442.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Leptomycin B
CAS:87081-35-4
Leptomycin B (LMB) is a potent inhibitor of the nuclear export of proteins and is …
Formula:
C33H48O6
Purity:
99.71%
Color and Shape:
White Crystalline Solid
Molecular weight:
540.73
Ref: TM-T15735
1mg | 203.00 € | ||
2mg | 335.00 € | ||
5mg | 611.00 € | ||
10mg | 867.00 € | ||
25mg | 1,296.00 € | ||
50mg | 1,747.00 € | ||
100mg | 2,349.00 € | ||
1ml*10 (DMSO) | 277.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
PD-161570
CAS:192705-80-9
PD-161570 is a potent and ATP-competitive human FGF-1 receptor inhibitor with an IC50 of 39.9 …
Formula:
C26H35Cl2N7O
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
532.51
Ref: TM-T23127
1mg | 95.00 € | ||
2mg | 133.00 € | ||
5mg | 207.00 € | ||
10mg | 306.00 € | ||
25mg | 516.00 € | ||
50mg | 735.00 € | ||
100mg | 997.00 € | ||
1ml*10 (DMSO) | 241.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Almonertinib hydrochloride
CAS:2134096-03-8
Almonertinib hydrochloride (HS-10296 hydrochloride) is a small molecule inhibitor of EGFR-activating mutations and T790M-resistant mutation …
Formula:
C30H36ClN7O2
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
562.1
Ref: TM-T5675
1mg | 90.00 € | ||
5mg | 182.00 € | ||
10mg | 305.00 € | ||
25mg | 525.00 € | ||
50mg | 740.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Genistein
CAS:446-72-0
Genistein (NPI 031L) is an isoflavonoid derived from soy products. It inhibits protein-tyrosine kinase and …
Formula:
C15H10O5
Purity:
99.69%
Color and Shape:
Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether Solid
Molecular weight:
270.24
Ref: TM-T1737
50mg | 45.00 € | ||
100mg | 58.00 € | ||
500mg | 93.00 € | ||
1ml*10 (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Rostafuroxin
CAS:156722-18-8
Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.
Formula:
C23H34O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
374.51
Ref: TM-T2621
2mg | 43.00 € | ||
5mg | 64.00 € | ||
10mg | 105.00 € | ||
25mg | 184.00 € | ||
50mg | 345.00 € | ||
100mg | 510.00 € | ||
1ml*10 (DMSO) | 71.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Tyrphostin AG30
CAS:122520-79-0
Tyrphostin AG30 (AG30) (AG30) is a potent protein tyrosine kinases (PTK) inhibitor.
Formula:
C10H7NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
205.17
Ref: TM-T7101
2mg | 46.00 € | ||
5mg | 69.00 € | ||
10mg | 86.00 € | ||
25mg | 172.00 € | ||
50mg | 301.00 € | ||
100mg | 500.00 € | ||
1ml*10 (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Almonertinib mesylate
CAS:2134096-06-1
Almonertinib mesylate is an irreversible inhibitor of EGFR tyrosine kinase with high selectivity for EGFR-sensitizing …
Formula:
C31H39N7O5S
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
621.75
Ref: TM-T9865
1mg | 90.00 € | ||
5mg | 185.00 € | ||
10mg | 306.00 € | ||
25mg | 518.00 € | ||
50mg | 732.00 € | ||
100mg | 1,044.00 € | ||
500mg | 2,070.00 € | ||
1ml*10 (DMSO) | 270.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
(Rac)-JBJ-04-125-02
CAS:2140807-05-0
(Rac)-JBJ-04-125-02 (JBJ-04-125-02) is effective as a single agent in both in vitro and in vivo …
Formula:
C29H26FN5O3S
Purity:
95.85%
Color and Shape:
Solid
Molecular weight:
543.61
Ref: TM-T8872
1mg | 103.00 € | ||
5mg | 212.00 € | ||
10mg | 346.00 € | ||
25mg | 585.00 € | ||
50mg | 832.00 € | ||
100mg | 1,133.00 € | ||
1ml*10 (DMSO) | 257.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024
Mobocertinib
CAS:1847461-43-1
Mobocertinib (tak788) is a potent inhibitor of epidermal growth factor receptor (EGFR) and an antineoplastic …
Formula:
C32H39N7O4
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
585.7
Ref: TM-T8151
5mg | 35.00 € | ||
10mg | 51.00 € | ||
25mg | 78.00 € | ||
50mg | 118.00 € | ||
100mg | 185.00 € | ||
500mg | 479.00 € | ||
1ml*10 (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 15 Jul 2024