GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,003 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Nelonicline
CAS:Nelonicline is a selective agonist of neuronal nicotinic receptors.Formula:C17H19N3OSPurity:98%Color and Shape:SolidMolecular weight:313.42Zicronapine
CAS:Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.Formula:C22H27ClN2Color and Shape:SolidMolecular weight:354.92SB 714786
CAS:SB 714786 is a selective antagonist of 5-HT1D.Formula:C26H28N4OPurity:98%Color and Shape:SolidMolecular weight:412.53GR 113808
CAS:GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formula:C19H27N3O4SPurity:98.16% - 99.96%Color and Shape:SolidMolecular weight:393.5Thioproperazine
CAS:Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.Formula:C22H30N4O2S2Purity:99.45%Color and Shape:SolidMolecular weight:446.63BAY-u 9773
CAS:BAY-u9773 is a non-selective CysLT receptor antagonist with similar IC50 for CysLT1 and CysLT2, inhibiting LT responses.Formula:C27H36O5SColor and Shape:White OilMolecular weight:472.642-Iodomelatonin
CAS:2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.Formula:C13H15IN2O2Purity:99.7%Color and Shape:SolidMolecular weight:358.17Ref: TM-T10073
10mg46.00€25mg84.00€50mg125.00€100mg188.00€200mg283.00€500mgTo inquire1mL*10mM (DMSO)35.00€Povafonidine
CAS:Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.Formula:C11H13N5Color and Shape:SolidMolecular weight:215.252-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
CAS:2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.Formula:C20H37NOSPurity:98%Color and Shape:SolidMolecular weight:339.58Niperotidine
CAS:Niperotidine is an antagonist of histamine H2-receptor.Formula:C20H26N4O5SPurity:98%Color and Shape:SolidMolecular weight:434.51(RS)-Minesapride
CAS:Minesapride is a serotonin receptor agonist.Formula:C21H31ClN4O5Purity:98%Color and Shape:SolidMolecular weight:454.95LY 206130
CAS:LY 206130 is an antagonist of serotonin 5-HT1A.Formula:C17H24N2O2Color and Shape:SolidMolecular weight:288.38LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13(S)-(-)-Propranolol hydrochloride
CAS:(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。Formula:C16H22ClNO2Purity:99.02% - 99.91%Color and Shape:SolidMolecular weight:295.8Medroxalol hydrochloride
CAS:Medroxalol hydrochloride is an antihypertensive agent that possesses both alpha and beta-adrenergic antagonistic properties.Formula:C20H25ClN2O5Color and Shape:SolidMolecular weight:408.88AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purity:98%Color and Shape:SolidMolecular weight:504.53Y2 Antagonist 36
CAS:Y2 Antagonist 36 is a highly potent, soluble and selective antagonist of NPY Y2.Formula:C27H29ClN4O3Color and Shape:SolidMolecular weight:493EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Formula:C15H27N5O6Color and Shape:SolidMolecular weight:373.4PF2562
CAS:PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Formula:C19H17N5OPurity:98%Color and Shape:SolidMolecular weight:331.37Iso-SLR 080811
CAS:Iso-SLR 080811 is an isomer of SLR 080811, suitable for relevant research in the life sciences. SLR080811 is a selective SphK2 inhibitor (Ki=1.3 μM).Formula:C21H32ClN5OPurity:98.34%Color and Shape:SolidMolecular weight:405.97(R)-DOI hydrochloride
CAS:(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.Formula:C11H17ClINO2Purity:99.88% - >99.99%Color and Shape:SolidMolecular weight:357.62OMDM-6
CAS:OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.Formula:C28H42N2O3Purity:99.66%Color and Shape:SolidMolecular weight:454.64Ref: TM-T12307
1mg85.00€5mg170.00€10mg250.00€25mg371.00€50mg522.00€100mg712.00€200mg954.00€1mL*10mM (DMSO)187.00€A61603
CAS:A61603 is an alpha-1A adrenergic receptor.Formula:C14H19N3O3SColor and Shape:SolidMolecular weight:309.38hA2AAR antagonist 1
CAS:Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31Amibegron
CAS:Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formula:C22H26ClNO4Color and Shape:SolidMolecular weight:403.9HSK0935
CAS:HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.Formula:C22H25ClO7Purity:98%Color and Shape:SolidMolecular weight:436.88Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
Formula:C19H23N5O3SPurity:99.51%Color and Shape:SolidMolecular weight:401.48N,N-Dimethylsphingosine
CAS:N,N-Dimethylsphingosine,is a potent competitive SphK phosphorylation inhibitor.DMS is elevated in models of neuropathic pain by increasing IL-1β and MCP-1.Formula:C20H41NO2Purity:98%Color and Shape:Clear Colorless To Faint Yellow Liquid/White To Off-White PowderMolecular weight:327.55L 640033
CAS:L 640033 is a beta-agonist.Formula:C18H25N3OPurity:98%Color and Shape:SolidMolecular weight:299.41RUSKI-201 dihydrochloride
CAS:RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.Formula:C20H29Cl2N3OSColor and Shape:SolidMolecular weight:430.43Sigma-LIGAND-1
CAS:Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively.Formula:C27H33NO4Purity:99.89%Color and Shape:SolidMolecular weight:435.56Ref: TM-T13510
1mg48.00€5mg104.00€10mg156.00€25mg235.00€50mg316.00€100mg434.00€200mg585.00€1mL*10mM (DMSO)119.00€Isamoltane hemifumarate
CAS:5-HT1B antagonistFormula:C16H22N202C4H404Purity:98%Color and Shape:SolidMolecular weight:332.45-HT3 antagonist 3
CAS:5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).Formula:C20H21N3OPurity:99.9%Color and Shape:SolidMolecular weight:319.4Ref: TM-T10162
1mg109.00€2mg163.00€5mg243.00€10mg355.00€25mg532.00€50mg750.00€100mg1,009.00€500mgTo inquire2-Methylthioadenosine diphosphate trisodium
CAS:2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.Formula:C11H14N5Na3O10P2SColor and Shape:SolidMolecular weight:539.24SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:403.865-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Formula:C18H21N3OPurity:98%Color and Shape:SolidMolecular weight:295.38Afurolol Hydrochloride
CAS:Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.Formula:C15H22ClNO4Purity:98.86%Color and Shape:SolidMolecular weight:315.79PNU-96391
CAS:PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Formula:C15H23NO2SPurity:99.53%Color and Shape:SolidMolecular weight:281.41Ref: TM-T28435
1mg77.00€5mg155.00€10mg221.00€25mg338.00€50mg472.00€100mg632.00€200mg843.00€1mL*10mM (DMSO)145.00€GR 55562 dihydrochloride
CAS:5-HT1B (5-HT1Dβ) silent antagonistFormula:C23H27Cl2N3O2Purity:99.45%Color and Shape:SolidMolecular weight:448.39Salmefamol
CAS:Salmefamol is a beta-adrenergic agonist. It may also be used as a bronchodilator.Formula:C19H25NO4Purity:99.89%Color and Shape:SolidMolecular weight:331.41D2343
CAS:D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.Formula:C20H27NO3Purity:98%Color and Shape:SolidMolecular weight:329.43Sulfinalol
CAS:Sulfinalol is a compound that acts as an orally active β-adrenoceptor antagonist and directly induces vasodilation [1].Formula:C20H27NO4SColor and Shape:SolidMolecular weight:377.52-Methylthio-ATP tetrasodium
CAS:2-Methylthio-ATP tetrasodium is a non-specific P2 receptor agonist, which can activate P2X2 and P2Y1 receptors and inhibiti ADP-induced platelet aggregation.Formula:C11H14N5Na4O13P3SPurity:98%Color and Shape:SolidMolecular weight:641.2Laropiprant
CAS:Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(KiFormula:C21H19ClFNO4SPurity:98.24% - 99.89%Color and Shape:SolidMolecular weight:435.9Ref: TM-T15712
1mg38.00€5mg87.00€10mg113.00€25mg220.00€50mg338.00€100mg482.00€200mg658.00€1mL*10mM (DMSO)95.00€AS19
CAS:AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).Formula:C18H25N3Purity:98%Color and Shape:SolidMolecular weight:283.41ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Formula:C24H28ClNO2Purity:98%Color and Shape:SolidMolecular weight:397.94Efaroxan hydrochloride
CAS:Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.Formula:C13H17ClN2OPurity:98%Color and Shape:SolidMolecular weight:252.742-Arachidonoylglycerol
CAS:In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligandFormula:C23H38O4Purity:95%Color and Shape:LiquidMolecular weight:378.55SK1-I hydrochloride
CAS:SK1-I hydrochloride is a selective and competitive SphK1 inhibitor and sphingosine analog ,anti-leukemic to inhibit tumor cell growth and promote apoptosis.Formula:C17H28ClNO2Purity:99.80%Color and Shape:SolidMolecular weight:313.86Carboprost
CAS:Carboprost (15(S)-15-Methyl Prostaglandin F2α) is a synthetic prostaglandin analogue of PGF2α which has the effect of oxytocic.Formula:C21H36O5Purity:98.18%Color and Shape:White Or Almost White PowderMolecular weight:368.51Ref: TM-T22285
1mg43.00€5mg110.00€10mg166.00€25mg290.00€50mg425.00€100mg577.00€200mg778.00€1mL*10mM (DMSO)122.00€PNU-142633
CAS:PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.Formula:C24H30N4O3Purity:98%Color and Shape:SolidMolecular weight:422.52hGPR91 antagonist 3
CAS:hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study diseases in hypertension and retinal angiogenesis.Formula:C23H18F4N4O2Purity:98.82% - 99.347%Color and Shape:SolidMolecular weight:458.41Ref: TM-T62858
1mg123.00€5mg295.00€10mg490.00€25mg792.00€50mg1,071.00€100mg1,468.00€200mg1,972.00€1mL*10mM (DMSO)299.00€Reversan
CAS:Reversan(CBLC4H10) is a potent, nontoxic, and glioblastoma-associated inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp).Formula:C26H27N5O2Purity:99.05%Color and Shape:SolidMolecular weight:441.53Ref: TM-T12714
1mg44.00€5mg93.00€10mg130.00€25mg250.00€50mg401.00€100mg640.00€200mg884.00€1mL*10mM (DMSO)92.00€2-Methyl-5-HT maleate
CAS:2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.Formula:C15H18N2O5Purity:98%Color and Shape:SolidMolecular weight:306.31ML179
CAS:ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.Formula:C21H25F3N4O2Purity:99.77%Color and Shape:SolidMolecular weight:422.44Ref: TM-T8954
1mg34.00€5mg75.00€10mg110.00€25mg220.00€50mg321.00€100mg469.00€200mg645.00€1mL*10mM (DMSO)92.00€Etrasimod arginine
CAS:Etrasimod arginine is used in the Treatment of Autoimmune and Inflammatory Diseases.Formula:C32H40F3N5O5Color and Shape:SolidMolecular weight:631.69BRL 44408 Maleate Salt
CAS:BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.Formula:C17H21N3O4Purity:98.71%Color and Shape:SolidMolecular weight:331.37cis-Epoxysuccinic acid
CAS:cis-Epoxysuccinic acid is a potential agonist of Succinate receptor 1 and inhibitor of Isocitrate lyase 1 for use in biochemical experiments.Formula:C4H4O5Purity:99.81%Color and Shape:SolidMolecular weight:132.07Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formula:C20H29FN2O3Purity:98.97% - >99.99%Color and Shape:SolidMolecular weight:364.45Ref: TM-T70302
1mg359.00€5mg842.00€10mg1,035.00€25mg1,663.00€50mg2,072.00€100mg2,660.00€1mL*10mM (DMSO)677.00€Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Formula:C15H17Cl2NO2Purity:99.77%Color and Shape:SolidMolecular weight:314.21BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Formula:C12H19N5O2S2Purity:98%Color and Shape:SolidMolecular weight:329.44Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Formula:C17H26N4OPurity:98%Color and Shape:SolidMolecular weight:302.415-HT7 agonist 1
CAS:5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).Formula:C19H20ClN3Purity:98.61%Color and Shape:SolidMolecular weight:325.84Ref: TM-T10170
1mg109.00€2mg163.00€5mg241.00€10mg355.00€25mg532.00€50mg745.00€100mg1,018.00€1mL*10mM (DMSO)241.00€TSI-01
CAS:TSI-01,Pro-inflammatory phospholipid mediator. Inhibits LPCAT2 (IC50=0.47 μM). Suppresses PAF biosynthesis in macrophages.Formula:C14H11Cl2NO4Purity:99.87%Color and Shape:SolidMolecular weight:328.15Ref: TM-T24904
1mg83.00€5mg175.00€10mg305.00€25mg659.00€50mg1,046.00€100mg1,607.00€200mg2,164.00€1mL*10mM (DMSO)193.00€Repinotan HCl
CAS:Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.
Formula:C21H25ClN2O4SPurity:99.57%Color and Shape:SolidMolecular weight:436.95ZK-90055 hydrochloride
CAS:ZK-90055 hydrochloride is a β2 adrenergic receptor agonist used to study asthma.Formula:C16H23ClN2O4Purity:99.26%Color and Shape:SolidMolecular weight:342.82Apadenoson
CAS:Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.Formula:C23H30N6O6Purity:98%Color and Shape:SolidMolecular weight:486.52Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purity:98%Color and Shape:SolidMolecular weight:310.78Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFormula:C25H36N4O10Purity:98%Color and Shape:SolidMolecular weight:552.581EP3 antagonist 3
CAS:EP3 antagonist 3, potent and selective oral, inhibited GR63799- or acetic acid-induced reduction in bladder capacity and PGE2-induced overactive bladder model.Formula:C21H18N2O4Color and Shape:SolidMolecular weight:362.38ONO-8713
CAS:ONO-8713 is a selective prostaglandin E receptor subtype EP1 antagonist that can be used to study diseases of the biblical system and metabolism-relatedFormula:C25H24F3NO6SPurity:99.97%Color and Shape:SolidMolecular weight:523.52CP-226269
CAS:CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.
Formula:C18H19FN4Purity:99.08%Color and Shape:SolidMolecular weight:310.37L-740093
CAS:L-740093 is a specific antagonist of CCK-B receptor.Formula:C26H31N5O2Purity:98%Color and Shape:SolidMolecular weight:445.56S 16924
CAS:S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful in the study of neurologic disorders.Formula:C22H24FNO4Purity:99.35% - 99.6%Color and Shape:SolidMolecular weight:385.43ESI-08
CAS:ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 μM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation.Formula:C20H23N3OSPurity:97.17%Color and Shape:SolidMolecular weight:353.48Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3Aganepag
CAS:Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and scar/wrinkle treatment research.Formula:C24H31NO4SPurity:98%Color and Shape:SolidMolecular weight:429.57Atrasentan hydrochloride
CAS:Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for ETA).Formula:C29H39ClN2O6Purity:99.75%Color and Shape:SolidMolecular weight:547.08A2AR-agonist-1
CAS:A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Formula:C20H22N6O4Purity:99.9%Color and Shape:SolidMolecular weight:410.43Ref: TM-T10212
1mg90.00€2mg127.00€5mg178.00€10mg269.00€25mg427.00€50mg610.00€100mg820.00€500mg1,603.00€1mL*10mM (DMSO)207.00€SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Formula:C18H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:352.49WS 009A
CAS:WS 009A is an antagonist of the endothelin receptor.Formula:C24H25NO10SPurity:98%Color and Shape:SolidMolecular weight:519.52VNA-932
CAS:VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).Formula:C23H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:402.88GBR 13069 dihydrochloride
CAS:GBR 13069 dihydrochloride is a dopamine uptake inhibitor.Formula:C28H32Cl2F2N2OPurity:98%Color and Shape:SolidMolecular weight:521.47(R)-SLV 319
CAS:(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.Formula:C23H20Cl2N4O2SColor and Shape:SolidMolecular weight:487.4DS-3801b
CAS:DS-3801b is a non-macrolide GPR38 agonist with an N-methylaniline structure for the study of functional gastrointestinal disorders.Formula:C28H39N3O3Purity:99.21%Color and Shape:SolidMolecular weight:465.63GSK1059865
CAS:GSK1059865 is a potent antagonist of the orexin 1 receptor.Formula:C20H23BrFN3O2Color and Shape:SolidMolecular weight:436.32MC-4R Agonist 1
CAS:MC-4R Agonist 1 is an agonist of human melanocortin-4 receptor (MC-4R) and can be used in the research of sexual dysfunction, obesity, and diabetes.Formula:C30H38ClF2N3O2Purity:98%Color and Shape:SolidMolecular weight:546.09TSHR antagonist S37b
CAS:S37b, a less effective enantiomer of TSHR antagonist S37a, offers minor thyrotropin receptor inhibition, useful for thyroid research.Formula:C25H20N2O3S2Color and Shape:SolidMolecular weight:460.57Indisetron Dihydrochloride
CAS:Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia.Formula:C17H24ClN5OColor and Shape:SolidMolecular weight:349.86TC-G 1004
CAS:adenosine A2A receptors antagonistFormula:C22H27N7O2Purity:98%Color and Shape:SolidMolecular weight:421.5PNU-282987 S enantiomer hydrochloride
CAS:(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.Formula:C14H18Cl2N2OPurity:98%Color and Shape:SolidMolecular weight:301.21Irindalone
CAS:IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.Formula:C24H29FN4OPurity:98%Color and Shape:SolidMolecular weight:408.51MPCI
CAS:MPCI is a selective melanocortin-4 receptor antagonist.Formula:C25H32BrFN4O2Purity:98%Color and Shape:SolidMolecular weight:519.45LH 21
CAS:LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.Formula:C20H20Cl3N3Color and Shape:SolidMolecular weight:408.75Lenperone HCl
CAS:Lenperone HCl is a dopamine antagonist and an antipsychotic agent.Formula:C22H24ClF2NO2Purity:98%Color and Shape:SolidMolecular weight:407.88Sch412348
CAS:Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.Formula:C22H21F2N9OPurity:98%Color and Shape:SolidMolecular weight:465.46Pruvanserin hydrochloride
CAS:Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.Formula:C22H22ClFN4OPurity:99.6%Color and Shape:SolidMolecular weight:412.89(-)-GSK598809
CAS:(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.Formula:C22H23F4N5OSPurity:98%Color and Shape:SolidMolecular weight:481.51Butanserin
CAS:Butanserin is a 5-hydroxytryptamine S2-antagonist.Formula:C24H26FN3O3Purity:98%Color and Shape:SolidMolecular weight:423.48NIDA 41020
CAS:NIDA 41020 is a CB1 receptor antagonist.Formula:C23H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:459.37
