GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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6-hydroxy Buspirone
CAS:6-Hydroxy Buspirone, an active metabolite of the anxiolytic compound buspirone, is produced via the cytochrome P450 (CYP) isoform CYP3A4.Formula:C21H31N5O3Color and Shape:SolidMolecular weight:401.50Litorin
CAS:Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.Formula:C51H68N14O11SColor and Shape:White PowderMolecular weight:1085.24Ridazolol HCl
CAS:Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.Formula:C15H19Cl3N4O3Purity:99.48%Color and Shape:SoildMolecular weight:409.7AR244555
CAS:AR244555 is a bioactive chemical.Formula:C23H23ClF2N2OColor and Shape:SolidMolecular weight:416.897-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene
CAS:7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).Formula:C42H44N2O6SPurity:98%Color and Shape:SolidMolecular weight:704.87Atenolol Hydrochloride
CAS:Atenolol Hydrochloride is a selective antagonist of ß1 receptor.Formula:C14H23ClN2O3Purity:98%Color and Shape:SolidMolecular weight:302.80MCI-225 dehydratase
CAS:MCI-225 dehydratase is an oral, selective inhibitor of noradrenaline reuptake, and functions as a 5-HT3 antagonist, exhibiting antidepressant effects in vivo .Formula:C17H18ClFN4SColor and Shape:SolidMolecular weight:364.87SB 271046 hydrochloride
CAS:SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Formula:C20H22ClN3O3S2·HClPurity:99.77%Color and Shape:SolidMolecular weight:488.45Ticlopidine
CAS:Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.Formula:C14H14ClNSPurity:99.67%Color and Shape:SolidMolecular weight:263.797-Desmethyl-3-hydroxyagomelatine
CAS:7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formula:C14H15NO3Purity:98%Color and Shape:SolidMolecular weight:245.27Dolasetron Mesylate
CAS:Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormula:C20H24N2O6SPurity:99.05%Color and Shape:White PowderMolecular weight:420.48MK-5046
CAS:MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formula:C20H18F6N4OPurity:98.56%Color and Shape:SolidMolecular weight:444.37LY 344864
CAS:LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formula:C21H22FN3OPurity:98%Color and Shape:SolidMolecular weight:351.42Lodoxamide tromethamine
CAS:Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormula:C19H28ClN5O12Purity:98.8%Color and Shape:SolidMolecular weight:553.91Paroxetine hydrochloride hemihydrate
CAS:Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formula:C38H44Cl2F2N2O7Purity:99.949%Color and Shape:SolidMolecular weight:749.67Guacetisal
CAS:Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.
Formula:C16H14O5Purity:99.18%Color and Shape:SolidMolecular weight:286.28Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Formula:C25H31NOPurity:98%Color and Shape:SolidMolecular weight:361.52HSK0935
CAS:HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.Formula:C22H25ClO7Purity:98%Color and Shape:SolidMolecular weight:436.88Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
Formula:C19H23N5O3SPurity:99.51%Color and Shape:SolidMolecular weight:401.48N,N-Dimethylsphingosine
CAS:N,N-Dimethylsphingosine,is a potent competitive SphK phosphorylation inhibitor.DMS is elevated in models of neuropathic pain by increasing IL-1β and MCP-1.Formula:C20H41NO2Purity:98%Color and Shape:Clear Colorless To Faint Yellow Liquid/White To Off-White PowderMolecular weight:327.55
![7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT10189.webp&w=3840&q=75)
