
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(36 products)
- Cysteine Protease(110 products)
- DPP-4(23 products)
- Glutaminase(44 products)
- HIV Protease(495 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(88 products)
- Serine Protease(51 products)
- p97(15 products)
Show 3 more subcategories
Found 993 products of "Proteases/Proteasome"
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Saxagliptin
CAS:Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.Formula:C18H25N3O2Purity:99.17% - 99.95%Color and Shape:SolidMolecular weight:315.41Efegatran
CAS:Efegatran is a hematologic agent and platelet aggregation inhibitor.
Formula:C21H32N6O3Color and Shape:SolidMolecular weight:416.52Tenofovir alafenamide hemifumarate
CAS:Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.
Formula:C21H29N6O5PC4H4O4Purity:99.33% - 99.96%Color and Shape:SolidMolecular weight:534.51Enfuvirtide acetate
CAS:Enfuvirtide acetate salt is a linear synthetic peptide made of 36 amino acids. It has an acetylated N-terminus and a carboxamide C-terminus.
Formula:C206H305N51O66Purity:99.34%Color and Shape:SolidMolecular weight:4552S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFormula:C13H16O3SPurity:97.33%Color and Shape:SolidMolecular weight:252.33Ref: TM-T4282
1mg88.00€5mg210.00€10mg338.00€25mg625.00€50mg938.00€100mg1,264.00€1mL*10mM (DMSO)188.00€Bortezomib-pinanediol
CAS:Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.Formula:C29H39BN4O4Purity:97.5%Color and Shape:Yellow SolidMolecular weight:518.46TAPI-1 trifluoroacetate (163847-77-6(free base))
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.Formula:C28H38F3N5O7Purity:98.06%Color and Shape:SolidMolecular weight:613.62HCV-IN-31
CAS:HCV-IN-31 is a HCV inhibitor with an EC50/EC95 of 15.7 μM.Formula:C12H17FN6O3Purity:99.83%Color and Shape:SolidMolecular weight:312.3Ivachtin
CAS:Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining
Formula:C20H21N3O7SPurity:99.74%Color and Shape:SolidMolecular weight:447.46Batimastat
CAS:Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.Formula:C23H31N3O4S2Purity:98.15% - 99.5%Color and Shape:SolidMolecular weight:477.64Boceprevir
CAS:Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.Formula:C27H45N5O5Purity:95% - 99.16%Color and Shape:SolidMolecular weight:519.68Ref: TM-T4988
1mg34.00€5mg66.00€10mg90.00€25mg137.00€50mg177.00€100mg260.00€200mg358.00€1mL*10mM (DMSO)75.00€Fulacimstat
CAS:Fulacimstat (BAY1142524) (BAY1142524) is a chymase inhibitor, with IC50s of 3, 4 nM for hamster and human chymase enzyme, respectively.Formula:C23H16F3N3O6Purity:99.77%Color and Shape:SolidMolecular weight:487.38Ref: TM-TQ0035
1mg101.00€5mg215.00€10mg313.00€25mg512.00€50mg737.00€100mg973.00€1mL*10mM (DMSO)230.00€Velpatasvir
CAS:Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.Formula:C49H54N8O8Purity:99.17% - 99.83%Color and Shape:SolidMolecular weight:883Ref: TM-T3334
5mg34.00€10mg49.00€25mg79.00€50mg98.00€100mg152.00€200mg219.00€500mg358.00€1mL*10mM (DMSO)54.00€EIDD-1931
CAS:EIDD-1931 (Beta-d-N4-hydroxycytidine) is a ribonucleoside analog with antiviral activity. It inhibits replication of SARS-CoV, MERS-CoV, and SARS-CoV-2.
Formula:C9H13N3O6Purity:99.14% - 99.73%Color and Shape:SolidMolecular weight:259.22Lersivirine
CAS:Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.Formula:C17H18N4O2Purity:98.01%Color and Shape:SolidMolecular weight:310.35T-26c
CAS:T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibitor (IC50: 6.75 pM).Formula:C24H21N3O6SPurity:>99.99%Color and Shape:SolidMolecular weight:479.51Ref: TM-T5361
1mg48.00€2mg64.00€5mg96.00€10mg153.00€25mg250.00€50mg424.00€100mg613.00€1mL*10mM (DMSO)97.00€Grazoprevir
CAS:Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.Formula:C38H50N6O9SPurity:99.36% - >99.99%Color and Shape:SolidMolecular weight:766.9STK16-IN-1
CAS:STK16-IN-1 is an inhibitor of STK16 kinase (IC50: 295 nM).Formula:C17H12FN3OPurity:99.52%Color and Shape:SolidMolecular weight:293.3Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purity:98.75%Color and Shape:SolidMolecular weight:300.837-Amino-4-methylcoumarin-3-acetic acid
CAS:7-Amino-4-methylcoumarin-3-acetic acid (7-Amino-4-methylcoumarin) is more suitable as a substrate for enteropeptidase than GD(4)K-NA.Formula:C12H11NO4Purity:98.38%Color and Shape:SolidMolecular weight:233.22
