GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5960 products of "GPCR/G-Protein"
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Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purity:98.1%Color and Shape:SolidMolecular weight:1269.45Nelociguat
CAS:Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formula:C19H17FN8O2Purity:99.19%Color and Shape:SolidMolecular weight:408.39Neurokinin A
CAS:Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.Formula:C50H80N14O14SPurity:>99.99%Color and Shape:White To Off-White Lyophilized SolidMolecular weight:1133.32Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formula:C8H11N5Purity:99.54%Color and Shape:SolidMolecular weight:177.21Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and
Formula:C52H77N13O13Purity:99.93%Color and Shape:SolidMolecular weight:1092.27I-191
CAS:I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formula:C23H26FN5O2Purity:99.8%Color and Shape:SolidMolecular weight:423.48Diquafosol tetrasodium
CAS:Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormula:C18H22N4Na4O23P4Purity:98.25% - 99.97%Color and Shape:SolidMolecular weight:878.23CAY10526
CAS:CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formula:C12H7BrO3SPurity:98.75%Color and Shape:SolidMolecular weight:311.15Velneperit
CAS:Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.Formula:C17H24F3N3O3SPurity:99.70%Color and Shape:SolidMolecular weight:407.45Ref: TM-T17222
1mg34.00€2mg49.00€5mg74.00€10mg113.00€25mg245.00€50mg416.00€100mg613.00€1mL*10mM (DMSO)82.00€Hemokinin 1 (human) acetate(491851-53-7 free base)
Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.Formula:C56H88N14O16SPurity:97.82%Color and Shape:SolidMolecular weight:1245.45Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formula:C18H20N4Purity:99.15% - 99.82%Color and Shape:SolidMolecular weight:292.38Plecanatide
CAS:Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.Formula:C65H104N18O26S4Purity:97.51%Color and Shape:SolidMolecular weight:1681.89Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purity:99.33%Color and Shape:SolidMolecular weight:354.27TY-52156
CAS:TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).Formula:C18H19Cl2N3OPurity:99.91% - 99.91%Color and Shape:SolidMolecular weight:364.27Ref: TM-T17183
2mg40.00€5mg60.00€10mg87.00€25mg166.00€50mg298.00€100mg510.00€200mg683.00€1mL*10mM (DMSO)66.00€BD-1047 dihydrobromide
CAS:BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormula:C13H22Br2Cl2N2Purity:98.13% - 99.39%Color and Shape:SolidMolecular weight:437.04Ref: TM-T1740
1mg37.00€2mg48.00€5mg73.00€10mg95.00€25mg168.00€50mg290.00€100mg490.00€1mL*10mM (DMSO)74.00€Amperozide
CAS:Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formula:C23H29F2N3OPurity:99.68%Color and Shape:SolidMolecular weight:401.49Ref: TM-T23733
1mg87.00€5mg178.00€10mg295.00€25mg497.00€50mg708.00€100mg964.00€500mg1,918.00€1mL*10mM (DMSO)321.00€Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formula:C35H47FN10O8Purity:97.97%Color and Shape:SolidMolecular weight:754.85Carazolol
CAS:Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.Formula:C18H22N2O2Purity:99% - 99.53%Color and Shape:Yellowish SolidMolecular weight:298.38L-732138
CAS:L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)Formula:C22H18F6N2O3Purity:99.77%Color and Shape:SolidMolecular weight:472.38Ref: TM-T8235
5mg50.00€10mg80.00€25mg135.00€50mg192.00€100mg286.00€200mg416.00€1mL*10mM (DMSO)To inquireIndophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formula:C19H15BrClF3N2O3SPurity:99.76%Color and Shape:SolidMolecular weight:523.75Ref: TM-T8946
1mg42.00€5mg82.00€10mg116.00€25mg188.00€50mg260.00€100mg366.00€200mg497.00€1mL*10mM (DMSO)95.00€
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