
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Donitriptan
CAS:Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。
Formula:C23H25N5O2Purity:98.76%Color and Shape:SolidMolecular weight:403.48Levoprotiline hydrochloride
CAS:Levoprotiline hydrochloride is an antidepressant.Formula:C20H24ClNOPurity:98%Color and Shape:SolidMolecular weight:329.86Tranterol hydrochloride
CAS:Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.Formula:C13H19Cl2F3N2OPurity:98%Color and Shape:SolidMolecular weight:347.2JPC-211
CAS:JPC-211 is an agonist of dopamine-receptor.Formula:C17H27NO2Purity:98%Color and Shape:SolidMolecular weight:277.4PGD2-IN-1
CAS:PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit prostaglandin D2 (PGD2) signaling.Formula:C23H23Cl2N3O3Purity:98.21%Color and Shape:SolidMolecular weight:460.35Ref: TM-T4624
1mg66.00€5mg150.00€1mL*10mM (DMSO)159.00€10mg245.00€25mg414.00€50mg610.00€100mg867.00€500mg1,738.00€Captodiame
CAS:Captodiame is an antihistamine agent.Formula:C21H29NS2Purity:98%Color and Shape:SolidMolecular weight:359.59NVP-QAV-680
CAS:NVP-QAV-680: Powerful, selective CRTh2 antagonist with nM potency inhibiting eosinophil/Th2 activation.Formula:C18H18N2O4SPurity:98%Color and Shape:SolidMolecular weight:358.41Felypressin acetate
CAS:Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.Formula:C48H69N13O13S2Purity:97.06%Color and Shape:SolidMolecular weight:1100.27Aminaftone
CAS:Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.Formula:C18H15NO4Purity:96.31% - 99.39%Color and Shape:SolidMolecular weight:309.32Tulopafant
CAS:Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.Formula:C25H19N3O2SPurity:99.38%Color and Shape:SolidMolecular weight:425.5A1AR antagonist 2
CAS:Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.Formula:C17H12N4OColor and Shape:SolidMolecular weight:288.3Isoproterenol-d7 HCl
CAS:Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.Formula:C11H18ClNO3Color and Shape:SolidMolecular weight:254.76Cicloprolol hydrochloride
CAS:Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.Formula:C18H30ClNO4Purity:97.26%Color and Shape:SolidMolecular weight:359.89Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFormula:C31H37N5O3Purity:96.68%Color and Shape:SolidMolecular weight:527.66L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59L-803087
CAS:L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Formula:C25H29F2N5O3Purity:99.37%Color and Shape:SolidMolecular weight:485.53Ref: TM-T11800
1mg50.00€5mg112.00€1mL*10mM (DMSO)126.00€10mg175.00€25mg366.00€50mg585.00€100mg928.00€200mg1,234.00€TD-5471 hydrochloride
CAS:TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (Formula:C32H32ClN3O4Purity:99.57%Color and Shape:SolidMolecular weight:558.07Napitane
CAS:napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the
Formula:C22H25NO2Purity:99.77% - 99.89%Color and Shape:SolidMolecular weight:335.44Daledalin tosylate
CAS:Daledalin tosylate is an antidepressant.Formula:C26H32N2O3SColor and Shape:SolidMolecular weight:452.61Trebenzomine
CAS:Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.Formula:C12H17NOPurity:98%Color and Shape:SolidMolecular weight:191.27
