GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(444 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
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Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Formula:C19H16F3N3O3Purity:99.33% - 99.8%Color and Shape:SolidMolecular weight:391.34Ref: TM-T16999
1mg81.00€5mg170.00€10mg274.00€25mg502.00€50mg705.00€100mg938.00€1mL*10mM (DMSO)188.00€ICI 118,551 hydrochloride
CAS:ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3Formula:C17H28ClNO2Purity:99.296% - 99.76%Color and Shape:SolidMolecular weight:313.86ARN272
CAS:ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formula:C27H20N4O2Purity:98.23%Color and Shape:SolidMolecular weight:432.47Exenatide
CAS:Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.Formula:C186H286N50O62SPurity:99.42%Color and Shape:SolidMolecular weight:4247Talnetant
CAS:Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.Formula:C25H22N2O2Purity:97.88%Color and Shape:SolidMolecular weight:382.45Ref: TM-T7549
1mg43.00€2mg56.00€5mg92.00€10mg130.00€25mg265.00€50mg490.00€100mg743.00€1mL*10mM (DMSO)142.00€Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formula:C17H25N3O5SPurity:99.65%Color and Shape:SolidMolecular weight:383.46Canagliflozin
CAS:Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.Formula:C24H25FO5SPurity:98.01% - >99.99%Color and Shape:SolidMolecular weight:444.52Ref: TM-T1782
2mg35.00€5mg50.00€10mg66.00€25mg87.00€50mg96.00€100mg123.00€500mg274.00€1mL*10mM (DMSO)52.00€Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83Gastrin I (human) acetate
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (Formula:C99H128N20O33SPurity:98.84%Color and Shape:SolidMolecular weight:2158.25CYM2503
CAS:<p>CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.</p>Formula:C45H55N5O7Purity:97.04%Color and Shape:SolidMolecular weight:777.95Bindarit
CAS:Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.Formula:C19H20N2O3Purity:98.35% - 98.55%Color and Shape:SolidMolecular weight:324.37Ref: TM-T6413
1mg38.00€2mg49.00€5mg80.00€10mg116.00€25mg188.00€50mg330.00€100mg520.00€200mgTo inquire1mL*10mM (DMSO)88.00€Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C145H240N44O48S2Purity:99.29%Color and Shape:SolidMolecular weight:3431.85VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35Ref: TM-T29112
1mg51.00€5mg92.00€10mg131.00€25mg235.00€50mg325.00€100mg462.00€200mg625.00€1mL*10mM (DMSO)94.00€Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormula:C43H77N17O12S2Purity:99.79%Color and Shape:SolidMolecular weight:1088.32Vercirnon sodium
CAS:Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.Formula:C22H21ClN2NaO4SColor and Shape:SolidMolecular weight:467.92[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formula:C69H108N22O16SPurity:99.71%Color and Shape:SolidMolecular weight:1533.8Talnetant hydrochloride
CAS:Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.Formula:C25H23ClN2O2Color and Shape:SolidMolecular weight:418.92Tiprenolol
CAS:Tiprenolol is a beta adrenergic receptor antagonist.[1]Formula:C13H21NO2SPurity:99.43%Color and Shape:SolidMolecular weight:255.38Ref: TM-T50081
1mg50.00€5mg103.00€10mg155.00€25mg248.00€50mg338.00€100mg472.00€200mg620.00€1mL*10mM (DMSO)95.00€AZD-4818
CAS:AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.Formula:C27H32Cl2N2O7Purity:99.01%Color and Shape:SolidMolecular weight:567.46
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