
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(36 products)
- Cysteine Protease(110 products)
- DPP-4(24 products)
- Glutaminase(44 products)
- HIV Protease(496 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(87 products)
- Serine Protease(51 products)
- p97(15 products)
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Found 991 products of "Proteases/Proteasome"
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NVP DPP 728 dihydrochloride
CAS:NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.Formula:C15H18N6OColor and Shape:SolidMolecular weight:298.34GLS1 Inhibitor
CAS:GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.Formula:C19H21N7O2SColor and Shape:SolidMolecular weight:411.48Nucleoside-Analog-2
CAS:Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.Formula:C9H11N5O6Purity:98%Color and Shape:SolidMolecular weight:285.21LY 806303
CAS:LY 806303 is a highly selective thrombin inhibitor.Formula:C16H14O5SPurity:98%Color and Shape:SolidMolecular weight:318.34Evogliptin HCl
CAS:Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.Formula:C19H27ClF3N3O3Color and Shape:SolidMolecular weight:437.88PSI-7409 tetrasodium
CAS:PSI-7409 tetrasodium, a sofosbuvir metabolite, inhibits GT 1b, 2a, 3a, 4a NS5B polymerases with IC50s of 1.6, 2.8, 0.7, 2.6 μM.Formula:C10H16FN2Na4O14P3Purity:98%Color and Shape:SolidMolecular weight:592.117Thrombin Inhibitor 2
CAS:Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.Formula:C19H16ClF3N6O2Purity:98%Color and Shape:SolidMolecular weight:452.82Alvelestat tosylate
CAS:Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.Formula:C32H30F3N5O7S2Purity:98%Color and Shape:SolidMolecular weight:717.73DPP-4-IN-2
CAS:DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.Formula:C18H18N6OColor and Shape:SolidMolecular weight:334.38Tyrosinase-IN-8
Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity whileFormula:C16H12O4Color and Shape:SolidMolecular weight:268.26SQ 32602
CAS:SQ 32602 is a cathepsin E inhibitor.Formula:C32H52N3O7PColor and Shape:SolidMolecular weight:621.74SJA6017
CAS:SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.Formula:C17H25FN2O4SPurity:98%Color and Shape:SolidMolecular weight:372.45CP-471474
CAS:MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.Formula:C16H17FN2O5SPurity:98%Color and Shape:SolidMolecular weight:368.38Sheng Gelieting
CAS:CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.Formula:C17H16F6N4OColor and Shape:SolidMolecular weight:406.33Tec-IN-21
CAS:Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).Formula:C16H15ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:362.83Cysteine Protease inhibitor hydrochloride
CAS:Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.Formula:C18H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:338.79JNJ-10329670
CAS:JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.Formula:C30H34ClF3N6O3SColor and Shape:SolidMolecular weight:651.14HCV-IN-33
CAS:HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.Formula:C31H36ClN5Color and Shape:SolidMolecular weight:514.1Gü2602
CAS:Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for matureFormula:C16H22N4O3Color and Shape:SolidMolecular weight:318.37Tyrosinase-IN-3
CAS:Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41
