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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1045 products of "Proteases/Proteasome"

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  • Sucunamostat

    CAS:
    <p>Sucunamostat is an L-aspartic acid enteropeptidase inhibitor.</p>
    Formula:C22H22N4O8
    Color and Shape:Solid
    Molecular weight:470.438
  • MMP-9/10-IN-2


    <p>MMP-9/10-IN-2 (compound 6e) serves as a potent inhibitor of MMP10 and MMP9, with an IC50 value for MMP10 at 0.076 μM and an inhibition concentration for MMP9 at 0.5 μM, achieving an inhibition rate of 93.18%. It plays a significant role in antitumor activities.</p>
    Formula:C17H12F3N5O3
    Color and Shape:Solid
    Molecular weight:391.3
  • Cajaninstilbene acid

    CAS:
    <p>Cajaninstilbene acid is a useful organic compound for research related to life sciences. The catalog number is T124035 and the CAS number is 87402-84-4.</p>
    Formula:C21H22O4
    Color and Shape:Solid
    Molecular weight:338.403
  • Z-Leu-Leu-Tyr-COCHO

    CAS:
    <p>Z-Leu-Leu-Tyr-COCHO is a potent inhibitor of chymotrypsin-like activity, exhibiting a Ki value of 3.0 nM [1].</p>
    Formula:C30H39N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.65
  • Fibrinopeptide B, human

    CAS:
    <p>Fibrinopeptide B (FPB) is produced during the cleavage of fibrinogen, by thrombin, to fibrin monomer.</p>
    Formula:C66H93N19O25
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1552.56
  • Cepeginterferon alfa-2b

    CAS:
    <p>Cepeginterferon alfa-2b: pegylated interferon with 20 kDa PEG for HCV, PV, ET research.</p>
    Color and Shape:Liquid
  • SL44


    <p>SL44 is an agonist of human caseinolytic protease P (HsClpP) with an EC50 of 1.30 μM. It inhibits LM3 proliferation with an IC50 of 3.1 μM and induces apoptosis in liver cancer cells by degrading respiratory chain complex subunits. In mouse models, SL44 demonstrates antitumor activity without significant toxicity (LD50=400 mg/kg) and exhibits favorable pharmacokinetic properties in rat models.</p>
    Formula:C22H20ClFN4O
    Molecular weight:410.13097
  • Dutogliptin tartrate

    CAS:
    <p>Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.</p>
    Formula:C14H26BN3O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.18
  • AE-3763

    CAS:
    <p>AE-3763 is a peptide-based human neutrophil elastase inhibitor (IC50: 29 nM).</p>
    Formula:C23H34F3N5O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:549.54
  • MK-6169

    CAS:
    <p>MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.</p>
    Formula:C54H62FN9O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1016.2
  • Tyrosinase-IN-15


    <p>Tyrosinase-IN-15 (Compound 39), with an IC50 of 7.12 μM and a Ki of 11.8 μM, functions as a tyrosinase inhibitor [1].</p>
    Purity:98%
    Color and Shape:Odour Solid
  • Sofigatran

    CAS:
    <p>Sofigatran (MCC-977) is an oral anticoagulant targeting thrombin for cardiovascular research.</p>
    Formula:C24H44N4O4S
    Color and Shape:Solid
    Molecular weight:484.7
  • Elastatinal

    CAS:
    <p>Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.</p>
    Formula:C21H36N8O7
    Color and Shape:Yellowish Solid
    Molecular weight:512.56
  • JC-10

    CAS:
    <p>JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.</p>
    Formula:C25H29Cl2IN4
    Purity:95%
    Color and Shape:Solid
    Molecular weight:583.34
  • Linagliptin Methyldimer

    CAS:
    <p>Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.</p>
    Formula:C50H56N16O4
    Purity:97.23%
    Color and Shape:Solid
    Molecular weight:945.08
  • (Z)-SU14813

    CAS:
    <p>(Z)-SU14813 is a tyrosine kinase inhibitor with anticardiogenic and antitumor activity.</p>
    Formula:C23H27FN4O4
    Purity:98.18%
    Color and Shape:Solid
    Molecular weight:442.48
  • Ecallantide TFA


    <p>Ecallantide (DX-88) TFA, a specific recombinant plasma kallikrein inhibitor, directly inhibits bradykinin production and is indicated for the prevention of</p>
    Color and Shape:Odour Solid
  • L-Methionine-DL-sulfoximine

    CAS:
    <p>MSO blocks glutamine synthetase, impacts astroglia, and is used in convulsant research.</p>
    Formula:C5H12N2O3S
    Purity:99.56% - ≥98%
    Color and Shape:White Crystalline Powder
    Molecular weight:180.23
  • Z-Leu-Tyr-Chloromethylketone

    CAS:
    <p>Z-Leu-Tyr-Chloromethylketone is a calpain inhibitor [1].</p>
    Formula:C24H29ClN2O5
    Color and Shape:Solid
    Molecular weight:460.95
  • Proteasome-IN-7


    <p>Proteasome-IN-7 (Compound 6f) is a macrolactam-based epoxyketone proteasome inhibitor with an IC50 value of 37.92 nM against the 20S proteasome ChT-L subunit. It exhibits potent antiproliferative effects on multiple myeloma, acute lymphoblastic leukemia, and non-small cell lung cancer.</p>
    Formula:C48H56N6O10S
    Color and Shape:Solid
    Molecular weight:909.06
  • Sofosbuvir impurity A

    CAS:
    <p>Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.</p>
    Formula:C22H29FN3O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.45
  • Recombinant Proteinase K


    <p>Recombinant Proteinase K: serine protease, cleaves carboxy-terminus peptides, digests proteins, purifies nucleic acids.</p>
    Color and Shape:Solid
  • Cathepsin L-IN-3

    CAS:
    <p>Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.</p>
    Formula:C41H49N7O4S
    Color and Shape:Solid
    Molecular weight:735.94
  • VPLSLYSG

    CAS:
    <p>VPLSLYSG, an octapeptide, degraded by MMP-9, MMP-1, MMP-2; potential MMP substrate uses.</p>
    Formula:C39H62N8O12
    Color and Shape:Solid
    Molecular weight:834.96
  • STK33-IN-1

    CAS:
    <p>STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.</p>
    Formula:C24H27N7O2
    Color and Shape:Solid
    Molecular weight:445.527
  • TAPI1 acetate


    <p>TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .</p>
    Formula:C28H41N5O7
    Purity:98.82% - 99.94%
    Color and Shape:Solid
    Molecular weight:559.65
  • Z-Arg-Arg-βNA acetate

    CAS:
    <p>Z-Arg-Arg-βNA acetate serves as a sensitive dipeptide substrate for Cathepsin B protease, while demonstrating resistance to proteases H and L. This compound is crucial for differentiating non-Cathepsin B type proteins.</p>
    Formula:C32H43N9O6
    Color and Shape:Solid
    Molecular weight:649.74
  • TMC647055 Choline salt


    <p>TMC647055 choline salt is a selective and cell-permeating inhibitor of HCV NS5B (IC50: 34 nM).</p>
    Formula:C37H53N5O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:727.91
  • Cathepsin C-IN-6


    <p>Cathepsin C-IN-6 (compound 2), an E-64c-hydrazideas-derived inhibitor of cathepsin C, possesses anti-inflammatory properties and impedes neutrophil elastase</p>
    Formula:C24H35N5O4·xC2HF3O2
    Color and Shape:Solid
  • GPLGLAGGWGERDGS

    CAS:
    <p>GPLGLAGGWGERDGS is a polypeptide with MMP enzyme responsiveness and tumor-targeting properties, suitable for research on enzyme-guided nanoparticle assembly within tumors.</p>
    Formula:C61H93N19O21
    Color and Shape:Solid
    Molecular weight:1428.51
  • GCPII-IN-1

    CAS:
    <p>GCPII-IN-1, a potent PSMA inhibitor, binds with 44.3 nM affinity.</p>
    Formula:C12H21N3O7
    Color and Shape:Solid
    Molecular weight:319.314
  • Neutrophil elastase inhibitor 4


    <p>Neutrophil elastase inhibitor 4 (compound 4f) is a competitive inhibitor of human neutrophil elastase (HNE) with IC50 of 42.30 nM and Ki of 8.04 nM.</p>
    Formula:C20H21N3O5
    Color and Shape:Solid
    Molecular weight:383.4
  • SFTI-1

    CAS:
    <p>SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.</p>
    Formula:C67H104N18O18S2
    Color and Shape:Solid
    Molecular weight:1513.78
  • Pirmitegravir

    CAS:
    <p>Pirmitegravir (STP0404) is a potent ALLINI, blocks LEDGF/p75 site, shows antiviral action against HIV.</p>
    Formula:C27H31ClN4O3
    Purity:99.79% - 99.79%
    Color and Shape:Solid
    Molecular weight:495.01
  • Z-Gly-Pro-Phe-Leu-CHO

    CAS:
    <p>Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde serving as a selective and potent proteasome inhibitor, demonstrating inhibition constants (Ki) of</p>
    Formula:C30H38N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:550.65
  • TNO211

    CAS:
    <p>TNO211 is a bioactive peptide that functions as a highly soluble fluorogenic substrate for select Matrix Metalloproteinases (MMPs)—specifically MMP-2, 8, 12, 13</p>
    Formula:C63H88N16O14S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1325.54
  • Sofosbuvir impurity J

    CAS:
    <p>Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C22H30FN4O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:528.47
  • WYRGRL

    CAS:
    <p>WYRGRL is a peptide that targets collagen II α1 (collagen II α1) through binding interaction. This short chondro-targeting peptide sequence enhances the targeting efficiency of peptide-functionalized nanoplatforms for cartilage in vivo, increasing it by approximately 72 times.</p>
    Formula:C40H59N13O8
    Color and Shape:Solid
    Molecular weight:849.98
  • BMS 180742

    CAS:
    <p>BMS 180742 is an exosite inhibitor of thrombin.</p>
    Formula:C67H93N11O22
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1404.52
  • Tilpisertib fosmecarbil TFA

    CAS:
    <p>Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.</p>
    Formula:C37H37ClF3N8O9P
    Color and Shape:Solid
    Molecular weight:861.16
  • Sofosbuvir impurity H


    <p>Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.</p>
    Formula:C29H33FN3O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:633.56
  • Dansyl-Glu-Gly-Arg-Chloromethylketone

    CAS:
    <p>Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activated</p>
    Formula:C26H36ClN7O7S
    Color and Shape:Solid
    Molecular weight:626.12
  • Sofosbuvir impurity L


    <p>Sofosbuvir impurity L is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C22H29FN3O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:545.45
  • PF 00356231

    CAS:
    <p>PF 00356231 is a selectivity inhibitor MMP-12 and can be used in studies about the treatment of emphysema and chronic obstructive pulmonary disease (COPD).</p>
    Formula:C25H20N2O3S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:428.5
  • CL 82198 hydrochloride

    CAS:
    <p>CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.</p>
    Formula:C17H23ClN2O3
    Color and Shape:Solid
    Molecular weight:338.83
  • EP 171

    CAS:
    <p>EP 171 is a potent agonist of TP-receptors.</p>
    Formula:C23H29FO5
    Color and Shape:Solid
    Molecular weight:404.47
  • MMP-9/MMP-13 Inhibitor I

    CAS:
    <p>MMP-9/MMP-13 Inhibitor I is a dual inhibitor of MMP-9 and MMP-13 with IC50 of both 0.9 nM.</p>
    Formula:C25H25N3O6S
    Color and Shape:Solid
    Molecular weight:495.55
  • AL-611

    CAS:
    <p>AL-611 is an HCV NS5B polymerase inhibitor ( EC 50 = 5 nM).</p>
    Formula:C25H33F2N6O8P
    Color and Shape:Solid
    Molecular weight:614.544
  • Cathepsin K inhibitor 7


    <p>Cathepsin K Inhibitor7 (compound 7) is an inhibitor of Cathepsin K, exhibiting a pKi value of 7.3. It is utilized in research on osteoporosis.</p>
    Color and Shape:Odour Solid
  • Nostosin G


    <p>Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).</p>
    Formula:C25H33N5O6
    Color and Shape:Solid
    Molecular weight:499.56
  • Thrombin (MW 37kDa)

    CAS:
    <p>Thrombin (MW 37kDa) is a trypsin-like allosteric serine protease.</p>
    Purity:98%
    Color and Shape:Solid
    Molecular weight:37kDa
  • APC-6860

    CAS:
    <p>APC-6860, a serine protease inhibitor, targets multiple enzymes; most potent against human urokinase (Ki: 0.1 µM). Used in cancer research.</p>
    Formula:C9H7IN2S
    Color and Shape:Solid
    Molecular weight:302.13
  • BPHA

    CAS:
    <p>BPHA is a selective oral inhibitor of MMP-2/9/14 (IC50: 12/16/17 nM), not affecting MMP-1/3/7, with anti-angiogenic and anti-tumor properties.</p>
    Formula:C21H20N2O4S
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:396.46
  • Obtusifolin-2-O-glucoside

    CAS:
    <p>Obtusifolin-2-O-glucoside (compound 7), a tyrosinase inhibitor with an IC50 value of 9.2 μM, can be isolated from cassia seed [1].</p>
    Formula:C22H22O10
    Color and Shape:Solid
    Molecular weight:446.4
  • HCV-IN-7 hydrochloride

    CAS:
    <p>HCV-IN-7 hydrochloride: Oral, potent HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.</p>
    Formula:C40H50Cl2N8O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:841.85
  • Sadopeptins B


    <p>Sadopeptins B, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].</p>
    Formula:C48H69N9O13S
    Color and Shape:Solid
    Molecular weight:1012.18
  • (Iso)-Fosdevirine

    CAS:
    <p>(Iso)-Fosdevirine ( (Iso)-GSK2248761), a reverse transcriptase (NNRTI) inhibitor with anti-HIV activity, is used in the study of neurological diseases.</p>
    Formula:C20H17ClN3O3P
    Purity:99.93%
    Color and Shape:Soild
    Molecular weight:413.79
  • PSI-353661

    CAS:
    <p>PSI-353661 (GS-558093), inhibits HCV's NS5B polymerase; EC90: 8nM (wild-type), 11nM (S282T); active in human hepatocytes.</p>
    Formula:C24H32FN6O8P
    Color and Shape:Solid
    Molecular weight:582.52
  • GSK2336805

    CAS:
    <p>GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.</p>
    Formula:C42H52N8O8
    Color and Shape:Solid
    Molecular weight:796.91
  • Cathepsin D and E FRET Substrate

    CAS:
    <p>Mca-GKPILFFRL-Dpa-r-amide, FRET substrate for cathepsin D and E. Also cleaved by napsin A.</p>
    Formula:C85H122N22O19
    Color and Shape:Solid
    Molecular weight:1756.046
  • Ledipasvir D-tartrate

    CAS:
    <p>Ledipasvir D-tartrate (GS-5885 D-tartrate) is an HCV NS5A inhibitor that suppresses viral overphosphorylation and replication</p>
    Formula:C53H60F2N8O12
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:1039.09
  • Clathrin-IN-1

    CAS:
    <p>Pitstop 2 inhibits clathrin-mediated endocytosis, targeting clathrin's terminal domain, with potential in cancer research.</p>
    Formula:C20H13BrN2O3S2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:473.36
  • (-)-Sitagliptin Carbamoyl Glucuronide

    CAS:
    <p>Minor phase II metabolite of DPP-4 inhibitor sitagliptin, found in rat and dog plasma.</p>
    Formula:C23H23F6N5O9
    Color and Shape:Solid
    Molecular weight:627.453
  • Tyrosinase-IN-36


    <p>Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.</p>
    Color and Shape:Odour Solid
  • Acetyl-Calpastatin (184-210)(human) acetate


    <p>Acetyl-Calpastatin acetate inhibits µ-calpain (Ki=0.2nM) and cathepsin L (Ki=6μM) selectively and reversibly.</p>
    Formula:C144H234N36O46S
    Purity:97.84% - 98.16%
    Color and Shape:Solid
    Molecular weight:3237.68
  • Dazcapistat

    CAS:
    <p>Dazcapistat is a potent calpain inhibitor, with IC50s of &lt;3 μM for calpain 1, calpain 2 and calpain 9, respectively.</p>
    Formula:C21H18FN3O4
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:395.38
  • CP-346086 dihydrate

    CAS:
    <p>CP-346086 dihydrate is a strong oral MTP inhibitor with 2.0 nM IC50, reducing cholesterol and triglycerides in vivo.</p>
    Formula:C26H26F3N5O3
    Color and Shape:Solid
    Molecular weight:513.521
  • MMP-3 Inhibitor acetate


    <p>MMP-3 Inhibitor acetate is a cell-permeable and potent inhibitor of human MMP-3.</p>
    Formula:C29H50N10O11S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:746.83
  • Sofosbuvir impurity M

    CAS:
    <p>Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C22H30N3O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.467
  • Sofosbuvir impurity N

    CAS:
    <p>Sofosbuvir impurity N is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C20H25FN3O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.404
  • MMP-12 Inhibitor

    CAS:
    <p>MMP-12 Inhibitor is a selective inhibitor of MMP-12 with IC50s of 2, 160, 320, and 22.3 nM for human, mouse, rat, and sheep MMP-12.</p>
    Formula:C19H20N2O7S
    Purity:97.51% - 99.96%
    Color and Shape:Soild
    Molecular weight:420.44
  • α 1 Antichymotrypsin, Human Plasma

    CAS:
    <p>Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.</p>
    Color and Shape:Solid
  • Sofosbuvir impurity I


    <p>Sofosbuvir impurity I is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.</p>
    Formula:C21H27FN3O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.43
  • ZG36


    <p>ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrial</p>
    Color and Shape:Odour Solid
  • Talabostat

    CAS:
    <p>Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.</p>
    Formula:C9H19BN2O3
    Color and Shape:Solid
    Molecular weight:214.07
  • Befovacimab

    CAS:
    <p>Befovacimab, a human IgG2 antibody, targets TFPI for hemophilia A/B research.</p>
    Color and Shape:Liquid
  • Pentosan Polysulfate

    CAS:
    <p>Pentosan Polysulfate: anti-HIV, anti-inflammatory, supports cartilage, treats interstitial cystitis.</p>
    Purity:98%
    Color and Shape:Solid
    Molecular weight:N/A
  • MMP-9-IN-7

    CAS:
    <p>N-[2-[(5-Cl-2-methoxyphenyl)amino]-4'-methyl[4,5'-bithiazol]-2'-yl]acetamide inhibits pro-MMP activation, treats MMP9/MMP13 syndromes.</p>
    Formula:C16H15ClN4O2S2
    Purity:97.35%
    Color and Shape:Solid
    Molecular weight:394.9
  • Apovincamine

    CAS:
    <p>Apovincamine is a vinca alkaloid and a chemical precursor of Vinpocetine, which is a derivative of Vincamine with vasodilating activity.</p>
    Formula:C21H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.44
  • Ac-PAL-AMC

    CAS:
    <p>Ac-PAL-AMC is a β1i/LMP2-specific substrate that fluoresces when cleaved; useful for measuring immunoproteasome activity.</p>
    Formula:C26H34N4O6
    Color and Shape:Solid
    Molecular weight:498.57
  • 6,6′-Dihydroxythiobinupharidine

    CAS:
    <p>6,6′-Dihydroxythiobinupharidine, a cysteine proteases inhibitor, amplifies DNA cleavage facilitated by human topoisomerase IIα and IIβ by approximately 8-fold</p>
    Formula:C30H42N2O4S
    Color and Shape:Solid
    Molecular weight:526.73
  • Z-FG-NHO-Bz

    CAS:
    <p>Z-FG-NHO-Bz is a selective inhibitor of cathepsin [1].</p>
    Formula:C26H25N3O6
    Color and Shape:Solid
    Molecular weight:475.49
  • Sadopeptins A


    <p>Sadopeptins A, a natural product isolated from Streptomyces sp., is a potent proteasome inhibitor [1].</p>
    Formula:C49H71N9O13S
    Color and Shape:Solid
    Molecular weight:1026.21
  • Grazoprevir potassium salt

    CAS:
    <p>Grazoprevir, a drug for hepatitis C, is a second-gen NS3/4a protease inhibitor.</p>
    Formula:C38H49KN6O9S
    Color and Shape:Solid
    Molecular weight:805
  • Rivulariapeptolides 1155


    <p>Rivulariapeptolides 1155 inhibits chymotrypsin (41.84 nM), elastase (4.94 nM), and proteinase K (56.54 nM).</p>
    Formula:C59H81N9O15
    Color and Shape:Solid
    Molecular weight:1156.33
  • MeOSuc-AAPA-CMK


    <p>MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].</p>
    Formula:C20H31ClN4O8
    Color and Shape:Solid
    Molecular weight:490.94
  • 15,16-Dihydrotanshindiol C


    <p>15,16-Dihydrotanshindiol C is a useful organic compound for research related to life sciences and the catalog number is T123985.</p>
    Formula:C18H18O5
    Color and Shape:Solid
    Molecular weight:314.337
  • HIV-1 Rev (34-50)

    CAS:
    <p>HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) is a 17 amino acid peptide with anti-HIV-1 activity.</p>
    Formula:C97H173N51O24
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:2437.74
  • PROTAC CG167


    <p>PROTAC CG167 is a potent and selective PROTAC degrader of CypA. It degrades CypA in a dose-dependent manner in Jurkat cells, with a DC50 of 123 nM. Additionally, PROTAC CG167 exhibits antiviral activity by inhibiting HIV-1 and HCV. (Pink: CypA Ligand; Black: Linker; Blue: E3LigaseLigand)</p>
    Formula:C65H79N13O11S
    Color and Shape:Solid
    Molecular weight:1250.47
  • H-Gly-Pro-Hyp-OH

    CAS:
    <p>H-Gly-Pro-Hyp-OH is a potent and oral anti-photoaging collagen peptide and improves the hydration of human skin, elasticity and anti-wrinkle properties.</p>
    Formula:C12H19N3O5
    Purity:98.47%
    Color and Shape:Solid
    Molecular weight:285.3
  • 5-epi-Arvestonate A

    CAS:
    <p>5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.</p>
    Formula:C16H26O5
    Color and Shape:Solid
    Molecular weight:298.37
  • VD2173

    CAS:
    <p>VD2173: a macrocyclic peptide that inhibits HGF serine proteases, matriptase, and hepsin, potentially for lung cancer research.</p>
    Formula:C31H45N9O6S
    Color and Shape:Solid
    Molecular weight:671.81
  • Bortezomib analog


    <p>Bortezomibanalog (Compound 13) is an analog of Bortezomib, functioning as an active control ligand for the 20S proteasome subunit β5.</p>
    Color and Shape:Odour Solid
  • NIM811

    CAS:
    <p>NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.</p>
    Formula:C62H111N11O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1202.635
  • MMP Inhibitor 4


    <p>MMP Inhibitor4 (compound 4 B) is an effective MMP inhibitor with anti-proliferative properties. It induces cell cycle arrest at the subG1 phase and reduces the mRNA expression of MMP2, MMP9, and VEGFA.</p>
    Formula:C16H18BrClN2O5
    Color and Shape:Solid
    Molecular weight:433.68
  • Tyrosinase/elastase-IN-1


    <p>Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastase</p>
    Formula:C33H52O5
    Color and Shape:Solid
    Molecular weight:528.76
  • Iso-VQA-ACC acetate


    <p>Iso-VQA-ACC acetate serves as a substrate for the constitutive proteasome.</p>
    Color and Shape:Odour Solid
  • FFAGLDD


    <p>"FFAGLDD: MMP9 peptide for controlled DOX delivery inside cells."</p>
    Formula:C37H49N7O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:783.82
  • Hepcidin-1 (mouse)

    CAS:
    <p>Hepcidin-1 (mouse) is a peptide hormone that regulates iron balance, elevates mRNA for TRAP, cathepsin K, and MMP-9, and promotes TRAP-5b protein secretion.</p>
    Formula:C111H169N31O35S8
    Color and Shape:Solid
    Molecular weight:2754.24
  • Leptosphaerodione

    CAS:
    <p>Leptosphaerodione from Remotididymella sp.: a potent UPS inhibitor with 3.2 μM IC50 in HeLa cells; anti-tumor.</p>
    Formula:C21H22O5
    Color and Shape:Solid
    Molecular weight:354.4
  • PROTAC 20S proteasome subunit β5 degrader 2


    <p>PROTAC 20S proteasome subunit β5 degrader 2 is a PROTAC degrader targeting the 20S proteasome subunit β5 (20Sproteasomesubunit β5), with a DC50 of 0.16 μM. It inhibits the proliferation of FaDu cancer cells, showcasing an IC50 of 0.23 μM. Additionally, PROTAC20Sproteasomesubunit β5 degrader 2 demonstrates antitumor activity in a mouse model.</p>
    Color and Shape:Odour Solid
  • GSK2818713

    CAS:
    <p>GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.</p>
    Formula:C46H56N8O8
    Color and Shape:Solid
    Molecular weight:849.002
  • Procizumab


    <p>Procizumab is a humanized IgG1 antibody that targets dipeptidyl peptidase 3 (DPP3). It shows potential for investigating sepsis. For the isotype control, refer to HumanIgG1kappa, Isotype Control.</p>
    Color and Shape:Odour Liquid
  • BI-1230

    CAS:
    <p>BI-1230 is a potent inhibitor of HCV NS3 protease, exhibiting efficacy in the low nanomolar range, and notably suppresses viral replication.</p>
    Formula:C42H52N6O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:816.96
  • Ellipyrone B


    <p>Ellipyrone B, a γ-pyrone-based macrocyclic polyketide with antihyperglycemic properties, demonstrates inhibitory activity against dipeptidyl peptidase-4 (IC 50</p>
    Formula:C25H38O7
    Color and Shape:Solid
    Molecular weight:450.57
  • MMP-3 Inhibitor

    CAS:
    <p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>
    Formula:C27H46N10O9S
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:686.78
  • HCV-IN-4

    CAS:
    <p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>
    Formula:C52H58FN9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:956.07
  • DPP-4-IN-14


    <p>DPP-4-IN-14 (compound 30) is an inhibitor of DPP-4, with an IC50 value of 12.82 nM.</p>
    Formula:C33H27N7O3
    Color and Shape:Solid
    Molecular weight:569.613
  • HIV-1 protease-IN-14


    <p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>
    Color and Shape:Odour Solid
  • Bictegravir Sodium

    CAS:
    <p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>
    Formula:C21H17F3N3NaO5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:471.36
  • LXE408 fumarate


    <p>LXE408 fumarate: orally available, selective kinetoplastid proteasome inhibitor with IC50/EC50 of 0.04 μM for L. donovani; potentially aids in VL research.</p>
    Formula:C27H22FN7O6
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:559.51
  • PS 915

    CAS:
    <p>PS 915 is a substrate for colorimetric assay. It was used for plasma antithrombin.</p>
    Formula:C27H36ClN7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.08
  • Ichorcumab

    CAS:
    <p>Ichorcumab (JNJ-375) is a fully human IgG4 antibody that targets thrombin. It binds to exosite 1 of thrombin, inhibiting substrate binding without affecting its catalytic activity. For isotype control, refer to HumanIgG1kappa, Isotype Control.</p>
    Color and Shape:Liquid
  • KKI-5

    CAS:
    <p>KKI 5: Serine protease inhibitor, blocks kallikrein &amp; plasmin, potential for cancer therapy &amp; angioedema treatment.</p>
    Formula:C35H55N11O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:773.88
  • Histargin

    CAS:
    <p>Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis.</p>
    Formula:C14H25N7O4
    Color and Shape:Solid
    Molecular weight:355.39
  • Relacatib

    CAS:
    <p>Relacatib (SB-462795) is a potent cathepsins K, L, V inhibitor with high affinity (Ki: 41-68 pM) and reduces bone resorption effectively.</p>
    Formula:C27H32N4O6S
    Color and Shape:Solid
    Molecular weight:540.64
  • Tyrosinase-IN-38


    <p>Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.</p>
    Color and Shape:Odour Solid
  • Aristololactam IIIa

    CAS:
    <p>Aristololactam IIIa inhibits superoxide and elastase generation; IC50: 0.12 μg/mL and 0.20 μg/mL.</p>
    Formula:C16H9NO4
    Color and Shape:Solid
    Molecular weight:279.25
  • Tiprelestat

    CAS:
    <p>Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.</p>
    Formula:C254H416N72O75S10
    Color and Shape:Solid
    Molecular weight:5999.09
  • Lonodelestat TFA


    <p>Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.</p>
    Formula:C73H112F3N15O21
    Color and Shape:Solid
    Molecular weight:1592.75
  • Cathepsin D and E FRET Substrate acetate(839730-93-7 Free base)


    <p>Fluorogenic substrate for cathepsins D &amp; E; cleaves at Phe-Phe bond; not for B, H, L. Useful for assays and studies.</p>
    Color and Shape:Odour Solid
  • Paritaprevir dihydrate

    CAS:
    <p>Paritaprevir dihydrate: potent oral HCV NS3/4A inhibitor (EC50: 0.21-1 nM), SARS-CoV-3CL blocker (IC50: 1.31 μM), metabolized by CYP3A, boosted by Ritonavir.</p>
    Formula:C40H47N7O9S
    Color and Shape:Solid
    Molecular weight:801.91
  • ADAM8-IN-1

    CAS:
    <p>ADAM8-IN-1 is a potent ADAM8 inhibitor with an IC 50 value of 73 nM.</p>
    Formula:C44H44Br4N6O12S2
    Color and Shape:Solid
    Molecular weight:1232.6
  • Ac-Phe-Gly-pNA

    CAS:
    <p>Ac-Phe-Gly-pNA is the chymotrypsin specific substrate [1] .</p>
    Formula:C19H20N4O5
    Color and Shape:Solid
    Molecular weight:384.39
  • Sulodexide

    CAS:
    <p>Sulodexide is an orally administered combination of glycosaminoglycans, consisting of low molecular weight heparin (80%) and dermatan sulfate (20%). It demonstrates antithrombotic properties by interacting with antithrombin III (AT III) and heparin cofactor II (HC II), and by inhibiting thrombin formation. Additionally, sulodexide enhances profibrinolytic activity by releasing tissue plasminogen activator (tPA). It also offers endothelial protection, possesses anti-inflammatory effects, and alleviates chronic venous disease.</p>
    Color and Shape:Solid
  • Cerpegin

    CAS:
    <p>Cerpegin, a pyridine ketone fused c-lactone, acts as an inhibitor of the 20S proteasome. It possesses pharmacological properties as a neuropsychiatric sedative, anti-inflammatory, analgesic, and exhibits anti-ulcer activity.</p>
    Formula:C10H11NO3
    Color and Shape:Solid
    Molecular weight:193.2
  • Carboxypeptidase C

    CAS:
    <p>Carboxypeptidase C removes COOH-terminal amino acids and others in peptides for biochemical studies.</p>
    Color and Shape:Solid
  • MMP-9-IN-6

    CAS:
    <p>MMP-9-IN-6: MMP-9 inhibitor, IC50 of 50 µM, anti-ulcer, potential anti-tumor, for tissue repair studies.</p>
    Formula:C25H19NO2
    Purity:99.75%
    Color and Shape:Soild
    Molecular weight:365.42
  • VAMP


    <p>VAMP is a tetrapeptide that acts as a competitive dipeptidyl peptidase IV (DPP-IV) inhibitor, exhibiting an IC50 of 1.00 μM and a Kd of 6.89 μM. It effectively targets the DPP-IV-GLP-1 axis and is utilized in the research of type 2 diabetes.</p>
    Formula:C18H32N4O5S
    Color and Shape:Solid
    Molecular weight:416.535
  • Ala-Phe-Pro-pNA TFA


    <p>Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.</p>
    Color and Shape:Odour Solid
  • Chymotrypsinogen

    CAS:
    <p>Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .</p>
    Color and Shape:Solid
  • CTTHWGFTLC, CYCLIC

    CAS:
    <p>CTT Gelatinase Inhibitor peptide blocks MMP-2/9, hindering cancer by stopping tumor growth.</p>
    Formula:C52H71N13O14S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1166.33
  • Alisporivir

    CAS:
    <p>Alisporivir (Debio-025) is a cyclophilin A inhibitor that disrupts the interaction between CypA and NS5A. HCV activity in vivo and in vitro.</p>
    Formula:C63H113N11O12
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:1216.64
  • Histatin 5 TFA


    <p>Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μM</p>
    Formula:C135H196N51F3O35
    Color and Shape:Solid
    Molecular weight:3150.31
  • Acetyl-Calpastatin(184-210)(human) TFA


    <p>Acetyl-Calpastatin(184-210)(human) TFA inhibits μ-calpain (Ki 0.2 nM) and cathepsin L (Ki 6 μM) selectively and reversibly.</p>
    Formula:C144H231F3N36O46S
    Color and Shape:Solid
    Molecular weight:3291.65
  • Gly-Pro-pNA hydrochloride

    CAS:
    <p>Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidase</p>
    Formula:C13H17ClN4O4
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:328.75
  • Suc-AAP-Abu-pNA

    CAS:
    <p>Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,</p>
    Formula:C25H34N6O9
    Color and Shape:Solid
    Molecular weight:562.57
  • TR-107

    CAS:
    <p>TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.</p>
    Formula:C22H19ClN4O
    Color and Shape:Soild
    Molecular weight:390.87
  • LMP7/LMP2-IN-1

    CAS:
    <p>LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.</p>
    Formula:C16H27BN4O3
    Color and Shape:Soild
    Molecular weight:334.22
  • Anticancer agent 114


    <p>Anticancer agent 114: oral dipeptide boronic acid, proteasome inhibitor, IC 50 = 2.2 nM, halts RPMI-8226 cell growth, for multiple myeloma research.</p>
    Formula:C28H33BF6N2O7
    Color and Shape:Solid
    Molecular weight:634.37
  • Phepropeptin C

    CAS:
    <p>Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with an IC50 of 12.5 μg/mL.</p>
    Formula:C38H60N6O6
    Color and Shape:Solid
    Molecular weight:696.92
  • PD150606

    CAS:
    <p>PD150606 is a calpain inhibitor with neuroprotective activity that inhibits μ-calpains and interferes with excitotoxicity-dependent motor neuron death.</p>
    Formula:C9H7IO2S
    Purity:98.19%
    Color and Shape:Solid
    Molecular weight:306.12
  • TWH106


    <p>TWH106 is an inhibitor of the cyclophilin (Cyp) enzyme, exhibiting strong affinity for CypA and CypB with dissociation constants (KD) of 53 nM and 139 nM, respectively. It effectively inhibits the replication of HIV and HCV, demonstrating antiviral activity.</p>
    Color and Shape:Odour Solid
  • BMS-767778

    CAS:
    <p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>
    Formula:C19H20Cl2N4O2
    Color and Shape:Solid
    Molecular weight:407.29
  • Roseltide rT1

    CAS:
    <p>Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.</p>
    Formula:C110H177N31O31S6
    Color and Shape:Solid
    Molecular weight:2622.16
  • α 1(I) Collagen (614-639), human

    CAS:
    <p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>
    Formula:C134H189N37O39
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2942.16
  • MMP-2 Inhibitor-4


    <p>MMP-2Inhibitor-4 (Compound 5g) is an MMP-2 inhibitor with an IC50 of 152.62 nM. It effectively reduces MMP-2 levels in K562 cell lines by stably binding to the active site of MMP-2 and exhibits strong anti-angiogenic effects in ACHN cell lines. MMP-2Inhibitor-4 shows potential for research in chronic myelogenous leukemia (CML).</p>
    Formula:C19H23N3O5S
    Color and Shape:Solid
    Molecular weight:405.468
  • NVP-DPP728 dihydrochloride

    CAS:
    <p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>
    Formula:C15H20Cl2N6O
    Color and Shape:Solid
    Molecular weight:371.27
  • RJS308


    <p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>
    Formula:C63H75N13O11S
    Color and Shape:Solid
    Molecular weight:1222.42
  • Stevia Powder


    <p>Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.</p>
    Color and Shape:Odour Solid
  • PR 39 (porcine) acetate


    <p>PR 39 (porcine) acetate is a noncompetitive, reversible and allosteric proteasome inhibitor.</p>
    Purity:98%
    Color and Shape:Liquid
    Molecular weight:N/A
  • 6-Acetylnimbandiol

    CAS:
    <p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>
    Formula:C28H34O8
    Color and Shape:Solid
    Molecular weight:498.56
  • Zetomipzomib maleate

    CAS:
    <p>Zetomipzomib maleate (KZR-616) selectively targets LMP7/2 in immunoproteasomes, potential for autoimmune research.</p>
    Formula:C34H46N4O12
    Color and Shape:Solid
    Molecular weight:702.758
  • Rivulariapeptolides 988


    <p>Rivulariapeptolides 988 inhibits serine proteases: chymotrypsin (IC50 = 95.46 nM), elastase (15.29 nM), proteinase K (85.50 nM).</p>
    Formula:C50H68N8O13
    Color and Shape:Solid
    Molecular weight:989.12
  • L 659286

    CAS:
    <p>L 659286 is one kind of cephalosporin derivative.</p>
    Formula:C17H21N5O7S2
    Color and Shape:Solid
    Molecular weight:471.51
  • Pseudostellarin G

    CAS:
    <p>Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.</p>
    Formula:C42H56N8O9
    Color and Shape:Solid
    Molecular weight:816.94
  • CRA-2059

    CAS:
    <p>CRA-2059 is a potent and selective inhibitor of tryptase, particularly targeting recombinant human tryptase-β (rHTβ), with a K i of 620 pM.</p>
    Formula:C34H46N12O8
    Purity:97.68%
    Color and Shape:Solid
    Molecular weight:750.818
  • Ellipyrone A


    <p>Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).</p>
    Formula:C25H34O8
    Color and Shape:Solid
    Molecular weight:462.53
  • Leptosin D

    CAS:
    <p>Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)</p>
    Formula:C25H24N4O3S2
    Color and Shape:Solid
    Molecular weight:492.61
  • Emtricitabine S-oxide

    CAS:
    <p>Emtricitabine treats HIV; its degradation byproduct is Emtricitabine S-oxide.</p>
    Formula:C8H10FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:263.25
  • Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2

    CAS:
    <p>Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effect</p>
    Formula:C47H64N14O10
    Color and Shape:Solid
    Molecular weight:985.1
  • Peptide 74

    CAS:
    <p>Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.</p>
    Formula:C62H107N23O20S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1558.79
  • Fotagliptin

    CAS:
    <p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>
    Formula:C17H19FN6O
    Color and Shape:Solid
    Molecular weight:342.37
  • Rivulariapeptolides 1121


    <p>Rivulariapeptolides 1121 inhibits serine proteases: chymotrypsin (IC50=35.52 nM), elastase (13.24 nM), proteinase K (48.05 nM).</p>
    Formula:C56H83N9O15
    Color and Shape:Solid
    Molecular weight:1122.31
  • E-64d [for Biochemical Research]

    CAS:
    Formula:C17H30N2O5
    Purity:>95.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:342.44

    Ref: 3B-E1337

    5mg
    127.00€
    25mg
    402.00€
  • CTS-1027

    CAS:
    <p>CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has &gt; 1,000 fold selectivity over MMP1.</p>
    Formula:C19H20ClNO6S
    Color and Shape:Solid
    Molecular weight:425.88
  • Tenofovir hydrate

    CAS:
    <p>Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.</p>
    Formula:C9H16N5O5P
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:305.23
  • Ilomastat

    CAS:
    Formula:C20H28N4O4
    Purity:>95.0%(HPLC)(qNMR)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:388.47

    Ref: 3B-I1202

    10mg
    189.00€
  • S-Methylglutathione

    CAS:
    <p>S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.</p>
    Formula:C11H19N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.35
  • Retagliptin

    CAS:
    <p>Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.</p>
    Formula:C19H18F6N4O3
    Color and Shape:Solid
    Molecular weight:464.36
  • PSI-6206 13C,d3

    CAS:
    <p>PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.</p>
    Formula:C10H13FN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.23
  • Tripeptide-32

    CAS:
    <p>Tripeptide-32 is a bioactive peptide recognized for its anti-aging properties, commonly utilized as an ingredient in cosmetics [1].</p>
    Formula:C12H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.33
  • Glutaminase-IN-3

    CAS:
    <p>Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.</p>
    Formula:C19H19F3N6O2S
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:452.45
  • MMP-8 Inhibitor I

    CAS:
    <p>MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.</p>
    Formula:C17H18N2O5S
    Color and Shape:Solid
    Molecular weight:362.4
  • Tilpisertib

    CAS:
    <p>Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).</p>
    Formula:C33H33ClN8O
    Color and Shape:Solid
    Molecular weight:593.13
  • Teneligliptin hydrobromide hydrate

    CAS:
    <p>Teneligliptin hydrobromide hydrate: potent, long-lasting DPP-4 inhibitor with ~1 nM IC50.</p>
    Formula:C22H33BrN6O2S
    Color and Shape:Solid
    Molecular weight:525.51
  • Sitagliptin fenilalanil

    CAS:
    <p>Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.</p>
    Formula:C25H24F6N6O2
    Color and Shape:Solid
    Molecular weight:554.49
  • PKSI-527

    CAS:
    <p>PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.</p>
    Formula:C25H32ClN3O4
    Color and Shape:Solid
    Molecular weight:473.99
  • H-Arg-4MβNA

    CAS:
    <p>H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.</p>
    Formula:C17H23N5O2
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:329.4
  • BAY-677

    CAS:
    <p>BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.</p>
    Formula:C20H15F3N4O2
    Color and Shape:Solid
    Molecular weight:400.35
  • 5-Amino-8-hydroxyquinoline

    CAS:
    <p>5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.</p>
    Formula:C9H8N2O
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:160.17
  • 6-Chloro-7-deazapurine-2F-β-D-arabinofuranose

    CAS:
    <p>6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.</p>
    Formula:C11H11ClFN3O3
    Color and Shape:Solid
    Molecular weight:287.67
  • (Arg)9

    CAS:
    <p>(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).</p>
    Formula:C54H110N36O10
    Color and Shape:Solid
    Molecular weight:1423.69
  • Ubenimex Hydrochloride [for Biochemical Research]

    CAS:
    Formula:C16H24N2O4·HCl
    Purity:>97.0%(HPLC)
    Color and Shape:White to Almost white powder to crystal
    Molecular weight:344.84

    Ref: 3B-B4000

    25mg
    196.00€
  • Dabigatran ethyl ester

    CAS:
    <p>Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.</p>
    Formula:C27H29N7O3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:499.56
  • Saquinavir mesylate

    CAS:
    <p>Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapy</p>
    Formula:C39H54N6O8S
    Purity:99.19%
    Color and Shape:White Or Pale Yellow Powder
    Molecular weight:766.9
  • Teneligliptin D8

    CAS:
    <p>Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.</p>
    Formula:C22H30N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.63
  • PD-166793

    CAS:
    <p>PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.</p>
    Formula:C17H18BrNO4S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:412.3
  • Tomeglovir

    CAS:
    <p>Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).</p>
    Formula:C23H27N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.54
  • DMP 777

    CAS:
    <p>DMP 777 is an orally active inhibitor of human leukocyte elastase.</p>
    Formula:C31H40N4O6
    Color and Shape:Solid
    Molecular weight:564.67
  • Thrombin inhibitor 5

    CAS:
    <p>Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.</p>
    Formula:C11H9FN4O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:264.21
  • H-Pro-Lys-OH TFA


    <p>H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.</p>
    Formula:C13H22F3N3O5
    Color and Shape:Solid
    Molecular weight:357.33
  • 2'-β-C-Ethynyladenosine

    CAS:
    <p>2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.</p>
    Formula:C12H13N5O4
    Color and Shape:Solid
    Molecular weight:291.26
  • Sivelestat Sodium Tetrahydrate

    CAS:
    Formula:C20H21N2NaO7S·4H2O
    Purity:>95.0%(T)(HPLC)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:528.50

    Ref: 3B-I1240

    25mg
    318.00€
  • Urokinase

    CAS:
    <p>Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.</p>
    Color and Shape:Solid
  • Pentosan Polysulfate Sodium (W/W 43%)

    CAS:
    <p>Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.</p>
    Purity:98%
    Color and Shape:Solid
    Molecular weight:N/A
  • Anguizole

    CAS:
    <p>Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.</p>
    Formula:C17H11ClF2N4O2S
    Color and Shape:Solid
    Molecular weight:408.81
  • Pepstatin A

    CAS:
    Formula:C34H63N5O9
    Purity:>90.0%(HPLC)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:685.90

    Ref: 3B-P3041

    10mg
    102.00€
  • (-)-Gallocatechin Gallate

    CAS:
    Formula:C22H18O11
    Purity:>95.0%(HPLC)
    Color and Shape:White to Light yellow powder to crystal
    Molecular weight:458.38

    Ref: 3B-G0628

    25mg
    290.00€
  • Tanaproget

    CAS:
    <p>Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.</p>
    Formula:C16H15N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.38