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Neuroscience

Neuroscience

Neuroscience inhibitors are compounds designed to modulate the activity of specific proteins, enzymes, or receptors within the nervous system. These inhibitors are crucial for studying the molecular mechanisms underlying neural function, synaptic transmission, and neurodegenerative diseases. By targeting neurotransmitter receptors, ion channels, and signaling pathways, neuroscience inhibitors aid in the exploration of brain function and the development of therapeutic strategies for neurological disorders such as Alzheimer's, Parkinson's, and epilepsy. At CymitQuimica, we offer a comprehensive range of high-quality neuroscience inhibitors to support your research in neurobiology, neuropharmacology, and cognitive sciences.

Subcategories of "Neuroscience"

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Found 5389 products of "Neuroscience"

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  • Tasimelteon

    CAS:
    <p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>
    Formula:C15H19NO2
    Purity:98.93% - 99.93%
    Color and Shape:Solid
    Molecular weight:245.32
  • 4F 4PP oxalate

    CAS:
    <p>4F 4PP oxalate is a 5-HT2A antagonist.</p>
    Formula:C22H26FNO·C2H2O4
    Purity:97.34%
    Color and Shape:Solid
    Molecular weight:429.49
  • Aripiprazole monohydrate

    CAS:
    <p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>
    Formula:C23H29Cl2N3O3
    Color and Shape:Solid
    Molecular weight:466.4
  • NS3861

    CAS:
    <p>NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.</p>
    Formula:C12H14BrNS
    Purity:99.853%
    Color and Shape:Solid
    Molecular weight:284.22
  • MCI-225

    CAS:
    <p>MCI-225 is a selective inhibitor of NA reuptake with 5-HT3 receptor antagonism.</p>
    Formula:C17H17FN4S
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:328.4
  • Puerarin

    CAS:
    <p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>
    Formula:C21H20O9
    Purity:98.90% - 99.21%
    Color and Shape:Yellow Brown Fine Powder
    Molecular weight:416.38
  • JLK6

    CAS:
    <p>JLK6 was a gamma-secretase inhibitor that does not interfere with Notch signalling</p>
    Formula:C10H8ClNO3
    Purity:96.50%
    Color and Shape:Solid
    Molecular weight:225.63
  • SB 204741

    CAS:
    SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.
    Formula:C14H14N4OS
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:286.35
  • Tacrine hydrochloride (hydrate)

    CAS:
    <p>Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.</p>
    Formula:C13H14N2·XHCl·XH2O
    Purity:99.01% - 99.89%
    Color and Shape:Solid
    Molecular weight:234.72
  • FK 3311

    CAS:
    <p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>
    Formula:C15H13F2NO4S
    Purity:97.98%
    Color and Shape:Solid
    Molecular weight:341.33
  • Isocarboxazid

    CAS:
    <p>Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.</p>
    Formula:C12H13N3O2
    Purity:98.32% - 99.94%
    Color and Shape:Solid
    Molecular weight:231.25
  • Acotiamide monohydrochloride trihydrate

    CAS:
    <p>Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.</p>
    Formula:C21H37ClN4O8S
    Purity:98% - 99.54%
    Color and Shape:Solid
    Molecular weight:541.06
  • TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Formula:C23H23F3N2O4
    Purity:99.66% - ≥95%
    Color and Shape:Solid
    Molecular weight:448.43
  • CX516

    CAS:
    <p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>
    Formula:C14H15N3O
    Purity:99.04% - ≥95%
    Color and Shape:Tan Solid
    Molecular weight:241.29
  • p-Hydroxybenzaldehyde

    CAS:
    1.
    Formula:C7H6O2
    Purity:99.05% - 99.86%
    Color and Shape:Solid
    Molecular weight:122.12
  • Idalopirdine Hydrochloride

    CAS:
    <p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>
    Formula:C20H20ClF5N2O
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:434.83
  • GNE0877

    CAS:
    <p>GNE0877 (GNE 0877) is a highly effective and specific leucine-rich repeat kinase 2 (LRRK2) inhibitor (Ki: 0.7 nM).</p>
    Formula:C14H16F3N7
    Purity:98.01% - 99.97%
    Color and Shape:Solid
    Molecular weight:339.32
  • Loxapine hydrochloride

    CAS:
    <p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>
    Formula:C18H19Cl2N3O
    Color and Shape:Solid
    Molecular weight:364.27
  • NH125

    CAS:
    <p>NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, &gt;125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.</p>
    Formula:C27H45IN2
    Purity:98.60%
    Color and Shape:Solid
    Molecular weight:524.56
  • Mosapride Citrate

    CAS:
    <p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>
    Formula:C21H25ClFN3O3·C6H8O7
    Purity:99.70%
    Color and Shape:White Powder
    Molecular weight:614.02
  • Ondansetron hydrochloride

    CAS:
    <p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>
    Formula:C18H19N3O·HCl
    Purity:99.78%
    Color and Shape:White Powder
    Molecular weight:329.82
  • Dicyclomine

    CAS:
    <p>Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.</p>
    Formula:C19H35NO2
    Color and Shape:Solid
    Molecular weight:309.49
  • Dolasetron Mesylate hydrate

    CAS:
    <p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>
    Formula:C20H26N2O7S
    Purity:99.86% - 99.9%
    Color and Shape:Solid
    Molecular weight:438.49
  • Gabazine free base

    CAS:
    <p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>
    Formula:C15H17N3O3
    Color and Shape:Solid
    Molecular weight:287.31
  • Tandospirone hydrochloride

    CAS:
    <p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>
    Formula:C21H30ClN5O2
    Color and Shape:Solid
    Molecular weight:419.95
  • Trihexyphenidyl hydrochloride

    CAS:
    <p>Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.</p>
    Formula:C20H32ClNO
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:337.927
  • Harmine

    CAS:
    <p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>
    Formula:C13H12N2O
    Purity:98.29% - 99.92%
    Color and Shape:Off-White Solid
    Molecular weight:212.25
  • Ramosetron hydrochloride

    CAS:
    <p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>
    Formula:C17H18ClN3O
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:315.8
  • Sarpogrelate

    CAS:
    <p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>
    Formula:C24H31NO6
    Color and Shape:Solid
    Molecular weight:429.51
  • GNE-7915 tosylate

    CAS:
    <p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>
    Formula:C26H29F4N5O6S
    Color and Shape:Solid
    Molecular weight:615.6
  • LP-211

    CAS:
    LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and >300-fold selectivity over the 5-HT1A receptor.
    Formula:C30H34N4O
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:466.62
  • Acamprosate calcium

    CAS:
    Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
    Formula:C10H20CaN2O8S2
    Purity:98% - 99.93%
    Color and Shape:White Odorless Or Nearly Odorless Powder
    Molecular weight:400.48
  • PU02

    CAS:
    <p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>
    Formula:C16H12N4S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:292.36
  • Bitopertin

    CAS:
    <p>Bitopertin (Paliflutine) (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nM</p>
    Formula:C21H20F7N3O4S
    Purity:98.57% - 98.71%
    Color and Shape:Solid
    Molecular weight:543.46
  • S26131

    CAS:
    <p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>
    Formula:C31H34N2O4
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:498.61
  • (S)-Amisulpride

    CAS:
    (S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.
    Formula:C17H27N3O4S
    Purity:98.38%
    Color and Shape:Solid
    Molecular weight:369.48
  • CALP1 acetate


    <p>CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.</p>
    Formula:C42H79N9O12
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:902.13
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Formula:C14H30N2O4·2Cl·2H2O
    Purity:99.87%
    Color and Shape:White Solid
    Molecular weight:397.34
  • (-)-Dizocilpine maleate

    CAS:
    <p>(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.</p>
    Formula:C20H19NO4
    Purity:>99.99%
    Color and Shape:White Solid
    Molecular weight:337.37
  • TCN238

    CAS:
    <p>TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with an EC50 of 1 μM).</p>
    Formula:C12H11N3
    Purity:99.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:197.24
  • Eslicarbazepine Acetate

    CAS:
    <p>Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.</p>
    Formula:C17H16N2O3
    Purity:99.58% - >99.99%
    Color and Shape:White To Off-White Solid
    Molecular weight:296.32
  • ST034307

    CAS:
    <p>ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).</p>
    Formula:C10H4Cl4O2
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:297.95
  • 1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide

    CAS:
    <p>1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide is the inhibitor of human erythrocyte AChE.</p>
    Formula:C20H30Br2N2
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:458.27
  • Mofezolac

    CAS:
    <p>Mofezolac (formerly known as Disopain or N-22) is a highly selective COX-1 (cyclooxygenase-1) inhibitor with COXs selectivity index &gt; 6000</p>
    Formula:C19H17NO5
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:339.34
  • VU0467154

    CAS:
    <p>VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.</p>
    Formula:C17H15F3N4O3S2
    Purity:98.28% - 99.51%
    Color and Shape:Solid
    Molecular weight:444.45
  • Sarpogrelate hydrochloride

    CAS:
    <p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>
    Formula:C24H32ClNO6
    Purity:99.73%
    Color and Shape:Colorless Liquid
    Molecular weight:465.97
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Formula:C19H26ClNOS
    Purity:99.53% - 99.56%
    Color and Shape:Almost White To White Crystalline Powder
    Molecular weight:351.93
  • Almotriptan

    CAS:
    Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.
    Formula:C17H25N3O2S
    Purity:99.85%
    Color and Shape:Light Yellow Or White Power
    Molecular weight:335.46
  • (S)-Flurbiprofen

    CAS:
    <p>Esflurbiprofen is an inhibitor of COX-1 and COX-2.</p>
    Formula:C15H13FO2
    Purity:99.99%
    Color and Shape:White To Yellowish Crystalline Powder
    Molecular weight:244.26
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Formula:C21H29Cl2N3O4S
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:490.44
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Formula:C21H30N4O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:402.49
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Formula:C20H25N3O2
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:339.43
  • DNQX disodium salt

    CAS:
    <p>DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor</p>
    Formula:C8H2N4Na2O6
    Purity:98.93%
    Color and Shape:Solid
    Molecular weight:296.1
  • BPAM344

    CAS:
    BPAM344 is a potent positive allosteric modulator (PAM) of the KAR subunits GluK1b, GluK2a, and GluK3a.
    Formula:C10H11FN2O2S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:242.27
  • STO-609

    CAS:
    <p>STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.</p>
    Formula:C19H10N2O3
    Purity:97.14% - 98.8%
    Color and Shape:Solid
    Molecular weight:314.29
  • Gefapixant

    CAS:
    <p>Gefapixant (AF219) is a P2X3 receptor (P2X3R) antagonist with IC50 of ~30 nM at recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors</p>
    Formula:C14H19N5O4S
    Purity:99.28% - 99.50%
    Color and Shape:Solid
    Molecular weight:353.4
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Formula:C4H10N2
    Color and Shape:Solid
    Molecular weight:86.14
  • Eptapirone

    CAS:
    <p>Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.</p>
    Formula:C16H23N7O2
    Purity:99.39% - 99.65%
    Color and Shape:Solid
    Molecular weight:345.4
  • Rotigotine-

    CAS:
    <p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>
    Formula:C19H25NOS
    Purity:98.08% - 99.59%
    Color and Shape:Solid
    Molecular weight:315.47
  • Nor-benzetimide

    CAS:
    <p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>
    Formula:C16H20N2O2
    Purity:98.63%
    Color and Shape:Solid
    Molecular weight:272.34
  • Frovatriptan Succinate

    CAS:
    <p>Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.</p>
    Formula:C18H25N3O6
    Color and Shape:Solid
    Molecular weight:379.41
  • OXA (17-33) acetate


    <p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>
    Formula:C79H125N23O22
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:1748.98
  • Piperacetazine

    CAS:
    <p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>
    Formula:C24H30N2O2S
    Purity:99.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.57
  • NGB 2904

    CAS:
    <p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>
    Formula:C28H29Cl2N3O
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:494.46
  • Chlorprothixene

    CAS:
    <p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>
    Formula:C18H18ClNS
    Purity:98.77% - 99.756%
    Color and Shape:Pale Yellow Crystals Solid
    Molecular weight:315.86
  • MTEP hydrochloride

    CAS:
    <p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>
    Formula:C11H9ClN2S
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:236.72
  • 5-BDBD

    CAS:
    <p>5-BDBD is a potent and selective P2X4 receptor antagonist.</p>
    Formula:C17H11BrN2O2
    Purity:97.78%
    Color and Shape:Solid
    Molecular weight:355.19
  • FITM

    CAS:
    <p>FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).</p>
    Formula:C18H18FN5OS
    Purity:97.25%
    Color and Shape:Solid
    Molecular weight:371.43
  • Gabazine

    CAS:
    <p>Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)</p>
    Formula:C15H18BrN3O3
    Purity:98.51% - 99.24%
    Color and Shape:Solid
    Molecular weight:368.23
  • Tiprenolol

    CAS:
    <p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>
    Formula:C13H21NO2S
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:255.38
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Formula:C18H22Cl4N4
    Purity:97.52%
    Color and Shape:Solid
    Molecular weight:436.21
  • PNU-282987

    CAS:
    <p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>
    Formula:C14H18Cl2N2O
    Purity:99% - >99.99%
    Color and Shape:Solid
    Molecular weight:301.21
  • N-Desmethylclozapine

    CAS:
    N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.
    Formula:C17H17ClN4
    Purity:97.25% - 99.83%
    Color and Shape:Yellow Crystalline Solid
    Molecular weight:312.8
  • Pergolide mesylate

    CAS:
    <p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>
    Formula:C20H30N2O3S2
    Purity:99.70%
    Color and Shape:White To Off-White Solid
    Molecular weight:410.59
  • Guvacine hydrochloride

    CAS:
    <p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>
    Formula:C6H10ClNO2
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:163.602
  • Clozapine N-Oxide

    CAS:
    View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.
    Formula:C18H19ClN4O
    Purity:98.65% - 99.94%
    Color and Shape:Solid
    Molecular weight:342.82
  • Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Formula:C22H25ClN4O4S2
    Color and Shape:Solid
    Molecular weight:509.04
  • Dasotraline hydrochloride

    CAS:
    Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.
    Formula:C16H16Cl3N
    Purity:98.92% - 99.6%
    Color and Shape:Solid
    Molecular weight:328.66
  • CGP52432

    CAS:
    CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
    Formula:C15H24Cl2NO4P
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:384.24
  • 5-Benzyloxygramine

    CAS:
    5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
    Formula:C18H20N2O
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:280.36
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Formula:C6H6N2O2
    Purity:99.94%
    Color and Shape:Soild
    Molecular weight:138.1238
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Formula:C35H47FN10O8
    Purity:97.97%
    Color and Shape:Solid
    Molecular weight:754.85
  • AZ 11645373

    CAS:
    <p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>
    Formula:C24H21N3O5S
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:463.51
  • pep2-EVKI acetate(1315378-67-6 free base)


    <p>Pep2-EVKI acetate, a cell-permeable peptide, disrupts PICK1-GluR2 AMPA receptor binding.</p>
    Formula:C64H99N13O21
    Purity:97.63%
    Color and Shape:Solid
    Molecular weight:1386.55
  • SR 57227 hydrochloride

    CAS:
    <p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>
    Formula:C10H14ClN3·HCl
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:248.15
  • Lurasidone

    CAS:
    <p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>
    Formula:C28H36N4O2S
    Purity:99.78% - 99.91%
    Color and Shape:Solid
    Molecular weight:492.68
  • VUF 10166

    CAS:
    <p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>
    Formula:C13H15ClN4
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:262.74
  • 4-Acetamidobutanoic acid

    CAS:
    <p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>
    Formula:C6H11NO3
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:145.16
  • γ-Mangostin

    CAS:
    <p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>
    Formula:C23H24O6
    Purity:98.55% - 99.08%
    Color and Shape:Solid
    Molecular weight:396.43
  • Tariquidar

    CAS:
    <p>Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.</p>
    Formula:C38H38N4O6
    Purity:98.07% - 99.45%
    Color and Shape:Solid
    Molecular weight:646.73
  • Edonerpic maleate

    CAS:
    Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).
    Formula:C20H25NO6S
    Purity:98.24%
    Color and Shape:Solid
    Molecular weight:407.48
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Formula:C22H28BrN
    Purity:97.99%
    Color and Shape:Solid
    Molecular weight:386.37
  • AVN-492

    CAS:
    AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
    Formula:C17H21N5O2S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:359.45
  • Oxyphencyclimine Hydrochloride

    CAS:
    <p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>
    Formula:C20H29ClN2O3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:380.91
  • AC-90179 HCl

    CAS:
    <p>AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.</p>
    Formula:C23H31ClN2O2
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:402.96
  • Opiranserin hydrochloride

    CAS:
    <p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>
    Formula:C21H35ClN2O5
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:430.97
  • SB 242084 dihydrochloride

    CAS:
    SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.
    Formula:C21H21Cl3N4O2
    Color and Shape:Solid
    Molecular weight:467.78
  • NPS ALX Compound 4a

    CAS:
    NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)
    Formula:C25H25N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.55
  • MK 212 hydrochloride

    CAS:
    <p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>
    Formula:C8H11ClN4·HCl
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:235.12
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Formula:C14H17ClN2
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:248.75