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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5984 products of "GPCR/G-Protein"

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  • C-021 dihydrochloride

    CAS:
    C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.
    Formula:C27H43Cl2N5O2
    Purity:98.67%
    Color and Shape:Solid
    Molecular weight:540.57

    Ref: TM-T10639

    1mg
    52.00€
    5mg
    97.00€
    1mL*10mM (DMSO)
    115.00€
    10mg
    154.00€
    25mg
    249.00€
    50mg
    374.00€
  • Calhex 231 hydrochloride

    CAS:
    Calhex 231 hydrochloride a potent CaSR negative-conversion modulator that blocks the increase in [3H]inositol phosphate, inhibits mir-208a-mediated .
    Formula:C25H28Cl2N2O
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:443.41

    Ref: TM-T10666

    25mg
    To inquire
    50mg
    To inquire
    1mg
    47.00€
    5mg
    92.00€
    1mL*10mM (DMSO)
    101.00€
    10mg
    152.00€
  • Dacopafant

    CAS:
    Dacopafant is an antagonist of platlet activationg factor receptor.
    Formula:C12H11N3OS
    Color and Shape:Solid
    Molecular weight:245.3

    Ref: TM-T23951

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BMS-466442

    CAS:
    BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.
    Formula:C31H30N4O5
    Color and Shape:Solid
    Molecular weight:538.59

    Ref: TM-T23806

    10mg
    884.00€
  • SNAP 5089

    CAS:
    α1A-adrenoceptor antagonist
    Formula:C36H40N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:608.73

    Ref: TM-T23374

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bopindolol (malonate)

    CAS:
    Bopindolol is a non-selective β-adrenergic receptor antagonist.
    Formula:C26H32N2O7
    Color and Shape:Solid
    Molecular weight:484.549

    Ref: TM-T35871

    100mg
    298.00€
    500mg
    1,035.00€
  • Phenindamine Tartrate

    CAS:
    Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.
    Formula:C23H25NO6
    Color and Shape:Solid
    Molecular weight:411.454

    Ref: TM-T33978

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Flestolol sulfate

    CAS:
    Flestolol sulfate is an anti-adrenergic beta-receptor.
    Formula:C15H24FN3O8S
    Color and Shape:Solid
    Molecular weight:425.43

    Ref: TM-T27332

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BRD5814

    CAS:
    BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.
    Formula:C21H23ClF3NO2
    Color and Shape:Solid
    Molecular weight:413.86

    Ref: TM-T70040

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AP-521 (Free base)

    CAS:
    AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.
    Formula:C20H18N2O3S
    Color and Shape:Solid
    Molecular weight:366.43

    Ref: TM-T26640

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CP19

    CAS:
    CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].
    Formula:C26H30N2O5
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T73571

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CB2R agonist 1

    CAS:
    CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.
    Formula:C22H32N2O
    Color and Shape:Solid
    Molecular weight:340.5

    Ref: TM-T72849

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Iodophenpropit dihydrobromide

    CAS:
    Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).
    Formula:C15H20BrIN4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:495.22

    Ref: TM-T15590

    5mg
    386.00€
    10mg
    577.00€
  • Ono 1301

    CAS:
    Ono 1301 mimics prostaglandin I2, inhibits thromboxane A2 synthase, reduces pancreatic fibrosis, and boosts cAMP via IP receptor.
    Formula:C26H24N2O4
    Color and Shape:Solid
    Molecular weight:428.48

    Ref: TM-T28240

    25mg
    690.00€
    50mg
    898.00€
    100mg
    1,566.00€
  • Latanoprost ethyl amide

    CAS:
    Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.
    Formula:C25H39NO4
    Color and Shape:Solid
    Molecular weight:417.58

    Ref: TM-T37627

    1mg
    239.00€
    5mg
    1,018.00€
    10mg
    1,783.00€
  • PPTN

    CAS:
    PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.
    Formula:C29H24F3NO2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:475.5

    Ref: TM-T12530

    1mg
    47.00€
    5mg
    92.00€
    10mg
    152.00€
    25mg
    289.00€
    50mg
    432.00€
    100mg
    618.00€
    200mg
    859.00€
  • CCX777

    CAS:
    CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer research.
    Formula:C31H43N7O3S
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:593.78

    Ref: TM-T23866

    1mg
    269.00€
  • CB1R Allosteric modulator 1

    CAS:
    CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.
    Formula:C24H24ClN3O
    Color and Shape:Solid
    Molecular weight:405.92

    Ref: TM-T62016

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CUMI-101

    CAS:
    CUMI-101 is an agonist of 5-HT1A receptor.
    Formula:C19H27N5O3
    Color and Shape:Solid
    Molecular weight:373.45

    Ref: TM-T27100

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Naronapride

    CAS:
    Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.
    Formula:C27H41ClN4O5
    Color and Shape:Solid
    Molecular weight:537.09

    Ref: TM-T63785

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€