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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • [Lys5,MeLeu9,Nle10]-NKA(4-10)

    CAS:
    Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
    Formula:C39H65N9O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:803.99

    Ref: TM-TP1883

    1mg
    96.00€
    5mg
    231.00€
    10mg
    343.00€
    25mg
    532.00€
    50mg
    735.00€
    100mg
    982.00€
    200mg
    1,333.00€
  • BWX 46 Acetate


    BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
    Formula:C118H190N36O30S2
    Purity:96.86%
    Color and Shape:Solid
    Molecular weight:2657.12

    Ref: TM-T21611L

    1mg
    240.00€
    2mg
    335.00€
    5mg
    500.00€
    10mg
    722.00€
    25mg
    1,121.00€
    50mg
    1,501.00€
    100mg
    2,023.00€
  • Metoclopramide hydrochloride hydrate

    CAS:
    Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.
    Formula:C14H25Cl2N3O3
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:354.27

    Ref: TM-T8385

    1g
    126.00€
    50mg
    38.00€
    100mg
    52.00€
    500mg
    87.00€
  • Ralinepag

    CAS:
    Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human and
    Formula:C23H26ClNO5
    Purity:99.79% - 99.85%
    Color and Shape:Solid
    Molecular weight:431.91

    Ref: TM-T4635

    1mg
    52.00€
    2mg
    To inquire
    5mg
    111.00€
    10mg
    170.00€
    25mg
    301.00€
    50mg
    424.00€
    100mg
    605.00€
    200mg
    848.00€
    1mL*10mM (DMSO)
    124.00€
  • Rolapitant hydrochloride hydrate

    CAS:
    Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.
    Formula:C25H29ClF6N2O3
    Color and Shape:Solid
    Molecular weight:554.95

    Ref: TM-T68371

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Puerarin

    CAS:
    Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.
    Formula:C21H20O9
    Purity:98.90% - 99.21%
    Color and Shape:Yellow Brown Fine Powder
    Molecular weight:416.38

    Ref: TM-T2815

    5mg
    51.00€
    10mg
    88.00€
    25mg
    160.00€
    50mg
    235.00€
    100mg
    354.00€
    500mg
    825.00€
    1mL*10mM (DMSO)
    87.00€
  • Histrelin acetate

    CAS:
    Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.
    Formula:C68H90N18O14
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:1383.55

    Ref: TM-TP2107L

    1mg
    84.00€
    5mg
    166.00€
    10mg
    260.00€
    25mg
    440.00€
    50mg
    617.00€
    100mg
    873.00€
  • Ciliobrevin A

    CAS:
    Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.
    Formula:C17H9Cl2N3O2
    Purity:98.54% - 99.57%
    Color and Shape:Solid
    Molecular weight:358.18

    Ref: TM-T3156

    2mg
    42.00€
    5mg
    59.00€
    10mg
    85.00€
    25mg
    168.00€
    50mg
    235.00€
    100mg
    331.00€
    200mg
    492.00€
    1mL*10mM (DMSO)
    69.00€
  • Plecanatide

    CAS:
    Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.
    Formula:C65H104N18O26S4
    Purity:97.51%
    Color and Shape:Solid
    Molecular weight:1681.89

    Ref: TM-T9080

    1mg
    79.00€
    5mg
    180.00€
    10mg
    298.00€
    25mg
    590.00€
    50mg
    835.00€
    100mg
    1,121.00€
  • SAG

    CAS:
    <p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>
    Formula:C28H28ClN3OS
    Purity:97.37% - 98.88%
    Color and Shape:Solid
    Molecular weight:490.06

    Ref: TM-T1779

    1mg
    48.00€
    2mg
    62.00€
    5mg
    90.00€
    10mg
    120.00€
    25mg
    234.00€
    50mg
    323.00€
    100mg
    477.00€
    200mg
    682.00€
  • MCL0020

    CAS:
    MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.
    Formula:C34H39N7O4
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:609.72

    Ref: TM-TP1889

    1mg
    110.00€
    5mg
    269.00€
    10mg
    371.00€
    25mg
    572.00€
    50mg
    783.00€
    100mg
    1,035.00€
    200mg
    1,404.00€
  • Triprolidine hydrochloride

    CAS:
    Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.
    Formula:C19H23ClN2
    Color and Shape:Solid
    Molecular weight:314.852

    Ref: TM-T21112

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Clozapine HCl

    CAS:
    Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.
    Formula:C18H20Cl2N4
    Color and Shape:Solid
    Molecular weight:363.29

    Ref: TM-T69129

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Glasdegib

    CAS:
    Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.
    Formula:C21H22N6O
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:374.44

    Ref: TM-T6514

    1mg
    43.00€
    5mg
    87.00€
    10mg
    145.00€
    25mg
    303.00€
    50mg
    512.00€
    100mg
    740.00€
    1mL*10mM (DMSO)
    96.00€
  • BX471

    CAS:
    BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.
    Formula:C21H24ClFN4O3
    Purity:98% - 99.98%
    Color and Shape:Solid
    Molecular weight:434.89

    Ref: TM-T2375

    1mg
    38.00€
    5mg
    90.00€
    10mg
    124.00€
    25mg
    212.00€
    50mg
    329.00€
    100mg
    515.00€
    200mg
    782.00€
    1mL*10mM (DMSO)
    90.00€
  • Ro 46-2005

    CAS:
    Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).
    Formula:C23H27N3O6S
    Purity:98.02% - 98.8%
    Color and Shape:Solid
    Molecular weight:473.54

    Ref: TM-T3194

    5mg
    43.00€
    10mg
    75.00€
    25mg
    124.00€
    50mg
    200.00€
    100mg
    288.00€
    200mg
    414.00€
    1mL*10mM (DMSO)
    47.00€
  • Emedastine

    CAS:
    Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
    Formula:C17H26N4O
    Purity:97.1% - 97.76%
    Color and Shape:Oil
    Molecular weight:302.41

    Ref: TM-T3979

    1mg
    34.00€
    5mg
    74.00€
    10mg
    109.00€
    25mg
    177.00€
    50mg
    264.00€
    100mg
    394.00€
    500mg
    883.00€
    1mL*10mM (DMSO)
    82.00€
  • Bavisant dihydrochloride hydrate

    CAS:
    Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.
    Formula:C19H31Cl2N3O3
    Color and Shape:Solid
    Molecular weight:420.38

    Ref: TM-T10462L

    2mg
    87.00€
    50mg
    750.00€
    100mg
    1,179.00€
  • AM095

    CAS:
    AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.
    Formula:C27H23N2NaO5
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:478.47

    Ref: TM-T2000

    1mg
    35.00€
    2mg
    47.00€
    5mg
    66.00€
    10mg
    97.00€
    25mg
    180.00€
    50mg
    283.00€
    100mg
    439.00€
    1mL*10mM (DMSO)
    70.00€
  • SORT-PGRN interaction inhibitor 1

    CAS:
    SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
    Formula:C15H18N2O2
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:258.32

    Ref: TM-T9044

    10mg
    33.00€
    1mL*10mM (DMSO)
    33.00€