GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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Tripelennamine
CAS:Tripelennamine: ethylenediamine derivative, H1-receptor blocker, reduces allergic reactions, treats rhinitis and conjunctivitis.Formula:C16H21N3Color and Shape:SolidMolecular weight:255.36CYM-5520
CAS:CYM-5520 is a noncompetitive allosteric agonist of S1P2Formula:C21H19N3O2Purity:99.47%Color and Shape:SolidMolecular weight:345.39Ref: TM-T22703
1mg46.00€2mg60.00€5mg88.00€10mg135.00€25mg236.00€50mg354.00€100mg528.00€1mL*10mM (DMSO)98.00€Cloprostenol sodium salt
CAS:Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.Formula:C22H28ClNaO6Purity:97.17% - 98.47%Color and Shape:White To Almost White Hygroscopic PowderMolecular weight:446.9Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formula:C17H25N3O5SPurity:99.65%Color and Shape:SolidMolecular weight:383.46Ablukast
CAS:Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.Formula:C28H34O8Purity:98.58%Color and Shape:SolidMolecular weight:498.56[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purity:97.68%Color and Shape:SolidMolecular weight:1576.91Ambrisentan sodium
CAS:Ambrosentan (BSF 208075) sodium is a selective and oral effective antagonist of ET type A receptor ( ETAR ).Formula:C22H21N2NaO4Color and Shape:SolidMolecular weight:400.41TCS 1102
CAS:TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).Formula:C27H26N4O2SPurity:99.35% - 99.52%Color and Shape:SolidMolecular weight:470.59Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formula:C32H51F3N8O9Purity:99.88%Color and Shape:SolidMolecular weight:748.79Midodrine
CAS:Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.Formula:C12H18N2O4Purity:99.89%Color and Shape:SolidMolecular weight:254.28Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55Ipsapirone hydrochloride
CAS:Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formula:C19H24ClN5O3SColor and Shape:SolidMolecular weight:437.94LM11A-31 dihydrochloride
CAS:LM11A-31 dihydrochloride is a water-soluble, BBB-penetrating p75NTR ligand and proNGF antagonist.Formula:C12H27Cl2N3O2Purity:99.47% - 99.9%Color and Shape:SolidMolecular weight:316.27Praliciguat
CAS:Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.Formula:C21H14F8N6O2Purity:98.82%Color and Shape:SolidMolecular weight:534.36Ref: TM-T16569
1mg142.00€2mg207.00€5mg349.00€10mg537.00€25mg858.00€50mg1,161.00€100mg1,558.00€1mL*10mM (DMSO)409.00€Isoxsuprine Free Base
CAS:Isoxsuprine Free Base relaxes uterine/vascular muscles, dilates arteries, treats peripheral vascular disease, and premature labor.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12Ref: TM-T16980
2mg34.00€5mg49.00€10mg84.00€25mg114.00€50mg166.00€100mg236.00€200mg353.00€1mL*10mM (DMSO)54.00€Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purity:98.95% - 99.13%Color and Shape:SolidMolecular weight:269.73Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFormula:C21H28N2O2Purity:99.53%Color and Shape:White Or Similar To White PowderMolecular weight:340.46Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Ref: TM-T5389
1mg39.00€5mg84.00€10mg117.00€25mg220.00€50mg285.00€100mg371.00€200mg530.00€1mL*10mM (DMSO)92.00€
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1931L1.webp&w=3840&q=75)
