GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Bilastine
CAS:Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration ofFormula:C28H37N3O3Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:463.616-fluoro-DL-Tryptophan
CAS:6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formula:C11H11FN2O2Purity:99.25%Color and Shape:Off-White PowderMolecular weight:222.22Pranlukast hemihydrate
CAS:Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.Formula:C27H23N5O40·5H2OPurity:99.28%Color and Shape:SolidMolecular weight:490.52MK 212 hydrochloride
CAS:MK 212 hydrochloride is a 5-HT2C receptor agonistFormula:C8H11ClN4·HClPurity:99.88%Color and Shape:SolidMolecular weight:235.12carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.
Formula:C24H31N3O2SPurity:98.06%Color and Shape:SolidMolecular weight:425.59Plecanatide
CAS:Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.Formula:C65H104N18O26S4Purity:97.51%Color and Shape:SolidMolecular weight:1681.89HS 014 acetate(207678-81-7 free base)
HS 014 acetate is a potent MC4R antagonist with Ki: 3.16 nM (MC4), and boosts food intake and nociception in animals.Formula:C73H98N20O19S2Purity:>99.99%Color and Shape:SolidMolecular weight:1623.83Sertindole
CAS:Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).
Formula:C24H26ClFN4OPurity:99.87% - 99.92%Color and Shape:Off-White To Pale Yellow SolidMolecular weight:440.94Ipsapirone hydrochloride
CAS:Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formula:C19H24ClN5O3SColor and Shape:SolidMolecular weight:437.94GLPG2938
CAS:GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent andFormula:C20H19F6N7O2Purity:98.25%Color and Shape:SolidMolecular weight:503.4Ref: TM-T9199
1mg84.00€2mg97.00€5mg144.00€10mg250.00€25mg550.00€50mg792.00€100mg1,093.00€1mL*10mM (DMSO)160.00€Donitriptan Mesylate
CAS:Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.Formula:C24H29N5O5SColor and Shape:SolidMolecular weight:499.58Bucindolol hydrochloride
CAS:Bucindolol, a 4th-gen β-blocker, prevents onset AF; effectiveness varies with β₁/α(2c) genes; best in β₁389 Arg homozygotes.Formula:C22H26ClN3O2Color and Shape:SolidMolecular weight:399.91Dioxopromethazine hydrochloride
CAS:Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.Formula:C17H20N2O2S·HClPurity:99.58%Color and Shape:SolidMolecular weight:352.88Albiglutide TFA (782500-75-8 free base)
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
Formula:C150H225F3N40O47Purity:>99.99%Color and Shape:SolidMolecular weight:3397.63Jatrorrhizine
CAS:Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formula:C20H20NO4Purity:97.18% - 99.06%Color and Shape:SolidMolecular weight:338.38Talastine HCl
CAS:Talastine is an antihistamine drug.Formula:C19H22ClN3OPurity:98%Color and Shape:SolidMolecular weight:343.86LY 78335
CAS:LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.Formula:C8H10Cl3NPurity:99.30% - 99.81%Color and Shape:SolidMolecular weight:226.539-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.37%Color and Shape:SolidMolecular weight:163.18TS-011
CAS:N-(3-Chloro-4-morpholinophenyl)-N'-hydroxyformimidamide (TS-011) is a selective 20-Hydroxyeicosatetraenoic acid synthesis inhibitor.Formula:C11H14ClN3O2Purity:99.48%Color and Shape:SolidMolecular weight:255.72-ATHBI
CAS:2-ATHBI is a S1P lyase inhibitor.Formula:C9H14N2O5Purity:99.10%Color and Shape:SolidMolecular weight:230.22
