Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,715 products)
- Apoptosis(6,164 products)
- Cell Cycle/Checkpoint(4,727 products)
- Chromatin/Epigenetics(2,400 products)
- Cytoskeletal Signaling(1,492 products)
- DNA Damage/DNA Repair(2,928 products)
- Endocrinology/Hormones(3,653 products)
- Enzyme(3,661 products)
- GPCR/G-Protein(8,861 products)
- Immunology and Inflammation(3,801 products)
- Influenza Virus(299 products)
- JAK/STAT signaling(412 products)
- MAPK Signaling(1,239 products)
- Membrane Transporter/Ion Channel(2,979 products)
- Metabolism(10,029 products)
- Microbiology/Virology(7,445 products)
- Neuroscience(10,281 products)
- Other Inhibitors(36,478 products)
- Oxidation-Reduction(44 products)
- PI3K/Akt/mTOR Signaling(1,443 products)
- Proteases/Proteasome(1,695 products)
- Stem Cell and Derivatives(829 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,693 products)
Show 16 more subcategories
Found 66676 products of "Inhibitors"
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MC-VA-PAB-Exatecan
CAS:MC-VA-PAB-Exatecan is an agent-linker conjugate designed for Antibody-Drug Conjugate (ADC) applications, comprising the ADC linker (peptide MC-VA-PAB) and theFormula:C50H54FN7O11Color and Shape:SolidMolecular weight:948.02TG6-129
CAS:<p>TG6-129 is an EP2 receptor antagonist, blocking PGE2 effects, reducing inflammatory markers with 1.6 µM IC50.</p>Formula:C20H18FN5O3S3Purity:99.55%Color and Shape:SolidMolecular weight:491.58(R)-MALT1-IN-7
CAS:(R)-MALT1-IN-7 (compound 142a) is a potent inhibitor of MALT1 protease and has potential for cancer research.Formula:C19H17F3N8O2SColor and Shape:SolidMolecular weight:478.45JH-131e-153
CAS:JH-131e-153, a diacylglycerol (DAG)-lactone, serves as a small molecule activator for the C1 domain of Munc13-1, exhibiting an activation hierarchy of WT>I590≈Formula:C22H38O5Color and Shape:SolidMolecular weight:382.53Dothiepin
CAS:Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFormula:C19H21NSPurity:98%Color and Shape:SolidMolecular weight:295.44Sirt2-IN-5
CAS:Sirt2-IN-5 is a potent inhibitor of SIRT2.Formula:C26H27Cl2N5O3Color and Shape:SolidMolecular weight:528.43Hydroxyphenyllactic acid
CAS:<p>Hydroxyphenyllactic acid is an antifungal metabolite, fungi such as Lactobacillus sp. SK007.</p>Formula:C9H10O4Purity:99.75%Color and Shape:SolidMolecular weight:182.17ZM 260384
CAS:ZM 260384 is a potassium channel opener.Formula:C15H11F4N3O4Color and Shape:SolidMolecular weight:373.26m-Se3
CAS:m-Se3 is a potent, selective inhibitor of c-MYC transcription with demonstrated capability to inhibit tumor growth and exhibit anti-cancer activity [1].Formula:C29H23IN2SePurity:98%Color and Shape:SolidMolecular weight:605.37SARS-CoV-2-IN-62
CAS:<p>SARS-CoV-2-IN-62 (Compound R3b) effectively inhibits SARS-CoV-2 replication in Vero E6 and Calu-3 cells, demonstrating low cytotoxicity and EC50 values of 2.97</p>Formula:C17H21N3O3SePurity:98%Color and Shape:SolidMolecular weight:394.33KRAS G12D modulator-1
CAS:KRAS G12D modulator-1 (compound 6), a potent modulator of KRAS G12D, exhibits IC50 values ranging from 1-10 μM against NEA-G12D, PPI-G12D, and p ERK-AGS, and isFormula:C30H36FN5O4Purity:98%Color and Shape:SolidMolecular weight:549.64Fecosterol
CAS:Fecosterol, a metabolite derived from Saccharomyces cerevisiae, is utilized in phytosterolemia research.Formula:C28H46OColor and Shape:SolidMolecular weight:398.66EAD1 TFA(1644388-26-0 Free base)
CAS:<p>EAD1 HCL is a potent autophagy inhibitor with antiproliferative activity in lung and pancreatic cancer cells. EAD1 HCL also induces apoptosis</p>Formula:C26H28Cl2F3N7O2Purity:97.41%Color and Shape:SolidMolecular weight:598.453-Bromocytisine
CAS:3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).Formula:C11H13BrN2OPurity:99.974%Color and Shape:SolidMolecular weight:269.14eeAChE-IN-2
CAS:eeAChE-IN-2 is a potent inhibitor of eeAChE, exhibiting inhibitory potency with an IC50 of 2 nM.Formula:C37H40N8O5SColor and Shape:SolidMolecular weight:708.83ARN 11391
CAS:<p>ARN 11391 enhances the function of the IP3-gated calcium channel ITPR1 (Inositol 1,4,5-trisphosphate (IP3) receptor type 1), boosting intracellular calcium ion</p>Formula:C22H29N3O3Color and Shape:SolidMolecular weight:383.49AM-156
CAS:AM-156 is a bio-active chemical.Formula:C23H24F3NNaO4Color and Shape:SolidMolecular weight:458.433FR-186054
CAS:FR-186054, a potent ACAT inhibitor with high oral efficacy, outperforms others in vitro regardless of dosage.Formula:C26H27N5OS2Purity:98%Color and Shape:SolidMolecular weight:489.66Proteasome-IN-5
CAS:<p>Proteasome-IN-5, also known as compound 5, acts as a proteasome inhibitor [1].</p>Formula:C20H30BN5O7Purity:98%Color and Shape:SolidMolecular weight:463.29WAY-659873
CAS:<p>WAY-659873 is an active molecule.</p>Formula:C19H17FN2O4S2Color and Shape:SolidMolecular weight:420.48Velagliflozin
CAS:Velagliflozin is an orally available inhibitor of sodium-glucose cotransporter 2.Formula:C23H25NO5Purity:98%Color and Shape:SolidMolecular weight:395.45D1N8
CAS:<p>D1N8 is a potent inhibitor of the SARS-CoV-2 3CL protease, displaying an IC50 value of 0.44 μM and a CC50 value of greater than 20 μM.</p>Formula:C19H14ClN5O3Purity:98%Color and Shape:SolidMolecular weight:395.8DS-1558
CAS:<p>DS-1558 is a potent and orally available GPR40 agonist.DS-1558 was found to have potent glucose lowering effects during an oral glucose tolerance test in ZDF</p>Formula:C21H21F3O4Color and Shape:SolidMolecular weight:394.38RR-RJW100
RR-RJW100: potent LRH-1 & SF-1 agonist; studies metabolic disorders, diabetes, liver disease, IBD.Formula:C28H34OColor and Shape:SolidMolecular weight:386.57ω-3 Arachidonic acid ethyl ester
CAS:Omega-3 Arachidonic Acid ethyl ester, a rare polyunsaturated fatty acid with limited presence in dietary sources, is crucial for infant growth and developmentFormula:C22H36O2Color and Shape:SolidMolecular weight:332.52Vitamin CK3
CAS:Vitamin CK3 is the combination of Vitamin C and vitamin K3 and has been shown to inhibit tumor growth and lung metastasis.Formula:C17H18Na2O11SPurity:98%Color and Shape:SolidMolecular weight:476.36Risevistinel
CAS:Risevistinel (NYX-783), a positive allosteric modulator of the N-methyl-D-aspartate (NMDA) receptor, may mitigate cognitive deficits in neurodegenerativeFormula:C14H23N3O4Purity:98%Color and Shape:SolidMolecular weight:297.35Nesuparib
CAS:Nesuparib, a potent PARP/TNKS1 inhibitor, has antitumor properties and potential for treating various diseases.Formula:C23H24N6OPurity:99.94%Color and Shape:SolidMolecular weight:400.48HD-2a
CAS:HA-2a inhibits the JAK2/STAT3 pathway by downregulating circDcbld2 expression in RAW264.7 cells [1].Formula:C18H18O6Color and Shape:SolidMolecular weight:330.33CCPG
CAS:CCPG is an agonist of excitatory Amino Acid.Formula:C6H9NO4Purity:98%Color and Shape:SolidMolecular weight:159.14JBI-589
CAS:<p>JBI-589 is an isoform-selective, non-covalent inhibitor of PAD4 that diminishes CXCR2 expression and impedes neutrophil chemotaxis.</p>Formula:C29H28FN5OColor and Shape:SolidMolecular weight:481.56WAY-660222
CAS:WAY-660222 is an active molecule.Formula:C19H13FOColor and Shape:SolidMolecular weight:276.3PYZD-4409
CAS:<p>PYZD-4409 is a selective UBA1 inhibitor with an IC50 of 20 μM.</p>Formula:C14H7ClFN3O5Purity:99.71%Color and Shape:SolidMolecular weight:351.67JAK2 JH2 Tracer
CAS:<p>JAK2 JH2 Tracer is a fluorescent probe for the JAK2 JH2 domain (Kd: 0.2 μM).</p>Formula:C38H27F2N7O6SPurity:98%Color and Shape:SolidMolecular weight:747.73Glycolithocholic acid
CAS:Glycolithocholic acid (Lithocholic acid glycine conjugate) is a glycine conjugate of lithocholic acid.Formula:C26H43NO4Purity:99.75% - 99.83%Color and Shape:SolidMolecular weight:433.62CCG-63808
CAS:CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.Formula:C25H15FN4O2SPurity:90%Color and Shape:SolidMolecular weight:454.48WF-210
CAS:<p>WF-210 is an effective activator of procaspase-3 that acts by inducing apoptosis in cancer cells and reducing tumor growth.</p>Formula:C41H38FN7O7SPurity:98%Color and Shape:SolidMolecular weight:791.85Mtb-IN-4
CAS:Mtb-IN-4 (compound 17h) is a non-toxic isoxazole that exhibits anti-Mycobacterium tuberculosis (Mtb) activity, with an IC50 value of 0.70 μM.Formula:C24H18N2O4SColor and Shape:SolidMolecular weight:430.48PI5P4Ks-IN-3
CAS:<p>PI5P4Ks-IN-3 (compound 30) is a covalent inhibitor of PI5P4K, exhibiting inhibition constants (IC50s) of 1.34 μM for PI5P4Kα and 9.9 μM for PI5P4Kβ.</p>Formula:C32H31N7O2Color and Shape:SolidMolecular weight:545.63TNP-351
CAS:<p>Tnp 351 is a novel antifolate drug being assessed for chemotherapy of lung cancer.</p>Formula:C21H24N6O5Color and Shape:SolidMolecular weight:440.45Piperidione
CAS:Piperidione is a cough-suppressing agent [1].Formula:C9H15NO2Color and Shape:SolidMolecular weight:169.22KRAS G12C inhibitor 53
CAS:KRAS G12C inhibitor 53 (Compound 1) is a KRAS G12C inhibitor.Formula:C21H14ClF2N5O2Color and Shape:SolidMolecular weight:441.82NGD 98-2 hydrochloride
corticotropin-releasing factor receptor 1 (CRF1) antagonistFormula:C19H24F3N3O3·HClPurity:98%Color and Shape:SolidMolecular weight:435.87QR-0217
CAS:<p>QR-0217 is a potent inhibitor of both Aβ1-40 and α-synuclein aggregation, exhibiting an IC50 of 7.5 µM for Aβ1-40.</p>Formula:C19H13NO3Color and Shape:SolidMolecular weight:303.31WAY-271999
CAS:<p>WAY-271999 is an active molecule.</p>Formula:C11H7ClN2O3Color and Shape:SolidMolecular weight:250.64Foropafant
CAS:Foropafant (SR27417) is a highly potent and selective platelet-activating factor (PAF) receptor antagonist (Ki: 57 pM).Formula:C28H40N4SPurity:99.67%Color and Shape:SolidMolecular weight:464.71NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Formula:C36H45N5O5SPurity:98%Color and Shape:SolidMolecular weight:659.84Voruciclib hydrochloride
CAS:Voruciclib hydrochloride is an orally active and selective inhibitor of CDK (Ki: 0.626 nM-9.1 nM).Formula:C22H20Cl2F3NO5Purity:98%Color and Shape:SolidMolecular weight:506.3Me-Indoxam
CAS:Me-Indoxam is an inhibitor of sPLA2. It has no effect on arachidonic acid release and platelet activating factor synthesis.Formula:C26H22N2O5Purity:98%Color and Shape:SolidMolecular weight:442.46MN-05
CAS:MN-05 is a neuroprotective and vasodilator for neurodegenerative diseases.Formula:C13H22N2O3Color and Shape:SolidMolecular weight:254.33WAY-327131
CAS:<p>WAY-327131 is an active molecule.</p>Formula:C16H16F3N3O2Color and Shape:SolidMolecular weight:339.31TLR7 agonist 14
CAS:Compound 17b, a TLR7 agonist also known as TLR7 agonist 14, exhibits high potency with an EC50 of 18 nM.Formula:C29H36N6O3Color and Shape:SolidMolecular weight:516.63TCS 46b
CAS:<p>TCS 46b is a NR1A/NR2B NMDA receptor antagonist with oral activity.</p>Formula:C22H23N3OPurity:99.78% - 99.78%Color and Shape:SolidMolecular weight:345.44SJ1461
CAS:SJ1461 is a potent, orally active inhibitor of the BET family, selectively targeting and inhibiting BRD2 (BD1), BRD2 (BD2), BRD4 (BD1), and BRD4 (BD2) withFormula:C21H18ClN7OS2Purity:98%Color and Shape:SolidMolecular weight:484Etiroxate
CAS:<p>Etiroxate (CG-635) is a lipid-lowering agent utilized in hyperlipoproteinemia studies [1].</p>Formula:C18H17I4NO4Color and Shape:SolidMolecular weight:818.95BILR-355
CAS:BILR-355 is a reverse transcriptase inhibitor.Formula:C25H23N5O3Purity:98%Color and Shape:SolidMolecular weight:441.48RPC425 free base
CAS:RPC425 is a noncompetitive inhibitors of the Betaine-γ-Aminobutyric Acid Transporter 1 (BGT1).Formula:C22H27NO2S2Purity:98%Color and Shape:SolidMolecular weight:401.59TASP0376377
CAS:TASP0376377 is a potent antagonist of CRTH2.Formula:C25H16Cl2N2O4Color and Shape:SolidMolecular weight:479.31STING agonist-3
CAS:STING agonist-3: non-nucleotide, selective, anti-tumor with pEC50=7.5, pIC50=9.5, could enhance cancer therapy.Formula:C37H42N12O6Purity:98%Color and Shape:SolidMolecular weight:750.81EP1013
CAS:EP1013 is a broad-spectrum selective inhibitor of Caspase used in the study of type 1 diabetes.Formula:C18H23FN2O6Purity:98%Color and Shape:SolidMolecular weight:382.38K-Ras G12C-IN-1
CAS:K-Ras G12C-IN-1 is a novel and irreversible inhibitor of mutant K-ras G12C.Formula:C22H23Cl2N3O3Color and Shape:SolidMolecular weight:448.34JNJ-28583867
CAS:JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.Formula:C24H32N2O2SColor and Shape:SolidMolecular weight:412.59Tiotropium Bromide hydrate
CAS:Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.Formula:C19H24BrNO5S2Purity:98.44% - 99.41%Color and Shape:SolidMolecular weight:490.43SAR-260301
CAS:<p>SAR-260301 is an orally available and selective inhibitor of PI3Kβ (IC50: 23 nM).</p>Formula:C19H22N4O3Purity:99.74%Color and Shape:SolidMolecular weight:354.4Valecobulin hydrochloride
CAS:<p>Valecobulin hydrochloride (CKD-516 hydrochloride) is the valine prodrug and vasoblocker of S516.Cost-effective and quality-assured.</p>Formula:C26H29ClN6O5SPurity:99.52%Color and Shape:SolidMolecular weight:573.06PLK1/p38γ-IN-1
CAS:<p>PLK1/p38γ-IN-1 (compound 14) serves as a dual inhibitor targeting both PLK1 and p38γ kinases, effectively suppressing the proliferation of human hepatocellular</p>Formula:C21H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:387.9HDAC/BET-IN-1
CAS:<p>HDAC/BET-IN-1 inhibits HDAC1 (IC50: 0.163 μM), HDAC6 (IC50: 0.067 μM), BRD4 (Ki: 0.076 μM), and fights leukemia.</p>Formula:C29H40N4O8SPurity:98%Color and Shape:SolidMolecular weight:604.71Tamgiblimab
CAS:Tamgiblimab (IBI939) is a fully human monoclonal antibody that targets the T-cell immunoreceptor with immunoglobulin and ITIM domains (TIGIT), exhibitingPurity:95% - 95%Color and Shape:LiquidHER2-IN-5
CAS:<p>HER2-IN-5 is an effective inhibitor of orally active HER-2.</p>Formula:C27H33N7O3Color and Shape:SolidMolecular weight:503.6Kv3 modulator 3
CAS:Kv3 modulator 3 is a selective modulator of Kv3.1 and/or Kv3.2 and/or Kv3.3 channels .has analgesic activity for use in the prophylaxis o or treatment of pain.Formula:C19H18N4O3Purity:98%Color and Shape:SolidMolecular weight:350.37TrkA-IN-4
TrkA-IN-4, a potent, orally active and allosteric TrkA inhibitor, is a prodrug of TrkA-IN-3 . TrkA-IN-4 exhibits potent antinociceptive effects [1] .Formula:C27H21F3N4O5Color and Shape:SolidMolecular weight:538.47BRD4 Inhibitor-28
CAS:BRD4 Inhibitor-28 (Compound 18), an orally active molecule, selectively inhibits the bromodomains of BRD4 (BRD4-BD1 and BRD4-BD2) with IC50 values of 15 and 55Formula:C23H21N3O3Purity:98%Color and Shape:SolidMolecular weight:387.43SOS1/KRAS-IN-1
CAS:SOS1/KRAS-IN-1 (Compound 2) serves as an inhibitor of SOS1/KRAS, with potential application in the study of diseases mediated by SOS1/KRAS [1].Formula:C24H26F3N5OPurity:98%Color and Shape:SolidMolecular weight:457.49Lysophosphatidylcholine C19:0
CAS:Lysophosphatidylcholine C19:0 (1-Nonadecanoyl-2-hydroxy-sn-glycero-3-phosphocholine), an acyl chain lipid, enhances IL-1beta secretion [1].Formula:C27H56NO7PColor and Shape:SolidMolecular weight:537.71CID-50930756
CAS:CID-50930756 is a novel HCV NS3 helicase catalyzed ATP hydrolysis stimulator.Formula:C27H18N4O4S3Color and Shape:SolidMolecular weight:558.65PA-082
CAS:PA-082: PPARγ partial agonist, boosts coactivator-1α, reduces triglycerides, enhances insulin signaling.Formula:C33H38N2O5Color and Shape:SolidMolecular weight:542.67CV1808
CAS:CV-1808 is a coronary vasodilator, antihypertensive, and antipsychotic following systemic administration in vivo. CV-1808 is an adenosine A2 receptor agonist.Formula:C16H18N6O4Color and Shape:Off-White To Pale Yellow SolidMolecular weight:358.35HDAC-IN-55
CAS:<p>HDAC-IN-55(8j) is a small-molecule inhibitor that enhances E-cadherin expression and suppresses cancer cell proliferation [1].</p>Formula:C17H17N3O3Purity:98%Color and Shape:SolidMolecular weight:311.34Cholesterylamine
CAS:<p>Cholesterylamine, a cationic lipid, can be incorporated into PLGA to create particles with a charged surface, facilitating its use in drug delivery systems and</p>Formula:C27H47NColor and Shape:SolidMolecular weight:385.67PM-43I
CAS:PM-43I is a potent inhibitor of both STAT5- and STAT6-dependent allergic airway disease in mice.Formula:C38H50F2N3O10PColor and Shape:SolidMolecular weight:777.79JTE-952
CAS:<p>JTE-952: oral, selective Type II CSF-1R inhibitor, IC50 = 13 nM for CSF1R, 261 nM for TrkA, effective in mouse arthritis model.</p>Formula:C30H34N2O6Purity:98%Color and Shape:SolidMolecular weight:518.6GT-2394
CAS:GT-2394 is a histamine H3 receptor agonist.Formula:C14H21N3O2Color and Shape:SolidMolecular weight:263.34Emicerfont
CAS:<p>Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).</p>Formula:C22H24N6O2Purity:98%Color and Shape:SolidMolecular weight:404.46CBP/p300-IN-17
CAS:CBP/p300-IN-17 (compound 7) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.18 μM) and LK2 H3K27 (IC50: 0.69 μM).Formula:C25H28N4O3Color and Shape:SolidMolecular weight:432.51AG-28262 besylate
CAS:AG-28262 besylate is a VEGFR-2 Inhibitorwhich may affect alanine aminotransferase gene expression and enzymatic activity in the liver.Formula:C28H24N4O5S3Color and Shape:SolidMolecular weight:592.7ICMT-IN-42
CAS:<p>ICMT-IN-42 (compound 21) serves as an ICMT inhibitor, demonstrating potency with an IC50 of 0.054 μM [1].</p>Formula:C23H31NOColor and Shape:SolidMolecular weight:337.5CDK/HDAC-IN-3
CAS:<p>CDK/HDAC-IN-3 is an orally active dual inhibitor of HDACs and CDKs, offering potent and selective inhibition of CDK9, CDK12, CDK13, HDAC1, HDAC2, and HDAC3,</p>Formula:C24H18Cl2N6O3Purity:98%Color and Shape:SolidMolecular weight:509.34Propiolactone
CAS:<p>Propiolactone (β-propiolactone; 2-Oxetanone), a chemosterilant, effectively inactivates viruses, rendering them non-infectious.</p>Formula:C3H4O2Purity:98%Color and Shape:SolidMolecular weight:72.06RP-52770
CAS:RP-52770 is a bioactive chemical.Formula:C18H14ClN3OSColor and Shape:SolidMolecular weight:355.84Androgen receptor antagonist 5
CAS:AR antagonist 5 blocks AR (IC50: 6.17 μM), hinders LNCaP cell growth, and has anti-tumor effects in mouse models.Formula:C21H15F4N5O3SColor and Shape:SolidMolecular weight:493.43P11149
CAS:P11149: oral AChE inhibitor, crosses BBB, IC50 1.3 μM, based on Galanthamine, aims Alzheimer's research.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02Antimicrobial photosensitizer-1
CAS:<p>Photosensitizer-1 shows promise in treating infections, effective against S. aureus in mouse wounds.</p>Formula:C19H19BF2I3N3Color and Shape:SolidMolecular weight:718.9Topoisomerase inhibitor 2
CAS:<p>Topoisomerase Inhibitor 2 (18C) is a broad-spectrum bacterial topoisomerase inhibitor effective against multidrug-resistant Gram-negative bacteria [1].</p>Formula:C23H23N5O4Purity:98%Color and Shape:SolidMolecular weight:433.46BACE1-IN-13
CAS:<p>BACE1-IN-13 (Compound 36), an orally active inhibitor of BACE1, exhibits high potency with an IC50 of 2.9 nM and demonstrates greater efficacy in hAβ42 cells (</p>Formula:C20H17FN8O2Purity:98%Color and Shape:SolidMolecular weight:420.4Oxonantenine
CAS:Oxonantenine, an acetylcholinesterase inhibitor, is an oxoaporphine alkaloid from Annona glabra with plant metabolite roles.Formula:C19H13NO5Color and Shape:SolidMolecular weight:335.31OSI-296
CAS:OSI-296: potent cMET/RON inhibitor (IC50: 42/200 nM), effective in tumor models, tolerable, oral, reduces bone tumor growth.Formula:C21H19Cl2FN4O3Purity:98%Color and Shape:SolidMolecular weight:465.3αvβ1 integrin-IN-2
CAS:<p>αvβ1 integrin-IN-2 (compound 32) is a potent inhibitor of ανβ1 and α5β1 integrins, exhibiting IC50 values of 0.9 nM and 33 nM, respectively.</p>Formula:C29H38N4O4Purity:98%Color and Shape:SolidMolecular weight:506.64JAK-IN-4
CAS:JAK-IN-4 is a prodrug of a JAK inhibitor, effective in murine collagen induced arthritis model.Formula:C18H21N4Na2O6PPurity:98%Color and Shape:SolidMolecular weight:466.341IMD-biphenylC
CAS:IMD-biphenylC: New, dual-action imidazoquinolinone dimer; inhibits tumor growth, low inflammation/toxicity.Formula:C35H33N5O3Purity:98%Color and Shape:SolidMolecular weight:571.67MK-386
CAS:MK-386 is a potent and selective inhibitor of human type-1 5alpha-reductase.Formula:C28H49NOColor and Shape:SolidMolecular weight:415.69S07-1066
CAS:S07-1066, an aldo-keto reductase 1C3 (AKR1C3) inhibitor, enhances doxorubicin (DOX) cytotoxicity by selectively inhibiting AKR1C3-mediated reduction of DOX andFormula:C16H11Cl2FO2Purity:98%Color and Shape:SolidMolecular weight:325.16RB 104
CAS:<p>RB 104 is a potent inhibitor of EC 3.4.24.11 that is used to detect nanogram quantities of the enzyme by inhibitor gel electrophoresis.</p>Formula:C21H23IN2O6Color and Shape:SolidMolecular weight:526.32KRAS G12C mutant protein inhibitor A-1
CAS:KRAS G12C mutant protein inhibitor A-1 can be used in studies about Ras.Formula:C31H26ClF4N7O2Color and Shape:SolidMolecular weight:640.03RNA polymerase II-IN-1
CAS:RNA polymerase II-IN-1 (19iv), an amatoxin, inhibits Pol II at 36.66 nM IC50, is more toxic to cancer cells, less to normal cells than α-Amanitin.Formula:C38H53N11O12SPurity:98%Color and Shape:SolidMolecular weight:887.96SU-11752
CAS:SU-11752 selectively inhibits DNA-PK by competing with ATP, enhances ionizing radiation sensitivity without affecting cell cycle or ATM activity.Formula:C26H27N3O5SColor and Shape:SolidMolecular weight:493.57Methyl 12-methyltridecanoate
CAS:<p>Methyl 12-methyltridecanoate ((R)-betaxolol hydrochloride), a biosurfactant derived from Brevibacterium casei LS14, enhances the biocompatibility of</p>Formula:C15H30O2Purity:98%Color and Shape:SolidMolecular weight:242.4Diflumidone sodium
CAS:Diflumidone sodium is a non-steroidal agent with anti-inflammatory activity.Formula:C14H10F2NNaO3SColor and Shape:SolidMolecular weight:333.29PD-1/PD-L1-IN-22
CAS:PD-1/PD-L1-IN-22 is a small molecule inhibitor of PD-1/PD-L1 protein-protein interactions that blocks PD-1/PD-L1 interactions (IC50: 0.732 μM).Formula:C25H26BrClN2O3Color and Shape:SolidMolecular weight:517.84ZG1077
CAS:ZG1077, a covalent KRAS G12C inhibitor, is utilized in non-small cell lung cancer (NSCLC) research.Formula:C33H33F2N5O5SColor and Shape:SolidMolecular weight:649.71ICI 200355
CAS:ICI 200355 is an inhibitor of human neutrophil elastase.Formula:C30H34BrF3N4O7SPurity:98%Color and Shape:SolidMolecular weight:731.58Antiproliferative agent-39
CAS:<p>Antiproliferative Agent-39 (Compound 12) effectively inhibits the proliferation of various cancer cell lines, including A549, SNU-638, Col2, HT1080, and MCF-7,</p>Formula:C22H22N4O3Color and Shape:SolidMolecular weight:390.44Mu opioid receptor antagonist 7
CAS:Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91Tankyrase-IN-5
CAS:Tankyrase-IN-5 (Compound 30f), structurally related to MSC2504877, effectively inhibits tankyrase isoforms TNKS1 and TNKS2, with half-maximal inhibitoryFormula:C17H18N2O2Purity:98%Color and Shape:SolidMolecular weight:282.34TOP1362
CAS:<p>TOP1362: a kinase inhibitor for dry eye and ocular inflammation; targets p38α, Syk, Src, Lck; reduces cytokines and cell infiltration.</p>Formula:C43H51N7O8SColor and Shape:SolidMolecular weight:825.97Amedalin
CAS:Amedalin is a biochemical.Formula:C19H22N2OColor and Shape:SolidMolecular weight:294.398Octahydroaminoacridine succinate
CAS:Octahydroaminoacridine succinate, an acetylcholinesterase inhibitor, is used potentially for the treatment of Alzheimer's disease.Formula:C17H24N2O4Purity:99.91%Color and Shape:SolidMolecular weight:320.38Cremastranone
CAS:Cremastranone: natural homoisoflavanone that hinders human retinal cell proliferation, migration, and tube creation.Formula:C18H18O7Color and Shape:SolidMolecular weight:346.33Edobacomab
CAS:Edobacomab (E5), a monoclonal IgM antibody targeting endotoxin, is utilized in the study of sepsis stemming from Gram-negative bacterial infections [1].Color and Shape:LiquidPD-1/PD-L1-IN-33
CAS:PD-1/PD-L1-IN-33 (Compound N11), a PD-1/PD-L1 inhibitor, effectively impedes the interaction between PD-1 and PD-L1 with an IC50 of 6.3 nM.Formula:C26H27N5OPurity:98%Color and Shape:SolidMolecular weight:425.53Aurora kinase inhibitor-8
CAS:Aurora kinase inhibitor-8 is a highly selective inhibitor of Aurora kinase.Formula:C30H29N7O3Color and Shape:SolidMolecular weight:535.6GSK2256294A
CAS:<p>GSK2256294A (GSK 2256294) is potent, selective inhibitor of recombinant human, rat and mouse sEH with IC50 of 27 pM, 61 pM and 189 pM, respectively.</p>Formula:C21H24F3N7OPurity:99.86% - 99.86%Color and Shape:SolidMolecular weight:447.46TIS108
CAS:<p>TIS108为一种抑制三唑型独脚金内酯生物合成的化合物。它抑制拟南芥的胚胎发生并降低水稻中2′-epi-5-deoxystrigol (epi-5DS)的含量。</p>Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4GSK217
CAS:GSK217 is a potent and selective inhibitor of the bromo and extraterminal domain (BET) second bromodomain (BD2) with high solubility, utilized in oncology andFormula:C20H20N6OPurity:98%Color and Shape:SolidMolecular weight:360.41CBP/p300-IN-15
CAS:CBP/p300-IN-15 inhibits p300 (IC50: 2.5 nM) & CBP (28 nM), affects OVCAR-3 (EC50: 0.865 μM) & A2780 cells (2.71 μM) for ovarian cancer research.Formula:C26H28N4O5Color and Shape:SolidMolecular weight:476.52HBV-IN-17
CAS:<p>HBV-IN-17 (compound 8) is a potent regulator of HBV capsid assembly (EC50: 511 nM).</p>Formula:C17H15F6N5O2Color and Shape:SolidMolecular weight:435.327'-Hydroxy ABA
CAS:<p>7'-Hydroxy ABA (7'-OH ABA), a metabolite of Abscisic acid (ABA), arises from the hydroxylation at the 7'-carbon of ABA.</p>Formula:C15H20O5Color and Shape:SolidMolecular weight:280.32RSV L-protein-IN-4
CAS:<p>RSV L-protein-IN-4 (Compound C) is a noncompetitive inhibitor of the RSV polymerase with an IC50 of 0.88 μM.</p>Formula:C32H35N5O6Purity:98%Color and Shape:SolidMolecular weight:585.65TP0480066
CAS:TP0480066 inhibits topoisomerase II, DNA gyrase (IC50=1.1nM), topo IV (IC50=62.89nM), effective against drug-resistant bacteria and N. gonorrhoeae.Formula:C18H14FN3O5Color and Shape:SolidMolecular weight:371.32GSK1360707
CAS:GSK1360707 is a selective triple reuptake inhibitor (TRI).Formula:C14H17Cl2NOPurity:98%Color and Shape:SolidMolecular weight:286.2Oxophoebine
CAS:Oxophoebine has been identified as a DNA topoisomerase inhibitorFormula:C20H15NO6Purity:99.14%Color and Shape:SolidMolecular weight:365.34MTP
CAS:MTP, a PKM2 inhibitor, promotes apoptosis in cancer cells via caspase-3 activation while also inducing autophagy and enhancing ROS generation.Formula:C29H23F3N4O2Purity:98%Color and Shape:SolidMolecular weight:516.51APX2039
CAS:APX2039 is an orally active fungal Gwt1 enzyme inhibitor and a prodrug of the novel Gwt2096 inhibitor APX1.APX2039 exhibits potent anti-Kryptococcal activityFormula:C20H15FN4O2Purity:98.72% - 99.07%Color and Shape:SolidMolecular weight:362.36WRN inhibitor 1
CAS:WRN Inhibitor 1 (example 7) is an inhibitor of the Werner Syndrome ATP-dependent helicase enzyme (WRN), selectively targeting its helicase domain.Formula:C16H13FN2O4SPurity:98%Color and Shape:SolidMolecular weight:348.35VU6005649
CAS:VU6005649 is an agonist of CNS penetrant mGlu7/8 receptor (EC50s: 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively).Formula:C16H12F5N3OPurity:99.87%Color and Shape:SolidMolecular weight:357.28W-54011
CAS:W-54011: potent non-peptide C5a receptor blocker; binds 125I-C5a (Ki=2.2nM); stops Ca2+ movement, chemotaxis, ROS in neutrophils (IC50=1.6-3.1nM).Formula:C30H37ClN2O2Purity:96.8%Color and Shape:SolidMolecular weight:493.08CP21
CAS:CP21: Iron chelator (3:1 ratio), anti-malarial; inhibits prostaglandin I2, protects rat aorta, HT22 cells. Enhances iron excretion in rabbits.Formula:C8H11NO2Color and Shape:SolidMolecular weight:153.18MoTPS1-IN-1
CAS:MoTPS1-IN-1 is a potent MoTPS1 inhibitor with antifungal anti-inflammatory activity that acts through interaction with Glu396 study ulcerative colitis.Formula:C23H27F3N2O4Purity:99.76%Color and Shape:SoildMolecular weight:452.47Bicyclophenamine
CAS:Bicyclophenamine is a pharmaceutical active ingredient.Formula:C20H27NO2Color and Shape:SolidMolecular weight:313.43β-Lactamase-IN-2
CAS:β-Lactamase-IN-2 is an inhibitor of β-Lactamase with anti-microbial and anti-bacterial effects.Formula:C11H9FO3Purity:99.52%Color and Shape:SolidMolecular weight:208.19ICMT-IN-20
CAS:ICMT-IN-20 (compound 54) serves as an ICMT inhibitor with an IC50 value of 0.682 μM [1].Formula:C21H26N2O3Color and Shape:SolidMolecular weight:354.44DprE1-IN-9
CAS:DprE1-IN-9 (compound B18) is an efficient reversible inhibitor of DprE1, interacting with the enzyme's receptor cavity.Formula:C22H25F3N4O2Color and Shape:SolidMolecular weight:434.45PK68
CAS:PK68 selectively inhibits RIPK1 (IC50=90nM), potentially useful in inflammation and cancer metastasis studies.Formula:C22H24N4O3SPurity:98.09% - 99.64%Color and Shape:SolidMolecular weight:424.52GSK-2485852
CAS:GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.Formula:C27H25BF2N2O6SColor and Shape:SolidMolecular weight:554.37AGN-191129
CAS:AGN-191129 (PGF2α-OMe) is a PGF2α analog with C-1 carboxyl replaced by O-methyl; it lowers eye pressure, but its receptors are unclear.Formula:C21H38O4Color and Shape:SolidMolecular weight:354.523-Hydroxyxanthone
CAS:3-Hydroxyxanthone (3-Hydroxy-xanthen-9-one), a xanthone derivative, exhibits inhibitory effects on NADPH-catalyzed lipid peroxidation in human umbilical veinFormula:C13H8O3Purity:98%Color and Shape:SolidMolecular weight:212.2TMV-IN-2
CAS:TMV-IN-2, a chalcone, inhibits TMV with an EC50 of 89.9 μg/mL, used in infection and tumor studies.Formula:C27H23FO4Color and Shape:SolidMolecular weight:430.47PHD2/HDACs-IN-1
CAS:PHD2/HDACs-IN-1: strong PHD2/HDAC inhibitor (IC50: 1.15-26.60 μM), low-toxicity, protects kidneys from cisplatin-induced AKI.Formula:C18H19N9O4Color and Shape:SolidMolecular weight:425.4FTI 276
CAS:FTI-276 is an inhibitor of protein farnesyltransferase (PFT) (IC50s: 0.9 and 0.5 nM for Plasmodium falciparum and human).Formula:C21H27N3O3S2Purity:98%Color and Shape:SolidMolecular weight:433.59LM-1484
CAS:LM-1484 displays a higher affinity for 3H-LTC4 sites and is an antagonist of CysLT1 receptor.Formula:C28H24N4O3Purity:98%Color and Shape:SolidMolecular weight:464.52H3 receptor antagonist 1
CAS:H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.Formula:C20H28F2N2OPurity:98%Color and Shape:SolidMolecular weight:350.45S-Octylglutathione
CAS:S-Octylglutathione is a competitive inhibitor of glutathione S-transferase (GST) [1].Formula:C18H33N3O6SColor and Shape:SolidMolecular weight:419.543M-011
CAS:<p>3M-011: potent TLR7/8 agonist, cytokine inducer, enhances radiotherapy, fights H3N2, and has anti-tumor effects.</p>Formula:C18H25N5O3SPurity:98%Color and Shape:SolidMolecular weight:391.49MAO-IN-3
CAS:MAO-IN-3 (Compound 5), a reversible and competitive monoamine oxidase (MAO) inhibitor with inhibition constants (K i) of 0.6 μM for MAO A and 0.2 μM for MAO B,Formula:C42H54N4O4Purity:98%Color and Shape:SolidMolecular weight:678.9DPM-1001
CAS:<p>DPM-1001 is an orally bioavailable and non-competitive protein-tyrosine phosphatase (PTP1B) inhibitor (IC50: 100 nM) with the anti-diabetic property.</p>Formula:C35H57N3O3Purity:98%Color and Shape:SolidMolecular weight:567.85TRV-1387
CAS:<p>TRV-1387, a benzofurazan derivative, inhibits the aggregation of tau and amyloid-β [1].</p>Formula:C23H25F3N4O2Color and Shape:SolidMolecular weight:446.47TXNIP-IN-1
CAS:<p>TXNIP-IN-1: TXNIP-TRX complex inhibitor, targets diabetes, cardiovascular, and inflammatory diseases.</p>Formula:C12H12N2O4Purity:99.11%Color and Shape:SolidMolecular weight:248.23CYP17-IN-1
CAS:<p>CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM.</p>Formula:C18H17FN2SPurity:99.14% - 99.83%Color and Shape:SolidMolecular weight:312.4SCH79797 dihydrochloride
CAS:SCH79797 dihydrochloride is a PAR1 antagonist with IC50 70 nM, Ki 35 nM, antiproliferative, and pro-apoptotic properties.Formula:C23H27Cl2N5Purity:99.5%Color and Shape:SolidMolecular weight:444.4MS023 trihydrochloride
CAS:MS023 trihydrochloride (MS023 3HCl) is a PRMT inhibitor with potential anticancer activity against PRMT1, PRMT3, PRMT4, PRMT6, and PRMT8 for cancer research.Formula:C17H28Cl3N3OPurity:99.81%Color and Shape:SolidMolecular weight:396.78ACT-606559
ACT-606559, a metabolite of ACT451840, is a novel chemical compound exhibiting antimalarial properties. It is utilized in malaria research.Formula:C47H52N6O3Color and Shape:SolidMolecular weight:748.95GPR52 receptor modulator 1
CAS:GPR52 receptor modulator 1, a compound delineated as per Procedure 1, is a modulator of the GPR52 receptor, offering research potential in the investigation ofFormula:C19H14F4N4OPurity:98%Color and Shape:SolidMolecular weight:390.33Cbl-b-IN-13
CAS:<p>Cbl-b-IN-13 (Example 520) is a potent Cbl-b inhibitor exhibiting an IC50 of less than 100 nM and is capable of activating T-cells [1].</p>Formula:C29H30F3N5O2Purity:98%Color and Shape:SolidMolecular weight:537.58NIP-101
CAS:NIP-101 is a potent calcium antagonist.Formula:C38H45N4O7PColor and Shape:SolidMolecular weight:700.76Anticancer agent 113
CAS:Anticancer agent 113 possesses anticancer activity [1].Formula:C27H31ClN6O2Color and Shape:SolidMolecular weight:507.03FGFR-IN-11
CAS:<p>FGFR-IN-11 (compound I-5) is an orally active, covalent inhibitor of FGFR, exhibiting IC50 values of 9.9 nM (FGFR1), 3.1 nM (FGFR2), 16 nM (FGFR3), and 1.8 nM (</p>Formula:C28H29ClN4O4Purity:98%Color and Shape:SolidMolecular weight:521.01Cinsebrutinib
CAS:<p>Cinsebrutinib, a Bruton's tyrosine kinase inhibitor, holds potential for research in cancer treatment.</p>Formula:C22H26FN3O2Purity:98%Color and Shape:SolidMolecular weight:383.46PF-06459988
CAS:PF-06459988 is a novel, effective, orally active, irreversible, and selective epidermal growth factor receptor (EGFR) mutant inhibitor.Formula:C19H22ClN7O3Purity:98%Color and Shape:SolidMolecular weight:431.88NVS-SM2
CAS:NVS-SM2 boosts SMN2 splicing, enhances exon 7 inclusion, and raises SMN protein levels orally.Formula:C23H30N6OColor and Shape:SolidMolecular weight:406.52CT1113
CAS:CT1113, a potent inhibitor of both USP28 and USP25, effectively reduces MYC levels in vivo and demonstrates anti-tumor efficacy in a mouse pancreatic cancer CDXFormula:C25H29N5O2SColor and Shape:SolidMolecular weight:463.6p-NH2-CHX-A"-DTPA
CAS:<p>p-NH2-CHX-A"-DTPA is a bifunctional chelating agent [1].</p>Formula:C25H36N4O10Color and Shape:SolidMolecular weight:552.57Fervenulin
CAS:<p>Fervenulin, from Streptomyces sp. CMU-MH021, halts egg hatch (MIC: 30 μg/mL) and kills J2 larvae (MIC: 120 μg/mL) of M. incognita.</p>Formula:C7H7N5O2Purity:99.75%Color and Shape:SolidMolecular weight:193.16Cymipristone
CAS:Cymipristone, a progesterone receptor antagonist, is used potentially for termination of intrauterine pregnancy.Formula:C34H43NO2Purity:98%Color and Shape:SolidMolecular weight:497.71HDAC-IN-50
CAS:HDAC-IN-50, a potent FGFR/HDAC inhibitor (IC50: 0.18-13 nM), induces apoptosis, cell cycle arrest, and shows anti-tumor activity.Formula:C31H41N7O4Color and Shape:SolidMolecular weight:575.7Lanabecestat HCl
CAS:Lanabecestat (AZD3293/LY3314814) is a potent oral BACE1 inhibitor that crosses the BBB and reduces Aβ levels.Formula:C26H29ClN4OColor and Shape:SolidMolecular weight:448.995BTK-IN-17
BTK-IN-17: selective, oral BTK inhibitor, IC50=13.7 nM, reduces p-BTK Y223/p-PLCγ2 Y1217, anti-inflammatory.Formula:C26H23N7O2Color and Shape:SolidMolecular weight:465.51HIV-1 integrase inhibitor 3
CAS:HIV-1 integrase inhibitor 3 is an HIV-1 integrase strand transfer (INST) inhibitor (IC50: 2.7 nM).Formula:C21H22F2N4O4Purity:98%Color and Shape:SolidMolecular weight:432.42Resencatinib
CAS:Resencatinib is a potent tyrosine kinase inhibitor with antineoplastic activity .Formula:C30H29N7O3Color and Shape:SolidMolecular weight:535.6CNDAC
CAS:CNDAC, a nucleoside analog, is a major metabolite of oral drug sapacitabine.Formula:C10H12N4O4Purity:98%Color and Shape:SolidMolecular weight:252.23Methyl α-D-galactopyranoside monohydrate
CAS:<p>Methyl α-D-galactopyranoside monohydrate, an alpha-D-galactoside featuring a methyl substituent at the anomeric position, inhibits both extracellular and</p>Formula:C7H16O7Color and Shape:SolidMolecular weight:212.2Elastase LasB-IN-1
CAS:Elastase LasB-IN-1 (Compound 4b), a potent and selective inhibitor of elastase LasB, exhibits antibacterial activity and has been determined to possess an IC50Formula:C13H17F3NO4PColor and Shape:SolidMolecular weight:339.25CD73-IN-4
CAS:CD73-IN-4 is a potent and selective methylenephosphonic acid CD73 inhibitorFormula:C16H23ClN5O7PPurity:98.61%Color and Shape:SolidMolecular weight:463.81P2X3 antagonist 34
CAS:Potent P2X3 antagonist 34, oral, selective for human, rat, guinea pig receptors; IC50s: 25/92/126 nM; strong anti-tussive, no taste change.Formula:C24H26F2N4O3Purity:98%Color and Shape:SolidMolecular weight:456.48Targeting the bacterial sliding clamp peptide 46
CAS:Peptide 46 is a short peptide that inhibits SC-dependent DNA synthesis by targeting the bacterial sliding clamp (SC).Formula:C47H64N8O11Color and Shape:SolidMolecular weight:917.06ZL0513
CAS:<p>ZL0513: orally active, BRD4 BD1 inhibitor with strong in vivo results and good pharmacokinetics for treating inflammation.</p>Formula:C27H33NO6Color and Shape:SolidMolecular weight:467.55HSP70/SIRT2-IN-2
CAS:<p>HSP70/SIRT2-IN-2 (Compounds 1a), a dual inhibitor of SIRT2 and HSP70, exhibits an IC50 of 45.1±5.0 μM against SIRT2 and demonstrates antitumor activity [1].</p>Formula:C17H13N3S3Purity:98%Color and Shape:SolidMolecular weight:355.5KRM-II-81
CAS:KRM-II-81 is a GABAA receptor ligand with enhanced anxiolytic effects in mice and rats.Formula:C21H13N5OColor and Shape:SolidMolecular weight:351.36HIV-1 inhibitor-10
CAS:HIV-1 inhibitor-10 is a nanomolar HIV-1 maturation inhibitor.Formula:C39H54O6Color and Shape:SolidMolecular weight:618.84HE-S2
CAS:HE-S2, an antibody-drug conjugate, blocks PD-1/PD-L1 and activates TLR7/8, triggering strong antitumor effects.Formula:C38H45N9O6S2Purity:98%Color and Shape:SolidMolecular weight:787.95BF738735
CAS:<p>BF738735 is a selective inhibitor of phosphatidylinositol 4-kinase III beta (PI4KIIIβ, IC50 = 5.7 nM) showing higher activity over α(IC50 = 1.7 μM).</p>Formula:C21H19FN4O3SPurity:90%Color and Shape:SolidMolecular weight:426.46Ganfeborole HCl
CAS:<p>Ganfeborole HCl (GSK3036656 HCl) is a compound with anti-tuberculosis activity and is an inhibitor of Mycobacterium tuberculosis (Mtb) leucyl-tRNA synthetase.</p>Formula:C10H14BCl2NO4Purity:99.88%Color and Shape:SolidMolecular weight:293.94ICMT-IN-26
CAS:ICMT-IN-26 (compound 38) acts as an ICMT inhibitor with an IC50 value of 0.36 μM [1].Formula:C21H26ClNOColor and Shape:SolidMolecular weight:343.89p-fin4
CAS:p-fin4, a peptide, inhibits STEP-GluA2 interaction, Ki 0.4 μM; may enhance cognition, has anxiolytic and antidepressant effects.Formula:C39H53N8O18PColor and Shape:SolidMolecular weight:952.85TLR8 agonist 6
CAS:Compound A, a potent TLR8 agonist, exhibits an EC50 of 0.052 µM and promotes the production of IL-12p40 in human PBMCs with an EC50 of 0.031 µM.Formula:C19H29N7O2Color and Shape:SolidMolecular weight:387.48C 87
CAS:C 87: Small-molecule TNF-α inhibitor, binds TNFα, inhibits cytotoxicity with IC50 of 8.73 μM, blocks signaling.Formula:C24H15ClN6O3SPurity:≥98%Color and Shape:SolidMolecular weight:502.93BTZO-15
CAS:BTZO-15 is a novel ARE activator, ameliorating DSS- and TNBS-induced colitis in rats.Formula:C17H13ClN2O5S2Color and Shape:SolidMolecular weight:424.88PAK1-IN-1
CAS:<p>PAK1-IN-1: PAK1 inhibitor, IC50 9.8 nM, hinders tumor cell migration and invasion dose-dependently.</p>Formula:C26H20ClN5O2Color and Shape:SolidMolecular weight:469.92VER-00158411
CAS:VER-00158411 is a checkpoint kinase 1 and CHK2 inhibitor (IC50: 4.4 nM and 4.5 nM, respectively).Formula:C31H34N6O3Purity:98%Color and Shape:SolidMolecular weight:538.64Stafib-2
CAS:<p>Stafib-2 is a potent and selective inhibitor of the transcription factor STAT5b.Stafib-2 inhibits STAT5b and STAT5a with IC50 values of 82 nM and 1.7 μM,</p>Formula:C28H26N2O12P2Purity:98.48%Color and Shape:SolidMolecular weight:644.46PI3Kδ-IN-17
CAS:PI3Kδ-IN-17 (Compound S5) is a potent PI3K δ inhibitor, exhibiting an IC50 value of 2.82 nM and demonstrates significant efficacy in suppressing theFormula:C23H24F3N7O2Purity:98%Color and Shape:SolidMolecular weight:487.48
