
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(34 products)
- Cysteine Protease(96 products)
- DPP-4(20 products)
- Glutaminase(40 products)
- HIV Protease(447 products)
- PAI-1(25 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(54 products)
- Proteasome(94 products)
- Serine Protease(50 products)
- p97(14 products)
Show 3 more subcategories
Found 1045 products of "Proteases/Proteasome"
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Avoralstat
CAS:<p>Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.</p>Formula:C28H27N5O5Purity:99.77%Color and Shape:SolidMolecular weight:513.54Benzoic acid, 4-[(aminoiminomethyl)amino]-, 6-(aminoiminomethyl)-2-naphthalenyl ester, dimethanesulfonate
CAS:Formula:C20H21N5O5SPurity:98%Color and Shape:SolidMolecular weight:443.4762Flanvotumab
CAS:<p>Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.</p>Purity:> 95%Color and Shape:LiquidMolecular weight:145.42 kDaDenagliptin
CAS:<p>Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study of</p>Formula:C20H18F3N3OPurity:99.12%Color and Shape:SolidMolecular weight:373.37Sofosbuvir impurity G
CAS:<p>Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.</p>Formula:C22H29FN3O9PPurity:98.04%Color and Shape:SolidMolecular weight:529.453-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-, methanesulfonate (1:1)
CAS:Formula:C33H49N3O7S2Purity:96%Color and Shape:SolidMolecular weight:663.8881(2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanamido]-4-methylpentanoic acid
CAS:Formula:C16H24N2O4Purity:98%Color and Shape:SolidMolecular weight:308.3728Ref: IN-DA00370Q
1g132.00€5g223.00€10g532.00€25gTo inquire50gTo inquire100gTo inquire10mg29.00€250gTo inquire100mg44.00€250mg68.00€Benzenemethanesulfonyl fluoride
CAS:Formula:C7H7FO2SPurity:99%Color and Shape:SolidMolecular weight:174.1927Ref: IN-DA00I6AP
1g25.00€5g39.00€10g55.00€1kgTo inquire25g93.00€2kgTo inquire50g137.00€5kgTo inquire100g181.00€250g572.00€Anisindione
CAS:<p>Anisindione, a synthetic indanedione, inhibits vitamin K, blocking factors II, VII, IX, X, and proteins C, S.</p>Formula:C16H12O3Purity:98.25%Color and Shape:Pale Yellow Crystals From Acetic Acid Or Ethanol SolidMolecular weight:252.263-Isoquinolinecarboxamide, N-(1,1-dimethylethyl)decahydro-2-[(2R,3R)-2-hydroxy-3-[(3-hydroxy-2-methylbenzoyl)amino]-4-(phenylthio)butyl]-, (3S,4aS,8aS)-
CAS:Formula:C32H45N3O4SPurity:98%Color and Shape:SolidMolecular weight:567.7824Q-VD-OPH
CAS:<p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>Formula:C26H25F2N3O6Purity:97.8% - 98.95%Color and Shape:SolidMolecular weight:513.54-Chlorosalicylic acid
CAS:<p>4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) is antimicrobial compositions comprising a metal salt and a benzoic acid analog</p>Formula:C7H5ClO3Purity:98.59%Color and Shape:Off-White To Light Beige PowderMolecular weight:172.57BLT-1
CAS:<p>BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.</p>Formula:C12H23N3SPurity:97.97%Color and Shape:SolidMolecular weight:241.4Elsulfavirine
CAS:<p>Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.</p>Formula:C24H17BrCl2FN3O5SPurity:99.66%Color and Shape:SolidMolecular weight:629.28MK-0608
CAS:<p>MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).</p>Formula:C12H16N4O4Purity:98.48%Color and Shape:SolidMolecular weight:280.28Fostemsavir Tris
CAS:<p>Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.</p>Formula:C29H37N8O11PPurity:99.45%Color and Shape:SolidMolecular weight:704.62Fenofibric acid
CAS:<p>Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate with antihyperlipidemic activity.</p>Formula:C17H15ClO4Purity:99.36%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:318.75Dolutegravir intermediate-1
CAS:<p>Dolutegravir intermediate-1 is a synthetic precursor for HIV-1 treatment from patent WO 2016125192 A2.</p>Formula:C13H17NO8Purity:99.52%Color and Shape:SolidMolecular weight:315.28Ruzasvir
CAS:<p>Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.</p>Formula:C49H55FN10O7SPurity:96.87% - 96.88%Color and Shape:SolidMolecular weight:947.09Mecarbinate
CAS:<p>Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.</p>Formula:C13H15NO3Purity:99.28%Color and Shape:Off-White Crystalline PowderMolecular weight:233.26Trelagliptin
CAS:<p>Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.</p>Formula:C18H20FN5O2Purity:98.88%Color and Shape:SolidMolecular weight:357.38Retagliptin Phosphate
CAS:<p>Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.</p>Formula:C19H21F6N4O7PPurity:98.70%Color and Shape:SolidMolecular weight:562.36L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Formula:C26H41N3O5Purity:98%Color and Shape:SolidMolecular weight:475.6208LSP-249
CAS:<p>LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.</p>Formula:C24H22ClN5OPurity:99.51%Color and Shape:SolidMolecular weight:431.92LDN-27219
CAS:<p>LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.</p>Formula:C20H16N4O2S2Purity:99.01% - 99.38%Color and Shape:SolidMolecular weight:408.5Begelomab
CAS:<p>Begelomab (SAND-26) is a mouse-derived monoclonal antibody targeting DPP-4/CD26. Begelomab can be used to study severe refractory inflammatory myopathies.</p>Purity:97.8% (SDS-PAGE); 98.3% (SEC-HPLC) - 97.8% (SDS-PAGE); 98.3% (SEC-HPLC)Color and Shape:LiquidSalicylanilide
CAS:<p>Salicylanilide (2-Hydroxybenzanilide)s are a group of compounds with antiviral potency, antibacterial and antifungal activities.</p>Formula:C13H11NO2Purity:99.55%Color and Shape:White To Off-White Crystalline PowderMolecular weight:213.233-Deazaadenosine hydrochloride
CAS:<p>3-Deazaadenosine HCl blocks SAH hydrolase (Ki: 3.9 μM), with anti-inflammatory, anti-proliferative, and anti-HIV effects.</p>Formula:C11H15ClN4O4Purity:98.48%Color and Shape:SolidMolecular weight:302.71Sitagliptin
CAS:<p>Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.</p>Formula:C16H15F6N5OPurity:99.33% - 99.83%Color and Shape:Yellow GreaseMolecular weight:407.31Probenecid
CAS:<p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>Formula:C13H19NO4SPurity:98.95% - 99.84%Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Molecular weight:285.36ARP-100
CAS:<p>ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).</p>Formula:C17H20N2O5SPurity:97.18%Color and Shape:SolidMolecular weight:364.42BRD-6929
CAS:<p>BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.</p>Formula:C19H17N3O2SPurity:98.01% - 99.05%Color and Shape:SolidMolecular weight:351.42Hck-IN-1
CAS:<p>Hck-IN-1 selectively inhibits Nef:Hck, IC50: 2.8 μM; >20 μM for Hck alone. Potent HIV-1 Nef antagonist, IC50: 100-300 nM for HIV-1 replication.</p>Formula:C16H11ClN6O3SPurity:99.07%Color and Shape:SolidMolecular weight:402.81PF-3450074
CAS:<p>PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.</p>Formula:C27H27N3O2Purity:99.92%Color and Shape:SolidMolecular weight:425.52RA190
CAS:<p>RA190 inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.</p>Formula:C28H23Cl5N2O2Purity:97.7%Color and Shape:SolidMolecular weight:596.76RAMB4
CAS:<p>RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.</p>Formula:C19H13Cl4NOPurity:98.89% - 99.38%Color and Shape:SolidMolecular weight:413.12GSK2838232
CAS:<p>GSK2838232 inhibit HIV reverse transcriptase activity across a broad panel of HIV-1 isolates,GSK2838232 is novel human immune virus (HIV) maturation inhibitor.</p>Formula:C48H73ClN2O6Purity:97.97%Color and Shape:SolidMolecular weight:809.56DBPR108
CAS:<p>DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9.</p>Formula:C16H25FN4O2Purity:99.68%Color and Shape:SolidMolecular weight:324.393-Aminopropionitrile fumarate (2:1)
CAS:<p>3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.</p>Formula:C4H4O4·2C3H6N2Purity:99.76% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:256.262-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Formula:C17H30N2O5Purity:98%Color and Shape:SolidMolecular weight:342.4305Islatravir
CAS:<p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>Formula:C12H12FN5O3Purity:98.77%Color and Shape:SolidMolecular weight:293.25Sofosbuvir impurity F
CAS:<p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>Formula:C34H45FN4O13P2Purity:98.05%Color and Shape:SolidMolecular weight:798.69Bivalirudin acetate
<p>Bivalirudin acetate is a thrombin inhibitor, a peptide-based anticoagulant, used for research on acute coronary syndrome.</p>Formula:C100H142N24O35Purity:99.84%Color and Shape:SolidMolecular weight:2240.34BJJF078
CAS:<p>BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.</p>Formula:C27H29N3O6SPurity:98.19%Color and Shape:SoildMolecular weight:523.6Aprotinin
CAS:<p>Aprotinin (Traskolan) is a broad-spectrum serine protease (BPTI) inhibitor. Aprotinin is an antifibrinolytic agent. Cost-effective and quality-assured.</p>Formula:C284H432N84O79S7Purity:98%Color and Shape:SolidMolecular weight:6511.516-Acetylnimbandiol
CAS:<p>6-Acetylnimbandiol, a non-toxic agent, inhibits tyrosinase (IC50=69.85 μM), melanin, and MITF; useful in melanoma studies.</p>Formula:C28H34O8Color and Shape:SolidMolecular weight:498.56α 1(I) Collagen (614-639), human
CAS:<p>This is a peptide inhibitor of collagen fibrillar matrix assembly.</p>Formula:C134H189N37O39Purity:98%Color and Shape:SolidMolecular weight:2942.16EP 171
CAS:<p>EP 171 is a potent agonist of TP-receptors.</p>Formula:C23H29FO5Color and Shape:SolidMolecular weight:404.47Berotralstat
CAS:<p>Berotralstat (BCX7353) is an oral, low-toxicity, specific kallikrein inhibitor for hereditary angioedema research, blocking bradykinin release.</p>Formula:C30H26F4N6OColor and Shape:SolidMolecular weight:562.56


