
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(447 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
Show 3 more subcategories
Found 1045 products of "Proteases/Proteasome"
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Retagliptin Phosphate
CAS:<p>Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.</p>Formula:C19H21F6N4O7PPurity:98.70%Color and Shape:SolidMolecular weight:562.36Fenofibric acid
CAS:<p>Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.</p>Formula:C17H15ClO4Purity:99.36%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:318.75Dolutegravir intermediate-1
CAS:<p>Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.</p>Formula:C13H17NO8Purity:99.52%Color and Shape:SolidMolecular weight:315.28Ruzasvir
CAS:<p>Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.</p>Formula:C49H55FN10O7SPurity:96.87% - 96.88%Color and Shape:SolidMolecular weight:947.09Sitagliptin
CAS:<p>Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.</p>Formula:C16H15F6N5OPurity:99.33% - 99.83%Color and Shape:Yellow GreaseMolecular weight:407.31BLT-1
CAS:<p>BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.</p>Formula:C12H23N3SPurity:97.97%Color and Shape:SolidMolecular weight:241.4Sofosbuvir impurity G
CAS:<p>Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.</p>Formula:C22H29FN3O9PPurity:98.04%Color and Shape:SolidMolecular weight:529.45Islatravir
CAS:<p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>Formula:C12H12FN5O3Purity:98.77%Color and Shape:SolidMolecular weight:293.25BRD-6929
CAS:<p>BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.</p>Formula:C19H17N3O2SPurity:98.01% - 99.05%Color and Shape:SolidMolecular weight:351.42ARP-100
CAS:<p>ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).</p>Formula:C17H20N2O5SPurity:97.18%Color and Shape:SolidMolecular weight:364.42RAMB4
CAS:<p>RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.</p>Formula:C19H13Cl4NOPurity:98.89% - 99.38%Color and Shape:SolidMolecular weight:413.12Probenecid
CAS:<p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>Formula:C13H19NO4SPurity:98.95% - 99.84%Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Molecular weight:285.36ML604440
CAS:<p>ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.</p>Formula:C17H24BF3N2O4Purity:97.06%Color and Shape:SolidMolecular weight:388.19LSP-249
CAS:<p>LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.</p>Formula:C24H22ClN5OPurity:99.51%Color and Shape:SolidMolecular weight:431.922-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Formula:C17H30N2O5Purity:98%Color and Shape:SolidMolecular weight:342.4305L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Formula:C26H41N3O5Purity:98%Color and Shape:SolidMolecular weight:475.6208Q-VD-OPH
CAS:<p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>Formula:C26H25F2N3O6Purity:97.8% - 98.95%Color and Shape:SolidMolecular weight:513.5Denagliptin
CAS:<p>Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study of</p>Formula:C20H18F3N3OPurity:99.12%Color and Shape:SolidMolecular weight:373.37Hck-IN-1
CAS:<p>Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; >20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.</p>Formula:C16H11ClN6O3SPurity:99.07%Color and Shape:SolidMolecular weight:402.81Sofosbuvir impurity F
CAS:<p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>Formula:C34H45FN4O13P2Purity:98.05%Color and Shape:SolidMolecular weight:798.69

