GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,024 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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GPR183-IN-1
CAS:GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.Formula:C16H19BrN2O2Color and Shape:SolidMolecular weight:351.24GLP-1 Receptor modulator 1
CAS:GLP-1 Receptormodulator 1 (Compound 7) is an effective positive allosteric modulator of the GLP-1 receptor. It is utilized in the research of obesity and type 2 diabetes.Formula:C18H21NOSMolecular weight:299.43PF-610355
CAS:PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.
Formula:C34H39N3O6SPurity:99.73%Color and Shape:SolidMolecular weight:617.76Risperidone Mesylate
CAS:Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formula:C24H31FN4O5SPurity:98%Color and Shape:SolidMolecular weight:506.59Rocatinlimab
CAS:Rocatinlimab (AMG 451) (KHK4083) is a fully human, non-fucosylated IgG1 anti-OX40 monoclonal antibody indicated for atopic dermatitis (AD) research [1].Color and Shape:LiquidMeticillin
CAS:Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.Formula:C17H20N2O6SColor and Shape:SolidMolecular weight:380.42Eptinezumab
CAS:Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
Purity:95% - 95%Color and Shape:LiquidTriflupromazine
CAS:Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.Formula:C18H19F3N2SColor and Shape:SolidMolecular weight:352.4217-phenyl trinor Prostaglandin F2α isopropyl ester
CAS:17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the AllerganFormula:C26H38O5Color and Shape:SolidMolecular weight:430.58Keto Ziprasidone
CAS:Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.Formula:C21H19ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:426.92Arazasetron HCl
CAS:Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.Formula:C17H20ClN3O3Purity:98%Color and Shape:SolidMolecular weight:349.81Tulobuterol
CAS:Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.Formula:C12H18ClNOColor and Shape:Crystalline SolidMolecular weight:227.73Fremanezumab
CAS:Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.Purity:95% - 97.6% (SDS-PAGE); 95.9% (SEC-HPLC)Color and Shape:LiquidMolecular weight:145.49 kDaBuflomedil
CAS:Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38Amitriptyline-d6 Hydrochloride
CAS:Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.Formula:C20H18D6ClNColor and Shape:SolidMolecular weight:319.9015-keto Prostaglandin F2α
CAS:15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.Formula:C20H32O5Purity:98%Color and Shape:SolidMolecular weight:352.47Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formula:C18H17D3N2Color and Shape:SolidMolecular weight:267.38Dapagliflozin-d5
CAS:Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Formula:C21H25ClO6Purity:98%Color and Shape:SolidMolecular weight:413.9Brexpiprazole-d8
CAS:Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.Formula:C25H27N3O2SPurity:98%Color and Shape:SolidMolecular weight:441.62Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purity:98%Color and Shape:SolidMolecular weight:268.37
