
Proteases/Proteasome
Protease and proteasome inhibitors are compounds that block the activity of proteases and the proteasome, which are involved in protein degradation and turnover. These inhibitors are vital for studying the regulation of protein homeostasis, cell cycle control, and apoptosis. Protease and proteasome inhibitors are also used in the treatment of diseases such as cancer, where abnormal protein degradation plays a role in disease progression. By inhibiting proteases or the proteasome, these compounds can induce cell death in cancer cells and are critical tools in both basic research and therapeutic development. At CymitQuimica, we provide a wide range of high-quality protease and proteasome inhibitors to support your research in biochemistry, cell biology, and drug development.
Subcategories of "Proteases/Proteasome"
- Acetyl-CoA Carboxylase(35 products)
- Cysteine Protease(105 products)
- DPP-4(20 products)
- Glutaminase(41 products)
- HIV Protease(477 products)
- PAI-1(26 products)
- Protease Inhibitors(50 products)
- Protease-activated Receptor(53 products)
- Proteasome(95 products)
- Serine Protease(55 products)
- p97(15 products)
Show 3 more subcategories
Found 1079 products of "Proteases/Proteasome"
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MK-0608
CAS:MK-0608 is an orally bioavailable HCV replication inhibitor in vitro(EC50 = 0.3 μM and EC90=1.3 μM in the subgenomic-replicon assay).Formula:C12H16N4O4Purity:98.48%Color and Shape:SolidMolecular weight:280.28Trelagliptin
CAS:Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor.Formula:C18H20FN5O2Purity:98.88%Color and Shape:SolidMolecular weight:357.38Sitagliptin
CAS:Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.Formula:C16H15F6N5OPurity:99.33% - 99.83%Color and Shape:Yellow GreaseMolecular weight:407.31Elsulfavirine
CAS:Elsulfavirine (VM-1500) is an HIV-1 infection reverse transcriptase inhibitor. It is a new anti-HIV drug.Formula:C24H17BrCl2FN3O5SPurity:99.66%Color and Shape:SolidMolecular weight:629.28LDN-27219
CAS:<p>LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.</p>Formula:C20H16N4O2S2Purity:99.01% - 99.38%Color and Shape:SolidMolecular weight:408.5RAMB4
CAS:RAMB4 (PTP1B-IN-9) is a ubiquitin-proteasome system (UPS)-stressor,with anticancer activity.Formula:C19H13Cl4NOPurity:98.89% - 99.38%Color and Shape:SolidMolecular weight:413.12Sofosbuvir impurity G
CAS:Sofosbuvir impurity G is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA replication.Formula:C22H29FN3O9PPurity:98.04%Color and Shape:SolidMolecular weight:529.45BJJF078
CAS:<p>BJJF078, an aminopiperidine, inhibits human/mouse TG2 (IC50: 41/54 nM) and TG1 (IC50: 0.16 μM), may be used in MS studies.</p>Formula:C27H29N3O6SPurity:98.19%Color and Shape:SoildMolecular weight:523.6BRD-6929
CAS:BRD-6929, a brain-targeted HDAC1/2 inhibitor (IC50 1/8 nM), enhances gnidimacrin's anti-HIV effect, useful in mood behavior studies.Formula:C19H17N3O2SPurity:98.01% - 99.05%Color and Shape:SolidMolecular weight:351.42Islatravir
CAS:<p>Islatravir (MK-8591) is an effective anti-HIV-1 agent.</p>Formula:C12H12FN5O3Purity:98.77%Color and Shape:SolidMolecular weight:293.25Probenecid
CAS:<p>Probenecid (Benemid) is a benzoic acid derivative with antihyperuricemic property.</p>Formula:C13H19NO4SPurity:98.95% - 99.84%Color and Shape:Crystals From Dil Alcohol Pleasant Aftertaste (Ntp 1992)Molecular weight:285.36Ruzasvir
CAS:<p>Ruzasvir (MK-8408) is a novel and potent pan-genotypic inhibitor of hepatitis C virus NS5A with antiviral activity.</p>Formula:C49H55FN10O7SPurity:96.87% - 96.88%Color and Shape:SolidMolecular weight:947.09LSP-249
CAS:<p>LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.</p>Formula:C24H22ClN5OPurity:99.51%Color and Shape:SolidMolecular weight:431.92ML604440
CAS:ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.Formula:C17H24BF3N2O4Purity:97.06%Color and Shape:SolidMolecular weight:388.19Q-VD-OPH
CAS:<p>Q-VD-OPh is an irreversible caspase inhibitor with an IC50 value of 48 nM against caspase-7 and between 25 and 400 nM against caspase-1, 3, 8, 9, 10, 12.</p>Formula:C26H25F2N3O6Purity:97.8% - 98.95%Color and Shape:SolidMolecular weight:513.52-Oxiranecarboxylic acid, 3-[[[(1S)-3-methyl-1-[[(3-methylbutyl)amino]carbonyl]butyl]amino]carbonyl]-, ethyl ester, (2S,3S)-
CAS:Formula:C17H30N2O5Purity:98%Color and Shape:SolidMolecular weight:342.4305L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Formula:C26H41N3O5Purity:98%Color and Shape:SolidMolecular weight:475.6208Avoralstat
CAS:Avoralstat (BCX4161) is an oral plasma kallikrein (PKK) inhibitor. Which is used for the treatment of hereditary angioedema.Formula:C28H27N5O5Purity:99.77%Color and Shape:SolidMolecular weight:513.54Mecarbinate
CAS:<p>Mecarbinate (Dimecarbin) is arbidol hydrochloride's chemical intermediate.</p>Formula:C13H15NO3Purity:99.28%Color and Shape:Off-White Crystalline PowderMolecular weight:233.26Sofosbuvir impurity F
CAS:<p>Sofosbuvir impurity F (Sofosbuvir 3',5'-Bis-(S)-phosphate) is both a diastereomer of Sofosbuvir and an impurity of Sofosbuvir which is an inhibitor of HCV RNA</p>Formula:C34H45FN4O13P2Purity:98.05%Color and Shape:SolidMolecular weight:798.69

