
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
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C-021 dihydrochloride
CAS:C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.Formula:C27H43Cl2N5O2Purity:98.67%Color and Shape:SolidMolecular weight:540.57Calhex 231 hydrochloride
CAS:Calhex 231 hydrochloride a potent CaSR negative-conversion modulator that blocks the increase in [3H]inositol phosphate, inhibits mir-208a-mediated .Formula:C25H28Cl2N2OPurity:99.36%Color and Shape:SolidMolecular weight:443.41Dacopafant
CAS:Dacopafant is an antagonist of platlet activationg factor receptor.Formula:C12H11N3OSColor and Shape:SolidMolecular weight:245.3BMS-466442
CAS:BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.Formula:C31H30N4O5Color and Shape:SolidMolecular weight:538.59SNAP 5089
CAS:α1A-adrenoceptor antagonistFormula:C36H40N4O5Purity:98%Color and Shape:SolidMolecular weight:608.73Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Formula:C26H32N2O7Color and Shape:SolidMolecular weight:484.549Phenindamine Tartrate
CAS:Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.Formula:C23H25NO6Color and Shape:SolidMolecular weight:411.454Flestolol sulfate
CAS:Flestolol sulfate is an anti-adrenergic beta-receptor.Formula:C15H24FN3O8SColor and Shape:SolidMolecular weight:425.43BRD5814
CAS:BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.Formula:C21H23ClF3NO2Color and Shape:SolidMolecular weight:413.86AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Formula:C20H18N2O3SColor and Shape:SolidMolecular weight:366.43CP19
CAS:CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].Formula:C26H30N2O5Color and Shape:SolidMolecular weight:450.53CB2R agonist 1
CAS:CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.Formula:C22H32N2OColor and Shape:SolidMolecular weight:340.5Iodophenpropit dihydrobromide
CAS:Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).Formula:C15H20BrIN4SPurity:98%Color and Shape:SolidMolecular weight:495.22Ono 1301
CAS:Ono 1301 mimics prostaglandin I2, inhibits thromboxane A2 synthase, reduces pancreatic fibrosis, and boosts cAMP via IP receptor.Formula:C26H24N2O4Color and Shape:SolidMolecular weight:428.48Latanoprost ethyl amide
CAS:Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.Formula:C25H39NO4Color and Shape:SolidMolecular weight:417.58PPTN
CAS:PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.Formula:C29H24F3NO2Purity:99.86%Color and Shape:SolidMolecular weight:475.5CCX777
CAS:CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer research.Formula:C31H43N7O3SPurity:98.73%Color and Shape:SolidMolecular weight:593.78CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Formula:C24H24ClN3OColor and Shape:SolidMolecular weight:405.92CUMI-101
CAS:CUMI-101 is an agonist of 5-HT1A receptor.Formula:C19H27N5O3Color and Shape:SolidMolecular weight:373.45Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Color and Shape:SolidMolecular weight:537.09
