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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5963 products of "GPCR/G-Protein"

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  • KY 234

    CAS:
    KY 234 is a thromboxane synthetase antagonist.
    Formula:C33H35N5O2
    Color and Shape:Solid
    Molecular weight:533.676

    Ref: TM-T70241

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR 196429

    CAS:
    GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.
    Formula:C14H18N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.3

    Ref: TM-T27430

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CID1792197

    CAS:
    CID1792197 is a selective agonist of GPR55.
    Formula:C24H23N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.59

    Ref: TM-T27017

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Setastine HCl

    CAS:
    Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.
    Formula:C22H29Cl2NO
    Color and Shape:Solid
    Molecular weight:394.38

    Ref: TM-T71791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PM226

    CAS:
    CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.
    Formula:C22H31NO3
    Color and Shape:Solid
    Molecular weight:357.49

    Ref: TM-T37815

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-817,818

    CAS:
    somatostatin sst5 receptor agonist
    Formula:C33H36N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:536.66

    Ref: TM-T22907

    10mg
    1,279.00€
  • TC 1

    CAS:
    σ1 receptor ligand
    Formula:C19H20FNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.37

    Ref: TM-T23423

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • threo Ifenprodil hemitartrate

    CAS:
    σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist
    Formula:C21H27NO2C4H6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.49

    Ref: TM-T23457

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Vasopressin V2 receptor antagonist 1

    CAS:
    Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).
    Formula:C33H37ClN4O4
    Color and Shape:Solid
    Molecular weight:589.12

    Ref: TM-T64174

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • PA-9

    CAS:
    PA-9 is the first small-molecule PAC1 receptor antagonist.
    Formula:C17H18N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.36

    Ref: TM-T24585

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS1177

    CAS:
    MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).
    Formula:C20H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.79

    Ref: TM-T16137

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-PF-06256142

    CAS:
    (R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.
    Formula:C21H16N4O2
    Color and Shape:Solid
    Molecular weight:356.38

    Ref: TM-T72744

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • Vicagrel

    CAS:
    Vicagrel, an oral antiplatelet, boosts aspirin's effect, targeting P2Y12 and fights clots in heart and vessel diseases.
    Formula:C18H18ClNO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.86

    Ref: TM-T17231

    2mg
    217.00€
    25mg
    888.00€
    50mg
    1,224.00€
    100mg
    1,674.00€
  • Ibodutant

    CAS:
    Ibodutant is an effective and selective tachykinin NK2 receptor antagonist (pKi: 10.1).
    Formula:C37H48N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:644.87

    Ref: TM-T16039

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • APC-3316 tosylate

    CAS:
    APC-3316 tosylate is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.
    Formula:C39H46N4O7S2
    Color and Shape:Solid
    Molecular weight:746.94

    Ref: TM-T69183

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Benzoctamine

    CAS:
    Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.
    Formula:C18H19N
    Color and Shape:Solid
    Molecular weight:249.35

    Ref: TM-T60368

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • S20928

    CAS:
    S20928 is an antagonist of melatonin receptor.
    Formula:C17H19NO
    Color and Shape:Solid
    Molecular weight:253.34

    Ref: TM-T28644

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DV 7028 hydrochloride

    CAS:
    DV 7028 hydrochloride is a 5-HT2A receptor antagonist.
    Formula:C21H26ClFN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.91

    Ref: TM-T22753

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • hA2A/hCA XII modulator 1

    CAS:
    Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.
    Formula:C24H19N7O4S
    Color and Shape:Solid
    Molecular weight:501.52

    Ref: TM-T63400

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Efpeglenatide

    CAS:
    Efpeglenatide is a long-acting GLP-1 receptor agonist that improves insulin sensitivity, lowers blood glucose, delays weight gain, and supports metabolic disease research.
    Purity:100% - 100%
    Color and Shape:Solid

    Ref: TM-T64252

    1mg
    To inquire
    5mg
    To inquire
    10mg
    To inquire
    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • VPC12249

    CAS:
    VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity.
    Formula:C34H52NO6P
    Color and Shape:Solid
    Molecular weight:601.75

    Ref: TM-T29109

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • A2AAR antagonist 1

    CAS:
    Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.
    Formula:C12H8BrN3O
    Color and Shape:Solid
    Molecular weight:290.12

    Ref: TM-T60591

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carbinoxamine

    CAS:
    Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.
    Formula:C16H19ClN2O
    Purity:98%
    Color and Shape:Liquid
    Molecular weight:290.79

    Ref: TM-T21247

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EGIS-7625

    CAS:
    EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.
    Formula:C18H24Cl2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.32

    Ref: TM-T27249

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alprenolol hydrochloride, (S)-

    CAS:
    Alprenolol hydrochloride, (S)- is a nonselective β-blocker. It is also a serotonin 5HT1A receptor antagonist.
    Formula:C15H24ClNO2
    Color and Shape:Solid
    Molecular weight:285.81

    Ref: TM-T4560L1

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR-203040 HCl

    CAS:
    GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.
    Formula:C20H26Cl2N6O
    Color and Shape:Solid
    Molecular weight:437.37

    Ref: TM-T24102

    25mg
    1,738.00€
  • HEMADO

    CAS:
    HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).
    Formula:C17H23N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T15468

    1mg
    112.00€
    5mg
    388.00€
  • PF-592379

    CAS:
    PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).
    Formula:C13H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.33

    Ref: TM-T10080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Centanafadine

    CAS:
    Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).
    Formula:C15H15N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.29

    Ref: TM-T10758

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Clonidine

    CAS:
    Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.
    Formula:C9H9Cl2N3
    Purity:99.42% - 99.44%
    Color and Shape:Crystals Solid
    Molecular weight:230.09

    Ref: TM-T7045

    5mg
    35.00€
    10mg
    46.00€
    25mg
    64.00€
    50mg
    89.00€
    100mg
    130.00€
    500mg
    306.00€
  • UCSF678

    CAS:
    UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.
    Formula:C15H18N2O2S
    Color and Shape:Solid
    Molecular weight:290.38

    Ref: TM-T60597

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • S(-)-Bisoprolol

    CAS:
    S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.
    Formula:C18H31NO4
    Color and Shape:Solid
    Molecular weight:325.44

    Ref: TM-T60901

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Spirendolol

    CAS:
    Spirendolol is an antagonist of β adrenergic receptor.
    Formula:C21H31NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.48

    Ref: TM-T16919

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UP202-56

    CAS:
    UP202-56 is an adenosinergic agonist and is an adenosine analog.
    Formula:C33H37N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.69

    Ref: TM-T13256

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • A331440

    CAS:
    A331440 is an modulator of L-histidine and histamine H3 receptor.
    Formula:C22H27N3O
    Color and Shape:Solid
    Molecular weight:349.47

    Ref: TM-T26480

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TCS-OX2-29 HCl

    CAS:
    TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.
    Formula:C23H32ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.97

    Ref: TM-T4965L

    5mg
    316.00€
    10mg
    600.00€
    50mg
    2,502.00€
  • (R,R)-Reboxetine mesylate

    CAS:
    (R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.
    Formula:C20H27NO6S
    Color and Shape:Solid
    Molecular weight:409.5

    Ref: TM-T72209

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZD5213

    CAS:
    AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.
    Formula:C19H25N3O2
    Color and Shape:Solid
    Molecular weight:327.42

    Ref: TM-T71423

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-06256142

    CAS:
    PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).
    Formula:C21H16N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.38

    Ref: TM-T12423

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • MRS 1334

    CAS:
    antagonist for the human adenosine A3 receptor
    Formula:C31H26N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:522.55

    Ref: TM-T23017

    25mg
    2,232.00€
  • SB357134

    CAS:
    SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.
    Formula:C17H18Br2FN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.21

    Ref: TM-T28689

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AChE-IN-14

    CAS:
    AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.
    Formula:C28H35NO3
    Color and Shape:Solid
    Molecular weight:433.58

    Ref: TM-T62441

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • CP94253 hydrochloride

    CAS:
    CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).
    Formula:C15H20ClN3O
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:293.79

    Ref: TM-T22689

    5mg
    66.00€
    10mg
    90.00€
    25mg
    205.00€
    50mg
    334.00€
    100mg
    537.00€
    200mg
    745.00€
    1mL*10mM (DMSO)
    66.00€
  • YQA14

    CAS:
    YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.
    Formula:C23H27ClN4O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:442.94

    Ref: TM-T29195

    1mg
    77.00€
    5mg
    170.00€
    10mg
    262.00€
    25mg
    546.00€
    50mg
    855.00€
    100mg
    1,170.00€
  • (R)-(-)-α-Methylhistamine dihydrobromide

    CAS:
    (R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
    Formula:C6H13Br2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:287

    Ref: TM-T12630

    50mg
    2,585.00€
  • WIN 62,577

    CAS:
    WIN 62,577 is a allosteric antagonist of mAChR.
    Formula:C29H31N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:437.58

    Ref: TM-T29158

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ-39220675

    CAS:
    JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.
    Formula:C21H24FN3O2
    Purity:98.13% - 99.89%
    Color and Shape:Solid
    Molecular weight:369.43

    Ref: TM-T27678

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • LUF6000

    CAS:
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).
    Formula:C22H20Cl2N4
    Color and Shape:Solid
    Molecular weight:411.33

    Ref: TM-T15791

    5mg
    294.00€
    25mg
    690.00€
    50mg
    898.00€
    100mg
    1,575.00€
    1mL*10mM (DMSO)
    323.00€
  • Tacitin

    CAS:
    Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.
    Formula:C18H20ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.81

    Ref: TM-T26772

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Melatonin receptor agonist 1

    CAS:
    Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].
    Formula:C15H19N3O2
    Color and Shape:Solid
    Molecular weight:273.33

    Ref: TM-T60490

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • MAT2A-IN-2

    CAS:
    MAT2A-IN-2 is a potent inhibitor of MAT2A. MAT2A-IN-2 has potential for cancer disease research.
    Formula:C23H17F3N6O2
    Color and Shape:Solid
    Molecular weight:466.42

    Ref: TM-T62984

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fosnetupitant

    CAS:
    Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.
    Formula:C31H35F6N4O5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:688.6

    Ref: TM-T15341

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Proglumide sodium

    CAS:
    Non-selective cholecystokinin (CCK) antagonist
    Formula:C18H26N2NaO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:357.4

    Ref: TM-T23185

    50mg
    259.00€
  • Epanolol

    CAS:
    Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.
    Formula:C20H23N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:369.41

    Ref: TM-T11608

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OPC-14523 hydrochloride

    CAS:
    OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.
    Formula:C23H29Cl2N3O2
    Purity:99.60%
    Color and Shape:Solid
    Molecular weight:450.4

    Ref: TM-T62711

    5mg
    873.00€
    10mg
    1,160.00€
    25mg
    1,458.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
    1mL*10mM (DMSO)
    925.00€
  • A2A/A1 AR antagonist-1

    CAS:
    A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).
    Formula:C15H12N6O2
    Color and Shape:Solid
    Molecular weight:308.29

    Ref: TM-T60732

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GPR55 agonist 3

    CAS:
    Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.
    Formula:C19H16F4N4
    Color and Shape:Solid
    Molecular weight:376.35

    Ref: TM-T79721

    1mg
    175.00€
    5mg
    434.00€
    10mg
    622.00€
    25mg
    973.00€
    50mg
    1,341.00€
    100mg
    1,773.00€
  • LY 306669

    CAS:
    LY 306669 is an antagonist of leukotriene B4 receptor.
    Formula:C23H29FN4NaO2
    Color and Shape:Solid
    Molecular weight:435.499

    Ref: TM-T27916

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • Adriforant

    CAS:
    Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.
    Formula:C13H22N6
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:262.35

    Ref: TM-T68280

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • SNT-207858

    CAS:
    SNT-207858: selective, BBB-penetrating, oral MC-4 receptor antagonist with 22 nM IC50 (binding), 11 nM (function).
    Formula:C32H45Cl4N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:689.54

    Ref: TM-T12946

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Palmitoyl serinol

    CAS:
    Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.
    Formula:C19H39NO3
    Color and Shape:Solid
    Molecular weight:329.52

    Ref: TM-T60957

    5mg
    132.00€
    10mg
    254.00€
    50mg
    1,018.00€
    100mg
    1,783.00€
  • Orexin receptor antagonist 3

    CAS:
    Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist.
    Formula:C21H22N8O3
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T62453

    25mg
    1,459.00€
    50mg
    1,900.00€
    100mg
    2,690.00€
  • AGI-41998

    CAS:
    AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.
    Formula:C22H16BrF3N4O2
    Color and Shape:Solid
    Molecular weight:505.29

    Ref: TM-T9730

    25mg
    1,144.00€
    50mg
    1,485.00€
    100mg
    2,385.00€
  • LY 393558

    CAS:
    Dual 5-HT1B/1D receptor antagonist
    Formula:C26H31FN4O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.68

    Ref: TM-T22953

    1mg
    112.00€
    5mg
    294.00€
    10mg
    517.00€
  • SF 11

    CAS:
    SF 11 is a potent and brain penetrant neuropeptide Y Y2 receptor antagonist with IC50 of 199 nM. Antidepressant-like activity
    Formula:C27H30N2O2S
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:446.6

    Ref: TM-T23349

    2mg
    34.00€
    5mg
    52.00€
    10mg
    86.00€
    25mg
    156.00€
    50mg
    264.00€
    100mg
    408.00€
    200mg
    548.00€
  • LUF 5834

    CAS:
    A2A and A2B adenosine receptor partial agonist
    Formula:C17H12N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.38

    Ref: TM-T22937

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Anatibant

    CAS:
    Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.
    Formula:C34H36Cl2N6O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:711.66

    Ref: TM-T26627

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
    500mg
    To inquire
  • PROTAC(H-PGDS)-7

    CAS:
    PROTAC(H-PGDS)-7, a potent H-PGDS degrader, inhibits PGD2 in KU812 cells; DC50 is 17.3 pM. Potential DMD treatment.
    Formula:C40H38N8O7
    Color and Shape:Solid
    Molecular weight:742.78

    Ref: TM-T41267

    1mg
    948.00€
    500µg
    677.00€
  • Adrenaline sulfate

    CAS:
    Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.
    Formula:C9H15NO7S
    Color and Shape:Solid
    Molecular weight:281.279

    Ref: TM-T69151

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SDZ 21009

    CAS:
    β-adrenoceptor and 5-HT1A/1B receptor antagonist
    Formula:C19H28N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.44

    Ref: TM-T23343

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Midodrine (hydrochloride)

    CAS:
    Midodrine hydrochloride ((±)-Midodrine hydrochloride) is an α1-receptor agonist used in the treatment of dysautonomia and orthostatic hypotension.
    Formula:C12H19ClN2O4
    Molecular weight:290.74

    Ref: TM-T21671

    10mg
    To inquire
    25mg
    To inquire
  • ROS 234

    CAS:
    ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.
    Formula:C13H15N5
    Color and Shape:Solid
    Molecular weight:241.29

    Ref: TM-T60340

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5'-(N-Cyclopropyl)carboxamidoadenosine

    CAS:
    adenosine A2 receptor agonist
    Formula:C13H16N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.3

    Ref: TM-T22523

    5mg
    166.00€
    10mg
    305.00€
  • SM-130686

    CAS:
    SM-130,686: orally-active GHSR agonist, 50% as potent as ghrelin in stimulating growth hormone.
    Formula:C22H24Cl2F3N3O3
    Color and Shape:Solid
    Molecular weight:506.35

    Ref: TM-T28812

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • SKF83959

    CAS:

    SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.

    Formula:C18H20ClNO2
    Purity:98.68%
    Color and Shape:Solid
    Molecular weight:317.81

    Ref: TM-T60835

    1mg
    52.00€
    5mg
    103.00€
    10mg
    169.00€
    25mg
    359.00€
    50mg
    530.00€
    100mg
    758.00€
  • DW-1350

    CAS:
    DW-1350 is an antagonist of LTB4 receptor.
    Formula:C25H31N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.6

    Ref: TM-T15182

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Substance P Receptor Antagonist 1

    CAS:
    Substance P Receptor Antagonist 1 may aid in treating GI, inflammatory, respiratory, and CNS disorders.
    Formula:C24H29F3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.49

    Ref: TM-T10121

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ 10181457 dihydrochloride

    CAS:
    JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.
    Formula:C20H28N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.45

    Ref: TM-T22878

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CFM 1571 hydrochloride

    CAS:
    CFM 1571 hydrochloride stimulates sGC with EC50 of 5.49 μM; potential for cardiovascular research.
    Formula:C23H29ClN4O3
    Color and Shape:Solid
    Molecular weight:444.96

    Ref: TM-T22197

    25mg
    1,440.00€
    50mg
    1,882.00€
  • BMY-25271

    CAS:
    BMY-25271 is an antagonist of histamine H2 receptor.
    Formula:C12H19N5O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.44

    Ref: TM-T10575

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Broxaterol

    CAS:
    Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.
    Formula:C9H15BrN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:263.13

    Ref: TM-T23823

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • B-HT 933 dihydrochloride

    CAS:
    Azepexole (B-HT 933) dihydrochloride is an α2-adrenoceptor agonist, pKi: 8.3/α2A, 7.6/α2B, 7.5/α2C; IC50: 78.72 nM for peristalsis inhibition.
    Formula:C9H17Cl2N3O
    Color and Shape:Solid
    Molecular weight:254.16

    Ref: TM-T21787

    1mg
    105.00€
    5mg
    444.00€
    10mg
    650.00€
  • Levobunolol

    CAS:
    Levobunolol is a nonselective beta-blocker. It is used topically to treat glaucoma.
    Formula:C17H25NO3
    Color and Shape:White To Pink Powder
    Molecular weight:291.39

    Ref: TM-T32699

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • BMS-665053

    CAS:
    BMS-665053: CRF1 receptor antagonist, IC50 = 1.0 nM; inhibits cAMP in Y-79 cells, IC50 = 4.9 nM; anti-anxiety in rats, Cl = 17 mL/min/kg, t½ = 7.8 h.
    Formula:C16H14Cl3F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.66

    Ref: TM-T26855

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SNT-207858 free base

    CAS:
    SNT-207858: selective MC-4 receptor antagonist, passes blood-brain barrier, orally active, IC50: 22 nM (binding), 11 nM (function).
    Formula:C32H43Cl2N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:616.62

    Ref: TM-T12945

    5mg
    401.00€
    25mg
    1,288.00€
    50mg
    1,674.00€
    100mg
    2,250.00€
  • Mosapramine

    CAS:
    Mosapramine is a dopamine D2-receptor antagonist.
    Formula:C28H35ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.06

    Ref: TM-T28086

    25mg
    2,160.00€
    50mg
    2,700.00€
    100mg
    3,600.00€
  • Kadsurenone

    CAS:
    Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.
    Formula:C21H24O5
    Color and Shape:Solid
    Molecular weight:356.41

    Ref: TM-T68233

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Bufetolol

    CAS:
    Bufetolol is an antagonist of beta-adrenoceptor.
    Formula:C18H29NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.43

    Ref: TM-T23836

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MK-2894

    CAS:
    MK-2894 is a highly potent and selective antagonist of second generation EP4 .
    Formula:C25H22F3NO3S
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:473.51

    Ref: TM-T12061

    1mg
    57.00€
    5mg
    120.00€
    10mg
    205.00€
    25mg
    497.00€
    50mg
    879.00€
    100mg
    1,161.00€
    500mg
    2,367.00€
    1mL*10mM (DMSO)
    128.00€
  • (Rac)-WAY-161503

    CAS:
    (Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.
    Formula:C11H11Cl2N3O
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:272.13

    Ref: TM-T13332

    5mg
    89.00€
    10mg
    111.00€
    25mg
    172.00€
    50mg
    253.00€
    100mg
    374.00€
  • Sultopride

    CAS:
    Sultopride is a compound that an amino on the sulfamide group of sulpiride is replaced by an ethyl group.
    Formula:C17H26N2O4S
    Color and Shape:Solid
    Molecular weight:354.46

    Ref: TM-T7180L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alprenolol tartrate, (S)-

    CAS:
    Alprenolol tartrate, (S)- is an 5-HT1A antagonist.
    Formula:C19H29NO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.44

    Ref: TM-T4560L2

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Guanoxabenz hydrochloride

    CAS:
    Guanoxabenz hydrochloride, α2 adrenergic receptor agonist; Ki: 4000 nM, α2A form Ki: 40 nM.
    Formula:C8H9Cl3N4O
    Color and Shape:Solid
    Molecular weight:283.54

    Ref: TM-T60548

    25mg
    1,260.00€
    50mg
    1,639.00€
    1mL*10mM (DMSO)
    326.00€
  • PD 119819

    CAS:
    PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.
    Formula:C21H25Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.35

    Ref: TM-T28318

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BI-L 239

    CAS:
    BI-L 239 is an inhibition of 5-lipoxygenase products that cause bronchoconstriction.
    Formula:C16H15FO
    Color and Shape:Solid
    Molecular weight:242.29

    Ref: TM-T26811

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bifeprunox Mesylate

    CAS:
    Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.
    Formula:C25H27N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.56

    Ref: TM-T26807

    1mg
    114.00€
  • Penbutolol

    CAS:
    Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.
    Formula:C18H29NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.43

    Ref: TM-T12402L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DMP 696

    CAS:
    DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.
    Formula:C18H21Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.3

    Ref: TM-T15145

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • IMTPPE

    CAS:
    IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.
    Formula:C20H27N3O2S
    Color and Shape:Solid
    Molecular weight:373.51

    Ref: TM-T27601

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JMV3002

    CAS:
    JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.
    Formula:C35H34N6O3
    Color and Shape:Solid
    Molecular weight:586.68

    Ref: TM-T35793

    1mg
    1,485.00€
    5mg
    6,193.00€
    100µg
    195.00€
    500µg
    845.00€