Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,850 products)
- Apoptosis(6,367 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,631 products)
- Cytoskeletal Signaling(1,586 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,053 products)
- Immunology and Inflammation(3,946 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,671 products)
- Neuroscience(10,551 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,989 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66515 products of "Inhibitors"
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E7016
CAS:E7016 (GPI 21016) is an orally available PARP inhibitor. E7016 inhibits of DNA repair. E7016 can enhance tumor cell radiosensitivity in vitro and in vivo.
Formula:C20H19N3O3Purity:99.02%Color and Shape:SolidMolecular weight:349.38Iptacopan
CAS:Iptacopan (LNP023) is an inhibitor with high affinity to factor B, with a KD value of 7.9 nM and an IC50 value of 10 nM. Cost-effective and quality-assured.Formula:C25H30N2O4Purity:99.07% - >99.99%Color and Shape:SolidMolecular weight:422.52Ref: TM-T11864
1mg52.00€5mg114.00€1mL*10mM (DMSO)126.00€10mg185.00€25mg334.00€50mg557.00€100mg919.00€200mg1,243.00€ADS032
CAS:ADS032 (BT-032) is an NLRP1 and NLRP3 inhibitor with anti-inflammatory activity for the study of respiratory inflammation or infection.Formula:C22H29NO4SPurity:98.37%Color and Shape:SolidMolecular weight:403.54Enerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purity:99.7%Color and Shape:SoildMolecular weight:398.50Ref: TM-T67828
1mg49.00€2mg67.00€5mg102.00€1mL*10mM (DMSO)111.00€10mg166.00€25mg339.00€50mg439.00€100mg610.00€200mg827.00€Varespladib methyl
CAS:Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Formula:C22H22N2O5Purity:99.42% - 99.97%Color and Shape:SolidMolecular weight:394.42Ref: TM-T17218
1mg93.00€2mg123.00€5mg200.00€1mL*10mM (DMSO)220.00€10mg319.00€25mg528.00€50mg730.00€100mg999.00€200mg1,333.00€TPN171
CAS:TPN171 is potent PDE5 inhibitor with subnanomolar potency for PDE5 and good selectivity over PDE6, which has the potential for the treatment of pulmonary
Formula:C24H35N5O3Purity:>99.99%Color and Shape:SolidMolecular weight:441.57α-(difluoromethyl)-DL-Arginine
CAS:α-(difluoromethyl)-DL-Arginine (RMI 71897) is an enzyma-activated, irreversible inhibitor of arginine decarboxylase for E.Formula:C7H14F2N4O2Purity:99.77% - 99.78%Color and Shape:SolidMolecular weight:224.21STAT6-IN-2
CAS:STAT6-IN-2(R)-84 is a STAT6 inhibitor that inhibits the secretion of eotaxin-3 and the tyrosine phosphorylation of STAT6.Formula:C28H31N5O2Purity:99.67%Color and Shape:SolidMolecular weight:469.58H-1152 dihydrochloride
CAS:H-1152 2HCl: ROCK inhibitor, IC50=12 nM, Ki=1.6 nM. Blocks PKA, PKC, PKG, Aurora A, CaMKII with higher IC50s.Formula:C16H23Cl2N3O2SPurity:99.85%Color and Shape:SolidMolecular weight:392.34Ref: TM-T35328
1mg60.00€5mg135.00€1mL*10mM (DMSO)147.00€10mg215.00€25mg415.00€50mg655.00€100mg888.00€0990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormula:C21H21N5Purity:98.99%Color and Shape:SolidMolecular weight:343.42Ref: TM-T13983
1mg192.00€5mg485.00€1mL*10mM (DMSO)507.00€10mg700.00€25mg1,063.00€50mg1,459.00€100mg1,963.00€HBED-CC-tris(tert-butyl ester)
CAS:HBED-CC-tris(tert-butyl ester) is a monovalent variant of HBED-CC that can be used for tumor imaging.Formula:C38H56N2O10Purity:99.9%Color and Shape:SolidMolecular weight:700.859PP5-IN-1
CAS:PP5-IN-1 is a serine/threonine protein phosphatase-5 (PP5) inhibitor with potential anticancer activity that induces apoptosis in cancer cells.Formula:C18H18N2O3SPurity:99.13%Color and Shape:SolidMolecular weight:342.41RO5263397
CAS:RO5263397: TAAR1 agonist, orally active, studied as antidepressant, COX-2 inhibitor.Formula:C10H11FN2OPurity:98.58%Color and Shape:SolidMolecular weight:194.21PA452
CAS:PA452 is a selective antagonist of retinoic X receptor (RXR) and suppresses the effect of Retinoic acid on Th1/Th2 development.Formula:C26H37N3O3Purity:97.14%Color and Shape:SolidMolecular weight:439.59Ref: TM-T16425
1mg87.00€5mg236.00€1mL*10mM (DMSO)259.00€10mg380.00€25mg622.00€50mg888.00€100mg1,215.00€L-DABA hydrobromide
CAS:L-DABA hydrobromide (L-2,4-Diaminobutyric acid hydrobromide) , GABA transaminase inhibitor with antitumor and anticonvulsant activity.Formula:C4H11BrN2O2Purity:99.11%Color and Shape:SolidMolecular weight:199.05Lartesertib
CAS:Lartesertib (ATM Inhibitor-5) is an inhibitor of the serine/threonine protein kinase ATM with potential anticancer activity and can be used to study lung cancerFormula:C23H21FN6O3Purity:99.9%Color and Shape:SolidMolecular weight:448.45Ref: TM-T62684
1mg123.00€2mg177.00€5mg295.00€1mL*10mM (DMSO)326.00€10mg505.00€25mg982.00€50mg1,639.00€100mg2,538.00€CO23
CAS:CO23 is a blood-brain barrier penetrant and selective TRα agonist and can be used in studies about the regulation of growth and development.Formula:C19H18I2N2O4Purity:98.08%Color and Shape:SolidMolecular weight:592.17GW-803430
CAS:GW-803430: potent MCH R1 antagonist, pIC50=9.3, orally effective against obesity in animals.Formula:C25H24ClN3O3SPurity:98.07% - 98.97%Color and Shape:SolidMolecular weight:481.99Ranirestat
CAS:Ranirestat (AS-3201) is an AR inhibitor with neuroprotective properties that improves peripheral nerve dysfunction in rats with advanced diabetic polyneuropathyFormula:C17H11BrFN3O4Purity:96.10% - 99.44%Color and Shape:SolidMolecular weight:420.19Cis-N-Feruloyltyramine
CAS:Cis-N-Feruloyltyramine is a naturally occurring compound found in various plants that shows cytotoxicity against the P-388 cancer cell line.Formula:C18H19NO4Purity:97.43%Color and Shape:SolidMolecular weight:313.35LB42708
CAS:LB42708 is an orally active farnesyltransferase (FTase) inhibitor (IC50: 0.8/1.2/2.0 nM toward H/N/K-ras).Formula:C30H27BrN4O2Purity:99.36%Color and Shape:SolidMolecular weight:555.47Tenofovir amibufenamide
CAS:Tenofovir amibufenamide (HS-10234) 是一种 Tenofovir 前药，是一种具有口服活性的抗病毒化合物。Tenofovir amibufenamide 对乙型肝炎病毒 (HBV)具有抑制作用，可用于慢性乙型肝炎 (CHB) 研究。Formula:C22H31N6O5PPurity:99.19% - 99.87%Color and Shape:SolidMolecular weight:490.49KDM4-IN-4
CAS:KDM4-IN-4 is a KDM4 inhibitor with anticancer activity that inhibits the KDM4A-Tudor structural domain for cancer research.Formula:C16H23NOPurity:99.61%Color and Shape:SolidMolecular weight:245.36M2698
CAS:M2698 (MSC2363318A) is an inhibitor of p70S6K, Akt1 and Akt3 with IC50s of 1 nM. M2698 shows anti-cancer activity.Formula:C21H19ClF3N5OPurity:99.88%Color and Shape:SolidMolecular weight:449.86Ref: TM-T11928
1mg50.00€5mg105.00€1mL*10mM (DMSO)123.00€10mg170.00€25mg329.00€50mg475.00€100mg655.00€200mg883.00€Ertugliflozin L-pyroglutamic acid
CAS:Ertugliflozin is a potent oral hSGLT2 inhibitor (IC50: 0.877 nM) for type 2 diabetes treatment studies.Formula:C27H32ClNO10Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:566Ref: TM-T15244
5mg44.00€1mL*10mM (DMSO)50.00€10mg57.00€25mg85.00€50mg90.00€100mg133.00€200mg188.00€500mg323.00€Xinidamine
CAS:Xinidamine: antitumor agent for prostate hyperplasia, macular degeneration; inhibits PWR-1E cell growth, IC50=4μM.Formula:C17H16N2O2Purity:98.12%Color and Shape:SolidMolecular weight:280.32UC-764864
CAS:UC-764864, a UBE2N inhibitor, impedes the enzymatic activity of UBE2N and exhibits cytotoxic effects through the disruption of UBE2N-dependent signaling inFormula:C19H18N2OSPurity:99.3%Color and Shape:SolidMolecular weight:322.42TAK-020
CAS:TAK-020 is a potent covalent inhibitor of Btk with potential antitumor activity for the study of rheumatoid arthritis and immune-related diseases.Formula:C18H17N5O3Purity:98.66%Color and Shape:SolidMolecular weight:351.36Ref: TM-T9529
1mg138.00€5mg334.00€1mL*10mM (DMSO)358.00€10mg597.00€25mg1,234.00€50mg1,908.00€100mg2,952.00€Bupivacaine hydrochloride monohydrate
CAS:Bupivacaine hydrochloride monohydrate is an NMDA receptor inhibitor that inhibits SCN5A channels and is commonly used in the study of chronic pain.Formula:C18H31ClN2O2Purity:99.91%Color and Shape:SolidMolecular weight:342.9ST-1006
CAS:ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.Formula:C16H20Cl2N6Purity:99.96% - 99.98%Color and Shape:SolidMolecular weight:367.28Ref: TM-T34709
1mg86.00€1mL*10mM (DMSO)187.00€5mg188.00€10mg299.00€25mg487.00€50mg600.00€100mg743.00€200mg990.00€Roxifiban acetate
CAS:Roxifiban acetate（DMP 754 acetate） is a potent GP IIb / IIIa antagonist that exhibits antiplatelet aggregation activity via immune mediation and can be used inFormula:C23H33N5O8Purity:97.91% - 98.36%Color and Shape:SolidMolecular weight:507.54PAOPA
CAS:dopamine D2 receptor modulatorFormula:C11H18N4O3Purity:>99.99%Color and Shape:SolidMolecular weight:254.29Reldesemtiv
CAS:Reldesemtiv (CK-2127107) boosts exercise capacity, targeting fast muscle troponin, EC50 3.4 μM.Formula:C19H18F2N6OPurity:97.27%Color and Shape:SolidMolecular weight:384.38Toxoflavin
CAS:Toxoflavin (Xanthothricin) is an antagonist of transcription factor 4 (TCF4)/β-catenin complex. Toxoflavin also acts as an inhibitor of KDM4A.Formula:C7H7N5O2Purity:98.24% - 99.7%Color and Shape:SolidMolecular weight:193.16Didesmethyl cariprazine
CAS:Didesmethyl cariprazine, Cariprazine's active metabolite, treats schizophrenia/bipolar with D3/D2 affinity; half-life 1-3 weeks.Formula:C19H28Cl2N4OPurity:99.52%Color and Shape:SolidMolecular weight:399.36MB-07811
CAS:MB-07811 (VK-2809) is an orally active HepDirect prodrug of MB07344 with cholesterol and triglycerides lowering activity.Formula:C28H32ClO5PPurity:99.74% - 99.94%Color and Shape:SolidMolecular weight:514.98JNJ-42253432
CAS:JNJ-42253432 is an oral active P2X7 antagonist capable of penetrating the central nervous system with a pKi value of 9.1 for rat and 7.9 for human P2X7 channelsFormula:C28H38N4OPurity:99.98%Color and Shape:SolidMolecular weight:446.63Ref: TM-T27683
1mg73.00€5mg166.00€1mL*10mM (DMSO)182.00€10mg243.00€25mg376.00€50mg505.00€100mg668.00€200mg888.00€CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purity:99.40% - 99.58%Color and Shape:SolidMolecular weight:494.46Ref: TM-T30846
1mg315.00€5mg745.00€10mg1,018.00€25mg1,431.00€50mg1,783.00€100mg2,250.00€500mg4,410.00€Salicyl-AMS
CAS:Salicyl-AMS is an inhibitor of mycobacterium auxin biosynthesis that inhibits the growth of mycobacterium in the presence of iron deficiency in vitro.Formula:C17H18N6O8SPurity:98.19%Color and Shape:SolidMolecular weight:466.43Phos-tag Acrylamide AAL-107
CAS:Phos-tag Acrylamide AAL-107 is a polyacrylamide-conjugated phosphate-binding tag,visualizing phosphorylated proteins. High-Quality, Low-Cost!Formula:C33H38N8O3Purity:99.86% - >99.99%Color and Shape:SoildMolecular weight:594.71EGFR/ErbB-2 inhibitor-1
CAS:EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.Formula:C23H15ClFN3OS2Purity:98.93%Color and Shape:SolidMolecular weight:467.97LE135
CAS:LE135: RARα/RARβ antagonist (Ki: 1.4 μM/220 nM), favors RARβ, selective vs RARγ/RXRs; also activates TRPV1/TRPA1 (EC50s: 2.5/20 μM).Formula:C29H30N2O2Purity:97.94%Color and Shape:SolidMolecular weight:438.56Ref: TM-T22920
1mg44.00€2mg58.00€1mL*10mM (DMSO)92.00€5mg96.00€10mg128.00€25mg207.00€50mg308.00€100mg447.00€Ropsacitinib
CAS:Ropsacitinib (PF-06826647) is a selective TYK2 inhibitor, which binds to TYK2 catalytically active JH1 domain (IC50: 17 nM).Formula:C20H17N9Purity:99.87%Color and Shape:SolidMolecular weight:383.41HS94
CAS:HS94 (DAPK3 inhibitor HS94) is a selective and potent DAPK3 inhibitor with a Ki value of 126 nM for Pim kinase inhibition and can be used to study hypertension.
Formula:C15H15N5O2SPurity:95.04%Color and Shape:SolidMolecular weight:329.38Tefinostat
CAS:Tefinostat (CHR-2845) is a potent monocyte/macrophage-targeted histone deacetylase (HDAC) inhibitor.Formula:C28H37N3O5Purity:99.83%Color and Shape:SolidMolecular weight:495.61Ref: TM-T17028
1mg90.00€5mg215.00€1mL*10mM (DMSO)233.00€10mg319.00€25mg484.00€50mg640.00€100mg1,009.00€Ac-YVAD-AOM
CAS:Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.Formula:C33H42N4O10Purity:98%Color and Shape:SolidMolecular weight:654.71GW274150
CAS:GW274150: selective oral iNOS inhibitor (Kd=40 nM), low activity on eNOS/nNOS, protective in acute lung injury.Formula:C8H17N3O2SPurity:99.90%Color and Shape:SolidMolecular weight:219.3IMP-1710
CAS:IMP-1710 is a selective UCH-L1 inhibitor with an IC50 value of 38 nM in a fluorescence polarization assay.[1]Cost-effective and quality-assured.Formula:C23H19N5OPurity:99.3%Color and Shape:SolidMolecular weight:381.43KSQ-4279
CAS:KSQ-4279 (USP1-IN-1) is an inhibitor of USP1 and PARP.KSQ-4279 has anticancer activity and is used in the study of non-small cell lung cancer, osteosarcoma,Formula:C27H25F3N8OPurity:99.76% - 99.79%Color and Shape:SoildMolecular weight:534.54JAK-IN-3
CAS:JAK-IN-3 is a potent JAK inhibitor that inhibits JAK3, JAK1, TYK2, and JAK2, and can be used for the study of immune system disorders.Formula:C18H20N4O3Purity:98.04% - 98.19%Color and Shape:SolidMolecular weight:340.38Ref: TM-T11704
1mg126.00€2mg178.00€5mg304.00€1mL*10mM (DMSO)334.00€10mg492.00€25mg982.00€50mg1,558.00€100mg2,538.00€200mg3,402.00€
