
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Dobutamine tartrate
CAS:Dobutamine tartrate is a cardiotonic.Formula:C22H29NO9Color and Shape:SolidMolecular weight:451.472Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Formula:C25H37NO4Purity:98% - >99.99%Color and Shape:Crystalline SolidMolecular weight:415.57Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formula:C23H31FO5Purity:99.47%Color and Shape:CoaMolecular weight:406.49Ref: TM-T21335
2mg47.00€5mg71.00€10mg101.00€25mg188.00€50mg276.00€100mg394.00€200mg520.00€1mL*10mM (DMSO)85.00€Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Ref: TM-T21389
2mg44.00€5mg65.00€10mg93.00€25mg149.00€50mg226.00€100mg335.00€200mg465.00€1mL*10mM (DMSO)63.00€Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Ref: TM-T5389
1mg42.00€5mg88.00€10mg124.00€25mg233.00€50mg301.00€100mg393.00€200mg560.00€1mL*10mM (DMSO)96.00€Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formula:C114H174N34O31Purity:99.05%Color and Shape:SolidMolecular weight:2516.81Ref: TM-TP2279L
1mg77.00€2mg97.00€5mg156.00€10mg225.00€25mg375.00€50mg535.00€100mg730.00€200mg938.00€Sigma-LIGAND-1 hydrochloride
CAS:Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurity:98.64% - 99.97%Color and Shape:SolidMolecular weight:623.63Ref: TM-T3630
2mg42.00€5mg62.00€10mg87.00€25mg170.00€50mg264.00€100mg430.00€200mg618.00€1mL*10mM (DMSO)86.00€Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formula:C76H103N15O28SPurity:99.35% - 99.82%Color and Shape:SolidMolecular weight:1706.78Exo1
CAS:Exo1 is an inhibitor of the exocytic pathwayFormula:C15H12FNO3Purity:98.75%Color and Shape:SolidMolecular weight:273.26Pemirolast
CAS:Pemirolast: oral antiallergic, reduces paclitaxel reactions, inhibits neuropeptides, for asthma and conjunctivitis study.Formula:C10H8N6OColor and Shape:SolidMolecular weight:228.21Bupranolol
CAS:Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.Formula:C14H22ClNO2Purity:97.63%Color and Shape:SolidMolecular weight:271.78Ref: TM-T8580
1mg52.00€5mg105.00€10mg159.00€25mg309.00€50mg440.00€100mg583.00€200mg785.00€1mL*10mM (DMSO)96.00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Ref: TM-T5031
2mg35.00€5mg52.00€10mg80.00€25mg144.00€50mg227.00€100mg359.00€200mg532.00€1mL*10mM (DMSO)74.00€RO1138452
CAS:RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).Formula:C19H23N3OPurity:97.01% - 99.34%Color and Shape:SolidMolecular weight:309.41Ref: TM-T4436
1mg52.00€2mg69.00€5mg96.00€10mg153.00€25mg329.00€50mg567.00€100mg810.00€1mL*10mM (DMSO)96.00€Pimavanserin
CAS:Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formula:C25H34FN3O2Purity:97.84% - 99.69%Color and Shape:Pale Yellow To Pale Orange SolidMolecular weight:427.55Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formula:C24H30N2O2SPurity:99.9% - 99.92%Color and Shape:SolidMolecular weight:410.57Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formula:C17H19N3O4Color and Shape:SolidMolecular weight:329.356TRAP-6
CAS:TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).Formula:C34H56N10O9Purity:>99.99%Color and Shape:SolidMolecular weight:748.87Ref: TM-T7625
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg274.00€50mg411.00€100mg550.00€200mg785.00€1mL*10mM (DMSO)126.00€Atrasentan sodium
CAS:Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.Formula:C29H37N2NaO6Color and Shape:SolidMolecular weight:532.61
