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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • Donitriptan

    CAS:

    Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。

    Formula:C23H25N5O2
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:403.48

    Ref: TM-T11075

    1mg
    56.00€
    2mg
    81.00€
    5mg
    119.00€
    10mg
    188.00€
    25mg
    432.00€
    50mg
    638.00€
  • Levoprotiline hydrochloride

    CAS:
    Levoprotiline hydrochloride is an antidepressant.
    Formula:C20H24ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.86

    Ref: TM-T27820

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tranterol hydrochloride

    CAS:
    Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.
    Formula:C13H19Cl2F3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:347.2

    Ref: TM-T29001

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JPC-211

    CAS:
    JPC-211 is an agonist of dopamine-receptor.
    Formula:C17H27NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.4

    Ref: TM-T27693

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PGD2-IN-1

    CAS:
    PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.
    Formula:C23H23Cl2N3O3
    Purity:98.21%
    Color and Shape:Solid
    Molecular weight:460.35

    Ref: TM-T4624

    1mg
    66.00€
    5mg
    150.00€
    1mL*10mM (DMSO)
    159.00€
    10mg
    245.00€
    25mg
    414.00€
    50mg
    610.00€
    100mg
    867.00€
    500mg
    1,738.00€
  • Captodiame

    CAS:
    Captodiame is an antihistamine agent.
    Formula:C21H29NS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.59

    Ref: TM-T23851

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NVP-QAV-680

    CAS:
    NVP-QAV-680: Powerful, selective CRTh2 antagonist with nM potency inhibiting eosinophil/Th2 activation.
    Formula:C18H18N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.41

    Ref: TM-T28221

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Felypressin acetate

    CAS:
    Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.
    Formula:C48H69N13O13S2
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:1100.27

    Ref: TM-T2568L

    5mg
    44.00€
    10mg
    66.00€
    25mg
    119.00€
    50mg
    177.00€
    100mg
    281.00€
    200mg
    421.00€
    500mg
    677.00€
  • Aminaftone

    CAS:
    Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.
    Formula:C18H15NO4
    Purity:96.31% - 99.39%
    Color and Shape:Solid
    Molecular weight:309.32

    Ref: TM-T14219

    1mg
    190.00€
    5mg
    523.00€
    10mg
    648.00€
    25mg
    858.00€
  • Tulopafant

    CAS:
    Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.
    Formula:C25H19N3O2S
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:425.5

    Ref: TM-T17178

    1mg
    630.00€
    5mg
    1,620.00€
  • A1AR antagonist 2

    CAS:
    Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.
    Formula:C17H12N4O
    Color and Shape:Solid
    Molecular weight:288.3

    Ref: TM-T60580

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Isoproterenol-d7 HCl

    CAS:
    Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.
    Formula:C11H18ClNO3
    Color and Shape:Solid
    Molecular weight:254.76

    Ref: TM-T69598

    1mg
    359.00€
  • Cicloprolol hydrochloride

    CAS:
    Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
    Formula:C18H30ClNO4
    Purity:97.26%
    Color and Shape:Solid
    Molecular weight:359.89

    Ref: TM-T10812

    1mg
    630.00€
    5mg
    1,620.00€
  • Bamirastine

    CAS:
    Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on
    Formula:C31H37N5O3
    Purity:96.68%
    Color and Shape:Solid
    Molecular weight:527.66

    Ref: TM-T13566

    1mg
    630.00€
    5mg
    1,620.00€
  • L-771688

    CAS:
    L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign
    Formula:C28H33F2N5O5
    Purity:94.15%
    Color and Shape:Solid
    Molecular weight:557.59

    Ref: TM-T15688

    1mg
    356.00€
    5mg
    888.00€
  • L-803087

    CAS:
    L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.
    Formula:C25H29F2N5O3
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:485.53

    Ref: TM-T11800

    1mg
    50.00€
    5mg
    112.00€
    1mL*10mM (DMSO)
    126.00€
    10mg
    175.00€
    25mg
    366.00€
    50mg
    585.00€
    100mg
    928.00€
    200mg
    1,234.00€
  • TD-5471 hydrochloride

    CAS:
    TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (
    Formula:C32H32ClN3O4
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:558.07

    Ref: TM-T13106

    1mg
    630.00€
    5mg
    1,333.00€
  • Napitane

    CAS:

    napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the

    Formula:C22H25NO2
    Purity:99.77% - 99.89%
    Color and Shape:Solid
    Molecular weight:335.44

    Ref: TM-T26363L

    1mg
    313.00€
    5mg
    758.00€
    10mg
    1,074.00€
    25mg
    1,644.00€
    50mg
    2,262.00€
    100mg
    2,945.00€
  • Daledalin tosylate

    CAS:
    Daledalin tosylate is an antidepressant.
    Formula:C26H32N2O3S
    Color and Shape:Solid
    Molecular weight:452.61

    Ref: TM-T31196

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Trebenzomine

    CAS:
    Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.
    Formula:C12H17NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:191.27

    Ref: TM-T29004

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€