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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • QF0301B

    CAS:
    QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
    Formula:C23H28N2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:364.48

    Ref: TM-T10100

    1mg
    665.00€
    5mg
    1,710.00€
  • 5-HT7 receptor ligand 1

    CAS:
    Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.
    Formula:C21H23N7
    Color and Shape:Solid
    Molecular weight:373.45

    Ref: TM-T61515

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amibegron hydrochloride

    CAS:
    Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.
    Formula:C22H27Cl2NO4
    Color and Shape:Solid
    Molecular weight:440.36

    Ref: TM-T10302

    25mg
    837.00€
    50mg
    1,089.00€
    100mg
    1,648.00€
  • BRL 44408 Maleate Salt

    CAS:
    BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.
    Formula:C17H21N3O4
    Purity:98.71%
    Color and Shape:Solid
    Molecular weight:331.37

    Ref: TM-T26904

    1mg
    74.00€
    5mg
    163.00€
    10mg
    283.00€
    25mg
    467.00€
    50mg
    682.00€
    100mg
    1,004.00€
  • Setastine HCl

    CAS:
    Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.
    Formula:C22H29Cl2NO
    Color and Shape:Solid
    Molecular weight:394.38

    Ref: TM-T71791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ-26070109

    CAS:
    JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.
    Formula:C23H17BrF2N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:547.37

    Ref: TM-T27669

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CID1792197

    CAS:
    CID1792197 is a selective agonist of GPR55.
    Formula:C24H23N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.59

    Ref: TM-T27017

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Oxetorone fumarate

    CAS:
    Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.
    Formula:C25H25NO6
    Purity:99.809%
    Color and Shape:Solid
    Molecular weight:435.48

    Ref: TM-T24575

    1mg
    302.00€
    5mg
    730.00€
    10mg
    999.00€
    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • Isoproterenol-d7 HCl

    CAS:
    Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.
    Formula:C11H18ClNO3
    Color and Shape:Solid
    Molecular weight:254.76

    Ref: TM-T69598

    1mg
    359.00€
  • GR 196429

    CAS:
    GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.
    Formula:C14H18N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.3

    Ref: TM-T27430

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SKF83822 hydrobromide

    CAS:
    SKF83822 hydrobromide is a dopamine D1-like receptor agonist.
    Formula:C20H23BrClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.76

    Ref: TM-T23363

    50mg
    3,510.00€
  • Cicloprolol hydrochloride

    CAS:
    Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
    Formula:C18H30ClNO4
    Purity:97.26%
    Color and Shape:Solid
    Molecular weight:359.89

    Ref: TM-T10812

    1mg
    630.00€
    5mg
    1,620.00€
  • Bamirastine

    CAS:
    Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on
    Formula:C31H37N5O3
    Purity:96.68%
    Color and Shape:Solid
    Molecular weight:527.66

    Ref: TM-T13566

    1mg
    665.00€
    5mg
    1,710.00€
  • (4E)-SUN9221

    CAS:
    (4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in
    Formula:C25H31FN4O3
    Purity:97.79%
    Color and Shape:Solid
    Molecular weight:454.54

    Ref: TM-T12596

    1mg
    665.00€
    5mg
    1,710.00€
  • A-940894

    CAS:
    A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.
    Formula:C17H21N5
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T23597

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GW848687X

    CAS:
    GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.
    Formula:C24H18ClF2NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.85

    Ref: TM-T27517

    1mg
    537.00€
    5mg
    2,277.00€
    500µg
    290.00€
  • CB1/2 agonist 4

    CAS:
    CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.
    Formula:C27H45NO3
    Color and Shape:Solid
    Molecular weight:431.65

    Ref: TM-T62411

    25mg
    2,033.00€
    50mg
    2,645.00€
    100mg
    3,345.00€
  • ONO4057

    CAS:
    ONO4057 is a potent and orally active Leukotriene B4 receptor antagonist with an IC50 value of 0.7±0.3 μM.
    Formula:C27H34O7
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:470.55

    Ref: TM-T16395

    1mg
    630.00€
    5mg
    1,620.00€
  • PAF-AN-1

    CAS:
    PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of anaphylactic death.
    Formula:C28H28N2O3
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:440.53

    Ref: TM-T14007

    1mg
    665.00€
    5mg
    1,710.00€
  • CP-66948

    CAS:
    CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.
    Formula:C13H20N6S
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:292.4

    Ref: TM-T15005

    1mg
    665.00€
    5mg
    1,710.00€
  • Indanidine

    CAS:
    Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in the
    Formula:C11H13N5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:215.25

    Ref: TM-T11651

    1mg
    152.00€
    2mg
    197.00€
    5mg
    295.00€
  • RS-601

    CAS:
    RS-601 is a potent dual leukotriene D4/thromboxane A2 inhibitor that inhibits antigen-induced airway hyperresponsiveness (AHR) and shows asthmatic effects in a
    Formula:C22H23F6NO4S
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:511.48

    Ref: TM-T12771

    1mg
    665.00€
    5mg
    1,710.00€
  • LUF 6283

    CAS:
    partial agonist of hydroxycarboxylic acid receptor 2 (HCA2)
    Formula:C8H12N2O2
    Color and Shape:Solid
    Molecular weight:168.19

    Ref: TM-T22938

    1mg
    105.00€
    5mg
    304.00€
    10mg
    388.00€
  • Adenosine receptor A1 antagonist 5

    CAS:
    1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.
    Formula:C17H20N4O2
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:312.37

    Ref: TM-T22466

    1mg
    46.00€
    5mg
    94.00€
    10mg
    137.00€
    25mg
    226.00€
    50mg
    324.00€
    100mg
    447.00€
    200mg
    600.00€
  • JNJ-10191584

    CAS:
    JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation
    Formula:C13H15ClN4O
    Color and Shape:Solid
    Molecular weight:278.74

    Ref: TM-T27658

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sograzepide

    CAS:
    Sograzepide (Netazepide) is a gastrin/CCK-B antagonist, inhibits gastrin/CCK-A activity, and can induce regression of type 1 gastric neuroendocrine tumors
    Formula:C28H30N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58

    Ref: TM-T16906

    1mg
    248.00€
    5mg
    692.00€
  • SCH-202676 HBr

    CAS:
    SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.
    Formula:C15H13N3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.35

    Ref: TM-T24770

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TSHR antagonist S37a

    CAS:
    TSHR antagonist S37a is a selective, orally bioavailable TSHR antagonist that inhibits TSH-induced cAMP in TSHR-expressing HEK 293 cells.
    Formula:C25H20N2O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.57

    Ref: TM-T13217

    1mg
    141.00€
    5mg
    340.00€
    10mg
    537.00€
    25mg
    1,044.00€
    50mg
    1,558.00€
    100mg
    2,277.00€
    1mL*10mM (DMSO)
    346.00€
  • PF-03654764

    CAS:
    PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.
    Formula:C20H28F2N2O
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:350.45

    Ref: TM-T61213

    1mg
    311.00€
    5mg
    747.00€
  • Guanoxabenz

    CAS:
    Guanoxabenz is an α2 adrenergic receptor agonist.
    Formula:C8H8Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.08

    Ref: TM-T11512

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bavisant dihydrochloride

    CAS:
    Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.
    Formula:C19H29Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.36

    Ref: TM-T10462

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Methdilazine Hydrochloride

    CAS:
    Methdilazine Hydrochloride (Bristaline) is a histamine H1 receptor antagonist for dermatologic conditions and relief of itching by allergies or rhinitis.
    Formula:C18H21ClN2S
    Color and Shape:Light-Tan Crystalline Powder 4 8-6 (Ntp 1992)
    Molecular weight:332.89

    Ref: TM-T33319

    1mg
    278.00€
    5mg
    597.00€
    10mg
    901.00€
    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • Dopamine D4 receptor antagonist-1

    CAS:
    Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.
    Formula:C18H19ClN4
    Color and Shape:Solid
    Molecular weight:326.82

    Ref: TM-T60917

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • T-0509

    CAS:

    T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-

    Formula:C18H23NO5
    Purity:97.52% - 98.43%
    Color and Shape:Solid
    Molecular weight:333.38

    Ref: TM-T28895

    1mg
    200.00€
    5mg
    472.00€
    10mg
    645.00€
    25mg
    905.00€
  • MAT2A-IN-1

    CAS:
    MAT2A-IN-1 suppresses MAT2A, key for MTAP-deficient cancer cell growth; studied for gastric, colon, liver, pancreatic cancers.
    Formula:C29H28F2N6O4
    Color and Shape:Solid
    Molecular weight:562.57

    Ref: TM-T63975

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Norfenefrine HCl

    CAS:
    Norfenefrine HCl is an α1-adrenergic receptor agonist, an endogenous neurotransmitter and sympathomimetic drug for hypotension,glycerol adipose.
    Formula:C8H12ClNO2
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:189.64

    Ref: TM-T71821

    200mg
    42.00€
    1mL*10mM (DMSO)
    37.00€
  • p-MPPF dihydrochloride

    CAS:
    p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.
    Formula:C25H29Cl2FN4O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:507.43

    Ref: TM-T69750

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • Propiomazine HCl

    CAS:
    Propiomazine HCl is an analgesia adjunct.
    Formula:C20H25ClN2OS
    Color and Shape:Solid
    Molecular weight:376.94

    Ref: TM-T34152L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RP73870

    CAS:
    RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
    Formula:C27H30N4O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:554.61

    Ref: TM-T28613

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • MRS2298

    CAS:
    MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.
    Formula:C10H16ClN5O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.66

    Ref: TM-T28100

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PD 118717

    CAS:
    PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.
    Formula:C20H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T28316

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Org37684

    CAS:
    5-HT2 receptors agonist
    Formula:C14H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:269.77

    Ref: TM-T23112

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 60-0175 fumarate

    CAS:
    5-HT2 receptor agonist
    Formula:C15H16ClFN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:342.75

    Ref: TM-T23246

    1mg
    105.00€
    5mg
    268.00€
  • CAY10412

    CAS:
    Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.
    Formula:C25H36O2S
    Color and Shape:Solid
    Molecular weight:400.62

    Ref: TM-T37684

    5mg
    128.00€
    10mg
    233.00€
    50mg
    945.00€
    100mg
    1,648.00€
  • Trebenzomine

    CAS:
    Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.
    Formula:C12H17NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:191.27

    Ref: TM-T29004

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carcinine

    CAS:
    Carcinine ditrifluoroacetate is a H3 receptor antagonist.
    Formula:C8H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:182.22

    Ref: TM-T22624

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VK-II-86

    CAS:
    VK-II-86 is a non-β-blocking carvedilol analog. It prevents ouabain-Induced cardiotoxicity
    Formula:C25H28N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.5

    Ref: TM-T8965

    1mg
    118.00€
    5mg
    515.00€
    10mg
    888.00€
    25mg
    1,882.00€
  • L-Alprenolol

    CAS:
    L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.
    Formula:C15H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.35

    Ref: TM-T24386

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS1186

    CAS:
    MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
    Formula:C16H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.75

    Ref: TM-T16138

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Argiprestocin

    CAS:
    Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.
    Formula:C43H67N15O12S2
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:1050.22

    Ref: TM-T3443

    50mg
    59.00€
    100mg
    97.00€
    200mg
    170.00€
  • PF-4479745

    CAS:
    PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.
    Formula:C17H22N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.38

    Ref: TM-T28384

    1mg
    427.00€
  • Remoxipride

    CAS:
    Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.
    Formula:C16H23BrN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.27

    Ref: TM-T28514

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ATC0065

    CAS:
    ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
    Formula:C25H29BrF3N5O
    Color and Shape:Solid
    Molecular weight:552.43

    Ref: TM-T26676

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PGN-9856

    CAS:
    PGN-9856 is an EP2 receptor ligand and EP2 receptor agonist with anti-inflammatory and intraocular pressure-lowering properties, useful for glaucoma research.
    Formula:C21H15F2NO4
    Purity:99.27%
    Color and Shape:Solid
    Molecular weight:383.35

    Ref: TM-T68514

    1mg
    77.00€
    5mg
    163.00€
    10mg
    232.00€
    25mg
    382.00€
    50mg
    568.00€
    100mg
    823.00€
    200mg
    1,103.00€
  • Mabuterol, (S)-

    CAS:
    Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.
    Formula:C13H18ClF3N2O
    Color and Shape:Solid
    Molecular weight:310.74

    Ref: TM-T69085

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Alimemazine

    CAS:
    Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.
    Formula:C18H22N2S
    Purity:98%
    Color and Shape:Crystals Solid
    Molecular weight:298.45

    Ref: TM-T10281

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • GT 2016

    CAS:
    GT 2016 is a H3 receptor antagonist.
    Formula:C19H31N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:317.47

    Ref: TM-T22823

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • UCSF648

    CAS:
    UCSF648 (Compound 5A6-48) weakly activates MTNR1A and ADRA2A. UCSF648 is a chemical probe for the serotonin receptor 5-HT 5A [1].
    Formula:C15H19ClN2O2S
    Color and Shape:Solid
    Molecular weight:326.84

    Ref: TM-T60918

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Colterol HCl

    CAS:
    Colterol HCl, a β2-adrenoceptor agonist salt, is used for bronchospasm in asthma and COPD.
    Formula:C12H20ClNO3
    Color and Shape:Solid
    Molecular weight:261.75

    Ref: TM-T69148

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OX2R-IN-1

    CAS:
    OX2R-IN-1: OX2R antagonist, low cytotoxicity, blood-brain barrier permeable, short half-life.
    Formula:C20H28ClN3O5S
    Color and Shape:Solid
    Molecular weight:457.97

    Ref: TM-T62855

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (RS)-Butyryltimolol

    CAS:
    (RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.
    Formula:C17H30N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.51

    Ref: TM-T13439

    2mg
    66.00€
  • Acetylaszonalenin

    CAS:
    Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.
    Formula:C25H25N3O3
    Color and Shape:Solid
    Molecular weight:415.48

    Ref: TM-T71833

    500µg
    335.00€
    2500µg
    1,170.00€
  • LEI 101 hydrochloride

    CAS:
    LEI 101 hydrochloride is potent and selective CB2 partial agonist.
    Formula:C23H26ClFN4O4S
    Color and Shape:Solid
    Molecular weight:508.99

    Ref: TM-T69732

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ambucetamide

    CAS:
    Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.
    Formula:C17H28N2O2
    Color and Shape:Solid
    Molecular weight:292.42

    Ref: TM-T26614

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • BAY-386

    CAS:
    BAY-386 is a PAR1 receptor inhibitor which suppresses activation of thrombin and platelet activity.
    Formula:C22H25F3N4O5S
    Color and Shape:Solid
    Molecular weight:514.52

    Ref: TM-T71109

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Roxindole hydrochloride

    CAS:
    Dopamine D2 autoreceptor agonist
    Formula:C23H27ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.93

    Ref: TM-T23250

    25mg
    690.00€
    50mg
    895.00€
    100mg
    1,378.00€
  • Benzatropine

    CAS:
    Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.
    Formula:C21H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.43

    Ref: TM-T23781

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Fluphenazine Decanoate Dihydrochloride

    CAS:
    Fluphenazine Decanoate Dihydrochloride: antipsychotic that blocks D2 dopamine receptors in brain regions.
    Formula:C32H46Cl2F3N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:664.69

    Ref: TM-T0068L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PD168,077

    CAS:
    PD168,077 is an agonist of dopamine D4 receptor. It has a facilitatory effect on memory consolidation.
    Formula:C20H22N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.41

    Ref: TM-T19666

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • ST1936

    CAS:
    ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74

    Ref: TM-T23396

    1mg
    44.00€
    5mg
    111.00€
    10mg
    178.00€
    25mg
    316.00€
    50mg
    470.00€
    100mg
    682.00€
    200mg
    954.00€
    1mL*10mM (DMSO)
    123.00€
  • VUF14738

    CAS:
    VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.
    Formula:C25H32N4O2
    Color and Shape:Solid
    Molecular weight:420.55

    Ref: TM-T69774

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • γ-Linolenic acid ethyl ester

    CAS:
    γ-Linolenic acid ethyl ester (Ethyl γ-linolenate) is a leukotriene B 4 receptor 4 (LTB 4 ) antagonist which has a potential anti-inflammatory effect[1].
    Formula:C20H34O2
    Color and Shape:Solid
    Molecular weight:306.48

    Ref: TM-T41235

    1g
    1,288.00€
    50mg
    114.00€
    100mg
    208.00€
    250mg
    489.00€
  • Levomepromazine Maleate

    CAS:
    Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.
    Formula:C23H28N2O5S
    Color and Shape:Solid
    Molecular weight:444.546

    Ref: TM-T71773

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Alaproclate (hydrochloride)

    CAS:
    Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.
    Formula:C13H19Cl2NO2
    Color and Shape:Solid
    Molecular weight:292.2

    Ref: TM-T36521

    5mg
    230.00€
    10mg
    399.00€
  • ZD7114 free base

    CAS:
    ZD7114 (ICI-D7114) selectively activates brown fat, boosts thermogenesis, and aids in obesity and metabolic disorders.
    Formula:C22H30N2O6
    Color and Shape:Solid
    Molecular weight:418.48

    Ref: TM-T71033

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NGB 2904 hydrochloride

    CAS:
    dopamine D3 receptor antagonist
    Formula:C28H30Cl3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:530.92

    Ref: TM-T23065

    1mg
    132.00€
    5mg
    375.00€
  • GRK5-IN-4

    CAS:
    GRK5-IN-4: potent, selective covalent inhibitor of GRK5 (IC50=1.1 μM), 90x more specific than GRK2, useful for heart failure research.
    Formula:C26H25N7O3
    Color and Shape:Solid
    Molecular weight:483.52

    Ref: TM-T63203

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Arbutamine hydrochloride

    CAS:
    Arbutamine hydrochloride is a catecholamine which acts as a cardiac stimulant.
    Formula:C18H24ClNO4
    Color and Shape:Solid
    Molecular weight:353.84

    Ref: TM-T30119

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GBR-12935 maleate

    CAS:
    GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.
    Formula:C32H38N2O5
    Color and Shape:Solid
    Molecular weight:530.665

    Ref: TM-T70914

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ridazolol

    CAS:
    Ridazolol is a vasodilating and cardioselective beta adrenergic blocker.
    Formula:C15H18Cl2N4O3
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:373.23

    Ref: TM-T26081

    1mg
    167.00€
    5mg
    411.00€
    10mg
    562.00€
    25mg
    867.00€
    50mg
    1,121.00€
    100mg
    1,501.00€
  • Levemopamil HCl

    CAS:
    Levemopamil HCl is used as a calcium channel blocker.
    Formula:C23H31ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.96

    Ref: TM-T25692L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 19-1400

    CAS:
    Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.
    Formula:C31H56N2O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:616.85

    Ref: TM-T28564

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 206553 hydrochloride

    CAS:
    SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders
    Formula:C17H17ClN4O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:328.8

    Ref: TM-T23314

    1mg
    62.00€
    5mg
    130.00€
    10mg
    203.00€
    25mg
    408.00€
    50mg
    587.00€
  • Thiothixene hydrochloride

    CAS:
    Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.
    Formula:C23H30ClN3O2S2
    Color and Shape:Solid
    Molecular weight:480.08

    Ref: TM-T63592

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Isoetharine hydrochloride

    CAS:
    Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.
    Formula:C13H22ClNO3
    Color and Shape:Solid
    Molecular weight:275.77

    Ref: TM-T60502

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Nafadotride

    CAS:
    Nafadotride is a dopamine D3 receptor antagonist.
    Formula:C22H27N3O2
    Color and Shape:Solid
    Molecular weight:365.47

    Ref: TM-T70542

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • NVS-CRF38

    CAS:
    NVS-CRF38 is an antagonist of corticotropin-releasing factor receptor 1 (CRF1).
    Formula:C19H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.4

    Ref: TM-T12276

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Ro 23-3423

    CAS:
    Ro 23-3423 is a specific inhibitor of thromboxane synthetase.
    Formula:C23H22N4O2
    Color and Shape:Solid
    Molecular weight:386.45

    Ref: TM-T28569

    25mg
    1,369.00€
  • Midodrine D6 hydrochloride

    CAS:
    Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.
    Formula:C12H19ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.78

    Ref: TM-T12035

    1mg
    To inquire
    5mg
    To inquire
  • Modipafant

    CAS:
    Modipaafant is a potent dihydropyridine PAF (platelet activating factor) antagonist.
    Formula:C34H29ClN6O3
    Color and Shape:Solid
    Molecular weight:605.09

    Ref: TM-T33466

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Prasugrel (Maleic acid)

    CAS:
    Prasugrel Maleic acid: oral P2Y12 antagonist, thienopyridine prodrug, inhibits ADP-induced platelet aggregation.
    Formula:C24H24FNO7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.51

    Ref: TM-T16572

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • JPC-211

    CAS:
    JPC-211 is an agonist of dopamine-receptor.
    Formula:C17H27NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.4

    Ref: TM-T27693

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DH-97

    CAS:
    DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).
    Formula:C22H26N2O
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T69409

    1mg
    124.00€
  • SKF 77434 hydrobromide

    CAS:
    SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.
    Formula:C19H22BrNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.29

    Ref: TM-T23360

    5mg
    233.00€
  • AR-A 2

    CAS:
    AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).
    Formula:C27H36N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.6

    Ref: TM-T10360

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • CAY10590

    CAS:
    CAY10590 (GK115) inhibits sPLA2, used in chronic kidney inflammation research.
    Formula:C21H33NO3
    Color and Shape:Solid
    Molecular weight:347.49

    Ref: TM-T61168

    5mg
    512.00€
    10mg
    884.00€
    50mg
    3,718.00€
  • BFE-55

    CAS:
    BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptors
    Formula:C14H19NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.31

    Ref: TM-T26783

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bitolterol

    CAS:
    Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.
    Formula:C28H31NO5
    Color and Shape:Solid
    Molecular weight:461.55

    Ref: TM-T69485

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide

    CAS:
    5-HT1A serotonin receptor agonist
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29

    Ref: TM-T23218

    10mg
    735.00€
    50mg
    3,052.00€
  • A1AR antagonist 2

    CAS:
    Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.
    Formula:C17H12N4O
    Color and Shape:Solid
    Molecular weight:288.3

    Ref: TM-T60580

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€