GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,003 products)
- Adenosine Receptor(247 products)
- Adrenergic Receptor(3,010 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(60 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(215 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(435 products)
- Endothelin Receptor(83 products)
- GNRH Receptor(82 products)
- GPCR19(33 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(190 products)
- Hedgehog/Smoothened(48 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(321 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5838 products of "GPCR/G-Protein"
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SDZ-62-434
CAS:SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.Formula:C23H27Cl2N3Purity:98.38%Color and Shape:SolidMolecular weight:416.39Taprizosin
CAS:<p>Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.</p>Formula:C25H26N6O4SPurity:96.34% - 99.11%Color and Shape:SolidMolecular weight:506.58Tiospirone
CAS:Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Formula:C24H32N4O2SPurity:99.74%Color and Shape:SolidMolecular weight:440.6CL 316243
CAS:CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Formula:C20H18ClNNa2O7Purity:98.00% - 99.68%Color and Shape:SolidMolecular weight:465.79GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Formula:C28H34Cl2N2OPurity:98.08%Color and Shape:SolidMolecular weight:485.49Ex26
CAS:<p>Ex26 (S1P1-IN-Ex26) is an S1P1 antagonist used in experimental autoimmune encephalomyelitis, atherosclerosis, and gastric cancer.</p>Formula:C28H28ClFN2O3Purity:99.62%Color and Shape:SolidMolecular weight:494.99Pipoxazole
CAS:Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Formula:C14H20N4OPurity:98.58% - 99.53%Color and Shape:SolidMolecular weight:260.33rel-(1R,2R)-Vesamicol Hydrochloride
CAS:rel-(1R,2R)-Vesamicol Hydrochloride is a acetylcholine transport inhibitor.Formula:C17H26ClNOPurity:99.88%Color and Shape:SolidMolecular weight:295.85ORM-10921
CAS:ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formula:C18H23NO2Purity:99.46% - 99.98%Color and Shape:SolidMolecular weight:285.38Nemazoline Free Base
CAS:Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Formula:C10H11Cl2N3Purity:98.06% - 98.83%Color and Shape:SolidMolecular weight:244.12LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purity:98.58%Color and Shape:SolidMolecular weight:407.33Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purity:99.77%Color and Shape:SolidMolecular weight:304.43Rafabegron
CAS:<p>Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.</p>Formula:C21H23ClN2O4Purity:99.21%Color and Shape:SolidMolecular weight:402.87Rocepafant
CAS:Rocepafant (LAU8080), a PAF antagonist, reduces neonatal rat brain damage and inhibits TNF-α toxicity in L929 cells.Formula:C26H23ClN6OS2Purity:97.31% - 98.95%Color and Shape:SolidMolecular weight:535.08Compound C108
CAS:<p>Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).</p>Formula:C15H14N2O3Purity:99.77%Color and Shape:SolidMolecular weight:270.28Ticolubant
CAS:Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Formula:C23H19Cl2NO3SPurity:99.5%Color and Shape:SolidMolecular weight:460.37BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurity:99.97%Color and Shape:SolidMolecular weight:384.85PPTN hydrochloride
CAS:<p>PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), but no agonist or antagonist activity at</p>Formula:C29H25ClF3NO2Purity:99.80%Color and Shape:SolidMolecular weight:511.96SK609 HCl
CAS:<p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>Formula:C10H15Cl2NPurity:99.02%Color and Shape:SolidMolecular weight:220.14CB1 agonist 1
CAS:CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Formula:C24H24N2O5SPurity:98.56%Color and Shape:SolidMolecular weight:452.52Teniloxazine
CAS:Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formula:C16H19NO2SPurity:99.29%Color and Shape:SolidMolecular weight:289.39Immethridine dihydrobromide
CAS:<p>Immethridine dihydrobromide is a histamine H3 receptor agonist.</p>Formula:C9H11Br2N3Purity:97.61% - 98.14%Color and Shape:SolidMolecular weight:321.01CV-6209
CAS:CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.Formula:C34H60ClN3O6Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:642.31Sergliflozin etabonate
CAS:Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.Formula:C23H28O9Purity:97.88%Color and Shape:SolidMolecular weight:448.46KP136
CAS:<p>KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).</p>Formula:C16H18N4O3Purity:98.3% - 98.61%Color and Shape:SolidMolecular weight:314.34Clemastine
CAS:Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Formula:C21H26ClNOPurity:99.21%Color and Shape:SolidMolecular weight:343.89Lorglumide sodium salt
CAS:Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).Formula:C22H31Cl2N2NaO4Purity:99.32%Color and Shape:SolidMolecular weight:481.39EP2 receptor antagonist-2
CAS:<p>CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.</p>Formula:C15H14F3N3OPurity:99.95%Color and Shape:SolidMolecular weight:309.29MM 77 dihydrochloride
CAS:<p>MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.</p>Formula:C19H29Cl2N3O3Purity:99.91%Color and Shape:SolidMolecular weight:418.36Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Formula:C19H27N3O2Purity:99.21% - 99.65%Color and Shape:SolidMolecular weight:329.44Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormula:C25H34N4O5SPurity:99.62% - 99.67%Color and Shape:SolidMolecular weight:502.63Spizofurone
CAS:Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.Formula:C12H10O3Purity:>99.99%Color and Shape:SolidMolecular weight:202.21Dimethindene maleate
CAS:Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.Formula:C24H28N2O4Purity:99.79%Color and Shape:SolidMolecular weight:408.49A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formula:C20H27F3N6OSPurity:98.80%Color and Shape:SolidMolecular weight:456.53YIL 781
CAS:YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM).Formula:C24H28FN3O2Purity:98.8%Color and Shape:SolidMolecular weight:409.5Terbogrel
CAS:<p>Terbogrel is an antiplatelet drug, blocking thromboxane A2 receptor/synthase. Helps prevent clots.</p>Formula:C23H27N5O2Purity:98.95%Color and Shape:SolidMolecular weight:405.49H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formula:C11H15Cl2N3O2SPurity:97.3%Color and Shape:SolidMolecular weight:324.23Antalarmin hydrochloride
CAS:Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.Formula:C24H35ClN4Purity:99.84% - 99.85%Color and Shape:SolidMolecular weight:415.02VA-K-14 hydrochloride
CAS:VA-K-14 hydrochloride（VAK14 HCl） is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonalFormula:C18H16ClN3SPurity:99.37%Color and Shape:SolidMolecular weight:341.86Aplindore Fumarate
CAS:Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formula:C22H22N2O7Purity:99.66%Color and Shape:SolidMolecular weight:426.42Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurity:98.03% - 98.93%Color and Shape:SolidMolecular weight:346.47Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purity:99.99%Color and Shape:SolidMolecular weight:455.59LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purity:99.47%Color and Shape:SolidMolecular weight:372.89Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Formula:C24H40N2O3Purity:97.87% - >99.99%Color and Shape:SolidMolecular weight:404.59Repinotan
CAS:<p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>Formula:C21H24N2O4SPurity:99%Color and Shape:SolidMolecular weight:400.49Butofilolol
CAS:<p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>Formula:C17H26FNO3Purity:98.96% - >99.99%Color and Shape:SolidMolecular weight:311.392Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurity:99.67%Color and Shape:White Crystalline PowderMolecular weight:322.83Masilukast
CAS:Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated with inflammation.Formula:C31H32F3N3O5SPurity:99.23% - 99.62%Color and Shape:SolidMolecular weight:615.66Enerisant hydrochloride
CAS:<p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>Formula:C22H31ClN4O3Purity:99.95%Color and Shape:SolidMolecular weight:434.96Camonagrel
CAS:<p>Camonagrel is a compound that has inhibitory effects on Prostaglandin E2.</p>Formula:C15H16N2O3Purity:98.71% - 99.25%Color and Shape:SolidMolecular weight:272.3U 99194 maleate
CAS:U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formula:C21H31NO6Purity:99.45%Color and Shape:SolidMolecular weight:393.47Sitaxsentan
CAS:Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.Formula:C18H15ClN2O6S2Purity:97.99% - 98.71%Color and Shape:SolidMolecular weight:454.9Rilapine
CAS:<p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>Formula:C22H20ClN3Purity:97.76% - 99.20%Color and Shape:SolidMolecular weight:361.87Anpirtoline hydrochloride
CAS:<p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>Formula:C10H14Cl2N2SPurity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:265.20Remogliflozin etabonate
CAS:<p>Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.</p>Formula:C26H38N2O9Purity:98.98%Color and Shape:SolidMolecular weight:522.59L 674573
CAS:L 674573 is an inhibitor of leukotriene biosynthesis.Formula:C28H27NO3SPurity:99.51%Color and Shape:SolidMolecular weight:457.58MrgprX2 antagonist-8
CAS:<p>MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.</p>Formula:C24H24ClF3N4O3SPurity:98.61%Color and Shape:SolidMolecular weight:540.99SB228357
CAS:<p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>Formula:C22H17F4N3O2Purity:99.82%Color and Shape:SolidMolecular weight:431.38Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formula:C19H27N3OPurity:99.52%Color and Shape:SolidMolecular weight:313.44Efletirizine
CAS:<p>Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.</p>Formula:C21H24F2N2O3Purity:99.39%Color and Shape:SolidMolecular weight:390.42Amosulalol
CAS:<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Formula:C18H24N2O5SPurity:99.5%Color and Shape:SolidMolecular weight:380.46A2A receptor antagonist 1
CAS:<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Formula:C16H12FN5OPurity:99.52% - 99.93%Color and Shape:SolidMolecular weight:309.3GSK299115A
CAS:GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.Formula:C20H16Cl2N4O2Purity:99.81%Color and Shape:SolidMolecular weight:415.27ST 91
CAS:<p>ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.</p>Formula:C13H20ClN3Purity:99.83%Color and Shape:SolidMolecular weight:253.77Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:99.89%Color and Shape:SolidMolecular weight:483.56RG 7152
CAS:RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.Formula:C20H19N5O2Purity:98.45%Color and Shape:SolidMolecular weight:361.47-Hydroxy-DPAT hydrobromide
CAS:7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formula:C16H26BrNOPurity:99.73%Color and Shape:SolidMolecular weight:328.29LY-2624803
CAS:LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formula:C22H25N3O3Purity:99.78% - 99.97%Color and Shape:SolidMolecular weight:379.45Regrelor disodium
CAS:Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibitsFormula:C22H23N6Na2O8PPurity:99.89%Color and Shape:SolidMolecular weight:576.41DF-1111301
CAS:<p>DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.</p>Formula:C15H25Cl2N3OPurity:99.17%Color and Shape:SolidMolecular weight:334.29CB1 antagonist 1
CAS:CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, andFormula:C26H22Cl2N4Purity:98%Color and Shape:SolidMolecular weight:461.39TRAP-6-IN-1
CAS:<p>TRAP-6-IN-1 inhibits collagen/TRAP-6, IC50: 17.12/11.88 μM, blocks platelet aggregation.</p>Formula:C18H20O3Color and Shape:SolidMolecular weight:284.35LM-1484
CAS:LM-1484 displays a higher affinity for 3H-LTC4 sites and is an antagonist of CysLT1 receptor.Formula:C28H24N4O3Purity:98%Color and Shape:SolidMolecular weight:464.52LPA1 receptor antagonist 1
CAS:<p>LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a lysophosphatidic acid receptor antagonist for the study of idiopathic pulmonary fibrosis.</p>Formula:C28H26N4O4Purity:99.46% - 99.56%Color and Shape:SolidMolecular weight:482.53BAY 73-1449
CAS:BAY 73-1449 is a selective and potent antagonist of the prostacyclin receptor(IC50<0.1 nM).Formula:C26H23N3O3Purity:99.77%Color and Shape:SolidMolecular weight:425.48GR-127935
CAS:GR-127935 is a potent and selective 5-HT1B/1D receptor antagonist.Formula:C29H31N5O3Color and Shape:SolidMolecular weight:497.59SKF 81297
CAS:<p>SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].</p>Formula:C16H16ClNO2Purity:98%Color and Shape:SolidMolecular weight:289.765-HT2A&5-HT2C agonist-1
CAS:<p>5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.</p>Formula:C14H20N2OPurity:98%Color and Shape:SolidMolecular weight:232.32Timiperone
CAS:Timiperone exhibits a high affinity for cerebral dopamine D2 receptors, demonstrating antipsychotic activity as it mitigates stereotyped behavior.Formula:C22H24FN3OSPurity:98%Color and Shape:SolidMolecular weight:397.51Tachykinin angatonist 1
CAS:Tachykinin antagonist 1 is an antagonist of neurokinin receptors.Formula:C24H35Cl2N5O3SPurity:98%Color and Shape:SolidMolecular weight:544.54L-772,405
CAS:L-772,405 is a highly selective agonists of h5-HT(1D) receptor.Formula:C26H31FN6OPurity:98%Color and Shape:SolidMolecular weight:462.56DA-3934
CAS:DA-3934 targets gastrin/CCK-B receptors, not CCK-A, and reduces rat gastric acid secretion dose-dependently.Formula:C35H35N5O7Purity:98%Color and Shape:SolidMolecular weight:637.68ONO-0740556
CAS:ONO-0740556 is a potent agonist of the Gi-coupled human lysophosphatidic acid receptor 1 (LPA1), exhibiting an EC50 value of 0.26 nM.Formula:C20H34NO6PColor and Shape:SolidMolecular weight:415.46WLB-89462
CAS:WLB-89462 (Compound 20c) is a selective σ2 receptor ligand with a K i of 13 nM, exhibiting neuroprotective properties and the ability to ameliorate Aβ peptide-Formula:C21H29N5O3Purity:98%Color and Shape:SolidMolecular weight:399.49JNJ-28583867
CAS:JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.Formula:C24H32N2O2SColor and Shape:SolidMolecular weight:412.59Pronetalol
CAS:<p>Pronethalol ((±)-Pronethalol), a non-selective β-adrenergic antagonist, effectively inhibits Sox2 expression and offers protection against Digitalis-induced ventricular arrhythmias. Additionally, it can reverse such arrhythmias and limit the development of cerebral arteriovenous malformations (AVMs) [1] [2].</p>Formula:C15H19NOColor and Shape:SolidMolecular weight:229.32PF 514273
CAS:PF 514273 is a CB1 receptor antagonist.Formula:C21H17Cl2F2N3O2Purity:98%Color and Shape:SolidMolecular weight:452.28GSK494581A
CAS:GSK494581A is a GPR55 agonist and glycine transporter subtype 1 inhibitor.Formula:C27H28F2N2O4SPurity:98%Color and Shape:SolidMolecular weight:514.58ONO-2050297
CAS:ONO-2050297 is the first potent dual CysLT1 and CysLT2 antagonist with IC50 values of 0.017 μM (CysLT1) and 0.00087 μM (CysLT2), respectively.Formula:C31H34N2O7Color and Shape:SolidMolecular weight:546.61Wf-516
CAS:Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor and 5-HT2A receptor in humans, respectively), and with potent antidepressantFormula:C25H25Cl2N3O4Purity:98%Color and Shape:SolidMolecular weight:502.39Pentiapine
CAS:Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Formula:C15H17N5SPurity:99.35%Color and Shape:SolidMolecular weight:299.39AH13205
CAS:AH13205 is an agonist of EP2 prostanoid receptor.Formula:C24H36O4Purity:98%Color and Shape:SolidMolecular weight:388.54CP-293019
CAS:CP-293019 is a potent, selective antagonist of dopamine D4 receptor.Formula:C19H22F2N4OPurity:98%Color and Shape:SolidMolecular weight:360.4GSK-554418A
CAS:GSK-554418A, a novel azaindole CB(2) agonists, is used for the treatment of chronic pain. It is efficacious in the acute model and the chronic joint pain model.Formula:C19H19ClN4O2Color and Shape:SolidMolecular weight:370.83NH2-c[X-R-L-S-X]-K-G-P-(D-1Nal)
CAS:Compound 39, an APJ receptor agonist, has a K i of 0.6 nM, activates Gαi1 (EC50 0.8 nM), recruits β-arrestin2 (EC50 31 nM), and affects heart function.Formula:C49H73N13O11Color and Shape:SolidMolecular weight:1020.18RS 17053 hydrochloride
CAS:RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.Formula:C24H30Cl2N2O2Purity:99.27%Color and Shape:SolidMolecular weight:449.41Flesinoxan
CAS:Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Formula:C22H26FN3O4Color and Shape:SolidMolecular weight:415.46PD 165929
CAS:PD 165929 is a selective antagonist of Bombesin BB1.Formula:C37H47N5O2Purity:98%Color and Shape:SolidMolecular weight:593.82-Chloro-ATP
CAS:2-Chloro-ATP is a soluble inhibitor of guanylate cyclase (guanylate cyclase) that can increase intracellular calcium ion concentrations at low concentrations through a mechanism independent of inositol phosphate production.Formula:C10H15ClN5O13P3Color and Shape:SolidMolecular weight:541.63NBI-35965
CAS:<p>NBI-35965 is a CRF1 receptor antagonist.</p>Formula:C21H22Cl2N4Color and Shape:SolidMolecular weight:401.33
