GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5980 products of "GPCR/G-Protein"
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γ-Mangostin
CAS:<p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>Formula:C23H24O6Purity:98.55% - 99.08%Color and Shape:SolidMolecular weight:396.43VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Formula:C13H15ClN4Purity:99.66%Color and Shape:SolidMolecular weight:262.74Buclizine
CAS:Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Formula:C28H33ClN2Color and Shape:SolidMolecular weight:433.03Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formula:C28H36N4O2SPurity:99.78% - 99.91%Color and Shape:SolidMolecular weight:492.68Ramosetron
CAS:Ramosetron 是一种血清素 5-HT3 受体拮抗剂，用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。Formula:C17H17N3OPurity:98.84%Color and Shape:SolidMolecular weight:279.34Nonapeptide-1 acetate salt (158563-45-2 free base)
<p>Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH)</p>Formula:C63H91N15O11SPurity:98.26%Color and Shape:SolidMolecular weight:1266.58SR 57227 hydrochloride
CAS:SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Formula:C10H14ClN3·HClPurity:99.89%Color and Shape:SolidMolecular weight:248.15BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formula:C26H31N3O2Purity:99.44%Color and Shape:SolidMolecular weight:417.54Ref: TM-T9100
1mg80.00€5mg162.00€10mg227.00€25mg379.00€50mg540.00€100mg730.00€200mg938.00€1mL*10mM (DMSO)177.00€Alloxazine
CAS:Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formula:C10H6N4O2Purity:99.75%Color and Shape:SolidMolecular weight:214.18Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Formula:C5H81N13O14Purity:99.37%Color and Shape:SolidMolecular weight:1148.31Droxidopa
CAS:Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.Formula:C9H11NO5Purity:97.27% - 99.88%Color and Shape:SolidMolecular weight:213.19TC-G-1008
CAS:TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).Formula:C18H19ClN6O2SPurity:97.37% - 99%Color and Shape:SolidMolecular weight:418.9Ref: TM-T4648
1mg38.00€5mg80.00€10mg120.00€25mg215.00€50mg354.00€100mg588.00€200mg833.00€1mL*10mM (DMSO)88.00€NPS-2143 hydrochloride
CAS:NPS-2143 hydrochloride (NPS-2143 HCL) is a selective potent calcium ion-sensing receptor antagonist.Formula:C24H25ClN2O2·HClPurity:99.38% - 99.67%Color and Shape:SolidMolecular weight:445.38Ref: TM-T4967
1mg46.00€2mg59.00€5mg92.00€10mg126.00€25mg215.00€50mg339.00€100mg502.00€1mL*10mM (DMSO)90.00€AF38469
CAS:AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).Formula:C15H11F3N2O3Purity:99.18%Color and Shape:SolidMolecular weight:324.25Ref: TM-TQ0086
1mg87.00€2mg120.00€5mg180.00€10mg283.00€25mg550.00€50mg847.00€100mg1,159.00€200mg1,549.00€1mL*10mM (DMSO)188.00€Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Exenatide
CAS:Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.Formula:C186H286N50O62SPurity:99.42%Color and Shape:SolidMolecular weight:4247Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formula:C32H44F3N3O2SPurity:98.14%Color and Shape:SolidMolecular weight:591.77Amezinium methylsulfate
CAS:Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.Formula:C12H15N3O5SPurity:99.64% - 99.99%Color and Shape:SolidMolecular weight:313.33Levobetaxolol hydrochloride
CAS:Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.Formula:C18H29NO3·HClPurity:98.80% - 99.69%Color and Shape:SolidMolecular weight:343.89FAUC 213
CAS:<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Formula:C18H19ClN4Purity:99.84%Color and Shape:SolidMolecular weight:326.82
