
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).Formula:C39H65N9O9Purity:>99.99%Color and Shape:SolidMolecular weight:803.99BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.Formula:C118H190N36O30S2Purity:96.86%Color and Shape:SolidMolecular weight:2657.12Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purity:99.33%Color and Shape:SolidMolecular weight:354.27Ralinepag
CAS:Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human andFormula:C23H26ClNO5Purity:99.79% - 99.85%Color and Shape:SolidMolecular weight:431.91Ref: TM-T4635
1mg52.00€2mgTo inquire5mg111.00€10mg170.00€25mg301.00€50mg424.00€100mg605.00€200mg848.00€1mL*10mM (DMSO)124.00€Rolapitant hydrochloride hydrate
CAS:Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.Formula:C25H29ClF6N2O3Color and Shape:SolidMolecular weight:554.95Puerarin
CAS:Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.Formula:C21H20O9Purity:98.90% - 99.21%Color and Shape:Yellow Brown Fine PowderMolecular weight:416.38Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55Ciliobrevin A
CAS:Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.Formula:C17H9Cl2N3O2Purity:98.54% - 99.57%Color and Shape:SolidMolecular weight:358.18Ref: TM-T3156
2mg42.00€5mg59.00€10mg85.00€25mg168.00€50mg235.00€100mg331.00€200mg492.00€1mL*10mM (DMSO)69.00€Plecanatide
CAS:Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.Formula:C65H104N18O26S4Purity:97.51%Color and Shape:SolidMolecular weight:1681.89SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Formula:C28H28ClN3OSPurity:97.37% - 98.88%Color and Shape:SolidMolecular weight:490.06MCL0020
CAS:MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.Formula:C34H39N7O4Purity:99.18%Color and Shape:SolidMolecular weight:609.72Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852Clozapine HCl
CAS:Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.Formula:C18H20Cl2N4Color and Shape:SolidMolecular weight:363.29Glasdegib
CAS:Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.Formula:C21H22N6OPurity:98.72%Color and Shape:SolidMolecular weight:374.44BX471
CAS:BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.Formula:C21H24ClFN4O3Purity:98% - 99.98%Color and Shape:SolidMolecular weight:434.89Ref: TM-T2375
1mg38.00€5mg90.00€10mg124.00€25mg212.00€50mg329.00€100mg515.00€200mg782.00€1mL*10mM (DMSO)90.00€Ro 46-2005
CAS:Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).Formula:C23H27N3O6SPurity:98.02% - 98.8%Color and Shape:SolidMolecular weight:473.54Emedastine
CAS:Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.Formula:C17H26N4OPurity:97.1% - 97.76%Color and Shape:OilMolecular weight:302.41Ref: TM-T3979
1mg34.00€5mg74.00€10mg109.00€25mg177.00€50mg264.00€100mg394.00€500mg883.00€1mL*10mM (DMSO)82.00€Bavisant dihydrochloride hydrate
CAS:Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.Formula:C19H31Cl2N3O3Color and Shape:SolidMolecular weight:420.38AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:98.87%Color and Shape:SolidMolecular weight:478.47Ref: TM-T2000
1mg35.00€2mg47.00€5mg66.00€10mg97.00€25mg180.00€50mg283.00€100mg439.00€1mL*10mM (DMSO)70.00€SORT-PGRN interaction inhibitor 1
CAS:SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).Formula:C15H18N2O2Purity:98.72%Color and Shape:SolidMolecular weight:258.32
