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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5959 products of "GPCR/G-Protein"

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  • (S)-(+)-Dimethindene maleate

    CAS:
    (S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors
    Formula:C24H28N2O4
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:408.49

    Ref: TM-T23297

    1mg
    50.00€
  • Piribedil D8

    CAS:
    Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.
    Formula:C16H18N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.39

    Ref: TM-T12486

    1mg
    255.00€
    5mg
    To inquire
  • 4-Hydroxyatomoxetine D3

    CAS:
    4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.
    Formula:C17H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:274.37

    Ref: TM-T10144

    1mg
    329.00€
    5mg
    842.00€
  • Mozavaptan hydrochloride

    CAS:
    Mozavaptan is a vasopressin receptor antagonist.
    Formula:C27H30ClN3O2
    Color and Shape:Solid
    Molecular weight:464

    Ref: TM-T21465

    5mg
    43.00€
    1mL*10mM (DMSO)
    54.00€
  • Argipressin

    CAS:
    Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.
    Formula:C46H65N15O12S2
    Purity:98%
    Color and Shape:White Powder
    Molecular weight:1084.23

    Ref: TM-T7434

    1mg
    52.00€
    5mg
    94.00€
    10mg
    112.00€
  • SB-277011 hydrochloride

    CAS:
    SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.
    Formula:C28H31ClN4O
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:475.03

    Ref: TM-T63096

    2mg
    50.00€
  • L 888607

    CAS:
    L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).
    Formula:C19H15ClFNO2S
    Color and Shape:Solid
    Molecular weight:375.84

    Ref: TM-T15828

    5mg
    284.00€
    1mL*10mM (DMSO)
    281.00€
  • Nefazodone

    CAS:
    Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.
    Formula:C25H32ClN5O2
    Purity:99.85%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:470.01

    Ref: TM-T21451

    2mg
    42.00€
    5mg
    60.00€
    10mg
    87.00€
    25mg
    177.00€
    50mg
    276.00€
    100mg
    422.00€
    200mg
    604.00€
    1mL*10mM (DMSO)
    95.00€
  • SAR247799

    CAS:
    SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.
    Formula:C21H16ClN3O5
    Color and Shape:Solid
    Molecular weight:425.82

    Ref: TM-T38716

    5mg
    1,214.00€
  • Zaloglanstat

    CAS:
    Zaloglanstat (ISC-27864) is a selective, orally active mPGES-1 inhibitor with an IC50 of 5 nM, analgesic in osteoarthritis and inflammatory arthritis.
    Formula:C21H20ClF3N4O2
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:452.86

    Ref: TM-T39000

    1mg
    154.00€
    5mg
    371.00€
    10mg
    620.00€
    25mg
    1,305.00€
    50mg
    1,765.00€
    100mg
    2,367.00€
    1mL*10mM (DMSO)
    409.00€
  • Timapiprant sodium

    CAS:
    Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.
    Formula:C21H17FN2NaO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.367

    Ref: TM-T17099

    2mg
    34.00€
    1mL*10mM (DMSO)
    67.00€
  • TFLLR-NH2(TFA)

    CAS:
    TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)
    Formula:C33H54F3N9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:761.83

    Ref: TM-TP1334

    1mg
    163.00€
    5mg
    640.00€
  • Endothelin-3 (Rat,Human) (TFA)


    Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).
    Formula:C123H169F3N26O35S4·xC2HF3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2757.07 (free base)

    Ref: TM-TP1173

    1mg
    567.00€
  • Quetiapine-d8 Fumarate

    CAS:
    Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
    Formula:C25H21D8N3O6S
    Color and Shape:Solid
    Molecular weight:507.63

    Ref: TM-TMIJ-0315

    1mg
    To inquire
    5mg
    To inquire
  • Canagliflozin (Standard)

    CAS:
    Canagliflozin (Standard) is the standard substance of Canagliflozin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor that inhibits CHO cells expressing mSGLT2, rSGLT2, and hSGLT2 (IC50=2/3.7/4.4 nM). Canagliflozin can be used for the treatment of type II diabetes mellitus (T2DM).
    Formula:C24H25FO5S
    Color and Shape:Solid
    Molecular weight:444.52

    Ref: TM-TMSM-0636

    5mg
    63.00€
  • Aripiprazole (D8)

    CAS:
    Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).
    Formula:C23H27Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.44

    Ref: TM-T10368

    1mg
    254.00€
    5mg
    632.00€
  • GLP-1R modulator C5

    CAS:
    GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.
    Formula:C24H21NO3
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:371.43

    Ref: TM-T61483

    1mg
    39.00€
  • PD176252

    CAS:
    PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.
    Formula:C32H36N6O5
    Purity:99.00%
    Color and Shape:Solid
    Molecular weight:584.67

    Ref: TM-T16449

    1mg
    35.00€
    5mg
    67.00€
    10mg
    To inquire
    25mg
    To inquire
    1mL*10mM (DMSO)
    88.00€
  • Setiptiline maleate

    CAS:
    Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.
    Formula:C23H23NO4
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:377.43

    Ref: TM-T12900L

    10mg
    51.00€
    1mL*10mM (DMSO)
    51.00€
  • Cetirizine D4

    CAS:
    Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
    Formula:C21H25ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.91

    Ref: TM-T10769

    1mg
    258.00€
    5mg
    620.00€