Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,657 products)
- Apoptosis(6,058 products)
- Cell Cycle/Checkpoint(4,657 products)
- Chromatin/Epigenetics(2,354 products)
- Cytoskeletal Signaling(1,460 products)
- DNA Damage/DNA Repair(2,908 products)
- Endocrinology/Hormones(3,601 products)
- Enzyme(3,655 products)
- GPCR/G-Protein(8,703 products)
- Immunology and Inflammation(3,737 products)
- Influenza Virus(298 products)
- JAK/STAT signaling(403 products)
- MAPK Signaling(1,227 products)
- Membrane Transporter/Ion Channel(2,922 products)
- Metabolism(9,881 products)
- Microbiology/Virology(7,303 products)
- Neuroscience(10,209 products)
- Other Inhibitors(36,770 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,669 products)
- Stem Cell and Derivatives(828 products)
- Tyrosine Kinase/Adaptors(2,042 products)
- Ubiquitination(1,681 products)
Show 16 more subcategories
Found 66609 products of "Inhibitors"
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N-Acetylpurinomycin
CAS:<p>N-Acetylpurinomycin is a selective agonist of CB2 receptor.</p>Formula:C24H31N7O6Color and Shape:SolidMolecular weight:513.55Naloxonazine
CAS:<p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>Formula:C38H42N4O6Color and Shape:SolidMolecular weight:650.763-Oxo-5β-cholanoic acid
CAS:3-Oxo-5β-cholanoic acid (Dehydrolithocholic acid) (Dehydrolithocholic acid) is a bile acid metabolite and inhibits the differentiation of TH17 cells by directlyFormula:C24H38O3Purity:98.01% - 99.86%Color and Shape:SolidMolecular weight:374.56XDM-CBP
CAS:XDM-CBP is an effective and selective CBP/p300 bromodomain inhibitor.Formula:C21H22N2O4Purity:98%Color and Shape:SolidMolecular weight:366.41LY 106737
CAS:<p>LY 106737 is opioid antagonist in the class of phenylpiperidine.</p>Formula:C21H27NOPurity:98%Color and Shape:SolidMolecular weight:309.45Cyclophostin
CAS:Cyclophostin is an irreversible inhibitor of acetylcholinesterase (AChE).Formula:C8H11O6PPurity:98%Color and Shape:SolidMolecular weight:234.14ASP-4000 HCl
CAS:ASP-4000 HCl is an inhibitor of dipeptidyl peptidase 4 (DPP) with anti-hyperglycemic activity.Formula:C12H18ClN3O2Color and Shape:SolidMolecular weight:271.74PDE5-IN-42
CAS:PDE5-IN-42 is a selective inhibitor of second-generation phosphodiesterase type 5 (PDE5).Formula:C23H31N7O3Purity:98%Color and Shape:SolidMolecular weight:453.54DC_AC50
CAS:"DC_AC50 inhibits Atox1/CCS to reduce cancer cell growth and prevent chemotherapy resistance."Formula:C17H12BrF2N3OSPurity:99.84% - 99.9%Color and Shape:SolidMolecular weight:424.26Miglustat hydrochloride
CAS:Miglustat hydrochloride (N-Butyldeoxynojirimycin hydrochloride) is an inhibitor of glucosylceramide synthase and can be used for studies about Type I GaucherFormula:C10H22ClNO4Purity:99.85%Color and Shape:SolidMolecular weight:255.74BD-AcAc 2
CAS:BD-AcAc 2 (Ketone Ester) is a ketone monoester and can be used as a source of oral nutritional ketones.Formula:C8H16O4Purity:99.62%Color and Shape:SolidMolecular weight:176.21MEN-10612
CAS:<p>MEN-10612 is a cyclic pseudopeptide and potent tachykinin NK-2 receptor antagonist.</p>Formula:C43H60N8O6Color and Shape:SolidMolecular weight:784.99PDE4-IN-8
CAS:<p>PDE4-IN-8 is a potent PDE4 inhibitor with IC50 0.93 nM for PDE4B2 and minor impact on IL13, IL4, IFNy (IC50: 4.04, 36.33, 2394 nM).</p>Formula:C18H22BNO4Color and Shape:SolidMolecular weight:327.18MAO A/HSP90-IN-2
CAS:MAO A/HSP90-IN-2 (compound 4-C), a dual inhibitor of HSP90 and MAO A, exhibits IC50 values of 0.016 μM for MAO A and 4.58 μM for HSP90.Formula:C25H31ClN2O4Purity:98%Color and Shape:SolidMolecular weight:458.98MetAP2-IN-1
CAS:MetAP2-IN-1 is a selective inhibitor of MetAP2, a target involved in angiogenesis-related conditions, suitable for research applications [1].Formula:C8H6BrN3Purity:98%Color and Shape:SolidMolecular weight:224.06BMT-108908
CAS:BMT-108908 is a Negative Allosteric Modulator. It is selective for the NR2B Subtype of The NMDA Receptor Impair Cognition in Multiple Domains.Formula:C22H25FN2O2Color and Shape:SolidMolecular weight:368.44LY-338979
CAS:LY-338979 is an impurity of pemetrexedone.Formula:C20H21N5O7Purity:98%Color and Shape:SolidMolecular weight:443.41Dothiepin
CAS:<p>Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing</p>Formula:C19H21NSPurity:98%Color and Shape:SolidMolecular weight:295.44Biphenylindanone A
CAS:Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological disorders.Formula:C30H30O4Purity:98%Color and Shape:SolidMolecular weight:454.56Ciprostene (free base)
CAS:Ciprostene, a stable prostacyclin analog, lowers blood pressure, increases heart rate, and inhibits platelets; tested in vascular disease patients.Formula:C22H36O4Color and Shape:SolidMolecular weight:364.52L 363851
CAS:L 363851 is a neurokinin B agonist.Formula:C38H51N7O7SColor and Shape:SolidMolecular weight:749.93U 89843A
CAS:<p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>Formula:C16H23N5Purity:99.62%Color and Shape:SolidMolecular weight:285.39GLPG0259
CAS:<p>GLPG-0259 is an inhibitor of mitogen-activated protein kinase-activated protein kinase 5 (MAPKAPK5).</p>Formula:C24H28N8O2Color and Shape:SolidMolecular weight:460.53RyRs activator 4
CAS:<p>Compound B18 (RyRs activator 4) is an insect ryanodine receptor activator that exhibits larvicidal activity against Mythimna separata with an LC50 value of 1.32</p>Formula:C24H21Br2ClFN5O2Color and Shape:SolidMolecular weight:625.72MIN-117
CAS:MIN-117, a SSRI/5-HT receptor antagonist, is potentially used for the treatment of depression.Formula:C25H26Cl3N3O4Purity:98%Color and Shape:SolidMolecular weight:538.85Fosfluridine tidoxil
CAS:<p>Fosfluridine tidoxil, a thymidylate synthase inhibitor, is used potentially for the treatment of colorectal cancer, and breast cancer.</p>Formula:C34H62FN2O10PSColor and Shape:SolidMolecular weight:740.9PF-06459988
CAS:PF-06459988 is a novel, effective, orally active, irreversible, and selective epidermal growth factor receptor (EGFR) mutant inhibitor.Formula:C19H22ClN7O3Purity:98%Color and Shape:SolidMolecular weight:431.88Ro 41-5253
CAS:<p>Ro 41-5253 is a RARα antagonist with antitumor activity that inhibits the proliferation of ZR-75.1 estrogen receptor-positive breast cancer cells.</p>Formula:C28H36O5SPurity:98%Color and Shape:SolidMolecular weight:484.65L-ANAP
CAS:<p>L-ANAP is a polarity-sensitive and genetically encodable fluorescent unnatural amino acid.</p>Formula:C15H16N2O3Purity:98%Color and Shape:SolidMolecular weight:272.3TAK-659
CAS:TAK-659 is a spleen tyrosine kinase (SYK) inhibitor.Formula:C17H21FN6OPurity:98%Color and Shape:SolidMolecular weight:344.39VT-1598 tosylate
CAS:VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.Formula:C38H28F4N6O5SColor and Shape:SolidMolecular weight:756.72Metabutoxycaine
CAS:<p>Metabutoxycaine, a local anesthetic [1], serves to numb specific areas of the body.</p>Formula:C17H28N2O3Color and Shape:SolidMolecular weight:308.42TC ASK 10
CAS:<p>TC ASK 10 is a potent, selective and orally active inhibitor of apoptosis signal-regulating kinase 1 (ASK1,IC50 = 14 nM). The IC50 value for ASK2 is 0.51 μM.</p>Formula:C21H23Cl2N5OPurity:99.86%Color and Shape:SolidMolecular weight:432.35NGD9002
CAS:NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.Formula:C20H31N5OPurity:98%Color and Shape:SolidMolecular weight:357.49GW-813893
CAS:GW-813893: potent, selective oral factor Xa inhibitor; Ki 4.0 nM (FXa), 9.7 nM (prothrombinase).Formula:C17H22ClN3O5S2Purity:98%Color and Shape:SolidMolecular weight:447.96Brasofensine sulfate
CAS:Brasofensine sulfate is a dopamine reuptake inhibitor.Formula:C16H22Cl2N2O5SColor and Shape:SolidMolecular weight:425.33L-644,698
CAS:L-644,698 is a selective agonist of human prostanoid DP receptor.Formula:C21H31NO4SPurity:98%Color and Shape:SolidMolecular weight:393.54K-756
CAS:<p>K-756 is a direct and selective inhibitor of tankyrase (TNKS), which inhibits the ADP-ribosylation activity of TNKS1 (IC50 = 31 nM) and TNKS2 (IC50 = 36 nM).</p>Formula:C24H27N5O3Purity:99.81%Color and Shape:SolidMolecular weight:433.5L-Moses
CAS:L-45 is the first potent and cell-active bromodomain (Brd) inhibitor of p300/CBP-associated factor (PCAF) (Kd: 126±15 nM).Formula:C21H24N6Purity:98%Color and Shape:SolidMolecular weight:360.46Cipemastat
CAS:<p>Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).</p>Formula:C22H36N4O5Purity:98%Color and Shape:SolidMolecular weight:436.55LDC3140
CAS:<p>LDC3140 is a potent inhibitor of Cyclin-dependent kinase 7 (CDK7).</p>Formula:C23H33N7OPurity:98%Color and Shape:SolidMolecular weight:423.55MiTMAB
CAS:<p>MiTMAB, a selective dynamin inhibitor, targets the interaction between dynamin and phospholipids.</p>Formula:C17H38N·BrColor and Shape:SolidMolecular weight:336.39HBV-IN-17
CAS:<p>HBV-IN-17 (compound 8) is a potent regulator of HBV capsid assembly (EC50: 511 nM).</p>Formula:C17H15F6N5O2Color and Shape:SolidMolecular weight:435.32Carotegrast
CAS:Carotegrast, an orally available α4 integrin receptor inhibitor, has anti-inflammatories activities.Formula:C27H24Cl2N4O5Color and Shape:SolidMolecular weight:555.41THRX-144644
CAS:THRX-144644: lung-specific ALK5 inhibitor, 0.14 nM IC50, no systemic TGFβ toxicity.Formula:C26H28ClF2N7Color and Shape:SolidMolecular weight:512(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Formula:C21H20ClNO6Purity:98%Color and Shape:SolidMolecular weight:417.84AY 31906
CAS:<p>AY 31906: High ceiling diuretic, boosts sodium/chloride excretion without affecting potassium, GFR, or renal flow in dogs.</p>Formula:C15H24N6O3SColor and Shape:SolidMolecular weight:368.45P11149
CAS:P11149: oral AChE inhibitor, crosses BBB, IC50 1.3 μM, based on Galanthamine, aims Alzheimer's research.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02L 663581
CAS:L 663581 is the benzodiazepine receptor partial agonist.Formula:C17H16ClN5O2Purity:98%Color and Shape:SolidMolecular weight:357.79Fenpropidin
CAS:Fenpropidin (Ro-12-3049), a fungicide, is a specific inhibitor of sterol 14-reductase and biosynthesis.Formula:C19H31NPurity:98.58% - 99.54%Color and Shape:SolidMolecular weight:273.46LX-1031
CAS:<p>LX-1031 is an effective inhibitor of tryptophan 5-hydroxylase. LX-1031 decreases serotonin (5-HT) synthesis peripherally.</p>Formula:C28H25F3N4O4Purity:97.123% - 98.97%Color and Shape:SolidMolecular weight:538.52A-849519
CAS:<p>A-849519 is a reversible MetAP2 inhibitor with anti-angiogenic and anticancer properties, tested against prostate cancer and compared to TNP-470.</p>Formula:C22H25FN2O4SColor and Shape:SolidMolecular weight:432.51Pivanex
CAS:<p>Pivanex, an oral HDAC inhibitor, targets metastasis, angiogenesis, reduces Bcr-Abl protein, and promotes apoptosis.</p>Formula:C10H18O4Purity:≥98%Color and Shape:SolidMolecular weight:202.25GSK2850163
CAS:<p>GSK2850163 is a novel inhibitor of inositol-requiring enzyme-1 alpha (IRE1α) which can inhibit RNase activity and IRE1α kinase activity (IC50s: 200 and 20 nM).</p>Formula:C24H29Cl2N3OPurity:99.04%Color and Shape:SolidMolecular weight:446.41Ro 31-9790
CAS:<p>Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).</p>Formula:C15H29N3O4Purity:98%Color and Shape:SolidMolecular weight:315.41H4R antagonist 2
CAS:<p>H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid</p>Formula:C13H17N5OPurity:98%Color and Shape:SolidMolecular weight:259.31FGIN-1-27
CAS:<p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>Formula:C28H37FN2OPurity:99.86%Color and Shape:SolidMolecular weight:436.6TXNIP-IN-1
CAS:<p>TXNIP-IN-1: TXNIP-TRX complex inhibitor, targets diabetes, cardiovascular, and inflammatory diseases.</p>Formula:C12H12N2O4Purity:99.11%Color and Shape:SolidMolecular weight:248.23GSK3395879
CAS:<p>GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).</p>Formula:C20H15F4N3O5SPurity:98%Color and Shape:SolidMolecular weight:485.41ATM-IN-1
CAS:<p>ATM-IN-1 is a potent inhibitor of ATM. ATM-IN-1 has shown research potential in cancer and neurological diseases.</p>Formula:C30H36N6O3Color and Shape:SolidMolecular weight:528.656-Iodoamiloride
CAS:<p>6-Iodoamiloride is a potent inhibitor of acid-sensing ion channel 1 (ASIC1), exhibiting an IC50 value of 88 nM.</p>Formula:C6H8IN7OPurity:98%Color and Shape:SolidMolecular weight:321.08Binedaline
CAS:Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formula:C19H23N3Purity:98%Color and Shape:SolidMolecular weight:293.41LY-426965
CAS:<p>LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.</p>Formula:C28H38N2O2Color and Shape:SolidMolecular weight:434.61Cathepsin Inhibitor 2
CAS:<p>Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor (Ki: <20 nM).</p>Formula:C19H21F6N3OPurity:98%Color and Shape:SolidMolecular weight:421.383,4'-Dihydroxyflavone
CAS:3,4'-Dihydroxyflavone (3,4'-DHF) is an oral active flavonoid. 3,4'-Dihydroxyflavone (3,4'-DHF) shows antiviral activity against Influenza A virus.Formula:C15H10O4Purity:98.33%Color and Shape:SolidMolecular weight:254.24CUR61414
CAS:<p>CUR61414 is a cell-permeable inhibitor of Hedgehog signaling pathway (IC50 =100-200 nM) and selectively binds to smoothened (Ki = 44 nM).</p>Formula:C31H42N4O5Purity:97.34% - 98%Color and Shape:SolidMolecular weight:550.69β-catenin-IN-4
CAS:<p>β-Catenin-IN-4 is a β-catenin inhibitor characterized by a K_i value of 0.64 μM.</p>Formula:C38H33ClF3N5O9Color and Shape:SolidMolecular weight:796.14WAY-659873
CAS:<p>WAY-659873 is an active molecule.</p>Formula:C19H17FN2O4S2Color and Shape:SolidMolecular weight:420.48Alteconazole
CAS:Alteconazole is an antifungal drug.Formula:C17H12Cl3N3OPurity:98%Color and Shape:SolidMolecular weight:380.66KD-026
CAS:KD-026 (SLx 4090), a microsomal triglyceride transfer protein (MTP) inhibitor(IC50 = 8.0 nM), is used in type 2 diabetes studies.Formula:C31H25F3N2O4Purity:99.74%Color and Shape:SolidMolecular weight:546.54GSK2188764
CAS:GSK2188764 is an inhibitor of T. brucei IPMK, partially inhibits rTbIPMK activity.Formula:C17H16Cl2N6OPurity:98%Color and Shape:SolidMolecular weight:391.25ASGPR ligand-1
CAS:ASGPR ligand-1 is a compound that targets the asialoglycoprotein receptor (ASGPR) and is utilized in various disease research contexts [1].Formula:C61H110N10O27Color and Shape:SolidMolecular weight:1415.58KPZ560
CAS:KPZ560, a potent HDAC 1 and HDAC 2 inhibitor, exhibits IC50 values of 12 nM and 68 nM, respectively.Formula:C26H21N5O3S2Purity:98%Color and Shape:SolidMolecular weight:515.61Levocabastine hydrochloride
CAS:<p>Levocabastine HCl is an agent with antihistaminic activity.</p>Formula:C26H30ClFN2O2Color and Shape:SolidMolecular weight:456.98ICMT-IN-14
CAS:ICMT-IN-14 (compound 50) serves as an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting potent activity with an IC50 of 0.025 μM [1].Formula:C21H25ClFNOColor and Shape:SolidMolecular weight:361.88MNI-444
CAS:<p>MNI-444 is a PET radiotracer for adenosine 2A receptors.</p>Formula:C24H26FN9O2Color and Shape:SolidMolecular weight:491.52HR68
CAS:<p>HR68, a derivative of the peroxisome proliferator-activated receptor (PPAR) agonist fenofibric acid, serves as an anticancer agent.</p>Formula:C22H19ClN2O3Color and Shape:SolidMolecular weight:394.85P-1075
CAS:P-1075 activates SUR2-KIR6 channels at 45 nM; may open mitoKATP channels and protect the heart.Formula:C12H17N5Purity:99.85%Color and Shape:SolidMolecular weight:231.3FC 11
CAS:<p>FC 11 is a reversible FAK PROTAC Degrader with DC50 of 40-370 pM and degrades pFAKtyr397 in TM3 cells within 3 hours at 100 nM.</p>Formula:C41H42F3N13O9SColor and Shape:SolidMolecular weight:949.91Anticancer agent 103
CAS:<p>Compound 103 (Compound 2k) serves as a potent anticancer agent [1].</p>Formula:C18H20BrN3OColor and Shape:SolidMolecular weight:374.28GEM-IB
CAS:<p>Gemcitabine-ibandronate (GEM–IB), a conjugate of gemcitabine (GEM)-5'-phosphate with ibandronate (IB), exhibits efficacy both as a monotherapy and</p>Formula:C18H33F2N4O13P3Color and Shape:SolidMolecular weight:644.39AD-35
CAS:<p>AD-35 treats Alzheimer's by blocking TNF-α and IL-1β, curbing inflammation.</p>Formula:C24H27N3O3Color and Shape:SolidMolecular weight:405.49SARS-CoV-2 3CLpro-IN-2
CAS:<p>SARS-CoV-2 3CLpro-IN-2 is a potent inhibitor of the 3CL protease pair and has shown research potential for SARS-CoV-2 disease.</p>Formula:C21H18F5N5O4Color and Shape:SolidMolecular weight:499.39mTOR inhibitor 9b
CAS:<p>mTOR inhibitor 9b is an enzyme inhibitor of protein kinase mTOR he phosphatidylinositol 3-kinase PIK3CA with IC50s of 0.76 nm and 1.262 µM, respectively.mTOR</p>Formula:C21H23N5O2SPurity:99.52%Color and Shape:SoildMolecular weight:409.5CBP/p300-IN-21
CAS:CBP/p300-IN-21 (Compound 5d), a selective inhibitor of CBP/p300 with IC50 values of 0.07 μM for p300 and 1.755 μM for CBP, reduces H3K18Ac levels and inhibitsFormula:C19H16ClNO4Purity:98%Color and Shape:SolidMolecular weight:357.79eIF4A3-IN-18
CAS:eIF4A3-IN-18, a silvestrol analogue with EC50s: 0.8/35/2 nM, inhibits eIF4F complex and is cytotoxic (LC50: 0.06 nM) for cancer research.Formula:C29H28N2O6Color and Shape:SolidMolecular weight:500.54Sodium Channel inhibitor 4
CAS:<p>Sodium Channel Inhibitor 4 is a compound that functions as a sodium channel inhibitor [1].</p>Formula:C19H18ClN3O4S2Purity:98%Color and Shape:SolidMolecular weight:451.95NaPi2b-IN-2
CAS:<p>NaPi2b-IN-2 (compound 5) serves as a potent inhibitor of the sodium-dependent transport protein 2b (SLC34A2, NaPi2b), exhibiting an IC50 of 38 nM against human</p>Formula:C41H47ClF3N5O5SPurity:98%Color and Shape:SolidMolecular weight:814.36Ro 18-5364
CAS:Ro 18-5364 is a potent inhibitor of the gastric (H+ + K+)-ATPase with an apparent Ki of 0.1 μM at pH 6.Formula:C22H25N3O3SPurity:98%Color and Shape:SolidMolecular weight:411.52MAT2A-IN-12
CAS:<p>MAT2A Allosteric Inhibitor 2 is a potent, selective inhibitor exhibiting an IC50 of 5 nM and demonstrates nanomolar efficacy (IC50 = 5 μM) in proliferation</p>Formula:C20H17NO3Purity:98%Color and Shape:SolidMolecular weight:319.35RET-IN-5
CAS:<p>RET-IN-5 is a potent inhibitor of RET (IC50: 4.57 nM).</p>Formula:C29H26FN9OColor and Shape:SolidMolecular weight:535.57ALK/EGFR-IN-1
CAS:ALK/EGFR-IN-1 (Compound 8l) is a dual inhibitor targeting both ALK and EGFR, effectively blocking their phosphorylation.Formula:C27H34ClN7O3SPurity:98%Color and Shape:SolidMolecular weight:572.12Glucocorticoid receptor agonist
CAS:<p>Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.</p>Formula:C20H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:396.38Amedalin
CAS:Amedalin is a biochemical.Formula:C19H22N2OColor and Shape:SolidMolecular weight:294.398BCR-ABL-IN-4
CAS:BCR-ABL-IN-4: Anticancer BCR-ABL inhibitor; stops K562 cells (IC50: 0.67 nM), targets T315I Ba/F3 cells (IC50: 16 nM).Formula:C27H24ClF2N5O4Color and Shape:SolidMolecular weight:555.96NLRP3-IN-22
CAS:<p>NLRP3-IN-22 (Compound II-4) is an inhibitor of NLRP3, exhibiting a 67% inhibition rate at a concentration of 10 μM [1].</p>Formula:C19H12F3NO4SPurity:98%Color and Shape:SolidMolecular weight:407.36GT-2394
CAS:GT-2394 is a histamine H3 receptor agonist.Formula:C14H21N3O2Color and Shape:SolidMolecular weight:263.34Indacrinone
CAS:<p>Indacrinone is an investigational diuretic.</p>Formula:C18H14Cl2O4Purity:98%Color and Shape:SolidMolecular weight:365.21MC-Val-Cit-PAB-NH-C2-NH-Boc
CAS:<p>MC-Val-Cit-PAB-NH-C2-NH-Boc is a cathepsin-cleavable ADC linker utilized in constructing antibody-drug conjugates (ADCs) [1].</p>Formula:C36H54N8O10Color and Shape:SolidMolecular weight:758.86IRAK inhibitor 3
CAS:IRAK inhibitor 3 is an interleukin-1 (IL-1) receptor-associated kinase (IRAK) modulator.Formula:C21H21N5O4SPurity:98.86%Color and Shape:SolidMolecular weight:439.49Pomaglumetad methionil hydrochloride
CAS:<p>LY2140023 hydrochloride: oral methionine prodrug of LY404039, a selective mGlu2/3 agonist, studied for schizophrenia.</p>Formula:C12H19ClN2O7S2Purity:98.57%Color and Shape:SolidMolecular weight:402.87LDHA/PDKs-IN-1
CAS:Compound 20e inhibits PDKs (IC50: 0.8 μM) & LDHA (IC50: 0.15 μM), halts A549 cell growth, lowers lactate, boosts oxygen use.Formula:C19H21FN2O4Color and Shape:SolidMolecular weight:360.38CP-96486
CAS:<p>CP-96486 is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor (Kis: 20 and 24 nM).</p>Formula:C31H23ClN4OPurity:98%Color and Shape:SolidMolecular weight:502.99Cholesterylamine
CAS:<p>Cholesterylamine, a cationic lipid, can be incorporated into PLGA to create particles with a charged surface, facilitating its use in drug delivery systems and</p>Formula:C27H47NColor and Shape:SolidMolecular weight:385.671-Methoxyphaseollidin
CAS:1-Methoxyphaseollidin exhibits anti-Helicobacter pylori activity against the CLAR and AMOX-resistant strain as well as four CLAR (AMOX)-sensitive strains.Formula:C21H22O5Purity:98%Color and Shape:SolidMolecular weight:354.4Coelenterazine h
CAS:<p>Coelenterazine H, a Ca2+ sensitive synthetic derivative, is a luminescent biomolecule used to measure Ca2+ changes.</p>Formula:C26H21N3O2Purity:99.49%Color and Shape:Yellow To Brownish PowderMolecular weight:407.46BMS-561390
CAS:<p>BMS-561390, a reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Formula:C14H12ClF3N2OColor and Shape:SolidMolecular weight:316.71Dezapelisib
CAS:<p>Dezapelisib, an oral delta PI3K inhibitor, blocks PIP3 production and PI3K/AKT pathway, hindering tumor cell growth and survival.</p>Formula:C20H16FN7OSColor and Shape:SolidMolecular weight:421.45Brodimoprim
CAS:<p>Brodimoprim is an inhibitor of dihydrofolate reductase(DHFR).</p>Formula:C13H15BrN4O2Purity:98% - 98.33%Color and Shape:SolidMolecular weight:339.19KCL-286
CAS:KCL-286 is an available and potent retinoic acid receptor beta agonist for the amelioration of spinal cord injury (SCI).Formula:C19H14N2O4Purity:99.93%Color and Shape:SolidMolecular weight:334.33uPSEM 817 tartrate
CAS:<p>Potent α7L-GlyR & PSAM4-5-HT3 agonist (EC50: 0.3/0.5 nM). Reduces cortical neuron activity; induces contralateral rotation in mice (LED 0.1 mg/kg).</p>Formula:C20H25N3O7Color and Shape:SolidMolecular weight:419.434Quorum Sensing-IN-2
CAS:Quorum Sensing-IN-2 (compound 23e) is a quorum sensing inhibitor that curtails bacterial pathogenicity without impeding growth.Formula:C19H13F2NO3Color and Shape:SolidMolecular weight:341.31Cynandione A
CAS:Cynandione A is an acetophenone derived from Cynanchum wilfordii with anti-inflammatory activity.Formula:C16H14O6Purity:99.62%Color and Shape:SolidMolecular weight:302.28Agerafenib hydrochloride
CAS:Agerafenib hydrochloride is a highly potent inhibitor of BRAFV600E (Kd: 14 nM).Formula:C24H23ClF3N5O5Purity:98%Color and Shape:SolidMolecular weight:553.92L 687908
CAS:L 687908 is a potent inhibitor of hydroxyethylene-containing HIV protease.Formula:C40H51N5O5Purity:98%Color and Shape:SolidMolecular weight:681.86Fructose-arginine
CAS:<p>Fructose-arginine is a non-saponin molecule from Korean Red Ginseng that attenuates AIM2 inflammatory vesicle activation.</p>Formula:C12H24N4O7Purity:97.79% - 99.86%Color and Shape:SolidMolecular weight:336.34FEN1-IN-6
CAS:<p>FEN1-IN-6 (compound 9) is a potent Flap endonuclease-1 (FEN1, IC50 = 10 nM) inhibitor, crucial for DNA damage repair in mammalian cells, and additionally</p>Formula:C12H8N2O5S2Purity:98%Color and Shape:SolidMolecular weight:324.33EGFR mutant-IN-1
<p>EGFR mutant-in-1, a 5-methylpyrimidopyridone, selectively inhibits EGFRL858R/T790M/C797S mutants with an IC50 of 27.5 nM, lessening EGFRWT impact.</p>Formula:C34H39ClFN7O2Purity:98%Color and Shape:SolidMolecular weight:632.17Inixaciclib
CAS:Inixaciclib is a potent CDK inhibitor, can be used to research anticancer.Formula:C26H30F2N6OColor and Shape:SolidMolecular weight:480.55HBV-IN-41
CAS:HBV-IN-41 (compound 45) is a potent, orally active inhibitor of Hepatitis B Virus (HBV), exhibiting an EC50 value of 0.027μM [1].Formula:C18H19ClFN5O3Purity:98%Color and Shape:SolidMolecular weight:407.83(rel)-BMS-641988
CAS:(rel)-BMS-641988, a relative configuration of the potent nonsteroidal androgen receptor antagonist BMS-641988, holds potential for prostate cancer research.Formula:C20H20F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:471.45FGFR-IN-8
CAS:<p>FGFR-IN-8, potent oral FGFR inhibitor for wild-type/mutant types, induces apoptosis with anti-cancer properties.</p>Formula:C27H31Cl2N9O2Color and Shape:SolidMolecular weight:584.5Fasidotril
CAS:Fasidotril inhibits NEP/ACE, treats high blood pressure in rats, effective in humans with hypertension.Formula:C23H25NO6SPurity:98%Color and Shape:SolidMolecular weight:443.51Lp-PLA2-IN-14
CAS:Lp-PLA2-IN-14 (Compound 19), an inhibitor of rhLp-PLA2, exhibits a potent inhibitory effect with a pIC50 value of 8.4.Formula:C16H14F3N3O3Purity:98%Color and Shape:SolidMolecular weight:353.3VU0463271
CAS:<p>VU0463271: KCC2 antagonist, IC50 61 nM, >100x selective over NKCC1, inactive on other GPCRs, channels, transporters.</p>Formula:C19H18N4OS2Purity:97.84% - 99.55%Color and Shape:SolidMolecular weight:382.5U 66985
CAS:<p>U 66985 is a Platelet-activating factor (PAF) receptor antagonist that inhibit the electrophysiological effects of PAF.</p>Formula:C32H66NO7PColor and Shape:SolidMolecular weight:607.84VGD020
CAS:<p>VGD020 inhibits CD4/sortilin, reduces sortilin & hinders breast cancer stem cell growth.</p>Formula:C31H45N3O5S2Color and Shape:SolidMolecular weight:603.84(R)-Necrocide 1
CAS:<p>(R)-Necrocide 1 (compound (R)-38) is a potent anticancer agent with antiproliferative activity [1].</p>Formula:C23H27NO3Purity:98%Color and Shape:SolidMolecular weight:365.47(S)-(-)-Bay-K-8644
CAS:(S)-(-)-Bay-K-8644 ((S)-(-)-Bay K 8644) is an agonist of L-type Ca2+ channel and activates Ba2+ currents with an EC50 of 32 nM.Formula:C16H15F3N2O4Purity:98.28% - 99.37%Color and Shape:SolidMolecular weight:356.3Iganidipine
CAS:<p>Iganidipine（NKY 722） is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.</p>Formula:C28H38N4O6Purity:96.3%Color and Shape:SolidMolecular weight:526.62CJ-15161 (free base)
CAS:<p>CJ-15161 (free base), an opioid κ-receptor agonist, is undergoing development with Pfizer as an analgesic agent.</p>Formula:C23H31N3O2Color and Shape:SolidMolecular weight:381.51Clibucaine
CAS:Clibucaine, a piperidine derivative, exhibits local anesthetic properties and is employed as a local anesthetic agent [1].Formula:C15H20Cl2N2OColor and Shape:SolidMolecular weight:315.24RSV L-protein-IN-2
CAS:<p>RSV L-protein-IN-2 (Compound A), a noncompetitive inhibitor of the RSV polymerase (IC50: 4.5 μM), exhibits antiviral activity against long RSV strains (EC50: 1.</p>Formula:C32H36N4O5Purity:98%Color and Shape:SolidMolecular weight:556.65RET-IN-13
CAS:RET-IN-13: potent quinoline RET inhibitor; IC50 = 0.5 nM (WT), 0.9 nM (V804M); potential for RET-related tumor/intestinal disease research.Formula:C32H33F4N5O3Color and Shape:SolidMolecular weight:611.63IDH1 Inhibitor 3
CAS:IDH1 Inhibitor 3 is a mutant isocitric dehydrogenase 1 (IDH1) inhibitor (IC50: 45 nM for IDH1R132H).Formula:C31H25F4N5O3Purity:98%Color and Shape:SolidMolecular weight:591.56Tegeprotafib
CAS:<p>5-OP-RU is a MAIT-activating ligand, a major antigen of MAIT cells, a mucosal adjuvant, and can be used to study Mycobacterium tuberculosis infection.</p>Formula:C13H11FN2O5SPurity:99.69%Color and Shape:SolidMolecular weight:326.3Efipladib
CAS:<p>Efipladib is a phospholipase inhibitor. Efipladib decreases nociceptive responses without affecting PGE2 levels in the cerebral spinal fluid.</p>Formula:C40H35Cl3N2O4SColor and Shape:SolidMolecular weight:746.14S1p receptor agonist 2
CAS:<p>S1P5-selective agonist; less so for S1P1/S1P3; useful for CNS disorders.</p>Formula:C24H23ClN2O4Color and Shape:SolidMolecular weight:438.9STAT6-IN-3
CAS:STAT6-IN-3 (Compound 18a) serves as an inhibitor of STAT6 with an IC50 value of 44 nM, specifically targeting the Src Homology 2 (SH2) domain.Formula:C32H35IN3O7PPurity:98%Color and Shape:SolidMolecular weight:731.51E1R
CAS:<p>E1R is a positive sigma-1 receptor (Sig1R PAM) allosteric modulator. It has a cognition-enhancing activity.</p>Formula:C13H16N2O2Color and Shape:SolidMolecular weight:232.28CLB-016
CAS:CLB-016 is an inhibitor of hypoxia-inducible factor (HIF)-1.Formula:C17H20N6O3Purity:98%Color and Shape:SolidMolecular weight:356.38Potassium Channel Activator 1
CAS:<p>Potassium Channel Activator 1 aids treatment of ADHD, schizophrenia, and mood disorders by targeting the dopaminergic system.</p>Formula:C19H23N3O3Purity:99.86%Color and Shape:SolidMolecular weight:341.4Thrombin inhibitor 1
CAS:<p>Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).</p>Formula:C22H20Cl2F2N4O3Purity:98%Color and Shape:SolidMolecular weight:497.32TG 100572 Hydrochloride
CAS:<p>TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src kinases(IC50s of 2, 7, 2, 16, 13, 5, 0.5, 6, 0.</p>Formula:C26H27Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:512.43DNA gyrase B-IN-3
CAS:DNA gyrase B-IN-3 (Compound A), with an IC50 of less than 10 nM, acts as an inhibitor of bacterial DNA gyrase B and exhibits antibacterial activity against GramFormula:C14H9Cl2N3O4SPurity:98%Color and Shape:SolidMolecular weight:386.21Urease Inhibitor 07
CAS:Urease Inhibitor 07 is an isosubstituted metalloproteinase inhibitor with potential activity against Mycobacterium tuberculosis strain H37Rv.Formula:C7H5N3OSPurity:99.65%Color and Shape:SolidMolecular weight:179.2ICI 200355
CAS:ICI 200355 is an inhibitor of human neutrophil elastase.Formula:C30H34BrF3N4O7SPurity:98%Color and Shape:SolidMolecular weight:731.58Melafolone
CAS:Melafolone: natural COX-2/EGFR inhibitor, enhances PD-1 therapy by normalizing tumor vessels, lowers PD-L1.Formula:C22H24O7Color and Shape:SolidMolecular weight:400.42Lifirafenib
CAS:Lifirafenib (Beigene-283) is a potent inhibitor of RAF family kinases and EGFR in biochemical assays with IC50 of 23, 29 and 495 nM for the recombinantFormula:C25H17F3N4O3Purity:97.99% - 98%Color and Shape:SolidMolecular weight:478.42Limocrocin
CAS:Limocrocin is an inhibitor of reverse transcriptase.Formula:C26H26N2O6Purity:98%Color and Shape:SolidMolecular weight:462.49Me-Indoxam
CAS:Me-Indoxam is an inhibitor of sPLA2. It has no effect on arachidonic acid release and platelet activating factor synthesis.Formula:C26H22N2O5Purity:98%Color and Shape:SolidMolecular weight:442.46STAT3-IN-14
CAS:<p>STAT3-IN-14 is a STAT3 inhibitor and has STAT3 phosphorylation inhibitory activity. STAT3-IN-14 can directly bind to the hinge region of STAT3 .</p>Formula:C14H10O5Color and Shape:SolidMolecular weight:258.23Indimilast
CAS:<p>Indimilast blocks PDE4, reducing lung inflammation and bronchiectasis, possibly treating COPD.</p>Formula:C37H40FN7O3SColor and Shape:SolidMolecular weight:681.82α,β-Methylene-ATP
CAS:<p>α,β-Methylene ATP，一种ATP的膦酸酯类似物，充当P2X3和P2X7受体的配体。该化合物对P2X1和P2X3表现出高选择性激动剂活性，而在P2X2, 4, 7受体上无活性。</p>Formula:C11H18N5O12P3Color and Shape:SolidMolecular weight:505.21PVZB1194
CAS:<p>PVZB1194, a biphenyl-type inhibitor of Kinesin spindle protein Eg5 (KIF11), exhibits anticancer potential by inducing cell cycle arrest and apoptosis through</p>Formula:C13H9F4NO2SPurity:98%Color and Shape:SolidMolecular weight:319.28PYZD-4409
CAS:<p>PYZD-4409 is a selective UBA1 inhibitor with an IC50 of 20 μM.</p>Formula:C14H7ClFN3O5Purity:99.71%Color and Shape:SolidMolecular weight:351.67(Rac)-PF-06250112
CAS:(Rac)-PF-0625011 is a racemic mix, orally active, selective BTK inhibitor, also targeting BMX and TEC kinases.Formula:C22H20F2N6O2Purity:98%Color and Shape:SolidMolecular weight:438.43BT424
CAS:BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation and renal fibrosis in the UUO model [1].Formula:C22H15BCl2N2O2Purity:98%Color and Shape:SolidMolecular weight:421.08Emicerfont
CAS:<p>Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).</p>Formula:C22H24N6O2Purity:98%Color and Shape:SolidMolecular weight:404.46KRAS G12C inhibitor 40
CAS:KRAS G12C inhibitor 40 targets KRAS G12C in cancer research (WO2021129824A1, compound 70).Formula:C34H36ClFN10O2Color and Shape:SolidMolecular weight:671.17Setipafant
CAS:<p>Setipafant is an antagonist of the platelet-activating factor.</p>Formula:C26H23ClN6O2SPurity:98%Color and Shape:SolidMolecular weight:519.02Aceratioside
CAS:Aceratioside is a new tetralin glucoside. It may have antineoplastic activity.Formula:C17H22O9Purity:98%Color and Shape:SolidMolecular weight:370.35Befiradol
CAS:Befiradol (NLX-112) is an agonist of 5-HT1A receptor.Formula:C20H22ClF2N3OColor and Shape:SolidMolecular weight:393.86PF-05150122
CAS:<p>PF-05150122 is a novel potent and selective human Nav1.7 blocker.</p>Formula:C24H21ClN6O3S2Color and Shape:SolidMolecular weight:541.04Antibacterial agent 92
<p>Antibacterial agent 92 inhibits Salmonella's aaRS; IC50 of 0.58 μM for Se ThrRS. Exhibits antibacterial effects.</p>Formula:C30H28Cl2F3N5O4Color and Shape:SolidMolecular weight:650.48GPR52 receptor modulator 1
CAS:GPR52 receptor modulator 1, a compound delineated as per Procedure 1, is a modulator of the GPR52 receptor, offering research potential in the investigation ofFormula:C19H14F4N4OPurity:98%Color and Shape:SolidMolecular weight:390.33Camonsertib
CAS:<p>Camonsertib (RP-3500) is a novel, potent and selective ATR kinase inhibitor (ATRi) that exhibits potent antitumor effects with an IC50: 1.00 nM in biochemical assays.Cost-effective and quality-assured.</p>Formula:C21H26N6O3Purity:99.6% - 99.93%Color and Shape:SolidMolecular weight:410.47Ecopladib
CAS:<p>Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) & 0.11 μM (rat blood).</p>Formula:C39H33Cl3N2O5SPurity:95.15%Color and Shape:SolidMolecular weight:748.11Selvigaltin
CAS:Selvigaltin (GB1211) is a Gal-3 inhibitor with potential anticancer activity. Selvigaltin is used in the study of cirrhosis and cancer.Formula:C19H16BrF3N4O4SPurity:99.49%Color and Shape:SolidMolecular weight:533.32TP-10
CAS:<p>TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.</p>Formula:C26H19F3N4OPurity:99.21%Color and Shape:SolidMolecular weight:460.45Plogosertib
CAS:<p>Plogosertib (CYC140) is a PLK1 inhibitor with an IC50 value of 3 nM.Plogosertib is antiproliferative and can be used to study solid and hematologic tumors.</p>Formula:C34H48N8O3Purity:99.22% - 99.85%Color and Shape:SolidMolecular weight:616.797OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purity:99.79%Color and Shape:SolidMolecular weight:421.58ML400
CAS:<p>ML400 (CID73050863) is an allosteric inhibitor of LMPTP with an EC50 of 1μM. ML400 displays good cell-based activity and rodent pharmacokinetics.</p>Formula:C24H29N3OPurity:99.95%Color and Shape:SolidMolecular weight:375.51ALDH2 modulator 1
CAS:<p>ALDH2 modulator 1 is a potent and orally active modulator of acetaldehyde dehydrogenase-2 (ALDH2), which reduces blood alcohol levels in mice.</p>Formula:C18H18ClFN2O3Purity:99.68%Color and Shape:SoildMolecular weight:364.8CDC801
CAS:<p>CDC801 is an inhibitor of PDE4 and TNF-α with IC50s of 1.1 μM and 2.5 μM, respectively.</p>Formula:C23H24N2O5Purity:99.61%Color and Shape:SolidMolecular weight:408.45BI-2493
CAS:BI-2493 is a highly selective pan-KRAS inhibitor and structural analog of BI-2865.BI-2493 exhibits antitumor activity and inhibits tumor cell growth.Cost-effective and quality-assured.Formula:C24H27N7OSPurity:97.74% - 99.88%Color and Shape:SoildMolecular weight:461.58(-)-Anonaine
CAS:<p>(-)-Anonaine can be extracted from several species of Magnoliaceae and Annelidae and has antimalarial, antibacterial, antifungal, antioxidant, anticancer,</p>Formula:C17H15NO2Purity:98.21% - 98.63%Color and Shape:SolidMolecular weight:265.31γ-Glu-Tyr
CAS:<p>gamma-Glu-Tyr (gamma-Glutamyltyrosine) is a kokumi peptide against dipeptidyl peptidase-IV (DPP-IV) and is used in the study of diabetes mellitus.</p>Formula:C14H18N2O6Purity:98.92%Color and Shape:SolidMolecular weight:310.3Cdk1/2 Inhibitor III
CAS:<p>Cdk1/2 Inhibitor III is a selective Cdk1/2 inhibitor with an IC50 value of 2.1 μM against CDK1/cyclin B.</p>Formula:C15H13F2N7O2S2Purity:99.07%Color and Shape:SolidMolecular weight:425.44NMI 8739
CAS:<p>NMI 8739 (n-docosahexaenoyl dopamine) is an agonist of D2 autoreceptor.</p>Formula:C30H41NO3Purity:98.51%Color and Shape:SolidMolecular weight:463.65EGFR/ErbB-2 inhibitor-1
CAS:<p>EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.</p>Formula:C23H15ClFN3OS2Purity:98.93%Color and Shape:SolidMolecular weight:467.97EPZ031686
CAS:<p>EPZ031686 is an effective inhibitor of SMYD3 inhibitor with an IC50 of 3 nM and can be used in studies about cancer.</p>Formula:C26H34ClF3N4O4SPurity:99.67%Color and Shape:SolidMolecular weight:591.09VGSCs-IN-1
CAS:<p>VGSCs-IN-1, a VGSC inhibitor and Riluzole analog, exhibits good blocking activity on Nav1.4 and can be used to study cellular excitability disorders.</p>Formula:C12H12F3N3OSPurity:99.88%Color and Shape:SolidMolecular weight:303.3GI 181771
CAS:<p>GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.</p>Formula:C34H31N5O6Purity:95.02%Color and Shape:SolidMolecular weight:605.64Ranirestat
CAS:Ranirestat (AS-3201) is an AR inhibitor with neuroprotective properties that improves peripheral nerve dysfunction in rats with advanced diabetic polyneuropathyFormula:C17H11BrFN3O4Purity:96.10% - 99.44%Color and Shape:SolidMolecular weight:420.19Oditrasertib
CAS:<p>Oditrasertib, a RIPK1 inhibitor characterized by an IC50 value below 100 nM, is employed in inflammation research.</p>Formula:C14H15F2N3O2Purity:98.65% - 99.65%Color and Shape:SolidMolecular weight:295.28M2698
CAS:<p>M2698 (MSC2363318A) is an inhibitor of p70S6K, Akt1 and Akt3 with IC50s of 1 nM. M2698 shows anti-cancer activity.</p>Formula:C21H19ClF3N5OPurity:99.88%Color and Shape:SolidMolecular weight:449.86LTβR-IN-1
CAS:<p>LTβR-IN-1 is a potent and selective lymphin β receptor (LTβR) inhibitor.</p>Formula:C18H16N4O2Purity:98.93%Color and Shape:SolidMolecular weight:320.35PARP-1-IN-4
CAS:<p>PARP-1-IN-4 is a potent PARP-1 inhibitor with potential see anti-tumor activity, and inhibition of PARP-1 may be used in cancer development.</p>Formula:C22H15Cl2N3O2Purity:99.82%Color and Shape:SolidMolecular weight:424.28Calcium channel-modulator-1
CAS:<p>Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.</p>Formula:C26H24Cl2N2O7SPurity:99.95%Color and Shape:SolidMolecular weight:579.45CCR3 antagonist 1
CAS:<p>CCR3 antagonist 1 is a potent CCR3 antagonist, used for the research of inflammatory and immunologic diseases.</p>Formula:C19H21Cl2N3O4S2Purity:98.28%Color and Shape:SolidMolecular weight:490.42Alrizomadlin
CAS:Alrizomadlin is an orally active MDM2 inhibitor. APG-115 shows significant dose-dependent inhibitory effects on TP53wt AML cell lines.Cost-effective and quality-assured.Formula:C34H38Cl2FN3O4Purity:98.41% - 99.47%Color and Shape:SolidMolecular weight:642.59KB-74935
CAS:<p>KB-74935: enzyme inhibitor, mineralocorticoid blocker, treats cholesterol, hypolipidemia, neurological issues, Alzheimer's.</p>Formula:C19H18ClF4N3O3SPurity:99.4%Color and Shape:SolidMolecular weight:479.88Nrf2-IN-3
CAS:Nrf2-IN-3 is an NRF2 inhibitor that selectively sensitizes xenografts of mouse mKEAP1 cancer cells to cisplatin.Formula:C22H26N4O4SPurity:98.07%Color and Shape:SolidMolecular weight:442.53MMV688533
CAS:<p>MMV688533 has antimalarial activity.</p>Formula:C24H15F6N5O2Purity:99.12%Color and Shape:SoildMolecular weight:519.4L-DABA hydrobromide
CAS:<p>L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) , GABA transaminase inhibitor with antitumor and anticonvulsant activity.</p>Formula:C4H11BrN2O2Purity:99.11%Color and Shape:SolidMolecular weight:199.05CFI-402257
CAS:<p>CFI-402257 is a selective inhibitor of Mps1/TTK kinase (Mps1 Ki = 0.09 nM; EC50 = 6.5 nM)and can be used in studies about hepatocellular carcinoma diseases.</p>Formula:C28H30N6O3Purity:96.66% - 99.51%Color and Shape:SolidMolecular weight:498.58AZD4573
CAS:<p>AZD4573 is an effective and selective CDK9 inhibitor (IC50: <4 nM). It enables transient target engagement for the treatment of hematologic malignancies.</p>Formula:C22H28ClN5O2Purity:99% - 99.51%Color and Shape:SolidMolecular weight:429.94Nothofagin
CAS:Nothofagin: Antioxidant, anti-inflammatory, prevents clotting, inhibits leukocyte activity, may treat vascular inflammation.Formula:C21H24O10Purity:98.51%Color and Shape:SolidMolecular weight:436.41DS08210767
CAS:<p>DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM.</p>Formula:C31H39N5O2Purity:98.79%Color and Shape:SolidMolecular weight:513.67
