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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Dapagliflozin ((2S)-1,2-propanediol, hydrate)
    Targetmol
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    Dapagliflozin ((2S)-1,2-propanediol, hydrate)

    CAS:
    <p>Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-</p>
    Formula:C24H35ClO9
    Purity:99.88% - 99.94%
    Color and Shape:Solid
    Molecular weight:502.98

    Ref: TM-T4460

  • Hypidone hydrochloride
    Targetmol
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    Hypidone hydrochloride

    CAS:
    <p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>
    Formula:C18H23ClN2O2
    Purity:99.82% - 99.93%
    Color and Shape:Solid
    Molecular weight:334.84

    Ref: TM-T3648

  • Neuropeptide SF(mouse,rat) acetate
    Targetmol
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    Neuropeptide SF(mouse,rat) acetate

    <p>Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) &amp; 12.1 nM (NPFF2), enhancing ASIC3 current.</p>
    Formula:C42H69N13O12
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:948.08

    Ref: TM-TP1884L1

  • Quipazine maleate
    Targetmol
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    Quipazine maleate

    CAS:
    <p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>
    Formula:C17H19N3O4
    Color and Shape:Solid
    Molecular weight:329.36

    Ref: TM-T71792

  • Pridopidine
    Targetmol
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    Pridopidine

    CAS:
    <p>Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.</p>
    Formula:C15H23NO2S
    Purity:95.2% - 99.89%
    Color and Shape:Solid
    Molecular weight:281.41

    Ref: TM-T7352

  • lumateperone Tosylate
    Targetmol
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    lumateperone Tosylate

    CAS:
    <p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>
    Formula:C31H36FN3O4S
    Purity:95.83% - 99.95%
    Color and Shape:Solid
    Molecular weight:565.7

    Ref: TM-TQ0084

  • Tandospirone hydrochloride
    Targetmol
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    Tandospirone hydrochloride

    CAS:
    <p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>
    Formula:C21H30ClN5O2
    Color and Shape:Solid
    Molecular weight:419.95

    Ref: TM-T62215

  • GR 94800 acetate
    Targetmol
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    GR 94800 acetate

    <p>GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.</p>
    Formula:C51H65N9O10
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:964.12

    Ref: TM-T22811L

  • Myristicin
    Targetmol
    + Info

    Myristicin

    CAS:
    <p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>
    Formula:C11H12O3
    Purity:99.828%
    Color and Shape:Liquid
    Molecular weight:192.21

    Ref: TM-T9113

  • Peptide YY (PYY) (3-36), human
    Targetmol
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    Peptide YY (PYY) (3-36), human

    CAS:
    <p>Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.</p>
    Formula:C176H272N52O54
    Purity:97.76%
    Color and Shape:Solid
    Molecular weight:3980.42

    Ref: TM-TP1059

  • Chlorprothixene
    Targetmol
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    Chlorprothixene

    CAS:
    <p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>
    Formula:C18H18ClNS
    Purity:98.77% - 99.756%
    Color and Shape:Pale Yellow Crystals Solid
    Molecular weight:315.86

    Ref: TM-T0074

  • CJC-1295 acetate(863288-34-0 free base)
    Targetmol
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    CJC-1295 acetate(863288-34-0 free base)

    <p>CJC-1295 acetate is a synthetic GHRH analogue and GHS.</p>
    Formula:C154H256N44O44
    Purity:97.29%
    Color and Shape:Solid
    Molecular weight:3428.01

    Ref: TM-TP2328L

  • Nitrobenzylthioinosine
    Targetmol
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    Nitrobenzylthioinosine

    CAS:
    <p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>
    Formula:C17H17N5O6S
    Purity:99.69% - 99.74%
    Color and Shape:Off-White Solid
    Molecular weight:419.41

    Ref: TM-T8551

  • Doxazosin
    Targetmol
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    Doxazosin

    CAS:
    <p>Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.</p>
    Formula:C23H25N5O5
    Purity:99.47% - 99.87%
    Color and Shape:Solid
    Molecular weight:451.48

    Ref: TM-T22316

  • Nifenalol
    Targetmol
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    Nifenalol

    CAS:
    <p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>
    Formula:C11H16N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:224.26

    Ref: TM-T8663L

  • CP 376395
    Targetmol
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    CP 376395

    CAS:
    <p>CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.</p>
    Formula:C21H30N2O
    Purity:99.86% - 99.94%
    Color and Shape:Solid
    Molecular weight:326.48

    Ref: TM-T4329

  • Triptorelin acetate(57773-63-4 free base)
    Targetmol
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    Triptorelin acetate(57773-63-4 free base)

    CAS:
    <p>Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.</p>
    Formula:C66H86N18O15
    Purity:99.90%
    Color and Shape:White Powder
    Molecular weight:1371.53

    Ref: TM-T21410

  • Olcegepant
    Targetmol
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    Olcegepant

    CAS:
    <p>Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4</p>
    Formula:C38H47Br2N9O5
    Purity:96.08% - 97.24%
    Color and Shape:Solid
    Molecular weight:869.65

    Ref: TM-T12293L

  • Substance P 1-9 aceate
    Targetmol
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    Substance P 1-9 aceate

    <p>Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.</p>
    Formula:C54H81N15O14
    Purity:99.01%
    Color and Shape:Solid
    Molecular weight:1164.31

    Ref: TM-TP1819L

  • Sigma-LIGAND-1 hydrochloride
    Targetmol
    + Info

    Sigma-LIGAND-1 hydrochloride

    CAS:
    <p>Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.</p>
    Formula:C27H34ClNO4
    Color and Shape:Solid
    Molecular weight:472.02

    Ref: TM-T63048