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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • Dobutamine tartrate

    CAS:
    Dobutamine tartrate is a cardiotonic.
    Formula:C22H29NO9
    Color and Shape:Solid
    Molecular weight:451.472

    Ref: TM-T8149L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bimatoprost

    CAS:
    <p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>
    Formula:C25H37NO4
    Purity:98% - >99.99%
    Color and Shape:Crystalline Solid
    Molecular weight:415.57

    Ref: TM-T2538

    2mg
    35.00€
    5mg
    50.00€
    10mg
    80.00€
    25mg
    134.00€
    50mg
    230.00€
    100mg
    393.00€
    200mg
    577.00€
  • Fluorogestone acetate

    CAS:
    FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.
    Formula:C23H31FO5
    Purity:99.47%
    Color and Shape:Coa
    Molecular weight:406.49

    Ref: TM-T21335

    2mg
    47.00€
    5mg
    71.00€
    10mg
    101.00€
    25mg
    188.00€
    50mg
    276.00€
    100mg
    394.00€
    200mg
    520.00€
    1mL*10mM (DMSO)
    85.00€
  • Enprofylline

    CAS:
    Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.
    Formula:C8H10N4O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:194.19

    Ref: TM-T21389

    2mg
    44.00€
    5mg
    65.00€
    10mg
    93.00€
    25mg
    149.00€
    50mg
    226.00€
    100mg
    335.00€
    200mg
    465.00€
    1mL*10mM (DMSO)
    63.00€
  • Volinanserin

    CAS:
    Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.
    Formula:C22H28FNO3
    Purity:98.94% - 99.95%
    Color and Shape:Solid
    Molecular weight:373.46

    Ref: TM-T5389

    1mg
    42.00€
    5mg
    88.00€
    10mg
    124.00€
    25mg
    233.00€
    50mg
    301.00€
    100mg
    393.00€
    200mg
    560.00€
    1mL*10mM (DMSO)
    96.00€
  • Obestatin (rat) acetate


    Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).
    Formula:C114H174N34O31
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:2516.81

    Ref: TM-TP2279L

    1mg
    77.00€
    2mg
    97.00€
    5mg
    156.00€
    10mg
    225.00€
    25mg
    375.00€
    50mg
    535.00€
    100mg
    730.00€
    200mg
    938.00€
  • Sigma-LIGAND-1 hydrochloride

    CAS:
    Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.
    Formula:C27H34ClNO4
    Color and Shape:Solid
    Molecular weight:472.02

    Ref: TM-T63048

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Relugolix

    CAS:
    Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with
    Formula:C29H27F2N7O5S
    Purity:98.64% - 99.97%
    Color and Shape:Solid
    Molecular weight:623.63

    Ref: TM-T3630

    2mg
    42.00€
    5mg
    62.00€
    10mg
    87.00€
    25mg
    170.00€
    50mg
    264.00€
    100mg
    430.00€
    200mg
    618.00€
    1mL*10mM (DMSO)
    86.00€
  • Olcegepant

    CAS:
    Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4
    Formula:C38H47Br2N9O5
    Purity:96.08% - 97.24%
    Color and Shape:Solid
    Molecular weight:869.65

    Ref: TM-T12293L

    1mg
    37.00€
    5mg
    96.00€
    10mg
    136.00€
    25mg
    221.00€
    100mg
    487.00€
    1mL*10mM (DMSO)
    190.00€
  • Mini Gastrin I, human acetate


    Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.
    Formula:C76H103N15O28S
    Purity:99.35% - 99.82%
    Color and Shape:Solid
    Molecular weight:1706.78

    Ref: TM-TP1821L

    1mg
    77.00€
    5mg
    255.00€
    10mg
    410.00€
    25mg
    737.00€
    50mg
    990.00€
    100mg
    1,341.00€
    200mg
    1,800.00€
  • Exo1

    CAS:
    Exo1 is an inhibitor of the exocytic pathway
    Formula:C15H12FNO3
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:273.26

    Ref: TM-T4609

    10mg
    43.00€
    25mg
    81.00€
    50mg
    130.00€
    100mg
    177.00€
    1mL*10mM (DMSO)
    33.00€
  • Pemirolast

    CAS:
    Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.
    Formula:C10H8N6O
    Color and Shape:Solid
    Molecular weight:228.21

    Ref: TM-T60289

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bupranolol

    CAS:
    Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.
    Formula:C14H22ClNO2
    Purity:97.63%
    Color and Shape:Solid
    Molecular weight:271.78

    Ref: TM-T8580

    1mg
    52.00€
    5mg
    105.00€
    10mg
    159.00€
    25mg
    309.00€
    50mg
    440.00€
    100mg
    583.00€
    200mg
    785.00€
    1mL*10mM (DMSO)
    96.00€
  • Elagolix sodium

    CAS:
    Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
    Formula:C32H29F5N3NaO5
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:653.57

    Ref: TM-T5031

    2mg
    35.00€
    5mg
    52.00€
    10mg
    80.00€
    25mg
    144.00€
    50mg
    227.00€
    100mg
    359.00€
    200mg
    532.00€
    1mL*10mM (DMSO)
    74.00€
  • RO1138452

    CAS:
    RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).
    Formula:C19H23N3O
    Purity:97.01% - 99.34%
    Color and Shape:Solid
    Molecular weight:309.41

    Ref: TM-T4436

    1mg
    52.00€
    2mg
    69.00€
    5mg
    96.00€
    10mg
    153.00€
    25mg
    329.00€
    50mg
    567.00€
    100mg
    810.00€
    1mL*10mM (DMSO)
    96.00€
  • Pimavanserin

    CAS:
    Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.
    Formula:C25H34FN3O2
    Purity:97.84% - 99.69%
    Color and Shape:Pale Yellow To Pale Orange Solid
    Molecular weight:427.55

    Ref: TM-T2076

    25mg
    52.00€
    50mg
    74.00€
    100mg
    106.00€
    1mL*10mM (DMSO)
    34.00€
  • Piperacetazine

    CAS:
    Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.
    Formula:C24H30N2O2S
    Purity:99.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.57

    Ref: TM-T3085

    2mg
    42.00€
    5mg
    62.00€
    10mg
    86.00€
    25mg
    130.00€
    50mg
    187.00€
    100mg
    283.00€
    1mL*10mM (DMSO)
    67.00€
  • Quipazine maleate

    CAS:
    Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.
    Formula:C17H19N3O4
    Color and Shape:Solid
    Molecular weight:329.356

    Ref: TM-T71792

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • TRAP-6

    CAS:
    TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
    Formula:C34H56N10O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:748.87

    Ref: TM-T7625

    1mg
    40.00€
    2mg
    52.00€
    5mg
    88.00€
    10mg
    126.00€
    25mg
    274.00€
    50mg
    411.00€
    100mg
    550.00€
    200mg
    785.00€
    1mL*10mM (DMSO)
    126.00€
  • Atrasentan sodium

    CAS:
    Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.
    Formula:C29H37N2NaO6
    Color and Shape:Solid
    Molecular weight:532.61

    Ref: TM-T70198

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€