GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(155 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5971 products of "GPCR/G-Protein"
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Bay 59-3074
CAS:Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).
Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36Galanin (1-16), mouse, porcine, rat
CAS:Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.Formula:C78H116N20O21Purity:98.65%Color and Shape:White PowderMolecular weight:1669.88(+)-PD 128907 hydrochloride
CAS:(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Formula:C14H20ClNO3Purity:97.76%Color and Shape:SolidMolecular weight:285.77Montelukast sodium
CAS:Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.Formula:C35H35ClNNaO3SPurity:99.14% - 99.89%Color and Shape:White To Off-White Crystalline PowderMolecular weight:608.17RFRP3(human) acetate(311309-27-0 free base)
RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.Formula:C47H76N14O12Purity:97.09%Color and Shape:SolidMolecular weight:1029.19Dexmedetomidine
CAS:Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.Formula:C13H16N2Purity:99% - >99.99%Color and Shape:SolidMolecular weight:200.28Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formula:C18H26ClN3O3·C4H6O4Purity:99.24%Color and Shape:SolidMolecular weight:485.96AM211
CAS:AM211 (AM211 free acid) is a potent and orally bioavailable antagonist of prostaglandin D2 (PGD2) receptor type 2 (DP2)Formula:C27H27F3N2O4Purity:≥95%Color and Shape:SolidMolecular weight:500.51nifenalol.HCl
CAS:Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.Formula:C11H17ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:260.72GW627368
CAS:GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.Formula:C30H28N2O6SPurity:99.75% - 99.92%Color and Shape:SolidMolecular weight:544.62Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formula:C20H21F3N4OPurity:99.37% - 99.93%Color and Shape:White PowderMolecular weight:390.41-Oleoyl lysophosphatidic acid sodium
CAS:1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formula:C21H40O7P·NaPurity:98.75% - 99.24%Color and Shape:SolidMolecular weight:458.51BAY 41-2272
CAS:BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.Formula:C20H17FN6Purity:99.54%Color and Shape:SolidMolecular weight:360.39SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurity:99.61%Color and Shape:SolidMolecular weight:266.3Decloxizine dihydrochloride
CAS:Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.
Formula:C21H28N2O2·2ClHPurity:99.73%Color and Shape:SolidMolecular weight:413.39ML221
CAS:ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM inFormula:C17H11N3O6SPurity:97.74%Color and Shape:SolidMolecular weight:385.35Ref: TM-T4390
2mgTo inquire5mg52.00€10mg85.00€25mg144.00€50mg227.00€100mg369.00€200mgTo inquire1mL*10mM (DMSO)55.00€Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formula:C24H30N2O2SPurity:99.9% - 99.92%Color and Shape:SolidMolecular weight:410.57Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurity:98.64% - 99.97%Color and Shape:SolidMolecular weight:623.63Ref: TM-T3630
2mg39.00€5mg58.00€10mg93.00€25mg167.00€50mg250.00€100mg408.00€200mg585.00€1mL*10mM (DMSO)81.00€Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formula:C114H174N34O31Purity:99.05%Color and Shape:SolidMolecular weight:2516.81Ref: TM-TP2279L
1mg77.00€2mg97.00€5mg156.00€10mg225.00€25mg375.00€50mg535.00€100mg730.00€200mg938.00€Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formula:C76H117N19O22SPurity:95.43%Color and Shape:SolidMolecular weight:1680.94
