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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5984 products of "GPCR/G-Protein"

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  • GTS-21

    CAS:
    GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.
    Formula:C19H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.37

    Ref: TM-T19933

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OUP-186

    CAS:
    OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.
    Formula:C19H30ClN3S
    Color and Shape:Solid
    Molecular weight:367.98

    Ref: TM-T28275

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Clenproperol

    CAS:
    Clenproperol is a β2-adrenergic agonist.
    Formula:C11H16Cl2N2O
    Color and Shape:Solid
    Molecular weight:263.16

    Ref: TM-T40480

    25mg
    1,369.00€
  • Benzamide Derivative 1

    CAS:
    Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.
    Formula:C22H34ClN3O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:423.98

    Ref: TM-T13570

    1mg
    630.00€
    5mg
    1,620.00€
  • FR 139317

    CAS:
    highly potent and selective ETA endothelin receptor antagonist
    Formula:C33H44N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.74

    Ref: TM-T22791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • E2508

    CAS:
    E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.
    Formula:C36H47N3O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:665.84

    Ref: TM-T27227

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JTC-017

    CAS:
    JTC-017 is an antagonist of Corticotropin-releasing hormone receptor 1.
    Formula:C20H25Cl2N3O5S
    Color and Shape:Solid
    Molecular weight:490.4

    Ref: TM-T24216

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Denopamine

    CAS:
    Denopamine is an agonist of 1-Adrenoceptor.
    Formula:C18H23NO4
    Color and Shape:Solid
    Molecular weight:317.38

    Ref: TM-T19707

    25mg
    973.00€
    50mg
    1,269.00€
    100mg
    1,998.00€
  • DR4485 hydrochloride

    CAS:
    5-HT7 antagonist
    Formula:C26H29Cl3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:491.88

    Ref: TM-T22750

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-Methylurapidil

    CAS:
    5-Methylurapidil is an alpha1A-adrenoceptor antagonist.
    Formula:C21H31N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.5

    Ref: TM-T26393

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucagon receptor antagonists-5

    CAS:
    Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.
    Formula:C30H29ClF3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:572.02

    Ref: TM-T11416

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Mequitazine

    CAS:
    (R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.
    Formula:C20H22N2S
    Color and Shape:Solid
    Molecular weight:322.47

    Ref: TM-T26373

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ranitidine bismuth citrate

    CAS:
    Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.
    Formula:C19H27BiN4O10S
    Color and Shape:Solid
    Molecular weight:712.48

    Ref: TM-T71059

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AF40431

    CAS:
    AF40431 is the first reported small-molecule ligand of sortilin (IC50: 4.4 μM; Kd: 0.7 μM). AF40431 is bound in the neurotensin-binding site of sortilin.
    Formula:C17H21NO5
    Color and Shape:Solid
    Molecular weight:319.35

    Ref: TM-T13530

    2mg
    217.00€
    5mg
    268.00€
    25mg
    888.00€
    50mg
    1,224.00€
    100mg
    1,674.00€
  • Ro 363

    CAS:
    RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.
    Formula:C19H25NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.4

    Ref: TM-T16769

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MHP 133

    CAS:
    MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
    Formula:C17H20ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.83

    Ref: TM-T13772

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GB83

    CAS:
    GB83 is a selective human protease activated receptor 2 (PAR2) antagonist.
    Formula:C32H44N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.72

    Ref: TM-T27406

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ABT-239

    CAS:
    ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.
    Formula:C22H22N2O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:330.42

    Ref: TM-T14087

    1mg
    44.00€
    1mL*10mM (DMSO)
    90.00€
    5mg
    93.00€
    10mg
    133.00€
    25mg
    270.00€
    50mg
    409.00€
    100mg
    595.00€
    200mg
    833.00€
  • Zolantidine dimaleate

    CAS:
    H2 receptor antagonist
    Formula:C26H31N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.61

    Ref: TM-T23565

    10mg
    705.00€
    50mg
    2,907.00€
  • GSK-894490A

    CAS:
    GSK-894490A is an agonist of ghrelin receptor. GSK-894490A crosses the blood/brain barrier and elicit pro-cognitive effects.
    Formula:C24H30ClN3O4S
    Color and Shape:Solid
    Molecular weight:492.03

    Ref: TM-T27493

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€