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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • Orexin receptor antagonist 3

    CAS:
    Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist.
    Formula:C21H22N8O3
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T62453

    25mg
    1,459.00€
    50mg
    1,900.00€
    100mg
    2,690.00€
  • AGI-41998

    CAS:
    AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.
    Formula:C22H16BrF3N4O2
    Color and Shape:Solid
    Molecular weight:505.29

    Ref: TM-T9730

    25mg
    1,144.00€
    50mg
    1,485.00€
    100mg
    2,385.00€
  • DW-1350

    CAS:
    DW-1350 is an antagonist of LTB4 receptor.
    Formula:C25H31N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.6

    Ref: TM-T15182

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BMS-665053

    CAS:
    BMS-665053: CRF1 receptor antagonist, IC50 = 1.0 nM; inhibits cAMP in Y-79 cells, IC50 = 4.9 nM; anti-anxiety in rats, Cl = 17 mL/min/kg, t½ = 7.8 h.
    Formula:C16H14Cl3F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.66

    Ref: TM-T26855

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bifeprunox Mesylate

    CAS:
    Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.
    Formula:C25H27N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.56

    Ref: TM-T26807

    1mg
    114.00€
  • DMP 696

    CAS:
    DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.
    Formula:C18H21Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.3

    Ref: TM-T15145

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • IMTPPE

    CAS:
    IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.
    Formula:C20H27N3O2S
    Color and Shape:Solid
    Molecular weight:373.51

    Ref: TM-T27601

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OUP-186

    CAS:
    OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.
    Formula:C19H30ClN3S
    Color and Shape:Solid
    Molecular weight:367.98

    Ref: TM-T28275

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • FR 139317

    CAS:
    highly potent and selective ETA endothelin receptor antagonist
    Formula:C33H44N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.74

    Ref: TM-T22791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-trans-Prostaglandin E2

    CAS:
    5-trans-PGE2 speeds up fibrinolysis, boosts tissue-PA mediated plasminogen activation, and blocks platelet clumping in human PRP.
    Formula:C20H32O5
    Color and Shape:Solid
    Molecular weight:352.47

    Ref: TM-T71851

    1mg
    233.00€
    5mg
    1,035.00€
    10mg
    1,783.00€
  • SEP-363856

    CAS:
    SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.
    Formula:C9H13NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:183.27

    Ref: TM-T12899

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HEAT hydrochloride

    CAS:
    HEAT hydrochloride is an α1-adrenoceptor antagonist.
    Formula:C19H22ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.84

    Ref: TM-T22837

    10mg
    577.00€
  • S1P1 Agonist III

    CAS:
    S1P1 Agonist III is an orally active S1P1 receptor agonist (EC₅₀ = 18 nM) with applications in inflammation, immunology, and receptor signaling studies.
    Formula:C21H16F3N3O3
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:415.37

    Ref: TM-T16833

    1mg
    37.00€
    5mg
    72.00€
    1mL*10mM (DMSO)
    73.00€
    10mg
    92.00€
    25mg
    187.00€
    50mg
    309.00€
    100mg
    464.00€
  • A1AR antagonist 4

    CAS:
    Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.
    Formula:C23H25N3O2
    Color and Shape:Solid
    Molecular weight:375.46

    Ref: TM-T61536

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KUL-7211 racemate

    CAS:
    KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.
    Formula:C19H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.39

    Ref: TM-T11786

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY320135

    CAS:
    CB1 receptor antagonist/inverse agonist
    Formula:C24H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.4

    Ref: TM-T22951

    5mg
    325.00€
    10mg
    605.00€
  • TBC3711

    CAS:
    TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.
    Formula:C20H21N3O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.53

    Ref: TM-T15232

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 363

    CAS:
    RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.
    Formula:C19H25NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.4

    Ref: TM-T16769

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CCK-B Receptor Antagonist 1

    CAS:
    CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
    Formula:C28H30N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58

    Ref: TM-T13261

    2mg
    50.00€
  • TC-C 14G

    CAS:
    CB1 receptor inverse agonist
    Formula:C24H17Cl2F2NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:492.3

    Ref: TM-T23427

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€