
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(447 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
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Found 1045 products of "Proteases/Proteasome"
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Sucunamostat
CAS:<p>Sucunamostat is an L-aspartic acid enteropeptidase inhibitor.</p>Formula:C22H22N4O8Color and Shape:SolidMolecular weight:470.438MMP-9/10-IN-2
<p>MMP-9/10-IN-2 (compound 6e) serves as a potent inhibitor of MMP10 and MMP9, with an IC50 value for MMP10 at 0.076 μM and an inhibition concentration for MMP9 at 0.5 μM, achieving an inhibition rate of 93.18%. It plays a significant role in antitumor activities.</p>Formula:C17H12F3N5O3Color and Shape:SolidMolecular weight:391.3Cajaninstilbene acid
CAS:<p>Cajaninstilbene acid is a useful organic compound for research related to life sciences. The catalog number is T124035 and the CAS number is 87402-84-4.</p>Formula:C21H22O4Color and Shape:SolidMolecular weight:338.403Z-Leu-Leu-Tyr-COCHO
CAS:<p>Z-Leu-Leu-Tyr-COCHO is a potent inhibitor of chymotrypsin-like activity, exhibiting a Ki value of 3.0 nM [1].</p>Formula:C30H39N3O7Purity:98%Color and Shape:SolidMolecular weight:553.65Fibrinopeptide B, human
CAS:<p>Fibrinopeptide B (FPB) is produced during the cleavage of fibrinogen, by thrombin, to fibrin monomer.</p>Formula:C66H93N19O25Purity:98%Color and Shape:SolidMolecular weight:1552.56Cepeginterferon alfa-2b
CAS:<p>Cepeginterferon alfa-2b: pegylated interferon with 20 kDa PEG for HCV, PV, ET research.</p>Color and Shape:LiquidSL44
<p>SL44 is an agonist of human caseinolytic protease P (HsClpP) with an EC50 of 1.30 μM. It inhibits LM3 proliferation with an IC50 of 3.1 μM and induces apoptosis in liver cancer cells by degrading respiratory chain complex subunits. In mouse models, SL44 demonstrates antitumor activity without significant toxicity (LD50=400 mg/kg) and exhibits favorable pharmacokinetic properties in rat models.</p>Formula:C22H20ClFN4OMolecular weight:410.13097Dutogliptin tartrate
CAS:<p>Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>Formula:C14H26BN3O9Purity:98%Color and Shape:SolidMolecular weight:391.18AE-3763
CAS:<p>AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).</p>Formula:C23H34F3N5O7Purity:98%Color and Shape:SolidMolecular weight:549.54MK-6169
CAS:<p>MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.</p>Formula:C54H62FN9O8SPurity:98%Color and Shape:SolidMolecular weight:1016.2Tyrosinase-IN-15
<p>Tyrosinase-IN-15 (Compound 39), with an IC50 of 7.12 μM and a Ki of 11.8 μM, functions as a tyrosinase inhibitor [1].</p>Purity:98%Color and Shape:Odour SolidSofigatran
CAS:<p>Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.</p>Formula:C24H44N4O4SColor and Shape:SolidMolecular weight:484.7Elastatinal
CAS:<p>Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.</p>Formula:C21H36N8O7Color and Shape:Yellowish SolidMolecular weight:512.56JC-10
CAS:<p>JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.</p>Formula:C25H29Cl2IN4Purity:95%Color and Shape:SolidMolecular weight:583.34Linagliptin Methyldimer
CAS:<p>Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.</p>Formula:C50H56N16O4Purity:97.23%Color and Shape:SolidMolecular weight:945.08(Z)-SU14813
CAS:<p>(Z)-SU14813 is a tyrosine kinase inhibitor with anticardiogenic and antitumor activity.</p>Formula:C23H27FN4O4Purity:98.18%Color and Shape:SolidMolecular weight:442.48Ecallantide TFA
<p>Ecallantide (DX-88) TFA, a specific recombinant plasma kallikrein inhibitor, directly inhibits bradykinin production and is indicated for the prevention of</p>Color and Shape:Odour SolidL-Methionine-DL-sulfoximine
CAS:<p>MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.</p>Formula:C5H12N2O3SPurity:99.56% - ≥98%Color and Shape:White Crystalline PowderMolecular weight:180.23Z-Leu-Tyr-Chloromethylketone
CAS:<p>Z-Leu-Tyr-Chloromethylketone is a calpain inhibitor [1].</p>Formula:C24H29ClN2O5Color and Shape:SolidMolecular weight:460.95Proteasome-IN-7
<p>Proteasome-IN-7 (Compound 6f) is a macrolactam-based epoxyketone proteasome inhibitor with an IC50 value of 37.92 nM against the 20S proteasome ChT-L subunit. It exhibits potent antiproliferative effects on multiple myeloma, acute lymphoblastic leukemia, and non-small cell lung cancer.</p>Formula:C48H56N6O10SColor and Shape:SolidMolecular weight:909.06Sofosbuvir impurity A
CAS:<p>Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.</p>Formula:C22H29FN3O9PPurity:98%Color and Shape:SolidMolecular weight:529.45Recombinant Proteinase K
<p>Recombinant Proteinase K: serine protease, cleaves carboxy-terminus peptides, digests proteins, purifies nucleic acids.</p>Color and Shape:SolidCathepsin L-IN-3
CAS:<p>Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.</p>Formula:C41H49N7O4SColor and Shape:SolidMolecular weight:735.94VPLSLYSG
CAS:<p>VPLSLYSG, an octapeptide, degraded by MMP-9, MMP-1, MMP-2; potential MMP substrate uses.</p>Formula:C39H62N8O12Color and Shape:SolidMolecular weight:834.96STK33-IN-1
CAS:<p>STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.</p>Formula:C24H27N7O2Color and Shape:SolidMolecular weight:445.527TAPI1 acetate
<p>TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .</p>Formula:C28H41N5O7Purity:98.82% - 99.94%Color and Shape:SolidMolecular weight:559.65Z-Arg-Arg-βNA acetate
CAS:<p>Z-Arg-Arg-βNA acetate serves as a sensitive dipeptide substrate for Cathepsin B protease, while demonstrating resistance to proteases H and L. This compound is crucial for differentiating non-Cathepsin B type proteins.</p>Formula:C32H43N9O6Color and Shape:SolidMolecular weight:649.74TMC647055 Choline salt
<p>TMC647055 choline salt is a selective and cell-permeating inhibitor of HCV NS5B (IC50: 34 nM).</p>Formula:C37H53N5O8SPurity:98%Color and Shape:SolidMolecular weight:727.91Cathepsin C-IN-6
<p>Cathepsin C-IN-6 (compound 2), an E-64c-hydrazideas-derived inhibitor of cathepsin C, possesses anti-inflammatory properties and impedes neutrophil elastase</p>Formula:C24H35N5O4·xC2HF3O2Color and Shape:SolidGPLGLAGGWGERDGS
CAS:<p>GPLGLAGGWGERDGS is a polypeptide with MMP enzyme responsiveness and tumor-targeting properties, suitable for research on enzyme-guided nanoparticle assembly within tumors.</p>Formula:C61H93N19O21Color and Shape:SolidMolecular weight:1428.51GCPII-IN-1
CAS:<p>GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.</p>Formula:C12H21N3O7Color and Shape:SolidMolecular weight:319.314Neutrophil elastase inhibitor 4
<p>Neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (HNE) with IC50 of 42.30 nM and Ki of 8.04 nM.</p>Formula:C20H21N3O5Color and Shape:SolidMolecular weight:383.4SFTI-1
CAS:<p>SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.</p>Formula:C67H104N18O18S2Color and Shape:SolidMolecular weight:1513.78Pirmitegravir
CAS:<p>Pirmitegravir (STP0404) is a potent ALLINI, blocks LEDGF/p75 site, shows antiviral action against HIV.</p>Formula:C27H31ClN4O3Purity:99.79% - 99.79%Color and Shape:SolidMolecular weight:495.01Z-Gly-Pro-Phe-Leu-CHO
CAS:<p>Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde serving as a selective and potent proteasome inhibitor, demonstrating inhibition constants (Ki) of</p>Formula:C30H38N4O6Purity:98%Color and Shape:SolidMolecular weight:550.65TNO211
CAS:<p>TNO211 is a bioactive peptide that functions as a highly soluble fluorogenic substrate for select Matrix Metalloproteinases (MMPs)—specifically MMP-2, 8, 12, 13</p>Formula:C63H88N16O14SPurity:98%Color and Shape:SolidMolecular weight:1325.54Sofosbuvir impurity J
CAS:<p>Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formula:C22H30FN4O8PPurity:98%Color and Shape:SolidMolecular weight:528.47WYRGRL
CAS:<p>WYRGRL is a peptide that targets collagen II α1 (collagen II α1) through binding interaction. This short chondro-targeting peptide sequence enhances the targeting efficiency of peptide-functionalized nanoplatforms for cartilage in vivo, increasing it by approximately 72 times.</p>Formula:C40H59N13O8Color and Shape:SolidMolecular weight:849.98BMS 180742
CAS:<p>BMS 180742 is an exosite inhibitor of thrombin.</p>Formula:C67H93N11O22Purity:98%Color and Shape:SolidMolecular weight:1404.52Tilpisertib fosmecarbil TFA
CAS:<p>Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.</p>Formula:C37H37ClF3N8O9PColor and Shape:SolidMolecular weight:861.16Sofosbuvir impurity H
<p>Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.</p>Formula:C29H33FN3O10PPurity:98%Color and Shape:SolidMolecular weight:633.56Dansyl-Glu-Gly-Arg-Chloromethylketone
CAS:<p>Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activated</p>Formula:C26H36ClN7O7SColor and Shape:SolidMolecular weight:626.12Sofosbuvir impurity L
<p>Sofosbuvir impurity L is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formula:C22H29FN3O10PPurity:98%Color and Shape:SolidMolecular weight:545.45PF 00356231
CAS:<p>PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).</p>Formula:C25H20N2O3SPurity:99.35%Color and Shape:SolidMolecular weight:428.5CL 82198 hydrochloride
CAS:<p>CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.</p>Formula:C17H23ClN2O3Color and Shape:SolidMolecular weight:338.83EP 171
CAS:<p>EP 171 is a potent agonist of TP-receptors.</p>Formula:C23H29FO5Color and Shape:SolidMolecular weight:404.47MMP-9/MMP-13 Inhibitor I
CAS:<p>MMP-9/MMP-13 Inhibitor I is a dual inhibitor of MMP-9 and MMP-13 with IC50 of both 0.9 nM.</p>Formula:C25H25N3O6SColor and Shape:SolidMolecular weight:495.55AL-611
CAS:<p>AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).</p>Formula:C25H33F2N6O8PColor and Shape:SolidMolecular weight:614.544Cathepsin K inhibitor 7
<p>Cathepsin K Inhibitor7 (compound 7) is an inhibitor of Cathepsin K, exhibiting a pKi value of 7.3. It is utilized in research on osteoporosis.</p>Color and Shape:Odour SolidNostosin G
<p>Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).</p>Formula:C25H33N5O6Color and Shape:SolidMolecular weight:499.56Thrombin (MW 37kDa)
CAS:<p>Thrombin (MW 37kDa) is a trypsin-like allosteric serine protease.</p>Purity:98%Color and Shape:SolidMolecular weight:37kDaAPC-6860
CAS:<p>APC-6860, a serine protease inhibitor, targets multiple enzymes; most potent against human urokinase (Ki: 0.1 µM). Used in cancer research.</p>Formula:C9H7IN2SColor and Shape:SolidMolecular weight:302.13BPHA
CAS:<p>BPHA is a selective oral inhibitor of MMP-2/9/14 (IC50: 12/16/17 nM), not affecting MMP-1/3/7, with anti-angiogenic and anti-tumor properties.</p>Formula:C21H20N2O4SPurity:99.44%Color and Shape:SolidMolecular weight:396.46Obtusifolin-2-O-glucoside
CAS:<p>Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].</p>Formula:C22H22O10Color and Shape:SolidMolecular weight:446.4HCV-IN-7 hydrochloride
CAS:<p>HCV-IN-7 hydrochloride: Oral, potent HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.</p>Formula:C40H50Cl2N8O6SPurity:98%Color and Shape:SolidMolecular weight:841.85Sadopeptins B
<p>Sadopeptins B, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].</p>Formula:C48H69N9O13SColor and Shape:SolidMolecular weight:1012.18(Iso)-Fosdevirine
CAS:<p>(Iso)-Fosdevirine ( (Iso)-GSK2248761), a reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological diseases.</p>Formula:C20H17ClN3O3PPurity:99.93%Color and Shape:SoildMolecular weight:413.79PSI-353661
CAS:<p>PSI-353661 (GS-558093), inhibits HCV's NS5B polymerase; EC90: 8nM (wild-type), 11nM (S282T); active in human hepatocytes.</p>Formula:C24H32FN6O8PColor and Shape:SolidMolecular weight:582.52GSK2336805
CAS:<p>GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.</p>Formula:C42H52N8O8Color and Shape:SolidMolecular weight:796.91Cathepsin D and E FRET Substrate
CAS:<p>Mca-GKPILFFRL-Dpa-r-amide, FRET substrate for cathepsin D and E. Also cleaved by napsin A.</p>Formula:C85H122N22O19Color and Shape:SolidMolecular weight:1756.046Ledipasvir D-tartrate
CAS:<p>Ledipasvir D-tartrate (GS-5885 D-tartrate) is an HCV NS5A inhibitor that suppresses viral overphosphorylation and replication</p>Formula:C53H60F2N8O12Purity:99.83%Color and Shape:SolidMolecular weight:1039.09Clathrin-IN-1
CAS:<p>Pitstop 2 inhibits clathrin-mediated endocytosis, targeting clathrin's terminal domain, with potential in cancer research.</p>Formula:C20H13BrN2O3S2Purity:99.53%Color and Shape:SolidMolecular weight:473.36(-)-Sitagliptin Carbamoyl Glucuronide
CAS:<p>Minor phase II metabolite of DPP-4 inhibitor sitagliptin, found in rat and dog plasma.</p>Formula:C23H23F6N5O9Color and Shape:SolidMolecular weight:627.453Tyrosinase-IN-36
<p>Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.</p>Color and Shape:Odour SolidAcetyl-Calpastatin (184-210)(human) acetate
<p>Acetyl-Calpastatin acetate inhibits µ-calpain (Ki=0.2nM) and cathepsin L (Ki=6μM) selectively and reversibly.</p>Formula:C144H234N36O46SPurity:97.84% - 98.16%Color and Shape:SolidMolecular weight:3237.68Dazcapistat
CAS:<p>Dazcapistat is a potent calpain inhibitor, with IC50s of <3 μM for calpain 1, calpain 2 and calpain 9, respectively.</p>Formula:C21H18FN3O4Purity:99.11%Color and Shape:SolidMolecular weight:395.38CP-346086 dihydrate
CAS:<p>CP-346086 dihydrate is a strong oral MTP inhibitor with 2.0 nM IC50, reducing cholesterol and triglycerides in vivo.</p>Formula:C26H26F3N5O3Color and Shape:SolidMolecular weight:513.521MMP-3 Inhibitor acetate
<p>MMP-3 Inhibitor acetate is a cell-permeable and potent inhibitor of human MMP-3.</p>Formula:C29H50N10O11SPurity:98%Color and Shape:SolidMolecular weight:746.83Sofosbuvir impurity M
CAS:<p>Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formula:C22H30N3O10PPurity:98%Color and Shape:SolidMolecular weight:527.467Sofosbuvir impurity N
CAS:<p>Sofosbuvir impurity N is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formula:C20H25FN3O9PPurity:98%Color and Shape:SolidMolecular weight:501.404MMP-12 Inhibitor
CAS:<p>MMP-12 Inhibitor is a selective inhibitor of MMP-12 with IC50s of 2, 160, 320, and 22.3 nM for human, mouse, rat, and sheep MMP-12.</p>Formula:C19H20N2O7SPurity:97.51% - 99.96%Color and Shape:SoildMolecular weight:420.44α 1 Antichymotrypsin, Human Plasma
CAS:<p>Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.</p>Color and Shape:SolidSofosbuvir impurity I
<p>Sofosbuvir impurity I is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>Formula:C21H27FN3O9PPurity:98%Color and Shape:SolidMolecular weight:515.43ZG36
<p>ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrial</p>Color and Shape:Odour SolidTalabostat
CAS:<p>Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.</p>Formula:C9H19BN2O3Color and Shape:SolidMolecular weight:214.07Befovacimab
CAS:<p>Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.</p>Color and Shape:LiquidPentosan Polysulfate
CAS:<p>Pentosan Polysulfate: anti-HIV, anti-inflammatory, supports cartilage, treats interstitial cystitis.</p>Purity:98%Color and Shape:SolidMolecular weight:N/AMMP-9-IN-7
CAS:<p>N-[2-[(5-Cl-2-methoxyphenyl)amino]-4'-methyl[4,5'-bithiazol]-2'-yl]acetamide inhibits pro-MMP activation, treats MMP9/MMP13 syndromes.</p>Formula:C16H15ClN4O2S2Purity:97.35%Color and Shape:SolidMolecular weight:394.9Apovincamine
CAS:<p>Apovincamine is a vinca alkaloid and a chemical precursor of Vinpocetine, which is a derivative of Vincamine with vasodilating activity.</p>Formula:C21H24N2O2Purity:98%Color and Shape:SolidMolecular weight:336.44Ac-PAL-AMC
CAS:<p>Ac-PAL-AMC is a β1i/LMP2-specific substrate that fluoresces when cleaved; useful for measuring immunoproteasome activity.</p>Formula:C26H34N4O6Color and Shape:SolidMolecular weight:498.576,6′-Dihydroxythiobinupharidine
CAS:<p>6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-fold</p>Formula:C30H42N2O4SColor and Shape:SolidMolecular weight:526.73Z-FG-NHO-Bz
CAS:<p>Z-FG-NHO-Bz is a selective inhibitor of cathepsin [1].</p>Formula:C26H25N3O6Color and Shape:SolidMolecular weight:475.49Sadopeptins A
<p>Sadopeptins A, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].</p>Formula:C49H71N9O13SColor and Shape:SolidMolecular weight:1026.21Grazoprevir potassium salt
CAS:<p>Grazoprevir, a drug for hepatitis C, is a second-gen NS3/4a protease inhibitor.</p>Formula:C38H49KN6O9SColor and Shape:SolidMolecular weight:805Rivulariapeptolides 1155
<p>Rivulariapeptolides 1155 inhibits chymotrypsin (41.84 nM), elastase (4.94 nM), and proteinase K (56.54 nM).</p>Formula:C59H81N9O15Color and Shape:SolidMolecular weight:1156.33MeOSuc-AAPA-CMK
<p>MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].</p>Formula:C20H31ClN4O8Color and Shape:SolidMolecular weight:490.9415,16-Dihydrotanshindiol C
<p>15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.</p>Formula:C18H18O5Color and Shape:SolidMolecular weight:314.337HIV-1 Rev (34-50)
CAS:<p>HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) is a 17 amino acid peptide with anti-HIV-1 activity.</p>Formula:C97H173N51O24Purity:99.91%Color and Shape:SolidMolecular weight:2437.74PROTAC CG167
<p>PROTAC CG167 is a potent and selective PROTAC degrader of CypA. It degrades CypA in a dose-dependent manner in Jurkat cells, with a DC50 of 123 nM. Additionally, PROTAC CG167 exhibits antiviral activity by inhibiting HIV-1 and HCV. (Pink: CypA Ligand; Black: Linker; Blue: E3LigaseLigand)</p>Formula:C65H79N13O11SColor and Shape:SolidMolecular weight:1250.47H-Gly-Pro-Hyp-OH
CAS:<p>H-Gly-Pro-Hyp-OH is a potent and oral anti-photoaging collagen peptide and improves the hydration of human skin, elasticity and anti-wrinkle properties.</p>Formula:C12H19N3O5Purity:98.47%Color and Shape:SolidMolecular weight:285.35-epi-Arvestonate A
CAS:<p>5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.</p>Formula:C16H26O5Color and Shape:SolidMolecular weight:298.37VD2173
CAS:<p>VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.</p>Formula:C31H45N9O6SColor and Shape:SolidMolecular weight:671.81Bortezomib analog
<p>Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.</p>Color and Shape:Odour SolidNIM811
CAS:<p>NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.</p>Formula:C62H111N11O12Purity:98%Color and Shape:SolidMolecular weight:1202.635MMP Inhibitor 4
<p>MMP Inhibitor4 (compound 4 B) is an effective MMP inhibitor with anti-proliferative properties. It induces cell cycle arrest at the subG1 phase and reduces the mRNA expression of MMP2, MMP9, and VEGFA.</p>Formula:C16H18BrClN2O5Color and Shape:SolidMolecular weight:433.68Tyrosinase/elastase-IN-1
<p>Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastase</p>Formula:C33H52O5Color and Shape:SolidMolecular weight:528.76Iso-VQA-ACC acetate
<p>Iso-VQA-ACC acetate serves as a substrate for the constitutive proteasome.</p>Color and Shape:Odour SolidFFAGLDD
<p>"FFAGLDD: MMP9 peptide for controlled DOX delivery inside cells."</p>Formula:C37H49N7O12Purity:98%Color and Shape:SolidMolecular weight:783.82Hepcidin-1 (mouse)
CAS:<p>Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion.</p>Formula:C111H169N31O35S8Color and Shape:SolidMolecular weight:2754.24Leptosphaerodione
CAS:<p>Leptosphaerodione from Remotididymella sp.: a potent UPS inhibitor with 3.2 μM IC50 in HeLa cells; anti-tumor.</p>Formula:C21H22O5Color and Shape:SolidMolecular weight:354.4PROTAC 20S proteasome subunit β5 degrader 2
<p>PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.</p>Color and Shape:Odour SolidGSK2818713
CAS:<p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>Formula:C46H56N8O8Color and Shape:SolidMolecular weight:849.002Procizumab
<p>Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Color and Shape:Odour LiquidBI-1230
CAS:<p>BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.</p>Formula:C42H52N6O9SPurity:98%Color and Shape:SolidMolecular weight:816.96Ellipyrone B
<p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>Formula:C25H38O7Color and Shape:SolidMolecular weight:450.57MMP-3 Inhibitor
CAS:<p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>Formula:C27H46N10O9SPurity:98.87%Color and Shape:SolidMolecular weight:686.78HCV-IN-4
CAS:<p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>Formula:C52H58FN9O8Purity:98%Color and Shape:SolidMolecular weight:956.07DPP-4-IN-14
<p>DPP-4-IN-14 (compound 30) is an inhibitor of DPP-4, with an IC50 value of 12.82 nM.</p>Formula:C33H27N7O3Color and Shape:SolidMolecular weight:569.613HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Color and Shape:Odour SolidBictegravir Sodium
CAS:<p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>Formula:C21H17F3N3NaO5Purity:99.97%Color and Shape:SolidMolecular weight:471.36LXE408 fumarate
<p>LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.</p>Formula:C27H22FN7O6Purity:99.89%Color and Shape:SoildMolecular weight:559.51PS 915
CAS:<p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>Formula:C27H36ClN7O6Purity:98%Color and Shape:SolidMolecular weight:590.08Ichorcumab
CAS:<p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>Color and Shape:LiquidKKI-5
CAS:<p>KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.</p>Formula:C35H55N11O9Purity:98%Color and Shape:SolidMolecular weight:773.88Histargin
CAS:<p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>Formula:C14H25N7O4Color and Shape:SolidMolecular weight:355.39Relacatib
CAS:<p>Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.</p>Formula:C27H32N4O6SColor and Shape:SolidMolecular weight:540.64Tyrosinase-IN-38
<p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>Color and Shape:Odour SolidAristololactam IIIa
CAS:<p>Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.</p>Formula:C16H9NO4Color and Shape:SolidMolecular weight:279.25Tiprelestat
CAS:<p>Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.</p>Formula:C254H416N72O75S10Color and Shape:SolidMolecular weight:5999.09Lonodelestat TFA
<p>Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.</p>Formula:C73H112F3N15O21Color and Shape:SolidMolecular weight:1592.75Cathepsin D and E FRET Substrate acetate(839730-93-7 Free base)
<p>Fluorogenic substrate for cathepsins D & E; cleaves at Phe-Phe bond; not for B, H, L. Useful for assays and studies.</p>Color and Shape:Odour SolidParitaprevir dihydrate
CAS:<p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>Formula:C40H47N7O9SColor and Shape:SolidMolecular weight:801.91ADAM8-IN-1
CAS:<p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>Formula:C44H44Br4N6O12S2Color and Shape:SolidMolecular weight:1232.6Ac-Phe-Gly-pNA
CAS:<p>Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .</p>Formula:C19H20N4O5Color and Shape:SolidMolecular weight:384.39Sulodexide
CAS:<p>Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.</p>Color and Shape:SolidCerpegin
CAS:<p>Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.</p>Formula:C10H11NO3Color and Shape:SolidMolecular weight:193.2Carboxypeptidase C
CAS:<p>Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.</p>Color and Shape:SolidMMP-9-IN-6
CAS:<p>MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.</p>Formula:C25H19NO2Purity:99.75%Color and Shape:SoildMolecular weight:365.42VAMP
<p>VAMP is a tetrapeptide that acts as a competitive dipeptidyl peptidase IV (DPP-IV) inhibitor, exhibiting an IC50 of 1.00 μM and a Kd of 6.89 μM. It effectively targets the DPP-IV-GLP-1 axis and is utilized in the research of type 2 diabetes.</p>Formula:C18H32N4O5SColor and Shape:SolidMolecular weight:416.535Ala-Phe-Pro-pNA TFA
<p>Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.</p>Color and Shape:Odour SolidChymotrypsinogen
CAS:<p>Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .</p>Color and Shape:SolidCTTHWGFTLC, CYCLIC
CAS:<p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>Formula:C52H71N13O14S2Purity:98%Color and Shape:SolidMolecular weight:1166.33Alisporivir
CAS:<p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>Formula:C63H113N11O12Purity:99.95%Color and Shape:SolidMolecular weight:1216.64Histatin 5 TFA
<p>Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μM</p>Formula:C135H196N51F3O35Color and Shape:SolidMolecular weight:3150.31Acetyl-Calpastatin(184-210)(human) TFA
<p>Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.</p>Formula:C144H231F3N36O46SColor and Shape:SolidMolecular weight:3291.65Gly-Pro-pNA hydrochloride
CAS:<p>Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidase</p>Formula:C13H17ClN4O4Purity:99.84%Color and Shape:SolidMolecular weight:328.75Suc-AAP-Abu-pNA
CAS:<p>Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,</p>Formula:C25H34N6O9Color and Shape:SolidMolecular weight:562.57TR-107
CAS:<p>TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.</p>Formula:C22H19ClN4OColor and Shape:SoildMolecular weight:390.87LMP7/LMP2-IN-1
CAS:<p>LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.</p>Formula:C16H27BN4O3Color and Shape:SoildMolecular weight:334.22Anticancer agent 114
<p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>Formula:C28H33BF6N2O7Color and Shape:SolidMolecular weight:634.37Phepropeptin C
CAS:<p>Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with an IC50 of 12.5 μg/mL.</p>Formula:C38H60N6O6Color and Shape:SolidMolecular weight:696.92PD150606
CAS:<p>PD150606 is a calpain inhibitor with neuroprotective activity that inhibits μ-calpains and interferes with excitotoxicity-dependent motor neuron death.</p>Formula:C9H7IO2SPurity:98.19%Color and Shape:SolidMolecular weight:306.12TWH106
<p>TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.</p>Color and Shape:Odour SolidBMS-767778
CAS:<p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>Formula:C19H20Cl2N4O2Color and Shape:SolidMolecular weight:407.29Roseltide rT1
CAS:<p>Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.</p>Formula:C110H177N31O31S6Color and Shape:SolidMolecular weight:2622.16α 1(I) Collagen (614-639), human
CAS:<p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>Formula:C134H189N37O39Purity:98%Color and Shape:SolidMolecular weight:2942.16MMP-2 Inhibitor-4
<p>MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).</p>Formula:C19H23N3O5SColor and Shape:SolidMolecular weight:405.468NVP-DPP728 dihydrochloride
CAS:<p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>Formula:C15H20Cl2N6OColor and Shape:SolidMolecular weight:371.27RJS308
<p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>Formula:C63H75N13O11SColor and Shape:SolidMolecular weight:1222.42Stevia Powder
<p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>Color and Shape:Odour SolidPR 39 (porcine) acetate
<p>PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor.</p>Purity:98%Color and Shape:LiquidMolecular weight:N/A6-Acetylnimbandiol
CAS:<p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>Formula:C28H34O8Color and Shape:SolidMolecular weight:498.56Zetomipzomib maleate
CAS:<p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>Formula:C34H46N4O12Color and Shape:SolidMolecular weight:702.758Rivulariapeptolides 988
<p>Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).</p>Formula:C50H68N8O13Color and Shape:SolidMolecular weight:989.12L 659286
CAS:<p>L 659286 is one kind of cephalosporin derivative.</p>Formula:C17H21N5O7S2Color and Shape:SolidMolecular weight:471.51Pseudostellarin G
CAS:<p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>Formula:C42H56N8O9Color and Shape:SolidMolecular weight:816.94CRA-2059
CAS:<p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>Formula:C34H46N12O8Purity:97.68%Color and Shape:SolidMolecular weight:750.818Ellipyrone A
<p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>Formula:C25H34O8Color and Shape:SolidMolecular weight:462.53Leptosin D
CAS:<p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>Formula:C25H24N4O3S2Color and Shape:SolidMolecular weight:492.61Emtricitabine S-oxide
CAS:<p>Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.</p>Formula:C8H10FN3O4SPurity:98%Color and Shape:SolidMolecular weight:263.25Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS:<p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>Formula:C47H64N14O10Color and Shape:SolidMolecular weight:985.1Peptide 74
CAS:<p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>Formula:C62H107N23O20S2Purity:98%Color and Shape:SolidMolecular weight:1558.79Fotagliptin
CAS:<p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>Formula:C17H19FN6OColor and Shape:SolidMolecular weight:342.37Rivulariapeptolides 1121
<p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>Formula:C56H83N9O15Color and Shape:SolidMolecular weight:1122.31E-64d [for Biochemical Research]
CAS:Formula:C17H30N2O5Purity:>95.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:342.44CTS-1027
CAS:<p>CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has > 1,000 fold selectivity over MMP1.</p>Formula:C19H20ClNO6SColor and Shape:SolidMolecular weight:425.88Tenofovir hydrate
CAS:<p>Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.</p>Formula:C9H16N5O5PPurity:99.63%Color and Shape:SolidMolecular weight:305.23Ilomastat
CAS:Formula:C20H28N4O4Purity:>95.0%(HPLC)(qNMR)Color and Shape:White to Light yellow powder to crystalMolecular weight:388.47S-Methylglutathione
CAS:<p>S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.</p>Formula:C11H19N3O6SPurity:98%Color and Shape:SolidMolecular weight:321.35Retagliptin
CAS:<p>Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.</p>Formula:C19H18F6N4O3Color and Shape:SolidMolecular weight:464.36PSI-6206 13C,d3
CAS:<p>PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.</p>Formula:C10H13FN2O5Purity:98%Color and Shape:SolidMolecular weight:264.23Tripeptide-32
CAS:<p>Tripeptide-32 is a bioactive peptide recognized for its anti-aging properties, commonly utilized as an ingredient in cosmetics [1].</p>Formula:C12H22N4O5Purity:98%Color and Shape:SolidMolecular weight:302.33Glutaminase-IN-3
CAS:<p>Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.</p>Formula:C19H19F3N6O2SPurity:98.51%Color and Shape:SolidMolecular weight:452.45MMP-8 Inhibitor I
CAS:<p>MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.</p>Formula:C17H18N2O5SColor and Shape:SolidMolecular weight:362.4Tilpisertib
CAS:<p>Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).</p>Formula:C33H33ClN8OColor and Shape:SolidMolecular weight:593.13Teneligliptin hydrobromide hydrate
CAS:<p>Teneligliptin hydrobromide hydrate: potent, long-lasting DPP-4 inhibitor with ~1 nM IC50.</p>Formula:C22H33BrN6O2SColor and Shape:SolidMolecular weight:525.51Sitagliptin fenilalanil
CAS:<p>Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.</p>Formula:C25H24F6N6O2Color and Shape:SolidMolecular weight:554.49PKSI-527
CAS:<p>PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.</p>Formula:C25H32ClN3O4Color and Shape:SolidMolecular weight:473.99H-Arg-4MβNA
CAS:<p>H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.</p>Formula:C17H23N5O2Purity:99.98%Color and Shape:SolidMolecular weight:329.4BAY-677
CAS:<p>BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.</p>Formula:C20H15F3N4O2Color and Shape:SolidMolecular weight:400.355-Amino-8-hydroxyquinoline
CAS:<p>5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.</p>Formula:C9H8N2OPurity:99.69%Color and Shape:SolidMolecular weight:160.176-Chloro-7-deazapurine-2F-β-D-arabinofuranose
CAS:<p>6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.</p>Formula:C11H11ClFN3O3Color and Shape:SolidMolecular weight:287.67(Arg)9
CAS:<p>(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).</p>Formula:C54H110N36O10Color and Shape:SolidMolecular weight:1423.69Ubenimex Hydrochloride [for Biochemical Research]
CAS:Formula:C16H24N2O4·HClPurity:>97.0%(HPLC)Color and Shape:White to Almost white powder to crystalMolecular weight:344.84Dabigatran ethyl ester
CAS:<p>Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.</p>Formula:C27H29N7O3Purity:99.98%Color and Shape:SolidMolecular weight:499.56Saquinavir mesylate
CAS:<p>Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapy</p>Formula:C39H54N6O8SPurity:99.19%Color and Shape:White Or Pale Yellow PowderMolecular weight:766.9Teneligliptin D8
CAS:<p>Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.</p>Formula:C22H30N6OSPurity:98%Color and Shape:SolidMolecular weight:434.63PD-166793
CAS:<p>PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.</p>Formula:C17H18BrNO4SPurity:99.86%Color and Shape:SolidMolecular weight:412.3Tomeglovir
CAS:<p>Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).</p>Formula:C23H27N3O4SPurity:98%Color and Shape:SolidMolecular weight:441.54DMP 777
CAS:<p>DMP 777 is an orally active inhibitor of human leukocyte elastase.</p>Formula:C31H40N4O6Color and Shape:SolidMolecular weight:564.67Thrombin inhibitor 5
CAS:<p>Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.</p>Formula:C11H9FN4O3Purity:99.58%Color and Shape:SolidMolecular weight:264.21H-Pro-Lys-OH TFA
<p>H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.</p>Formula:C13H22F3N3O5Color and Shape:SolidMolecular weight:357.332'-β-C-Ethynyladenosine
CAS:<p>2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.</p>Formula:C12H13N5O4Color and Shape:SolidMolecular weight:291.26Sivelestat Sodium Tetrahydrate
CAS:Formula:C20H21N2NaO7S·4H2OPurity:>95.0%(T)(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:528.50Urokinase
CAS:<p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>Color and Shape:SolidPentosan Polysulfate Sodium (W/W 43%)
CAS:<p>Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.</p>Purity:98%Color and Shape:SolidMolecular weight:N/AAnguizole
CAS:<p>Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.</p>Formula:C17H11ClF2N4O2SColor and Shape:SolidMolecular weight:408.81Pepstatin A
CAS:Formula:C34H63N5O9Purity:>90.0%(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:685.90(-)-Gallocatechin Gallate
CAS:Formula:C22H18O11Purity:>95.0%(HPLC)Color and Shape:White to Light yellow powder to crystalMolecular weight:458.38Tanaproget
CAS:<p>Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.</p>Formula:C16H15N3OSPurity:98%Color and Shape:SolidMolecular weight:297.38


