
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(54 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5981 products of "GPCR/G-Protein"
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Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Geissoschizine methyl ether
CAS:Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Formula:C22H26N2O3Purity:99.24% - 99.68%Color and Shape:SolidMolecular weight:366.45Ref: TM-TN1032
1mg137.00€2mg197.00€5mg338.00€10mg512.00€25mg812.00€50mg1,093.00€100mg1,473.00€1mL*10mM (DMSO)344.00€Mecamylamine
CAS:Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formula:C11H21NColor and Shape:SolidMolecular weight:167.29Eptapirone
CAS:Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formula:C16H23N7O2Purity:99.39% - 99.65%Color and Shape:SolidMolecular weight:345.4LY255283
CAS:LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human PMNL and in monocytes.Formula:C19H28N4O3Purity:99.18%Color and Shape:SolidMolecular weight:360.45Ref: TM-T22946
2mg47.00€5mg88.00€10mg127.00€25mg250.00€50mg401.00€100mg645.00€200mg898.00€1mL*10mM (DMSO)87.00€Motilin (26-47), human, porcine
CAS:Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.Formula:C120H188N34O35SPurity:98%Color and Shape:SolidMolecular weight:2699.07Ref: TM-TP1425
1mg117.00€5mg353.00€10mg532.00€25mg787.00€50mg1,054.00€100mg1,415.00€200mg1,872.00€500µg90.00€Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurity:99.99%Color and Shape:Crystalline SolidMolecular weight:327.90Ref: TM-T4274
10mg47.00€25mg67.00€50mg87.00€100mg116.00€200mg170.00€500mg279.00€1mL*10mM (DMSO)50.00€Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purity:98.1%Color and Shape:SolidMolecular weight:1269.45R243
CAS:R243 is CCR8 signaling and chemotaxis inhibitor.Formula:C21H27NO4Purity:99.03%Color and Shape:SolidMolecular weight:357.44Ref: TM-T24700
1mg43.00€2mg56.00€5mg85.00€10mg124.00€25mg220.00€50mg350.00€100mg522.00€1mL*10mM (DMSO)95.00€Pipamperone HCl
CAS:Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formula:C21H31ClFN3O2Color and Shape:SolidMolecular weight:411.95SAG hydrochloride (912545-86-9(free base))
CAS:SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.Formula:C28H29Cl2N3OSPurity:99.19% - 99.97%Color and Shape:SolidMolecular weight:526.52Ref: TM-T4211
1mg49.00€2mg65.00€5mg90.00€10mg114.00€25mg222.00€50mg334.00€100mg502.00€200mg717.00€1mL*10mM (DMSO)105.00€Sonidegib
CAS:Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.Formula:C26H26F3N3O3Purity:98% - 99.97%Color and Shape:SolidMolecular weight:485.5Vercirnon
CAS:Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.Formula:C22H21ClN2O4SPurity:99.23%Color and Shape:SolidMolecular weight:444.93Ref: TM-T17225
1mg105.00€5mg259.00€10mg406.00€25mg680.00€50mg938.00€100mg1,301.00€500mg2,593.00€1mL*10mM (DMSO)363.00€Salmeterol Xinafoate
CAS:<p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>Formula:C36H45NO7Purity:98% - 98.24%Color and Shape:White SolidMolecular weight:603.75MK 571
CAS:<p>MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.</p>Formula:C26H27ClN2O3S2Purity:98.69% - 99.65%Color and Shape:SolidMolecular weight:515.09SDZ WAG 994
CAS:SDZ WAG 994 is an A1 adenosine receptor agonist.Formula:C17H25N5O4Purity:99.82%Color and Shape:SolidMolecular weight:363.41Ref: TM-T23347
1mg63.00€5mg114.00€10mg172.00€25mg299.00€50mg432.00€100mg587.00€200mg792.00€1mL*10mM (DMSO)120.00€AF38469
CAS:AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).Formula:C15H11F3N2O3Purity:99.18%Color and Shape:SolidMolecular weight:324.25Ref: TM-TQ0086
1mg87.00€2mg120.00€5mg180.00€10mg283.00€25mg550.00€50mg847.00€100mg1,159.00€200mg1,549.00€1mL*10mM (DMSO)188.00€MRT-81
CAS:MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.Formula:C31H29N3O5SPurity:99.72%Color and Shape:SolidMolecular weight:555.64Ref: TM-T9532
1mg48.00€5mg97.00€10mg145.00€25mg255.00€50mg368.00€100mg505.00€200mg692.00€1mL*10mM (DMSO)116.00€MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Formula:C24H23N3O5SPurity:99.73%Color and Shape:SolidMolecular weight:465.52RS102895
CAS:RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.Formula:C21H21F3N2O2Purity:97.64% - 99.80%Color and Shape:SolidMolecular weight:390.4
