
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
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GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purity:98%Color and Shape:SolidMolecular weight:308.37OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Formula:C19H30ClN3SColor and Shape:SolidMolecular weight:367.98Clenproperol
CAS:Clenproperol is a β2-adrenergic agonist.Formula:C11H16Cl2N2OColor and Shape:SolidMolecular weight:263.16Benzamide Derivative 1
CAS:Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.Formula:C22H34ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:423.98FR 139317
CAS:highly potent and selective ETA endothelin receptor antagonistFormula:C33H44N6O5Purity:98%Color and Shape:SolidMolecular weight:604.74E2508
CAS:E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.Formula:C36H47N3O7SPurity:98%Color and Shape:SolidMolecular weight:665.84JTC-017
CAS:JTC-017 is an antagonist of Corticotropin-releasing hormone receptor 1.Formula:C20H25Cl2N3O5SColor and Shape:SolidMolecular weight:490.4Denopamine
CAS:Denopamine is an agonist of 1-Adrenoceptor.Formula:C18H23NO4Color and Shape:SolidMolecular weight:317.38DR4485 hydrochloride
CAS:5-HT7 antagonistFormula:C26H29Cl3N2OPurity:98%Color and Shape:SolidMolecular weight:491.885-Methylurapidil
CAS:5-Methylurapidil is an alpha1A-adrenoceptor antagonist.Formula:C21H31N5O3Purity:98%Color and Shape:SolidMolecular weight:401.5Glucagon receptor antagonists-5
CAS:Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.Formula:C30H29ClF3N3O3Purity:98%Color and Shape:SolidMolecular weight:572.02(R)-Mequitazine
CAS:(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.Formula:C20H22N2SColor and Shape:SolidMolecular weight:322.47Ranitidine bismuth citrate
CAS:Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.Formula:C19H27BiN4O10SColor and Shape:SolidMolecular weight:712.48AF40431
CAS:AF40431 is the first reported small-molecule ligand of sortilin (IC50: 4.4 μM; Kd: 0.7 μM). AF40431 is bound in the neurotensin-binding site of sortilin.Formula:C17H21NO5Color and Shape:SolidMolecular weight:319.35Ro 363
CAS:RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.Formula:C19H25NO6Purity:98%Color and Shape:SolidMolecular weight:363.4MHP 133
CAS:MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).Formula:C17H20ClN5O3Purity:98%Color and Shape:SolidMolecular weight:377.83GB83
CAS:GB83 is a selective human protease activated receptor 2 (PAR2) antagonist.Formula:C32H44N4O4Purity:98%Color and Shape:SolidMolecular weight:548.72ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Formula:C22H22N2OPurity:99.94%Color and Shape:SolidMolecular weight:330.42Ref: TM-T14087
1mg44.00€1mL*10mM (DMSO)90.00€5mg93.00€10mg133.00€25mg270.00€50mg409.00€100mg595.00€200mg833.00€Zolantidine dimaleate
CAS:H2 receptor antagonistFormula:C26H31N3O5SPurity:98%Color and Shape:SolidMolecular weight:497.61GSK-894490A
CAS:GSK-894490A is an agonist of ghrelin receptor. GSK-894490A crosses the blood/brain barrier and elicit pro-cognitive effects.Formula:C24H30ClN3O4SColor and Shape:SolidMolecular weight:492.03
