GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Blarcamesine
CAS:Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.
Formula:C19H23NOPurity:99.87%Color and Shape:SolidMolecular weight:281.39Nomifensine maleate
CAS:Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
Formula:C20H22N2O4Purity:98.46%Color and Shape:SolidMolecular weight:354.4Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75Buserelin Acetate (57982-77-1 free base)
CAS:Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Formula:C62H90N16O15Purity:99.31% - 99.78%Color and Shape:SolidMolecular weight:1299.48SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formula:C21H21Cl3N4O2Color and Shape:SolidMolecular weight:467.781-(1-Naphthyl) piperazine hydrochloride
CAS:1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multipleFormula:C14H17ClN2Purity:98.27%Color and Shape:SolidMolecular weight:248.75HAEGTFTSDVSSYLE
HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.Formula:C71H103N17O28Purity:>99.99%Color and Shape:SolidMolecular weight:1642.71Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53CCR2 antagonist 4 hydrochloride
CAS:CCR2 antagonist 4 hydrochloride is a specific CCR2 antagonist (IC50s: 180 nM for CCR2b). It potently inhibits MCP-1-induced chemotaxis (IC50: 24 nM).Formula:C21H22Cl2F3N3O2Color and Shape:SolidMolecular weight:476.32CAY10444
CAS:CAY10444 is an S1P3 specific antagonist.Formula:C15H29NO2SPurity:99.15% - 99.61%Color and Shape:SolidMolecular weight:287.46Ref: TM-T23860
5mg44.00€10mg71.00€25mg137.00€50mg222.00€100mg371.00€200mg505.00€500mg795.00€1mL*10mM (DMSO)48.00€CYM-5520
CAS:CYM-5520 is a noncompetitive allosteric agonist of S1P2Formula:C21H19N3O2Purity:99.47%Color and Shape:SolidMolecular weight:345.39Ref: TM-T22703
1mg46.00€2mg60.00€5mg88.00€10mg135.00€25mg236.00€50mg354.00€100mg528.00€1mL*10mM (DMSO)98.00€ML 10302
CAS:ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formula:C15H21ClN2O3Color and Shape:SolidMolecular weight:312.79N-Cbz-DL-tryptophan
CAS:N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.Formula:C19H18N2O4Purity:99.97%Color and Shape:SolidMolecular weight:338.36Samelisant dihydrochloride
CAS:SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.Formula:C21H33Cl2N3O3Color and Shape:SolidMolecular weight:446.41Galnon TFA
CAS:Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).Formula:C42H47F3N4O8Purity:99.47%Color and Shape:SolidMolecular weight:792.84Ref: TM-T8559
1mg58.00€5mg116.00€10mg172.00€25mg281.00€50mg396.00€100mg537.00€200mg712.00€1mL*10mM (DMSO)86.00€CRT0273750
CAS:CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.Formula:C25H22ClF3N4O2Purity:99.91%Color and Shape:SolidMolecular weight:502.92Picotamide
CAS:Picotamide has anticoagulant and fibrinolytic properties.Formula:C21H20N4O3Purity:98.90%Color and Shape:SolidMolecular weight:376.41Ref: TM-T9153
1mg38.00€5mg92.00€10mg147.00€25mg241.00€50mg349.00€100mg479.00€200mg657.00€1mL*10mM (DMSO)94.00€Bevantolol
CAS:Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formula:C20H27NO4Color and Shape:SolidMolecular weight:345.43Lodoxamide
CAS:Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formula:C11H6ClN3O6Purity:99.13% - 99.96%Color and Shape:SolidMolecular weight:311.63Benorilate
CAS:Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formula:C17H15NO5Purity:98.39% - 99.85%Color and Shape:SolidMolecular weight:313.3
