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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5981 products of "GPCR/G-Protein"

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  • Adenosine amine congener

    CAS:
    Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
    Formula:C28H32N8O6
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:576.6

    Ref: TM-T7683

    1mg
    70.00€
    5mg
    152.00€
    10mg
    222.00€
    25mg
    403.00€
    50mg
    593.00€
    100mg
    845.00€
    1mL*10mM (DMSO)
    234.00€
  • Geissoschizine methyl ether

    CAS:
    Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.
    Formula:C22H26N2O3
    Purity:99.24% - 99.68%
    Color and Shape:Solid
    Molecular weight:366.45

    Ref: TM-TN1032

    1mg
    137.00€
    2mg
    197.00€
    5mg
    338.00€
    10mg
    512.00€
    25mg
    812.00€
    50mg
    1,093.00€
    100mg
    1,473.00€
    1mL*10mM (DMSO)
    344.00€
  • Mecamylamine

    CAS:
    Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.
    Formula:C11H21N
    Color and Shape:Solid
    Molecular weight:167.29

    Ref: TM-T69019

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Eptapirone

    CAS:
    Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.
    Formula:C16H23N7O2
    Purity:99.39% - 99.65%
    Color and Shape:Solid
    Molecular weight:345.4

    Ref: TM-T3179

    10mg
    52.00€
    25mg
    90.00€
    50mg
    145.00€
    100mg
    210.00€
    200mg
    304.00€
    1mL*10mM (DMSO)
    35.00€
  • LY255283

    CAS:
    LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human PMNL and in monocytes.
    Formula:C19H28N4O3
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:360.45

    Ref: TM-T22946

    2mg
    47.00€
    5mg
    88.00€
    10mg
    127.00€
    25mg
    250.00€
    50mg
    401.00€
    100mg
    645.00€
    200mg
    898.00€
    1mL*10mM (DMSO)
    87.00€
  • Motilin (26-47), human, porcine

    CAS:
    Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.
    Formula:C120H188N34O35S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2699.07

    Ref: TM-TP1425

    1mg
    117.00€
    5mg
    353.00€
    10mg
    532.00€
    25mg
    787.00€
    50mg
    1,054.00€
    100mg
    1,415.00€
    200mg
    1,872.00€
    500µg
    90.00€
  • Melitracen hydrochloride

    CAS:
    Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.
    Formula:C21H26ClN
    Purity:99.99%
    Color and Shape:Crystalline Solid
    Molecular weight:327.90

    Ref: TM-T4274

    10mg
    47.00€
    25mg
    67.00€
    50mg
    87.00€
    100mg
    116.00€
    200mg
    170.00€
    500mg
    279.00€
    1mL*10mM (DMSO)
    50.00€
  • Lecirelin acetate(61012-19-9 free base)


    Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts
    Formula:C61H88N16O14
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:1269.45

    Ref: TM-TP1434L

    1mg
    74.00€
    5mg
    131.00€
    10mg
    180.00€
    25mg
    269.00€
    50mg
    323.00€
    100mg
    487.00€
  • R243

    CAS:
    R243 is CCR8 signaling and chemotaxis inhibitor.
    Formula:C21H27NO4
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:357.44

    Ref: TM-T24700

    1mg
    43.00€
    2mg
    56.00€
    5mg
    85.00€
    10mg
    124.00€
    25mg
    220.00€
    50mg
    350.00€
    100mg
    522.00€
    1mL*10mM (DMSO)
    95.00€
  • Pipamperone HCl

    CAS:
    Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.
    Formula:C21H31ClFN3O2
    Color and Shape:Solid
    Molecular weight:411.95

    Ref: TM-T28417

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • SAG hydrochloride (912545-86-9(free base))

    CAS:
    SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.
    Formula:C28H29Cl2N3OS
    Purity:99.19% - 99.97%
    Color and Shape:Solid
    Molecular weight:526.52

    Ref: TM-T4211

    1mg
    49.00€
    2mg
    65.00€
    5mg
    90.00€
    10mg
    114.00€
    25mg
    222.00€
    50mg
    334.00€
    100mg
    502.00€
    200mg
    717.00€
    1mL*10mM (DMSO)
    105.00€
  • Sonidegib

    CAS:
    Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.
    Formula:C26H26F3N3O3
    Purity:98% - 99.97%
    Color and Shape:Solid
    Molecular weight:485.5

    Ref: TM-T1926

    5mg
    59.00€
    10mg
    84.00€
    25mg
    116.00€
    50mg
    161.00€
    100mg
    260.00€
    1mL*10mM (DMSO)
    64.00€
  • Vercirnon

    CAS:
    Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.
    Formula:C22H21ClN2O4S
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:444.93

    Ref: TM-T17225

    1mg
    105.00€
    5mg
    259.00€
    10mg
    406.00€
    25mg
    680.00€
    50mg
    938.00€
    100mg
    1,301.00€
    500mg
    2,593.00€
    1mL*10mM (DMSO)
    363.00€
  • Salmeterol Xinafoate

    CAS:
    <p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>
    Formula:C36H45NO7
    Purity:98% - 98.24%
    Color and Shape:White Solid
    Molecular weight:603.75

    Ref: TM-T6653

    5mg
    50.00€
    10mg
    79.00€
    25mg
    140.00€
    50mg
    227.00€
    100mg
    376.00€
  • MK 571

    CAS:
    <p>MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.</p>
    Formula:C26H27ClN2O3S2
    Purity:98.69% - 99.65%
    Color and Shape:Solid
    Molecular weight:515.09

    Ref: TM-T7841

    2mg
    35.00€
    5mg
    52.00€
    10mg
    86.00€
    25mg
    168.00€
    50mg
    301.00€
    100mg
    455.00€
    200mg
    652.00€
  • SDZ WAG 994

    CAS:
    SDZ WAG 994 is an A1 adenosine receptor agonist.
    Formula:C17H25N5O4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:363.41

    Ref: TM-T23347

    1mg
    63.00€
    5mg
    114.00€
    10mg
    172.00€
    25mg
    299.00€
    50mg
    432.00€
    100mg
    587.00€
    200mg
    792.00€
    1mL*10mM (DMSO)
    120.00€
  • AF38469

    CAS:
    AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
    Formula:C15H11F3N2O3
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:324.25

    Ref: TM-TQ0086

    1mg
    87.00€
    2mg
    120.00€
    5mg
    180.00€
    10mg
    283.00€
    25mg
    550.00€
    50mg
    847.00€
    100mg
    1,159.00€
    200mg
    1,549.00€
    1mL*10mM (DMSO)
    188.00€
  • MRT-81

    CAS:
    MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.
    Formula:C31H29N3O5S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:555.64

    Ref: TM-T9532

    1mg
    48.00€
    5mg
    97.00€
    10mg
    145.00€
    25mg
    255.00€
    50mg
    368.00€
    100mg
    505.00€
    200mg
    692.00€
    1mL*10mM (DMSO)
    116.00€
  • MRT-10

    CAS:
    <p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>
    Formula:C24H23N3O5S
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:465.52

    Ref: TM-T23027

    2mg
    48.00€
    5mg
    67.00€
    10mg
    95.00€
    25mg
    185.00€
    50mg
    264.00€
    100mg
    370.00€
    200mg
    504.00€
  • RS102895

    CAS:
    RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.
    Formula:C21H21F3N2O2
    Purity:97.64% - 99.80%
    Color and Shape:Solid
    Molecular weight:390.4

    Ref: TM-TQ0283

    2mg
    42.00€
    5mg
    62.00€
    10mg
    90.00€
    25mg
    166.00€
    50mg
    241.00€
    100mg
    359.00€
    1mL*10mM (DMSO)
    69.00€