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Proteases/Proteasome

Proteases/Proteasome

Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.

Subcategories of "Proteases/Proteasome"

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Found 1079 products of "Proteases/Proteasome"

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  • MK-0608

    CAS:
    MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).
    Formula:C12H16N4O4
    Purity:98.48%
    Color and Shape:Solid
    Molecular weight:280.28
  • Trelagliptin

    CAS:
    Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.
    Formula:C18H20FN5O2
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:357.38
  • Sitagliptin

    CAS:
    Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.
    Formula:C16H15F6N5O
    Purity:99.33% - 99.83%
    Color and Shape:Yellow Grease
    Molecular weight:407.31
  • Elsulfavirine

    CAS:
    Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.
    Formula:C24H17BrCl2FN3O5S
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:629.28
  • LDN-27219

    CAS:
    <p>LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.</p>
    Formula:C20H16N4O2S2
    Purity:99.01% - 99.38%
    Color and Shape:Solid
    Molecular weight:408.5
  • RAMB4

    CAS:
    RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.
    Formula:C19H13Cl4NO
    Purity:98.89% - 99.38%
    Color and Shape:Solid
    Molecular weight:413.12
  • Sofosbuvir impurity G

    CAS:
    Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.
    Formula:C22H29FN3O9P
    Purity:98.04%
    Color and Shape:Solid
    Molecular weight:529.45
  • BJJF078

    CAS:
    <p>BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.</p>
    Formula:C27H29N3O6S
    Purity:98.19%
    Color and Shape:Soild
    Molecular weight:523.6
  • BRD-6929

    CAS:
    BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.
    Formula:C19H17N3O2S
    Purity:98.01% - 99.05%
    Color and Shape:Solid
    Molecular weight:351.42
  • Islatravir

    CAS:
    <p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>
    Formula:C12H12FN5O3
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:293.25
  • Probenecid

    CAS:
    <p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>
    Formula:C13H19NO4S
    Purity:98.95% - 99.84%
    Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)
    Molecular weight:285.36
  • Ruzasvir

    CAS:
    <p>Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.</p>
    Formula:C49H55FN10O7S
    Purity:96.87% - 96.88%
    Color and Shape:Solid
    Molecular weight:947.09
  • LSP-249

    CAS:
    <p>LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.</p>
    Formula:C24H22ClN5O
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:431.92
  • ML604440

    CAS:
    ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.
    Formula:C17H24BF3N2O4
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:388.19
  • Q-VD-OPH

    CAS:
    <p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>
    Formula:C26H25F2N3O6
    Purity:97.8% - 98.95%
    Color and Shape:Solid
    Molecular weight:513.5
  • Ref: IN-DA0048C1

    1mg
    50.00€
    5mg
    50.00€
    25mg
    155.00€
    50mg
    197.00€
    100mg
    331.00€
    250mg
    531.00€
  • Ref: IN-DA0072SK

    1g
    To inquire
    5mg
    68.00€
    10mg
    90.00€
    25mg
    124.00€
    50mg
    168.00€
    100mg
    229.00€
    250mg
    500.00€
  • Avoralstat

    CAS:
    Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.
    Formula:C28H27N5O5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:513.54
  • Mecarbinate

    CAS:
    <p>Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.</p>
    Formula:C13H15NO3
    Purity:99.28%
    Color and Shape:Off-White Crystalline Powder
    Molecular weight:233.26
  • Sofosbuvir impurity F

    CAS:
    <p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>
    Formula:C34H45FN4O13P2
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:798.69