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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • GSK189254A
    Targetmol
    + Info

    GSK189254A

    CAS:
    <p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>
    Formula:C21H25N3O2
    Purity:98.71% - 99.858%
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-TQ0066

  • SDZ WAG 994
    Targetmol
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    SDZ WAG 994

    CAS:
    <p>SDZ WAG 994 is an A1 adenosine receptor agonist.</p>
    Formula:C17H25N5O4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:363.41

    Ref: TM-T23347

  • GSK2018682
    Targetmol
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    GSK2018682

    CAS:
    <p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>
    Formula:C22H21ClN4O4
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:440.88

    Ref: TM-T7360

  • LY255283
    Targetmol
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    LY255283

    CAS:
    LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human PMNL and in monocytes.
    Formula:C19H28N4O3
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:360.45

    Ref: TM-T22946

  • S 14506 HCl
    Targetmol
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    S 14506 HCl

    CAS:
    <p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), &lt;6.0 (5-HT3).</p>
    Formula:C24H26FN3O2
    Color and Shape:Solid
    Molecular weight:407.48

    Ref: TM-T28637

  • PD 168568
    Targetmol
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    PD 168568

    CAS:
    <p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>
    Formula:C22H27N3O
    Color and Shape:Solid
    Molecular weight:349.47

    Ref: TM-T73215

  • Xamoterol
    Targetmol
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    Xamoterol

    CAS:
    <p>Xamoterol is a cardiac stimulant.</p>
    Formula:C16H25N3O5
    Color and Shape:Solid
    Molecular weight:339.39

    Ref: TM-T35153

  • T-1095
    Targetmol
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    T-1095

    CAS:
    <p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>
    Formula:C26H28O11
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:516.49

    Ref: TM-T9590

  • Regadenoson hydrate
    Targetmol
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    Regadenoson hydrate

    CAS:
    <p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>
    Formula:C15H20N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.37

    Ref: TM-T26054

  • Neuromedin N acetate(92169-45-4 free base)
    Targetmol
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    Neuromedin N acetate(92169-45-4 free base)

    <p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>
    Formula:C40H67N7O10
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:805.9

    Ref: TM-TP1085L

  • Methyldopa hydrate
    Targetmol
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    Methyldopa hydrate

    CAS:
    <p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>
    Formula:C10H13NO4H2O
    Purity:99.67%
    Color and Shape:White Solid
    Molecular weight:238.24

    Ref: TM-T5954

  • Tiprenolol
    Targetmol
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    Tiprenolol

    CAS:
    <p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>
    Formula:C13H21NO2S
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:255.38

    Ref: TM-T50081

  • Geissoschizine methyl ether
    Targetmol
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    Geissoschizine methyl ether

    CAS:
    <p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>
    Formula:C22H26N2O3
    Purity:99.24% - 99.68%
    Color and Shape:Solid
    Molecular weight:366.45

    Ref: TM-TN1032

  • Litorin acetate(55749-97-8 Free base)
    Targetmol
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    Litorin acetate(55749-97-8 Free base)

    <p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>
    Formula:C53H72N14O13S
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:1145.29

    Ref: TM-T20604L

  • Rolapitant hydrochloride hydrate
    Targetmol
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    Rolapitant hydrochloride hydrate

    CAS:
    <p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>
    Formula:C25H29ClF6N2O3
    Color and Shape:Solid
    Molecular weight:554.95

    Ref: TM-T68371

  • GSK 789472 hydrochloride
    Targetmol
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    GSK 789472 hydrochloride

    CAS:
    GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.
    Formula:C15H22ClN3O
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:295.81

    Ref: TM-T22817

  • Brompheniramine
    Targetmol
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    Brompheniramine

    CAS:
    <p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>
    Formula:C16H19BrN2
    Color and Shape:Solid
    Molecular weight:319.24

    Ref: TM-T60843

  • Siponimod hemifumarate
    Targetmol
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    Siponimod hemifumarate

    CAS:
    <p>Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.</p>
    Formula:C62H74F6N4O10
    Color and Shape:Solid
    Molecular weight:1149.282

    Ref: TM-T64065

  • Desipramine
    Targetmol
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    Desipramine

    CAS:
    <p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>
    Formula:C18H22N2
    Color and Shape:Solid
    Molecular weight:266.38

    Ref: TM-T60445

  • AC-55541
    Targetmol
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    AC-55541

    CAS:
    <p>AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.</p>
    Formula:C25H20BrN5O3
    Purity:98% - 99.33%
    Color and Shape:Solid
    Molecular weight:518.36

    Ref: TM-T2370