GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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JNJ-31020028
CAS:JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68ML-031
CAS:ML-031 activated S1P2 with an EC50 value of 1 μM in an S1P reporter assay.Formula:C19H20N2O3Purity:99.21%Color and Shape:SolidMolecular weight:324.37CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formula:C154H256N44O44Purity:97.29%Color and Shape:SolidMolecular weight:3428.01Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Formula:C19H16F2N8O2Purity:98.86% - 99.93%Color and Shape:SolidMolecular weight:426.38PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein ProSAAS, is an endogenous ligand of GPR83.Formula:C99H163N27O34Purity:99.25%Color and Shape:SolidMolecular weight:2275.51Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formula:C24H29ClN4O4Color and Shape:SolidMolecular weight:472.97ACTH 11-24 acetate(4237-93-8 free base)
CAS:ACTH 11-24 acetate is a cortisol-stimulating adrenocorticotrophin fragment and a competitive antagonist of ACTH 1-39 and 1-10.Formula:C79H138N24O18Purity:>99.99%Color and Shape:SolidMolecular weight:1712.12CYM 50358 hydrochloride (1314212-39-9 free base)
CAS:CYM50358 HCl is an S1P4 antagonist.Formula:C20H19Cl3N2O2Purity:99.57%Color and Shape:SolidMolecular weight:425.73Laropiprant sodium
Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.Color and Shape:SolidPNU 22394 hydrochloride
CAS:PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonistFormula:C13H17ClN2Purity:97.83%Color and Shape:SolidMolecular weight:236.74ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Formula:C129H207N45O41S3Purity:98.24%Color and Shape:SolidMolecular weight:3140.5Ref: TM-TP1220L
1mg185.00€5mg459.00€10mg657.00€25mg1,026.00€50mg1,388.00€100mg1,872.00€200mg2,527.00€BAR501
CAS:BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。Formula:C26H46O3Purity:99.29% - 99.68%Color and Shape:SolidMolecular weight:406.64Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88Alosetron (Hydrochloride(1:X))
CAS:Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.Formula:C17H18ClN4OColor and Shape:SolidMolecular weight:329.11691TG6-10-1
CAS:TG6-10-1 is an EP2 antagonist.Formula:C23H23F3N2O4Purity:99.66% - ≥95%Color and Shape:SolidMolecular weight:448.43Bindarit
CAS:Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.Formula:C19H20N2O3Purity:98.35% - 98.55%Color and Shape:SolidMolecular weight:324.37Ref: TM-T6413
1mg38.00€2mg49.00€5mg80.00€10mg116.00€25mg188.00€50mg330.00€100mg520.00€200mgTo inquire1mL*10mM (DMSO)88.00€CID 16020046
CAS:<p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>Formula:C25H19N3O4Purity:99.03%Color and Shape:SolidMolecular weight:425.44Puerarin
CAS:Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.Formula:C21H20O9Purity:98.90% - 99.21%Color and Shape:Yellow Brown Fine PowderMolecular weight:416.38Evatanepag sodium
CAS:Evatanepag (CP-533536), an EP2-specific PGE2 agonist, promotes bone growth and heals fractures in rats with a single dose.Formula:C25H27N2NaO5SColor and Shape:SolidMolecular weight:490.55Betaxolol
CAS:Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formula:C18H29NO3Purity:99.01%Color and Shape:White Crystalline SolidMolecular weight:307.43
