GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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BGC-20-1531 hydrochloride(1186532-61-5 free base)
CAS:<p>BGC-20-1531 hydrochloride(1186532-61-5 free base) (GTPL3380 hydrochloride) is a EP4 antagonist for the treatment of acute migraine.</p>Formula:C26H25ClN2O6SPurity:98.94% - 99.85%Color and Shape:SolidMolecular weight:529GLP-1 receptor agonist 9
CAS:1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.Formula:C32H31ClFN3O5Purity:98%Color and Shape:SolidMolecular weight:592.06MK-0557
CAS:MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).Formula:C22H19FN4O3Purity:99.88%Color and Shape:SolidMolecular weight:406.41Ref: TM-TQ0286
1mg35.00€5mg71.00€10mg97.00€25mg170.00€50mg279.00€100mg393.00€200mg547.00€1mL*10mM (DMSO)80.00€Butyrophenone
CAS:Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.Formula:C10H12OPurity:99.84%Color and Shape:Colourless To Yellow LiquidMolecular weight:148.2Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Formula:C46H60F3N13O12SPurity:98.49%Color and Shape:SolidMolecular weight:1076.12Ref: TM-T7627L
1mg54.00€2mg71.00€5mg92.00€10mg152.00€25mg324.00€50mg485.00€100mg620.00€200mg897.00€1mL*10mM (DMSO)202.00€Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C128H219N45O36SPurity:94.61%Color and Shape:SolidMolecular weight:2996.45Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonistFormula:C37H48F6N8O11Purity:98.54%Color and Shape:SolidMolecular weight:894.81Ref: TM-T7740
1mg48.00€2mg60.00€5mg86.00€10mg138.00€25mg274.00€50mg411.00€100mg607.00€1mL*10mM (DMSO)170.00€PACAP 1-38 acetate
PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), not VIP1.Purity:98.16%Color and Shape:LiquidMolecular weight:N/AHS024
CAS:HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.Formula:C58H79N19O10S2Purity:>99.99%Color and Shape:SolidMolecular weight:1266.5OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formula:C79H125N23O22Purity:98.52%Color and Shape:SolidMolecular weight:1748.98Ablukast
CAS:Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.Formula:C28H34O8Purity:98.58%Color and Shape:SolidMolecular weight:498.56Ref: TM-T26519
2mgTo inquire5mg77.00€10mg111.00€25mg212.00€50mg298.00€100mg404.00€1mL*10mM (DMSO)85.00€Ipsapirone hydrochloride
CAS:Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formula:C19H24ClN5O3SColor and Shape:SolidMolecular weight:437.94GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:447.354-Methylhistamine hydrochloride
CAS:Compound with imidazole ring & amine group; inhibits copper enzymes, affects gene expression.Formula:C6H12ClN3Purity:95%Color and Shape:SolidMolecular weight:161.633Ref: TM-T50049
1mg74.00€2mg96.00€5mg156.00€10mg225.00€25mg379.00€50mg568.00€100mg810.00€500mg1,644.00€1mL*10mM (DMSO)126.00€4F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49GSK2018682 HCl
CAS:GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.Formula:C22H22Cl2N4O4Color and Shape:SolidMolecular weight:477.34Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purity:99.39%Color and Shape:SolidMolecular weight:386.4Evatanepag sodium
CAS:Evatanepag (CP-533536), an EP2-specific PGE2 agonist, promotes bone growth and heals fractures in rats with a single dose.Formula:C25H27N2NaO5SColor and Shape:SolidMolecular weight:490.55Epinastine
CAS:Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.Formula:C16H15N3Purity:99.94%Color and Shape:SolidMolecular weight:249.31Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formula:C24H29ClN4O4Color and Shape:SolidMolecular weight:472.97
