PI3K/Akt/mTOR Signaling

Subcategories of "PI3K/Akt/mTOR Signaling"

AMPK

ATM/ATR

DNA-PK

EGFR

gsk-3

MELK

mTOR

PDK

PI3K

S6 Kinase

Show 4 more subcategories

Products of "PI3K/Akt/mTOR Signaling"

100
- 20
- 50
- 200

products per page. 493 products on this category.

Product data	Purity	Price range	Estimated delivery
Olmutinib REF: TM-T8460CAS: 1802181-20-9	97.46%	110.00 € ~ 903.00 €	3 Feb 2022
SF1670 REF: TM-T6667CAS: 345630-40-2	98.54%	62.00 € ~ 900.00 €	3 Feb 2022
A 769662 REF: TM-T2468CAS: 844499-71-4	98.23%	65.00 € ~ 539.00 €	3 Feb 2022
XL147 analogue REF: TM-T2377CAS: 956958-53-5	99.72%	65.00 € ~ 534.00 €	3 Feb 2022
TDZD8 REF: TM-T6187CAS: 327036-89-5	97.13%	45.00 € ~ 219.00 €	3 Feb 2022
LJI308 REF: TM-T6878CAS: 1627709-94-7	98.86%	97.00 € ~ 496.00 €	3 Feb 2022
Palomid 529 REF: TM-T2706CAS: 914913-88-5	98.59%	48.00 € ~ 440.00 €	3 Feb 2022
XL388 REF: TM-T6030CAS: 1251156-08-7	99.53%	68.00 € ~ 1,109.00 €	3 Feb 2022
GSK2292767 REF: TM-T6850CAS: 1254036-66-2	- - -	90.00 € ~ 818.00 €	3 Feb 2022
GSK2636771 REF: TM-T2073CAS: 1372540-25-4	98.00%	65.00 € ~ 540.00 €	3 Feb 2022
PF4989216 REF: TM-T6938CAS: 1276553-09-3	99.73%	68.00 € ~ 762.00 €	3 Feb 2022
Gedatolisib REF: TM-T1970CAS: 1197160-78-3	98.99%	61.00 € ~ 737.00 €	3 Feb 2022
LY2090314 REF: TM-T1755CAS: 603288-22-8	98.00%	71.00 € ~ 714.00 €	3 Feb 2022
NIH12848 REF: TM-T3556CAS: 959551-10-1	100.00%	66.00 € ~ 797.00 €	3 Feb 2022
TBB REF: TM-T2695CAS: 17374-26-4	98.86%	62.00 € ~ 440.00 €	3 Feb 2022
Torin 1 REF: TM-T6045CAS: 1222998-36-8	98.00%	65.00 € ~ 715.00 €	3 Feb 2022
Avitinib REF: TM-T3024CAS: 1557267-42-1	99.87%	66.00 € ~ 630.00 €	3 Feb 2022
NU7026 REF: TM-T2433CAS: 154447-35-5	100.00%	48.00 € ~ 551.00 €	3 Feb 2022
Torin 2 REF: TM-T6100CAS: 1223001-51-1	98.31%	50.00 € ~ 720.00 €	3 Feb 2022
TGX221 REF: TM-T2661CAS: 663619-89-4	100.00%	65.00 € ~ 619.00 €	3 Feb 2022
CH5132799 REF: TM-T2619CAS: 1007207-67-1	99.87%	77.00 € ~ 1,116.00 €	3 Feb 2022
Genistein REF: TM-T1737CAS: 446-72-0	99.69%	36.00 € ~ 99.00 €	3 Feb 2022
Icotinib REF: TM-T6153CAS: 610798-31-7	98.83%	65.00 € ~ 172.00 €	3 Feb 2022
PF4708671 REF: TM-T2002CAS: 1255517-76-0	99.67%	65.00 € ~ 271.00 €	3 Feb 2022
Canertinib dihydrochloride REF: TM-T2501CAS: 289499-45-2	99.23%	46.00 € ~ 220.00 €	3 Feb 2022
AZ5104 REF: TM-T2491CAS: 1421373-98-9	99.59%	65.00 € ~ 482.00 €	3 Feb 2022
AS252424 REF: TM-T6208CAS: 900515-16-4	99.06%	65.00 € ~ 293.00 €	3 Feb 2022
NS1643 REF: TM-T3192CAS: 448895-37-2	98.37%	69.00 € ~ 891.00 €	3 Feb 2022
Serabelisib REF: TM-T3153CAS: 1268454-23-4	99.50%	66.00 € ~ 589.00 €	3 Feb 2022
CL387785 REF: TM-T2245CAS: 194423-06-8	96.68%	59.00 € ~ 715.00 €	3 Feb 2022
BX795 REF: TM-T1830CAS: 702675-74-9	98.00%	66.00 € ~ 563.00 €	3 Feb 2022
WAY600 REF: TM-T6730CAS: 1062159-35-6	98.0%	66.00 € ~ 1,114.00 €	3 Feb 2022
LY3023414 REF: TM-T6883CAS: 1386874-06-1	99.06%	85.00 € ~ 722.00 €	3 Feb 2022
Icotinib Hydrochloride REF: TM-T2307CAS: 1204313-51-8	- - -	75.00 € ~ 255.00 €	3 Feb 2022
WYE125132 REF: TM-T6346CAS: 1144068-46-1	98.0%	62.00 € ~ 1,154.00 €	3 Feb 2022
SB216763 REF: TM-T3077CAS: 280744-09-4	- - -	41.00 € ~ 372.00 €	3 Feb 2022
Cyanoacetohydrazide REF: TM-T0704CAS: 140-87-4	99.90%	65.00 €	3 Feb 2022
SodiumDichloroacetate REF: TM-T3604CAS: 2156-56-1	99.87%	50.00 € ~ 72.00 €	3 Feb 2022
Antrapurol REF: TM-T0800CAS: 117-10-2	99.03%	46.00 € ~ 79.00 €	3 Feb 2022
GNE317 REF: TM-T6845CAS: 1394076-92-6	99.42%	65.00 € ~ 860.00 €	3 Feb 2022
AG18 REF: TM-T2063CAS: 118409-57-7	99.19%	60.00 € ~ 538.00 €	3 Feb 2022
1-Azakenpaullone REF: TM-T6358CAS: 676596-65-9	98.0%	88.00 € ~ 618.00 €	3 Feb 2022
Dacomitinib REF: TM-T2483CAS: 1110813-31-4	98.00%	61.00 € ~ 489.00 €	3 Feb 2022
PIK294 REF: TM-T2297CAS: 900185-02-6	100.00%	66.00 € ~ 483.00 €	3 Feb 2022
Rociletinib REF: TM-T2369CAS: 1374640-70-6	98.00%	65.00 € ~ 219.00 €	3 Feb 2022
Voxtalisib REF: TM-T7014CAS: 934493-76-2	99.36%	65.00 € ~ 430.00 €	3 Feb 2022
Bikinin REF: TM-T1965CAS: 188011-69-0	100.00%	63.00 € ~ 421.00 €	3 Feb 2022
GDC0349 REF: TM-T6510CAS: 1207360-89-1	98.0%	69.00 € ~ 400.00 €	3 Feb 2022
OSI420 REF: TM-T6619CAS: 183320-51-6	98.0%	74.00 € ~ 551.00 €	3 Feb 2022
YM201636 REF: TM-T6110CAS: 371942-69-7	93.28%	63.00 € ~ 1,114.00 €	3 Feb 2022
TG100-115 REF: TM-T2672CAS: 677297-51-7	99.89%	73.00 € ~ 443.00 €	3 Feb 2022
BGT226 REF: TM-T6072CAS: 1245537-68-1	97.75%	68.00 € ~ 1,061.00 €	3 Feb 2022
GDC0326 REF: TM-T3985CAS: 1282514-88-8	100.00%	68.00 € ~ 1,266.00 €	3 Feb 2022
PHA767491 REF: TM-T6206CAS: 845714-00-3	98.0%	66.00 € ~ 800.00 €	3 Feb 2022
LY 303511 REF: TM-T2434CAS: 154447-38-8	- - -	72.00 € ~ 936.00 €	3 Feb 2022
BX912 REF: TM-T1837CAS: 702674-56-4	- - -	89.00 € ~ 735.00 €	3 Feb 2022
Sesamol REF: TM-T3676CAS: 533-31-3	99.90%	36.00 € ~ 72.00 €	3 Feb 2022
PIK293 REF: TM-T3348CAS: 900185-01-5	99.80%	74.00 € ~ 386.00 €	3 Feb 2022
WYE687 REF: TM-T6732CAS: 1062161-90-3	98.0%	73.00 € ~ 809.00 €	3 Feb 2022
EBE-A22 REF: TM-T3558CAS: 229476-53-3	99.69%	94.00 € ~ 1,101.00 €	3 Feb 2022
SNS032 REF: TM-T6049CAS: 345627-80-7	98.27%	65.00 € ~ 239.00 €	3 Feb 2022
AZD1080 REF: TM-T1741CAS: 612487-72-6	98.00%	61.00 € ~ 574.00 €	3 Feb 2022
TWS119 REF: TM-T2166CAS: 601514-19-6	99.13%	48.00 € ~ 458.00 €	3 Feb 2022
BAY1082439 REF: TM-T14511CAS: 1375469-38-7	100.00%	60.00 € ~ 569.00 €	3 Feb 2022
ICA-105574 REF: TM-T9009CAS: 316146-57-3	99.77%	100.00 € ~ 1,079.00 €	3 Feb 2022
EGFR-IN-1 hydrochloride REF: TM-T11157LCAS: 2227455-78-7	98.00%	To inquire	3 Feb 2022
9-ING-41 REF: TM-T14066CAS: 1034895-42-5	99.25%	78.00 € ~ 1,486.00 €	3 Feb 2022
Dactolisib REF: TM-T2235CAS: 915019-65-7	98.00%	50.00 € ~ 119.00 €	3 Feb 2022
PI3K-IN-1 REF: TM-T12462CAS: 1911564-39-0	98.00%	To inquire	3 Feb 2022
A 1070722 REF: TM-T10202CAS: 1384424-80-9	98.00%	To inquire	3 Feb 2022
ZSTK474 REF: TM-T6168CAS: 475110-96-4	98.29%	42.00 € ~ 158.00 €	3 Feb 2022
RG 13022 REF: TM-T3545CAS: 136831-48-6	99.42%	65.00 € ~ 530.00 €	3 Feb 2022
KenPaullone REF: TM-T2247CAS: 142273-20-9	98.99%	65.00 € ~ 633.00 €	3 Feb 2022
Autophinib REF: TM-T4219CAS: 1644443-47-9	99.41%	42.00 € ~ 478.00 €	3 Feb 2022
CHMFL-EGFR-202 REF: TM-T10802CAS: 2089381-40-6	98.00%	To inquire	3 Feb 2022
740 Y-P REF: TM-TQ0003CAS: 1236188-16-1	99.87%	106.00 € ~ 645.00 €	3 Feb 2022
Afatinib free base REF: TM-T21312CAS: 850140-72-6	99.90%	65.00 € ~ 201.00 €	3 Feb 2022
BI-4020 REF: TM-T10534	98.00%	297.00 € ~ 913.00 €	3 Feb 2022
Osimertinib dimesylate REF: TM-T10433CAS: 2070014-82-1	98.00%	65.00 € ~ 189.00 €	3 Feb 2022
PI3K inhibitor 1 REF: TM-T12464CAS: 1172118-03-4	98.00%	To inquire	3 Feb 2022
L-Leucine REF: TM-T3O2749CAS: 61-90-5	99.00%	50.00 € ~ 65.00 €	3 Feb 2022
SKI V REF: TM-T8461CAS: 24418-86-8	99.62%	245.00 € ~ 1,565.00 €	3 Feb 2022
GSK-3 inhibitor 1 REF: TM-T11467CAS: 187325-53-7	98.00%	182.00 € ~ 874.00 €	3 Feb 2022
CHIR 98024 REF: TM-T3074CAS: 556813-39-9	99.04%	65.00 € ~ 653.00 €	3 Feb 2022
Gomisin J REF: TM-T3904CAS: 66280-25-9	99.59%	65.00 € ~ 219.00 €	3 Feb 2022
3BDO REF: TM-T14033CAS: 890405-51-3	98.00%	To inquire	3 Feb 2022
Tideglusib REF: TM-T3067CAS: 865854-05-3	100.00%	65.00 € ~ 398.00 €	3 Feb 2022
LTURM34 REF: TM-T15789CAS: 1879887-96-3	99.91%	98.00 € ~ 992.00 €	3 Feb 2022
XMD-17-51 REF: TM-T22460CAS: 1628614-50-5	98.00%	120.00 € ~ 3,505.00 €	3 Feb 2022
Temsirolimus REF: TM-T2145CAS: 162635-04-3	97.76%	72.00 € ~ 797.00 €	3 Feb 2022
mTOR inhibitor-2 REF: TM-T12124CAS: 2219323-96-1	98.00%	To inquire	3 Feb 2022
Gefitinib-based PROTAC 3 REF: TM-T5437CAS: 2230821-27-7	98.25%	112.00 € ~ 177.00 €	3 Feb 2022
CC115 REF: TM-T3541CAS: 1228013-15-7	86.79%	66.00 € ~ 452.00 €	3 Feb 2022
TGR1202 REF: TM-T4976CAS: 1532533-67-7	99.56%	88.00 € ~ 843.00 €	3 Feb 2022
K-7174 dihydrochloride REF: TM-T11742LCAS: 191089-60-8	98.00%	78.00 € ~ 329.00 €	3 Feb 2022
O-Desmethyl gefitinib REF: TM-T16369CAS: 847949-49-9	98.00%	To inquire	3 Feb 2022
Idelalisib REF: TM-T1894CAS: 870281-82-6	98.00%	46.00 € ~ 157.00 €	3 Feb 2022
PQR-530 REF: TM-T16567CAS: 1927857-61-1	99.78%	144.00 € ~ 1,216.00 €	3 Feb 2022
CGS 15943 REF: TM-T14944CAS: 104615-18-1	98.00%	65.00 € ~ 285.00 €	3 Feb 2022
Buparlisib REF: TM-T1827CAS: 944396-07-0	98.00%	62.00 € ~ 239.00 €	3 Feb 2022

+ info

Olmutinib

CAS:1802181-20-9

Olmutinib is a Novel Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitor

Formula:

C₂₆H₂₆N₆O₂S

Purity:

97.46%

Color and Shape:

Solid

Molecular weight:

486.6

Ref: TM-T8460

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

SF1670

CAS:345630-40-2

SF1670 is a specific PTEN inhibitor with IC50 of 2 μM.

Formula:

C₁₉H₁₇NO₃

Purity:

98.54%

Color and Shape:

solid

Molecular weight:

307.34

Ref: TM-T6667

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

A 769662

CAS:844499-71-4

A-769662 is an effective, reversible AMPK activator(EC50=0.8 μM).

Formula:

C₂₀H₁₂N₂O₃S

Purity:

98.23%

Color and Shape:

solid

Molecular weight:

360.39

Ref: TM-T2468

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

XL147 analogue

CAS:956958-53-5

XL147 analogue is a selective and reversible class I PI3K inhibitor for PI3K//.

Formula:

C₂₁H₁₆N₆O₂S₂

Purity:

99.72%

Color and Shape:

solid

Molecular weight:

448.52

Ref: TM-T2377

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

TDZD8

CAS:327036-89-5

TDZD-8 is an inhibitor of GSK-3, with an IC50 of 2 μM; minimal inhibitory effect …

Formula:

C₁₀H₁₀N₂O₂S

Purity:

97.13%

Color and Shape:

White Solid

Molecular weight:

222.26

Ref: TM-T6187

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

LJI308

CAS:1627709-94-7

LJI308 is a potent, and pan-RSK (p90 ribosomal S6 kinase) inhibitor with IC50 of 6 …

Formula:

C₂₁H₁₈F₂N₂O₂

Purity:

98.86%

Color and Shape:

Solid

Molecular weight:

368.38

Ref: TM-T6878

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Palomid 529

CAS:914913-88-5

Palomid 529 has been used in trials studying the treatment of Age-Related Macular Degeneration.

Formula:

C₂₄H₂₂O₆

Purity:

98.59%

Color and Shape:

solid

Molecular weight:

406.43

Ref: TM-T2706

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

XL388

CAS:1251156-08-7

XL388 is a highly effective, specifc, ATP-competitive inhibitor of mTOR ( IC50: 9.9 nM), 1000-fold …

Formula:

C₂₃H₂₂FN₃O₄S

Purity:

99.53%

Color and Shape:

solid

Molecular weight:

455.5

Ref: TM-T6030

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

GSK2292767

CAS:1254036-66-2

GSK2292767 is a potent and selective PI3K inhibitor.

Formula:

C₂₄H₂₈N₆O₅S

Molecular weight:

512.58

Ref: TM-T6850

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

GSK2636771

CAS:1372540-25-4

GSK2636771, an effective, specific, orally bioavailable, PI3K inhibitor, has been used in cancer, lymphoma, solid …

Formula:

C₂₂H₂₂F₃N₃O₃

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

433.42

Ref: TM-T2073

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PF4989216

CAS:1276553-09-3

PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, …

Formula:

C₁₈H₁₃FN₆OS

Purity:

99.73%

Color and Shape:

solid

Molecular weight:

380.4

Ref: TM-T6938

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Gedatolisib

CAS:1197160-78-3

Gedatolisib is a highly effective dual inhibitor targeting the PI3K/ (IC50: 0.4/5.4 nM)and mTOR (IC50: …

Formula:

C₃₂H₄₁N₉O₄

Purity:

98.99%

Color and Shape:

solid

Molecular weight:

615.73

Ref: TM-T1970

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

LY2090314

CAS:603288-22-8

LY2090314, an effective GSK-3/ inhibitor (IC50: 1.5 nM/0.9 nM), may improve the efficacy of platinum-based …

Formula:

C₂₈H₂₅FN₆O₃

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

512.53

Ref: TM-T1755

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

NIH12848

CAS:959551-10-1

NIH-12848 is a putative inhibitor of phosphatidylinositol 5-phosphate 4-kinase (PI5P4K) with an IC50 of 1 …

Formula:

C₂₀H₁₄F₃N₃S

Purity:

100.00%

Color and Shape:

Solid

Molecular weight:

385.41

Ref: TM-T3556

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

TBB

CAS:17374-26-4

TBB(NSC 231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).

Formula:

C₆HBr₄N₃

Purity:

98.86%

Color and Shape:

Off-White Solid

Molecular weight:

434.71

Ref: TM-T2695

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Torin 1

CAS:1222998-36-8

Torin 1 is an effective inhibitor of mTORC1/2 with (IC50: 2 nM/10 nM); has 1000-fold …

Formula:

C₃₅H₂₈F₃N₅O₂

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

607.62

Ref: TM-T6045

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Avitinib

CAS:1557267-42-1

Avitinib, also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth factor …

Formula:

C₂₆H₂₆FN₇O₂

Purity:

99.87%

Color and Shape:

Solid

Molecular weight:

487.53

Ref: TM-T3024

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

NU7026

CAS:154447-35-5

NU7026 is an effective DNA-PK inhibitor (IC50: 0.23 μM, in cell-free assays), 60-fold selective for …

Formula:

C₁₇H₁₅NO₃

Purity:

100.00%

Color and Shape:

solid

Molecular weight:

281.31

Ref: TM-T2433

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Torin 2

CAS:1223001-51-1

Torin 2(IC50=0.25 nM), a specific and effective mTOR inhibitor, is the 800-fold greater specific activity …

Formula:

C₂₄H₁₅F₃N₄O

Purity:

98.31%

Color and Shape:

solid

Molecular weight:

432.4

Ref: TM-T6100

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

TGX221

CAS:663619-89-4

TGX-221, an effective, specific, and cell membrane permeable inhibitor of the PI3K p110 catalytic subunit, …

Formula:

C₂₁H₂₄N₄O₂

Purity:

100.00%

Color and Shape:

solid

Molecular weight:

364.44

Ref: TM-T2661

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

CH5132799

CAS:1007207-67-1

CH5132799 has been used in trials studying the treatment of Solid Tumors.

Formula:

C₁₅H₁₉N₇O₃S

Purity:

99.87%

Color and Shape:

solid

Molecular weight:

377.42

Ref: TM-T2619

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Genistein

CAS:446-72-0

Genistein is an isoflavonoid derived from soy products. It inhibits protein-tyrosine kinase and topoisomerase-II (DNA …

Formula:

C₁₅H₁₀O₅

Purity:

99.69%

Color and Shape:

Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether Solid

Molecular weight:

270.24

Ref: TM-T1737

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Icotinib

CAS:610798-31-7

Icotinib is an orally available quinazoline-based inhibitor of epidermal growth factor receptor (EGFR), with potential …

Formula:

C₂₂H₂₁N₃O₄

Purity:

98.83%

Color and Shape:

solid

Molecular weight:

391.42

Ref: TM-T6153

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PF4708671

CAS:1255517-76-0

PF-4708671 is a cell-permeable inhibitor of p70 ribosomal S6 kinase (S6K1 isoform) .In cell-free assays, …

Formula:

C₁₉H₂₁F₃N₆

Purity:

99.67%

Color and Shape:

solid

Molecular weight:

390.41

Ref: TM-T2002

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

Canertinib dihydrochloride

CAS:289499-45-2

Canertinib dihydrochloride is the hydrochloride salt of an orally bio-available quinazoline with potential antineoplastic and …

Formula:

C₂₄H₂₇Cl₃FN₅O₃

Purity:

99.23%

Color and Shape:

solid

Molecular weight:

558.86

Ref: TM-T2501

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

AZ5104

CAS:1421373-98-9

AZ5104 is a potent EGFR inhibitor.

Formula:

C₂₇H₃₁N₇O₂

Purity:

99.59%

Color and Shape:

Solid Powder

Molecular weight:

485.58

Ref: TM-T2491

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

AS252424

CAS:900515-16-4

AS-252424 is a potent and selective inhibitor of PI3K with IC50 of 33 nM; >10 …

Formula:

C₁₄H₈FNO₄S

Purity:

99.06%

Color and Shape:

solid

Molecular weight:

305.28

Ref: TM-T6208

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

NS1643

CAS:448895-37-2

NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator with EC50 of …

Formula:

C₁₅H₁₀F₆N₂O₃

Purity:

98.37%

Color and Shape:

solid

Molecular weight:

380.24

Ref: TM-T3192

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Serabelisib

CAS:1268454-23-4

MLN1117 (INK1117) is a p110/// inhibitor (IC50: 15/4.5/1.9/13.39 μM).

Formula:

C₁₉H₁₇N₆O₃

Purity:

99.50%

Color and Shape:

solid

Molecular weight:

363.37

Ref: TM-T3153

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

CL387785

CAS:194423-06-8

CL-387785(EKI785; WAY-EKI 785) is an irreversible inhibitor of EGFRIC50 370+/-120 pM; is able to overcome …

Formula:

C₁₈H₁₃BrN₄O

Purity:

96.68%

Color and Shape:

solid

Molecular weight:

381.23

Ref: TM-T2245

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

BX795

CAS:702675-74-9

BX795 is an effective and selective PDK1 inhibitor (IC50: 6 nM), and its selectivity is …

Formula:

C₂₃H₂₆IN₇O₂S

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

591.47

Ref: TM-T1830

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

WAY600

CAS:1062159-35-6

WAY-600 is a potent, ATP-competitive and selective inhibitor of mTOR with IC50 of 9 nM; …

Formula:

C₂₈H₃₀N₈O

Purity:

98.0%

Molecular weight:

494.59

Ref: TM-T6730

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

LY3023414

CAS:1386874-06-1

LY3023414 is an oral ATP competitive inhibitor of the class I PI3K isoforms, DNA-PK, and …

Formula:

C₂₃H₂₆N₄O₃

Purity:

99.06%

Color and Shape:

Solid

Molecular weight:

406.48

Ref: TM-T6883

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

Icotinib Hydrochloride

CAS:1204313-51-8

Icotinib Hydrochloride is the hydrochloride salt form of icotinib, an orally available quinazoline-based inhibitor of …

Formula:

C₂₂H₂₂ClN₃O₄

Molecular weight:

427.88

Ref: TM-T2307

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

WYE125132

CAS:1144068-46-1

WYE-125132 (WYE-132) is a highly potent, ATP-competitive mTOR inhibitor with IC50 of 0.19 nM; highly …

Formula:

C₂₇H₃₃N₇O₄

Purity:

98.0%

Molecular weight:

519.6

Ref: TM-T6346

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

SB216763

CAS:280744-09-4

SB216763 is an effective and specific GSK-3/ inhibitor (IC50: 34.3 nM).

Formula:

C₁₉H₁₂N₂O₂Cl₂

Color and Shape:

solid

Molecular weight:

371.22

Ref: TM-T3077

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

Cyanoacetohydrazide

CAS:140-87-4

Cyanoacetohydrazide is an anti-TB drug.

Formula:

C₃H₅N₃O

Purity:

99.90%

Color and Shape:

Stout Prisms From Alcohol Slightly Brown Powder

Molecular weight:

99.09

Ref: TM-T0704

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

SodiumDichloroacetate

CAS:2156-56-1

Dichloroacetate, a specific inhibitor of pyruvate dehydrogenase kinase (PDK) with IC50 values of 183 and …

Formula:

C₂HCl₂NaO₂

Purity:

99.87%

Color and Shape:

White Powder

Molecular weight:

150.92

Ref: TM-T3604

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Antrapurol

CAS:117-10-2

Danthron is a natural product, regulates glucose, and lipid metabolism by activating AMPK.

Formula:

C₁₄H₈O₄

Purity:

99.03%

Color and Shape:

Red Or Red-Yellow Needles Or Leaves (From Alcohol) Physical Description Orange Crystalline Powder Almost Odorless And Tasteless

Molecular weight:

240.22

Ref: TM-T0800

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

GNE317

CAS:1394076-92-6

GNE-317, a PI3K/mTOR inhibitor, can pass through the blood-brain barrier (BBB).

Formula:

C₁₉H₂₂N₆O₃S

Purity:

99.42%

Color and Shape:

solid

Molecular weight:

414.48

Ref: TM-T6845

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

AG18

CAS:118409-57-7

AG-18 inhibits EGFR with IC50 of 35 μM.

Formula:

C₁₀H₆N₂O₂

Purity:

99.19%

Color and Shape:

Yellow-Tan Solid

Molecular weight:

186.17

Ref: TM-T2063

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

1-Azakenpaullone

CAS:676596-65-9

1-Azakenpaullone is a potent and selective GSK-3 inhibitor with IC50 of 18 nM, >100-fold selectivity …

Formula:

C₁₅H₁₀BrN₃O

Purity:

98.0%

Color and Shape:

Tan Solid

Molecular weight:

328.16

Ref: TM-T6358

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Dacomitinib

CAS:1110813-31-4

Dacomitinib(PF299804; PF-00299804) is a highly selective, orally bioavailable small-molecule inhibitor of the HER family of …

Formula:

C₂₄H₂₅ClFN₅O₂

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

469.94

Ref: TM-T2483

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PIK294

CAS:900185-02-6

PIK-294 is a excellently specific p110 inhibitor(IC50=10 nM).

Formula:

C₂₈H₂₃N₇O₂

Purity:

100.00%

Color and Shape:

solid

Molecular weight:

489.53

Ref: TM-T2297

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Rociletinib

CAS:1374640-70-6

Rociletinib is an orally available small molecule, irreversible inhibitor of epidermal growth factor receptor (EGFR) …

Formula:

C₂₇H₂₈F₃N₇O₃

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

555.55

Ref: TM-T2369

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Voxtalisib

CAS:934493-76-2

Voxtalisib (SAR245409, XL765) is a dual inhibitor of mTOR/PI3K, mostly for p110 with IC50 of …

Formula:

C₁₃H₁₄N₆O

Purity:

99.36%

Color and Shape:

solid

Molecular weight:

270.29

Ref: TM-T7014

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Bikinin

CAS:188011-69-0

Bikinin, a potent inhibitor of plant GSK-3/Shaggy-like kinase, activates BR signaling downstream of the BR …

Formula:

C₉H₉BrN₂O₃

Purity:

100.00%

Color and Shape:

solid

Molecular weight:

273.08

Ref: TM-T1965

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

GDC0349

CAS:1207360-89-1

GDC-0349 is a potent and selective ATP-competitive inhibitor of mTOR with Ki of 3.8 nM, …

Formula:

C₂₄H₃₂N₆O₃

Purity:

98.0%

Color and Shape:

solid

Molecular weight:

452.55

Ref: TM-T6510

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

OSI420

CAS:183320-51-6

OSI-420 (Desmethyl Erlotinib, CP-473420) is an active metabolite of erlotinib which is an orally active …

Formula:

C₂₁H₂₁N₃O₄·HCl

Purity:

98.0%

Molecular weight:

415.87

Ref: TM-T6619

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

YM201636

CAS:371942-69-7

YM201636 (IC50=33 nM), a specific PIKfyve inhibitor, is less effective to p110 and insensitive to …

Formula:

C₂₅H₂₁N₇O₃

Purity:

93.28%

Color and Shape:

solid

Molecular weight:

467.48

Ref: TM-T6110

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

TG100-115

CAS:677297-51-7

TG100-115 is a PI3K/ inhibitor (IC50: 83/235 nM), with fewer effects on PI3K/.

Formula:

C₁₈H₁₄N₆O₂

Purity:

99.89%

Color and Shape:

solid

Molecular weight:

346.34

Ref: TM-T2672

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

BGT226

CAS:1245537-68-1

BGT226 (NVP-BGT226) is a class I PI3K/mTOR inhibitor for PI3K// (IC50: 4/63/38 nM) .

Formula:

C₂₈H₂₅F₃N₆O₂·C₄H₄O₄

Purity:

97.75%

Color and Shape:

solid

Molecular weight:

650.6

Ref: TM-T6072

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

GDC0326

CAS:1282514-88-8

GDC-0326 is a potent and selective inhibitor of -Isoform of Phosphoinositide 3-Kinase (PI3Kalpha inhibitor).

Formula:

C₁₉H₂₂N₆O₃

Purity:

100.00%

Color and Shape:

Solid

Molecular weight:

382.18

Ref: TM-T3985

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PHA767491

CAS:845714-00-3

PHA-767491 is a potent ATP-competitive dual Cdc7/CDK9 inhibitor with IC50 of 10 nM and 34 …

Formula:

C₁₂H₁₁N₃O

Purity:

98.0%

Color and Shape:

solid

Molecular weight:

213.24

Ref: TM-T6206

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

LY 303511

CAS:154447-38-8

LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.

Formula:

C₁₉H₁₈N₂O₂

Color and Shape:

solid

Molecular weight:

306.36

Ref: TM-T2434

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

BX912

CAS:702674-56-4

BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM). The selectivity of …

Formula:

C₂₀H₂₃BrN₈O

Color and Shape:

solid

Molecular weight:

471.35

Ref: TM-T1837

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Sesamol

CAS:533-31-3

Sesamol could decrease lung inflammation and lipopolysaccharide (LPS)-induced lung injury in rats. Sesamol ameliorates inflammatory …

Formula:

C₇H₆O₃

Purity:

99.90%

Color and Shape:

White To Off-White Crystalline Powder

Molecular weight:

138.12

Ref: TM-T3676

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PIK293

CAS:900185-01-5

PIK-293 is a PI3K inhibitor, for PI3K( IC50=0.24 μM), and less potent for PI3K// .

Formula:

C₂₂H₁₉N₇O

Purity:

99.80%

Color and Shape:

solid

Molecular weight:

397.43

Ref: TM-T3348

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

WYE687

CAS:1062161-90-3

WYE-687 is an ATP-competitive and selective inhibitor of mTOR with IC50 of 7 nM; blocks …

Formula:

C₂₈H₃₂N₈O₃

Purity:

98.0%

Color and Shape:

solid

Molecular weight:

528.61

Ref: TM-T6732

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

EBE-A22

CAS:229476-53-3

EBE-A22 is a derivative of PD 153035 which can inhibit ErbB-1-phosphorylation, whereas EBE-A22 is inactive.

Formula:

C₁₇H₁₆BrN₃O₂

Purity:

99.69%

Color and Shape:

solid

Molecular weight:

374.23

Ref: TM-T3558

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

SNS032

CAS:345627-80-7

SNS-032 is a selective inhibitor of CDK2 (IC50: 48 nM ) and is 10- and …

Formula:

C₁₇H₂₄N₄O₂S₂

Purity:

98.27%

Color and Shape:

solid

Molecular weight:

380.53

Ref: TM-T6049

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

AZD1080

CAS:612487-72-6

AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor.

Formula:

C₁₉H₁₈N₄O₂

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

334.37

Ref: TM-T1741

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

TWS119

CAS:601514-19-6

TWS119 is a GSK-3 inhibitor; capable of inducing neuronal differentiation

Formula:

C₁₈H₁₄N₄O₂

Purity:

99.13%

Color and Shape:

solid

Molecular weight:

318.33

Ref: TM-T2166

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

BAY1082439

CAS:1375469-38-7

BAY1082439 is highly effective in inhibiting Pten-null prostate cancer growth[1][2] and it is an orally …

Formula:

C₂₅H₃₀N₆O₅

Purity:

100.00%

Color and Shape:

Solid

Molecular weight:

494.54

Ref: TM-T14511

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

ICA-105574

CAS:316146-57-3

ICA-105574 is an activator of hERG that binds to the channel to remove inactivation, thus …

Formula:

C₁₉H₁₄N₂O₄

Purity:

99.77%

Molecular weight:

334.33

Ref: TM-T9009

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

EGFR-IN-1 hydrochloride

CAS:2227455-78-7

EGFR-IN-1 hydrochloride displays strong antiproliferative activity against the H1975 cells and the first line mutant …

Formula:

C₂₈H₃₁ClN₆O₄

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

551.04

Ref: TM-T11157L

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

9-ING-41

CAS:1034895-42-5

9-ING-41 is a glycogen synthase kinase-3 inhibitor.

Formula:

C₂₂H₁₃FN₂O₅

Purity:

99.25%

Color and Shape:

solid

Molecular weight:

404.35

Ref: TM-T14066

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Dactolisib

CAS:915019-65-7

Dactolisib is an orally bioavailable inhibitor of PI3K and mTOR (IC50s: 4 nM/5 nM/7 nM/75 …

Formula:

C₃₀H₂₃N₅O

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

469.54

Ref: TM-T2235

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PI3K-IN-1

CAS:1911564-39-0

PI3K-IN-1 is an efficacious PI3K inhibitor (IC50 of 1.7 nM).

Formula:

C₂₂H₂₀F₃N₇O₂

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

471.44

Ref: TM-T12462

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

A 1070722

CAS:1384424-80-9

A 1070722 is a potent and selective GSK-3 inhibitor, with a Ki of 0.6 nM …

Formula:

C₁₇H₁₃F₃N₄O₂

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

362.31

Ref: TM-T10202

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

ZSTK474

CAS:475110-96-4

PI3K Inhibitor ZSTK474 is an orally available, s-triazine derivative, ATP-competitive phosphatidylinositol 3-kinase (PI3K) inhibitor with …

Formula:

C₁₉H₂₁F₂N₇O₂

Purity:

98.29%

Color and Shape:

White Powder

Molecular weight:

417.41

Ref: TM-T6168

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

RG 13022

CAS:136831-48-6

RG13022 is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF receptor (IC50: …

Formula:

C₁₆H₁₄N₂O₂

Purity:

99.42%

Color and Shape:

solid

Molecular weight:

266.29

Ref: TM-T3545

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

KenPaullone

CAS:142273-20-9

Kenpaullone, a potent CDK1, CDK2 and CDK5 inhibitor, as new enhancer for iTreg cell differentiation. …

Formula:

C₁₆H₁₁BrN₂O

Purity:

98.99%

Color and Shape:

Tan Solid

Molecular weight:

327.18

Ref: TM-T2247

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Autophinib

CAS:1644443-47-9

Autophinib is a potent autophagy inhibitor with a novel chemotype with IC50 values of 90 …

Formula:

C₁₄H₁₁ClN₆O₃

Purity:

99.41%

Color and Shape:

Solid

Molecular weight:

346.73

Ref: TM-T4219

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

CHMFL-EGFR-202

CAS:2089381-40-6

CHMFL-EGFR-202 is a potent, irreversible inhibitor of EGFR mutant kinase (IC50s: 5.3 nM and 8.3 …

Formula:

C₂₅H₂₄ClN₇O₂

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

489.96

Ref: TM-T10802

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

740 Y-P

CAS:1236188-16-1

740 Y-P is a potent and cell-permeable activator of PI3K.

Formula:

C₁₄₁H₂₂₂N₄₃O₃₉PS₃

Purity:

99.87%

Color and Shape:

Solid

Molecular weight:

3270.72

Ref: TM-TQ0003

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

Afatinib free base

CAS:850140-72-6

Afatinib is an irreversible inhibitor of EGFR family (EGFR-wt, EGFR-L858R, EGFR-L858R/T790M and HER2 with IC50s …

Formula:

C₂₄H₂₅ClFN₅O₃

Purity:

99.90%

Color and Shape:

Off-White Solid

Molecular weight:

485.94

Ref: TM-T21312

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

BI-4020

BI-4020 is a fourth-generation, non-covalent, and orally active inhibitor of EGFR tyrosine kinase.

Formula:

C₃₀H₃₈N₈O₂

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

542.68

Ref: TM-T10534

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

Osimertinib dimesylate

CAS:2070014-82-1

Osimertinib dimesylate is an irreversible and mutant selective EGFR inhibitor (IC50s: 12 and 1 nM …

Formula:

C₃₀H₄₁N₇O₈S₂

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

691.82

Ref: TM-T10433

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

PI3K inhibitor 1

CAS:1172118-03-4

PI3K inhibitor 1 is a inhibitor of PI3K and PI3K.

Formula:

C₃₂H₂₆N₈O₂S

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

586.67

Ref: TM-T12464

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

L-Leucine

CAS:61-90-5

Leucine is one of nine essential amino acids in humans (provided by food), Leucine is …

Formula:

C₆H₁₃NO₂

Purity:

99.00%

Color and Shape:

White Solid Crystalline

Molecular weight:

131.17

Ref: TM-T3O2749

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

SKI V

CAS:24418-86-8

SKI V is a potent and noncompetitive non-lipid sphingosine kinase (SPHK; SK) inhibitor (GST-hSK,IC50 : …

Formula:

C₁₅H₁₀O₄

Purity:

99.62%

Color and Shape:

Solid

Molecular weight:

254.24

Ref: TM-T8461

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

GSK-3 inhibitor 1

CAS:187325-53-7

GSK-3 inhibitor 1 is an inhibitor of GSK-3( IC50 of 4.9 nM) and demonstrates high …

Formula:

C₁₄H₁₀N₂O

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

222.24

Ref: TM-T11467

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

CHIR 98024

CAS:556813-39-9

CHIR 98024 is a potent GSK-3/ inhibitor with IC50 of 0.65 nM/0.58 nM in cell-free …

Formula:

C₂₀H₁₇Cl₂N₉O₂

Purity:

99.04%

Molecular weight:

486.31

Ref: TM-T3074

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Gomisin J

CAS:66280-25-9

Gomisin J is a natural product and have vasodilatory activity. Gomisin J suppresses lipid accumulation …

Formula:

C₂₂H₂₈O₆

Purity:

99.59%

Color and Shape:

solid

Molecular weight:

388.46

Ref: TM-T3904

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

3BDO

CAS:890405-51-3

3BDO is an activator of mTOR. It can also inhibit autophagy..

Formula:

C₁₈H₁₇NO₅

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

327.33

Ref: TM-T14033

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Tideglusib

CAS:865854-05-3

Tideglusib, a non-ATP competitive inhibitor of glycogen synthase kinase 3 (GSK-3), is with anti-inflammatory and …

Formula:

C₁₉H₁₄N₂O₂S

Purity:

100.00%

Color and Shape:

solid

Molecular weight:

334.39

Ref: TM-T3067

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

LTURM34

CAS:1879887-96-3

LTURM34 is an inhibitor of DNA-PK with IC50 of 34 nM. LTURM34 displays effective antiproliferative …

Formula:

C₂₄H₁₈N₂O₃S

Purity:

99.91%

Color and Shape:

Solid

Molecular weight:

414.48

Ref: TM-T15789

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

XMD-17-51

CAS:1628614-50-5

XMD-17-51 is a potent and highly selective NUAK1 inhibitor.

Formula:

C₂₁H₂₄N₈O

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

404.47

Ref: TM-T22460

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Temsirolimus

CAS:162635-04-3

Temsirolimus is a specific mTOR inhibitor ( IC50: 1.76 μM), used in the treatment of …

Formula:

C₅₆H₈₇NO₁₆

Purity:

97.76%

Color and Shape:

White Crystalline Powder

Molecular weight:

1030.29

Ref: TM-T2145

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

mTOR inhibitor-2

CAS:2219323-96-1

mTOR inhibitor-2 is an inhibitor of selective and oral mTOR (IC50 of 7 nM).

Formula:

C₂₃H₂₁N₇O

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

411.46

Ref: TM-T12124

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

Gefitinib-based PROTAC 3

CAS:2230821-27-7

Gefitinib-based PROTAC 3, conjugating an EGFR binding element to a VHL ligand via a linker, …

Formula:

C₄₇H₅₇ClFN₇O₈S

Purity:

98.25%

Color and Shape:

Solid

Molecular weight:

934.51

Ref: TM-T5437

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

CC115

CAS:1228013-15-7

CC-115 is a inhibitor of mTOR/DNA-PK (IC50= 21/ 13 nM).

Formula:

C₁₆H₁₆N₈O

Purity:

86.79%

Color and Shape:

solid

Molecular weight:

336.35

Ref: TM-T3541

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

TGR1202

CAS:1532533-67-7

TGR-1202 is a PI3K inhibitor.

Formula:

C₃₁H₂₄F₃N₅O₃

Purity:

99.56%

Color and Shape:

White Solid

Molecular weight:

571.55

Ref: TM-T4976

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

K-7174 dihydrochloride

CAS:191089-60-8

K-7174 dihydrochloride is a novel cell adhesion inhibitor; inhibits the expression of vascular cell adhesion …

Formula:

C₃₃H₅₀Cl₂N₂O₆

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

641.67

Ref: TM-T11742L

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

+ info

O-Desmethyl gefitinib

CAS:847949-49-9

O-Desmethyl gefitinib inhibits EGFR (IC50: 36 nM in subcellular assays). In human plasma, O-Desmethyl gefitinib …

Formula:

C₂₁H₂₂ClFN₄O₃

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

432.88

Ref: TM-T16369

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Idelalisib

CAS:870281-82-6

Idelalisib is a small molecule inhibitor of the PI3K catalytic subunit p110 (IC50: 2.5 nM). …

Formula:

C₂₂H₁₈FN₇O

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

415.42

Ref: TM-T1894

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

PQR-530

CAS:1927857-61-1

PQR530 is a highly potent dual pan-PI3K/mTORC1/2 inhibitor. PQR530 inhibited protein kinase B (PKB, pSer473) …

Formula:

C₁₈H₂₃F₂N₇O₂

Purity:

99.78%

Color and Shape:

Solid

Molecular weight:

407.42

Ref: TM-T16567

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

CGS 15943

CAS:104615-18-1

CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, …

Formula:

C₁₃H₈ClN₅O

Purity:

98.00%

Color and Shape:

Solid

Molecular weight:

285.69

Ref: TM-T14944

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info

Buparlisib

CAS:944396-07-0

Buparlisib is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: 52/166/116/nM …

Formula:

C₁₈H₂₁F₃N₆O₂

Purity:

98.00%

Color and Shape:

solid

Molecular weight:

410.39

Ref: TM-T1827

Estimated delivery in United States, on Thursday 3 Feb 2022

+ info