GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32CGP 71683 (free base)
CAS:CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formula:C26H29N5O2SColor and Shape:SolidMolecular weight:475.61Moxilubant
CAS:Moxilubant, a small molecule, blocks LTB4R to treat immune, skin, and joint disorders, may help in psoriasis and rheumatoid arthritis research.Formula:C26H37N3O4Purity:98%Color and Shape:SolidMolecular weight:455.59SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Formula:C10H14ClNColor and Shape:SolidMolecular weight:183.68Pizuglanstat
CAS:Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formula:C27H36N6O4Purity:99.62%Color and Shape:SolidMolecular weight:508.61SB-423562 HCl
CAS:SB-423562 is a calcium-sensing receptor antagonist.Formula:C26H33ClN2O4Purity:98%Color and Shape:SolidMolecular weight:473Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColor and Shape:SolidMolecular weight:228.74CID 1375606
CAS:CID 1375606: Surrogate agonist for GPR27, conserved in vertebrates, mainly in CNS.Formula:C20H14Cl2N2O2Purity:99.41%Color and Shape:SolidMolecular weight:385.24TFLLR-NH2 2TFA(197794-83-5(free base))
TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).Formula:C35H55F6N9O10Purity:99.56%Color and Shape:SolidMolecular weight:875.87Isoetharine mesylate salt
CAS:Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42GSK2018682 HCl
CAS:GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.Formula:C22H22Cl2N4O4Color and Shape:SolidMolecular weight:477.34Landiolol hydrochloride
CAS:Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05[Pyr1]-Apelin-13
CAS:[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.Formula:C69H108N22O16SPurity:99.71%Color and Shape:SolidMolecular weight:1533.8VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35Ref: TM-T29112
1mg49.00€5mg96.00€10mg124.00€25mg222.00€50mg309.00€100mg439.00€200mg592.00€1mL*10mM (DMSO)88.00€BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Ref: TM-T8512
1mg84.00€5mg161.00€10mg235.00€25mg420.00€50mg605.00€100mg842.00€200mg1,134.00€1mL*10mM (DMSO)172.00€[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C77H118N22O20Purity:98.41% - 99.14%Color and Shape:SolidMolecular weight:1671.9Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purity:99.83% - 99.97%Color and Shape:SolidMolecular weight:403.52BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.Formula:C118H190N36O30S2Purity:96.86%Color and Shape:SolidMolecular weight:2657.12CGP71683 hydrochloride
CAS:CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).Formula:C26H30ClN5O2SPurity:99.92%Color and Shape:SolidMolecular weight:512.07ZK 756326
CAS:ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formula:C21H28N2O3Purity:99.43%Color and Shape:SolidMolecular weight:356.46
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