CymitQuimica logo
Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

Show 3 more subcategories

Found 990 products of "Proteases/Proteasome"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Anticancer agent 82

    CAS:
    Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.
    Formula:C19H18Cl2N4O
    Color and Shape:Solid
    Molecular weight:389.28

    Ref: TM-T61746

    100mg
    1,224.00€
  • Tyrosinase-IN-6

    CAS:
    Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.
    Formula:C24H31N3O2
    Color and Shape:Solid
    Molecular weight:393.52

    Ref: TM-T61817

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alicapistat

    CAS:
    Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).
    Formula:C25H27N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.5

    Ref: TM-T14178

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • VEL-0230

    CAS:
    VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.
    Formula:C14H24NNaO5
    Color and Shape:Solid
    Molecular weight:309.33

    Ref: TM-T69793

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PK44 phosphate

    CAS:
    PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).
    Formula:C17H19F5N7O5P
    Color and Shape:Solid
    Molecular weight:527.349

    Ref: TM-T63698

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • BAY8040

    CAS:
    BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.
    Formula:C21H16F3N5O2
    Color and Shape:Solid
    Molecular weight:427.38

    Ref: TM-T30303

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AA10 TG2 inhibitor

    CAS:
    AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65

    Ref: TM-T26494

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DPP-4-IN-1

    CAS:
    DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.
    Formula:C19H19ClN6
    Color and Shape:Solid
    Molecular weight:366.85

    Ref: TM-T61422

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CAY10704

    CAS:
    CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.
    Formula:C18H20Cl2N2
    Color and Shape:Solid
    Molecular weight:335.27

    Ref: TM-T37463

    1mg
    166.00€
    5mg
    705.00€
    10mg
    1,234.00€
  • ASPER-29

    CAS:
    ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.
    Formula:C31H29BrN2O5S
    Color and Shape:Solid
    Molecular weight:621.54

    Ref: TM-T73395

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Elasnin

    CAS:
    Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.
    Formula:C24H40O4
    Color and Shape:Solid
    Molecular weight:392.57

    Ref: TM-T27251

    5mg
    863.00€
  • Tyrosinase-IN-5

    CAS:
    Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.
    Formula:C18H13N3O6
    Color and Shape:Solid
    Molecular weight:367.31

    Ref: TM-T61425

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BRD-8899

    CAS:
    BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].
    Formula:C17H22N4O3S
    Color and Shape:Solid
    Molecular weight:362.45

    Ref: TM-T61361

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HCV-IN-36

    CAS:
    HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.
    Formula:C30H36ClN5
    Color and Shape:Solid
    Molecular weight:502.09

    Ref: TM-T63407

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • GLS1 Inhibitor-3

    CAS:
    GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.
    Formula:C30H32N10O2S
    Color and Shape:Solid
    Molecular weight:596.71

    Ref: TM-T64211

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MMP-2/9-IN-1

    CAS:
    MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.
    Formula:C14H16IN7S
    Color and Shape:Solid
    Molecular weight:441.29

    Ref: TM-T62555

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • (R)-ND-336

    CAS:
    (R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.
    Formula:C16H18ClNO3S2
    Color and Shape:Solid
    Molecular weight:371.89

    Ref: TM-T61491

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • L-873724

    CAS:
    L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.
    Formula:C23H26F3N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.53

    Ref: TM-T16092

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JO146

    CAS:
    JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂,其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM,可应用于细菌感染的抑制。
    Formula:C31H44N3O7P
    Color and Shape:Solid
    Molecular weight:601.67

    Ref: TM-T73532

    25mg
    1,224.00€
    50mg
    1,594.00€
    100mg
    2,250.00€
  • Immunoproteasome inhibitor 1

    CAS:
    Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.
    Formula:C20H26N2O4
    Color and Shape:Solid
    Molecular weight:358.43

    Ref: TM-T61320

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€