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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • Retagliptin Phosphate

    CAS:
    <p>Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.</p>
    Formula:C19H21F6N4O7P
    Purity:98.70%
    Color and Shape:Solid
    Molecular weight:562.36
  • Fenofibric acid

    CAS:
    <p>Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.</p>
    Formula:C17H15ClO4
    Purity:99.36%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:318.75
  • Dolutegravir intermediate-1

    CAS:
    <p>Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.</p>
    Formula:C13H17NO8
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:315.28
  • Ruzasvir

    CAS:
    <p>Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.</p>
    Formula:C49H55FN10O7S
    Purity:96.87% - 96.88%
    Color and Shape:Solid
    Molecular weight:947.09
  • Sitagliptin

    CAS:
    <p>Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.</p>
    Formula:C16H15F6N5O
    Purity:99.33% - 99.83%
    Color and Shape:Yellow Grease
    Molecular weight:407.31
  • BLT-1

    CAS:
    <p>BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.</p>
    Formula:C12H23N3S
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:241.4
  • Sofosbuvir impurity G

    CAS:
    <p>Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.</p>
    Formula:C22H29FN3O9P
    Purity:98.04%
    Color and Shape:Solid
    Molecular weight:529.45
  • Islatravir

    CAS:
    <p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>
    Formula:C12H12FN5O3
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:293.25
  • BRD-6929

    CAS:
    <p>BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.</p>
    Formula:C19H17N3O2S
    Purity:98.01% - 99.05%
    Color and Shape:Solid
    Molecular weight:351.42
  • ARP-100

    CAS:
    <p>ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).</p>
    Formula:C17H20N2O5S
    Purity:97.18%
    Color and Shape:Solid
    Molecular weight:364.42
  • RAMB4

    CAS:
    <p>RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.</p>
    Formula:C19H13Cl4NO
    Purity:98.89% - 99.38%
    Color and Shape:Solid
    Molecular weight:413.12
  • Probenecid

    CAS:
    <p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>
    Formula:C13H19NO4S
    Purity:98.95% - 99.84%
    Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)
    Molecular weight:285.36
  • ML604440

    CAS:
    <p>ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.</p>
    Formula:C17H24BF3N2O4
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:388.19
  • LSP-249

    CAS:
    <p>LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.</p>
    Formula:C24H22ClN5O
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:431.92
  • Ref: IN-DA0048C1

    1mg
    50.00€
    5mg
    50.00€
    25mg
    155.00€
    50mg
    197.00€
    100mg
    331.00€
    250mg
    531.00€
  • Ref: IN-DA0072SK

    1g
    To inquire
    5mg
    68.00€
    10mg
    90.00€
    25mg
    124.00€
    50mg
    168.00€
    100mg
    229.00€
    250mg
    500.00€
  • Q-VD-OPH

    CAS:
    <p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>
    Formula:C26H25F2N3O6
    Purity:97.8% - 98.95%
    Color and Shape:Solid
    Molecular weight:513.5
  • Denagliptin

    CAS:
    <p>Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study of</p>
    Formula:C20H18F3N3O
    Purity:99.12%
    Color and Shape:Solid
    Molecular weight:373.37
  • Hck-IN-1

    CAS:
    <p>Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; &gt;20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.</p>
    Formula:C16H11ClN6O3S
    Purity:99.07%
    Color and Shape:Solid
    Molecular weight:402.81
  • Sofosbuvir impurity F

    CAS:
    <p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>
    Formula:C34H45FN4O13P2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:798.69