
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Orexin receptor antagonist 3
CAS:Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45AGI-41998
CAS:AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.Formula:C22H16BrF3N4O2Color and Shape:SolidMolecular weight:505.29DW-1350
CAS:DW-1350 is an antagonist of LTB4 receptor.Formula:C25H31N3O3SPurity:98%Color and Shape:SolidMolecular weight:453.6BMS-665053
CAS:BMS-665053: CRF1 receptor antagonist, IC50 = 1.0 nM; inhibits cAMP in Y-79 cells, IC50 = 4.9 nM; anti-anxiety in rats, Cl = 17 mL/min/kg, t½ = 7.8 h.Formula:C16H14Cl3F2N3O2Purity:98%Color and Shape:SolidMolecular weight:424.66Bifeprunox Mesylate
CAS:Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.Formula:C25H27N3O5SPurity:98%Color and Shape:SolidMolecular weight:481.56DMP 696
CAS:DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.Formula:C18H21Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:410.3IMTPPE
CAS:IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.Formula:C20H27N3O2SColor and Shape:SolidMolecular weight:373.51OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Formula:C19H30ClN3SColor and Shape:SolidMolecular weight:367.98FR 139317
CAS:highly potent and selective ETA endothelin receptor antagonistFormula:C33H44N6O5Purity:98%Color and Shape:SolidMolecular weight:604.745-trans-Prostaglandin E2
CAS:5-trans-PGE2 speeds up fibrinolysis, boosts tissue-PA mediated plasminogen activation, and blocks platelet clumping in human PRP.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.47SEP-363856
CAS:SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.Formula:C9H13NOSPurity:98%Color and Shape:SolidMolecular weight:183.27HEAT hydrochloride
CAS:HEAT hydrochloride is an α1-adrenoceptor antagonist.Formula:C19H22ClNO2Purity:98%Color and Shape:SolidMolecular weight:331.84S1P1 Agonist III
CAS:S1P1 Agonist III is an orally active S1P1 receptor agonist (EC₅₀ = 18 nM) with applications in inflammation, immunology, and receptor signaling studies.Formula:C21H16F3N3O3Purity:99.08%Color and Shape:SolidMolecular weight:415.37A1AR antagonist 4
CAS:Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.Formula:C23H25N3O2Color and Shape:SolidMolecular weight:375.46KUL-7211 racemate
CAS:KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.Formula:C19H23NO5Purity:98%Color and Shape:SolidMolecular weight:345.39LY320135
CAS:CB1 receptor antagonist/inverse agonistFormula:C24H17NO4Purity:98%Color and Shape:SolidMolecular weight:383.4TBC3711
CAS:TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.Formula:C20H21N3O5S2Purity:98%Color and Shape:SolidMolecular weight:447.53Ro 363
CAS:RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.Formula:C19H25NO6Purity:98%Color and Shape:SolidMolecular weight:363.4CCK-B Receptor Antagonist 1
CAS:CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.Formula:C28H30N6O3Purity:98%Color and Shape:SolidMolecular weight:498.58TC-C 14G
CAS:CB1 receptor inverse agonistFormula:C24H17Cl2F2NO4Purity:98%Color and Shape:SolidMolecular weight:492.3
